Pyrrolin-2-ylamino compounds for combating animal pests
    53.
    发明授权
    Pyrrolin-2-ylamino compounds for combating animal pests 失效
    用于对抗动物害虫的吡咯啉-2-基氨基化合物

    公开(公告)号:US08221775B2

    公开(公告)日:2012-07-17

    申请号:US13062531

    申请日:2009-09-08

    CPC分类号: C07D207/22 C07D209/54

    摘要: The present invention relates to pyrrolin-2-ylamino compounds for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to plant propagation material and to an agricultural composition comprising said compounds. The invention also relates to a method for treating or protecting an animal from infestation or infection by parasites by using said compounds: wherein: A is a radical of the formulae A.1 or A.2: n, m, R1, R2, R3, R4, R5a, R5b, R5c, R5d, R5e, and R5f are defined herein.

    摘要翻译: 本发明涉及用于对抗动物害虫的吡咯啉-2-基氨基化合物。 本发明还涉及通过使用这些化合物,植物繁殖材料和包含所述化合物的农业组合物来控制动物害虫的方法。 本发明还涉及通过使用所述化合物来治疗或保护动物免受寄生虫感染或感染的方法:其中:A是式A.1或A.2的基团:n,m,R1,R2,R3 ,R4,R5a,R5b,R5c,R5d,R5e和R5f如本文所定义。

    Pesticidal active mixtures comprising aminothiazoline compounds
    54.
    发明授权
    Pesticidal active mixtures comprising aminothiazoline compounds 失效
    包含氨基噻唑啉化合物的杀虫活性混合物

    公开(公告)号:US08153560B2

    公开(公告)日:2012-04-10

    申请号:US12528686

    申请日:2008-02-22

    IPC分类号: A01N43/78 C07D277/04

    摘要: Pesticidal mixtures comprising aminothiazoline compounds The present invention relates to pesticidal mixtures comprising as active compounds 1) at least one aminothiazoline compound I of the Formula (I) wherein R1, R2, R3, R4, R5 and R6 are defined in the description; and 2) at least one active compound II selected from a group A comprising acetylcholine esterase inhibitors, GABA-gated chloride channel antagonists, sodium channel modulators, nicotinic acetylcholine receptor agonists/antagonists, chloride channel activators, juvenile hormone mimics, compounds affecting the oxidative phosphorylation, inhibitors of the chitin biosynthesis, moulting disruptors, inhibitors of the MET, voltage-dependent sodium channel blockers, inhibitors of the lipidsynthesis and other compounds as defined in the description, in synergistically effective amounts. The invention relates further to methods and use of these mixtures for combating insects, arachnids or nematodes in and on plants, and for protecting such plants being infested with pests, especially also for protecting seeds.

    摘要翻译: 包含氨基噻唑啉化合物的杀虫混合物本发明涉及包含作为活性化合物的杀虫混合物1)至少一种式(I)的氨基噻唑啉化合物I,其中R 1,R 2,R 3,R 4,R 5和R 6在说明书中定义; 和2)选自包括乙酰胆碱酯酶抑制剂,GABA门控氯化物通道拮抗剂,钠通道调节剂,烟碱乙酰胆碱受体激动剂/拮抗剂,氯化物通道激活剂,幼年激素模拟物,影响氧化磷酸化的化合物的组A中的至少一种活性化合物II ,甲壳素生物合成抑制剂,蜕皮破坏剂,MET抑制剂,电压依赖性钠通道阻滞剂,脂质合成抑制剂和描述中定义的其它化合物,具有协同有效量。 本发明进一步涉及这些混合物用于防治植物中和植物上的昆虫,蜘蛛或线虫的方法和用途,并且还用于保护被害虫侵染的植物,特别是用于保护种子。

    Pyrrolin-2-ylamino Compounds For Combating Animal Pests
    55.
    发明申请
    Pyrrolin-2-ylamino Compounds For Combating Animal Pests 失效
    吡咯啉-2-基氨基化合物用于防治动物害虫

    公开(公告)号:US20110160269A1

    公开(公告)日:2011-06-30

    申请号:US13062531

    申请日:2009-09-08

    CPC分类号: C07D207/22 C07D209/54

    摘要: The present invention relates to pyrrolin-2-ylamino compounds for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to plant propagation material and to an agricultural composition comprising said compounds. The invention also relates to a method for treating or protecting an animal from infestation or infection by parasites by using said compounds. wherein n is 0, 1, 2, 3, 4 or 5; m is 0, 1, 2, 3, 4 or 5; R1, R2 are each independently selected from the group consisting of: halogen, CN, N3, NO2, C1-C6-alkyl, C2-C6-alkenyl and C2-C6-alkynyl, where the last 3 radicals mentioned may be partly or completely halogenated and/or may carry any combination of 1, 2 or 3 radicals R#, etc.; R3 and R4 are selected each independently of one another from hydrogen, halogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, wherein the last 3 radicals mentioned may be partly or completely halogenated and/or may carry any combination of 1, 2 or 3 radicals selected independently of one another from the group consisting of CN, NO2, —ORb, NRcRd, —SRe, —C(═O)Ra and —C(═O)ORb, etc.; A is a radical of the formulae A.1 or A.2, wherein * indicates the point of attachment to the remaining part of the compound; R5a, R5b, R5c, R5d, R5e and R5f are selected independently from one another from hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino, di(C1-C6-alkyl)amino, C3-C6-cycloalkyl and Ar2, etc.; R6 and R7 are selected each independently from one another from hydrogen, CN, NO2, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, saturated or partially unsaturated 5-, 6- or 7-membered heterocyclic radicals, Ar3, etc.

    摘要翻译: 本发明涉及用于对抗动物害虫的吡咯啉-2-基氨基化合物。 本发明还涉及通过使用这些化合物,植物繁殖材料和包含所述化合物的农业组合物来控制动物害虫的方法。 本发明还涉及通过使用所述化合物治疗或保护动物免受寄生虫感染或感染的方法。 其中n为0,1,2,3,4或5; m为0,1,2,3,4或5; R 1,R 2各自独立地选自:卤素,CN,N 3,NO 2,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基和C 2 -C 6 - 炔基,其中所述的最后3个基团可以部分或完全 卤化和/或可以携带1,2或3个基团R#等的任何组合; R 3和R 4彼此独立地选自氢,卤素,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基,C 2 -C 6 - 炔基,其中所述的最后3个基团可以部分或完全卤化和/或可以携带 CN,NO2,-ORb,NRcRd,-SRe,-C(= O)Ra和-C(= O)ORb等独立选自1,2或3个基团的任意组合; A是式A.1或A.2的基团,其中*表示与化合物的其余部分的连接点; R5a,R5b,R5c,R5d,R5e和R5f彼此独立地选自氢,卤素,C1-C6-烷基,C1-C6-烷氧基,C1-C6-烷基氨基,二(C1-C6-烷基)氨基, C3-C6-环烷基和Ar2等; R 6和R 7彼此独立地选自氢,CN,NO 2,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基,C 2 -C 6炔基,C 3 -C 8 - 环烷基,饱和或部分不饱和的5-, 或7元杂环基,Ar 3等

    Substituted Azolin-2-yl-Amino Compounds
    56.
    发明申请
    Substituted Azolin-2-yl-Amino Compounds 审中-公开
    取代的唑啉-2-基氨基化合物

    公开(公告)号:US20100167925A1

    公开(公告)日:2010-07-01

    申请号:US12376455

    申请日:2007-08-06

    IPC分类号: A01C1/06 A01N43/78 C07D417/02

    摘要: The present invention relates to azolin-2-yl-amino compounds of formulae (I. a) and (1.b) and their salts which are useful for combating animal pest, in particular arthropod and nematodes. The present invention also relates to a method for combating such pests and for protecting crops against infestation or infection by such pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests. Formula (I.a), formula (I.b) wherein n is 0 to 4; X is S, O or NR5; A is —C(R6a)(R6b)—, O, NR7, S, S(O) or S(O)2; B is a bond Or CH2; R1 is H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R2a, R2b are H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, (C1-C6-alkyl)-thiocarbonyl, C(O)NRaRb, C(S)NRaRb, (SO2)NRaRb, phenyl, benzyl, 5 or 6 membered heterocyclic ring etc.; or R1 together with R2a is C3-C5-alkandiyl; or R1 together with R2 are C(O); R3a, R3b, R3c, R3d are H, halogen, CN, C1-C6-alkyl, C1-C6-alkylamino, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R4a, R4b are H, halogen, C1-C6-alkyl, C2-C6-alkenyl, phenyl, benzyl, 5 or 6 membered hetaryl; or R4a together with Rb may also be ═O, ═NRC or ═CRdRe; or R2a together with R4a may form a bridging bivalent radical.

    摘要翻译: 本发明涉及用于对抗动物害虫,特别是节肢动物和线虫的式(Ⅰa)和(Ⅰb)的唑啉-2-基氨基化合物及其盐。 本发明还涉及一种防治这种害虫并防止作物抵抗这种害虫侵染或感染的方法。 此外,本发明涉及用于对抗动物害虫的兽用组合物。 式(Ⅰa),式(Ⅰb)其中n为0-4; X是S,O或NR5; A是-C(R6a)(R6b) - ,O,NR7,S,S(O)或S(O) B是键或CH2; R1是H,CN,C1-C6-烷基,C2-C6-烯基,C1-C6-烷基羰基,C3-C6-环烷基,苯基,苄基等; R2a,R2b是H,CN,C1-C6-烷基,C2-C6-烯基,C1-C6-烷基羰基,(C1-C6-烷基) - 硫代羰基,C(O)NRaRb,C(S)NRaRb,(SO2 )NRaRb,苯基,苄基,5或6元杂环等; 或R 1与R 2a一起为C 3 -C 5 - 烷二基; 或R 1与R 2一起为C(O); R3a,R3b,R3c,R3d是H,卤素,CN,C1-C6-烷基,C1-C6-烷基氨基,C3-C6-环烷基,苯基,苄基等; R4a,R4b是H,卤素,C1-C6-烷基,C2-C6-烯基,苯基,苄基,5或6元杂芳基; 或R 4a与R b一起也可以是= O,= NRC或= CRdRe; 或R 2a与R 4a一起形成桥连二价基团。

    Azoline Compounds for Combating Arthropod Pests
    58.
    发明申请
    Azoline Compounds for Combating Arthropod Pests 审中-公开
    用于防治节肢动物害虫的唑啉化合物

    公开(公告)号:US20100010058A1

    公开(公告)日:2010-01-14

    申请号:US12305267

    申请日:2007-05-25

    CPC分类号: C07D277/18

    摘要: The present invention relates to azoline compounds and their salts which are useful for combating arthropod pests. The present invention also relates to a method for combating arthropod pests and to agricultural compositions for combating said pests. It has been found that these objectives can be achieved by azoline compounds of the general formulae Ia or Ib, wherein X is S, O or NR4; Ar is phenyl or a 5 or 6 membered heteroaromatic ring; R1 is H, C1-C6-alkyl, C2-C6-alkenyl, phenyl, a heteroaromatic ring etc.; R2a, R2b are H, CN, C1-C6-alkyl etc.; R1 together with R2a may also form a linear C2-C4-alkandiyl; R3a-d are H, halogen, C1-C6-alkyl etc.

    摘要翻译: 本发明涉及可用于防治节肢动物害虫的唑啉化合物及其盐。 本发明还涉及一种防治节肢动物害虫的方法和用于对抗所述害虫的农业组合物。 已经发现,这些目的可以通过通式Ia或Ib的唑啉化合物来实现,其中X是S,O或NR 4; Ar是苯基或5或6元杂芳环; R1是H,C1-C6-烷基,C2-C6-烯基,苯基,杂芳环等; R2a,R2b是H,CN,C1-C6-烷基等; R1与R2a一起也可以形成直链C 2 -C 4 - 烷二基; R3a-d为H,卤素,C1-C6烷基等。