公开(公告)号：US20100280078A1

公开(公告)日：2010-11-04

申请号：US12667299

申请日：2008-07-02

申请人： Markus Kordes ,  Christopher Koradin ,  Ronan Le Vezouet ,  Ernst Baumann ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Cecile Ebuenga

发明人： Markus Kordes ,  Christopher Koradin ,  Ronan Le Vezouet ,  Ernst Baumann ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Cecile Ebuenga

IPC分类号： A01N43/78 ,  C07D277/18 ,  A61K31/426 ,  C07D417/12 ,  C07D417/14 ,  A61K31/427 ,  C07D263/28 ,  A01N43/76 ,  A61K31/421 ,  A61K31/4439 ,  A61P33/00 ,  A01P7/00 ,  A01P7/02 ,  A01P7/04 ,  A01P5/00

CPC分类号： C07D263/28 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N47/12 ,  A01N47/16 ,  C07D233/48 ,  C07D277/18 ,  C07D417/06 ,  C07D417/12

摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.

公开(公告)号：US20080312085A1

公开(公告)日：2008-12-18

申请号：US12158261

申请日：2006-12-11

申请人： Markus Kordes ,  Livio Tedeschi ,  Ronan Le Vezouet ,  Christopher Koradin ,  Deborah L. Culbertson

发明人： Markus Kordes ,  Livio Tedeschi ,  Ronan Le Vezouet ,  Christopher Koradin ,  Deborah L. Culbertson

IPC分类号： A01N43/78 ,  C07D417/12 ,  A01N43/40 ,  A01P7/04 ,  A01N43/42 ,  A01N43/836

CPC分类号： C07D417/12

摘要： The present invention relates to 1-(Azolin-2-yl)-amino-alkane compounds, which are useful for combating insects, arachnids and nematodes.The present invention also relates to a method for combating animal pests selected from insects, arachnids and nematodes, and to agricultural compositions for combating animal pests.It has been found that animal pests can be combated by 1-(Azolin-2-yl)-amino-alkane compounds of the general formula I: wherein A is a radical of the formulae A1 or A2: and wherein X is sulfur or oxygen and W, B and R1 to R6 are defined as in the description.

摘要翻译： 本发明涉及1-（唑啉-2-基） - 氨基 - 烷烃化合物，其可用于防治昆虫，蜘蛛和线虫。 本发明还涉及一种防治选自昆虫，蜘蛛和线虫的动物害虫的方法以及用于对抗动物害虫的农业组合物。 已经发现，可以通过通式I的1-（氮杂-2-基） - 氨基 - 烷烃化合物与动物害虫相抗衡：其中A是式A1或A2的基团：其中X是硫或氧 W，B，R 1〜R 6如说明书所述。

公开(公告)号：US08211924B2

公开(公告)日：2012-07-03

申请号：US12667299

申请日：2008-07-02

申请人： Markus Kordes ,  Christopher Koradin ,  Ronan Le Vezouet ,  Ernst Baumann ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Cecille Ebuenga

发明人： Markus Kordes ,  Christopher Koradin ,  Ronan Le Vezouet ,  Ernst Baumann ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Cecille Ebuenga

IPC分类号： A01N43/78 ,  A01N43/76 ,  A61K31/425 ,  A61K31/42 ,  C07D277/00 ,  C07D263/00

CPC分类号： C07D263/28 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N47/12 ,  A01N47/16 ,  C07D233/48 ,  C07D277/18 ,  C07D417/06 ,  C07D417/12

摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, —C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.

公开(公告)号：US08173675B2

公开(公告)日：2012-05-08

申请号：US12601017

申请日：2008-05-13

申请人： Christopher Koradin ,  Markus Kordes ,  Ernst Baumann ,  Ronan Le Vezouet ,  Deborah L. Culbertson

发明人： Christopher Koradin ,  Markus Kordes ,  Ernst Baumann ,  Ronan Le Vezouet ,  Deborah L. Culbertson

IPC分类号： A61K31/47 ,  C07D215/14

CPC分类号： A01N47/36 ,  A01N47/32 ,  C07C335/14 ,  C07C2602/08 ,  C07C2602/10 ,  C07D307/82 ,  C07D333/66

摘要： The invention relates to substituted amino-thiourea compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to the use of the substituted amino-thiourea compounds, of their salts or of compositions comprising them for combating animal pests. Furthermore the invention relates also to methods of applying such compounds. The substituted amino-thiourea compounds are defined by the following formula (I): wherein A, B, R1, R2, R3, R4, R5.1, R5.2 and R6 are defined as in the description.

摘要翻译： 本发明涉及式（I）的取代的氨基 - 硫脲化合物，其涉及其对映体，非对映异构体和盐以及包含这些化合物的组合物。 本发明还涉及取代的氨基 - 硫脲化合物，其盐或包含它们的组合物用于对抗动物害虫的用途。 此外，本发明还涉及应用这些化合物的方法。 取代的氨基 - 硫脲化合物由下式（I）定义：其中A，B，R1，R2，R3，R4，R5.1，R5.2和R6如说明书所定义。

公开(公告)号：US07981437B2

公开(公告)日：2011-07-19

申请号：US12094854

申请日：2006-11-15

申请人： Markus Kordes ,  Christopher Koradin ,  Deborah L. Culbertson

发明人： Markus Kordes ,  Christopher Koradin ,  Deborah L. Culbertson

IPC分类号： A61K31/4168 ,  A61K31/42 ,  A61K31/426 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  C07D277/04 ,  C07D277/18 ,  C07D233/02 ,  C07D233/50 ,  C07D263/04 ,  C07D263/28

CPC分类号： C07D277/18 ,  C07D233/50 ,  C07D263/28

摘要： The present invention relates to Indanyl- and Tetrahydronaphthyl-amino-azoline compounds of formula I wherein the variables R1 and R2 are as defined in description. The invention relates also to methods of combating or controlling insects, arachnids or nematodes, to methods for protecting growing plants from attack or infestation by insects, arachnids or nematodes, to methods for the protection of seeds from soil insects and of the seedlings' roots and shoots from soil and foliar insects and to methods for treating, controlling, preventing or protecting animals against infestation or infection by parasites.

摘要翻译： 本发明涉及式I的茚满基和四氢萘基 - 氨基 - 唑啉化合物，其中变量R1和R2如描述中所定义。 本发明还涉及防治昆虫，蜘蛛或线虫的方法，用于保护生长植物免受昆虫，蜘蛛或线虫侵袭或侵染的方法，用于保护种子免受土壤昆虫和幼苗根部和 来自土壤和叶面昆虫的芽，以及用于治疗，控制，预防或保护动物免受寄生虫感染或感染的方法。

公开(公告)号：US07871960B2

公开(公告)日：2011-01-18

申请号：US11914992

申请日：2006-05-18

申请人： Markus Kordes ,  Norbert Götz ,  Michael Rack ,  Christopher Koradin ,  Livio Tedeschi ,  Deborah L. Culbertson

发明人： Markus Kordes ,  Norbert Götz ,  Michael Rack ,  Christopher Koradin ,  Livio Tedeschi ,  Deborah L. Culbertson

IPC分类号： A01N43/50 ,  C07D233/04

CPC分类号： A01N43/50 ,  C07D233/48

摘要： The present invention relates to 1-(imidazolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and their agriculturally acceptable salts, wherein A is a radical of the formula A1 or A2. The invention relates also to agricultural compositions and to seed comprising at least one compound I and/or a salt thereof, as well as a method of combating animal pests, a method for protecting crops from attack or infestation by animal pests and a method for protecting non-living materials from attack or infestation by animal pests, a method for the protection of seeds from animal pests and of the seedlings' roots and shoots from animal pests by applying a pesticidally effective amount of at least one 1-(imidazolin-2-yl)amino-1,2-diphenylethane compound I and/or a salt thereof.

摘要翻译： 本发明涉及式I的1-（咪唑啉-2-基）氨基-1,2-二苯基乙烷化合物及其农业上可接受的盐，其中A是式A1或A2的基团。 本发明还涉及农业组合物和包含至少一种化合物I和/或其盐的种子，以及防治动物害虫的方法，用于保护作物免受动物害虫侵袭或侵染的方法和保护方法 通过施用杀虫有效量的至少一种1-（咪唑啉-2-酮）的动物害虫的攻击或感染的非生物材料，动物害虫的种子保护方法和来自动物害虫的幼苗的根和芽， 氨基-1,2-二苯基乙烷化合物I和/或其盐。

公开(公告)号：US07544637B2

公开(公告)日：2009-06-09

申请号：US11791398

申请日：2005-11-24

申请人： Wolfgang von Deyn ,  Henricus Maria Martinus Bastiaans ,  Matthias Pohlman ,  Michael Rack ,  Ernst Baumann ,  Michael Puhl ,  Michael Hofmann ,  Livio Tedeschi ,  Markus Kordes ,  Christopher Koradin ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Henry van Tuyl Cotter ,  Hassan Oloumi-Sadeghi

发明人： Wolfgang von Deyn ,  Henricus Maria Martinus Bastiaans ,  Matthias Pohlman ,  Michael Rack ,  Ernst Baumann ,  Michael Puhl ,  Michael Hofmann ,  Livio Tedeschi ,  Markus Kordes ,  Christopher Koradin ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Henry van Tuyl Cotter ,  Hassan Oloumi-Sadeghi

IPC分类号： C07C311/15 ,  A01N25/00 ,  A01N25/26 ,  A01P17/00 ,  A61K31/18

CPC分类号： C07C319/20 ,  A01N41/06 ,  C07C311/29 ,  C07C323/62

摘要： The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds I where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to the use of compounds I and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula I and/or at least one agriculturally acceptable salt thereof. a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula I

摘要翻译： 本发明涉及2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物I，其中变量Alk和R1至R5如权利要求1所定义，和/或其农业上有用的盐。 此外，本发明涉及化合物I和/或其盐对抗动物害虫的用途; 包含至少一种式I化合物和/或至少一种农业上可用的I盐和至少一种惰性液体和/或其农业上可接受的载体的农药组合物，其具有杀虫作用，如果需要 ，至少一种表面活性剂; 以及一种对抗动物害虫的方法，包括使动物有害生物，其习惯，繁殖地，食物供应，植物，种子，土壤，区域，动物害虫生长或可能生长的区域，材料或环境，或材料，植物 ，防止动物攻击或侵染的种子，土壤，表面或空间与杀虫有效量的式I的至少一个2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物和/或至少一种农业上可接受的盐 其中。 包括从土壤和叶面昆虫中保护种子免受土壤昆虫和所得植物的根和芽的方法，包括在种子播种前和/或后发芽后将种子与2-氰基-3-（卤代）烷氧基 - 苯磺酰胺 通式I的化合物

公开(公告)号：US20090131256A1

公开(公告)日：2009-05-21

申请号：US12305419

申请日：2007-06-29

申请人： Markus Kordes ,  Delphine Breuninger ,  Ronan Le Vezouet ,  Christopher Koradin ,  Livio Tedeschi ,  Michael Puhl ,  Deborah L. Culbertson

发明人： Markus Kordes ,  Delphine Breuninger ,  Ronan Le Vezouet ,  Christopher Koradin ,  Livio Tedeschi ,  Michael Puhl ,  Deborah L. Culbertson

IPC分类号： A01N25/26 ,  C07D333/20 ,  A01N43/10 ,  A01N43/56 ,  A01P7/00 ,  C07D231/12 ,  C07D213/36 ,  A01N43/40

CPC分类号： C07D333/20 ,  C07D213/40 ,  C07D231/12 ,  C07D307/52 ,  C07D413/12 ,  C07D417/12

摘要： The present invention relates to 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane compounds (I) and 1-(aminothiocarbonylamino)-2-aryl-1-hetaryl-ethane compounds (II) and their salts which are useful for combating animal pest, in particular insects, arachnids and nematodes. Furthermore, the present invention relates to a method for combating animal pests selected from insects, arachnids and nematodes, and to agricultural compositions for combating animal pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests.

摘要翻译： 本发明涉及1-（吡唑啉-2-基） - 氨基-2-芳基-1-杂芳基 - 乙烷化合物（I）和1-（氨基硫代羰基氨基）-2-芳基-1-杂芳基 - 乙烷化合物（II） 和它们的盐可用于对抗动物害虫，特别是昆虫，蜘蛛和线虫。 此外，本发明涉及一种防治选自昆虫，蜘蛛和线虫的动物害虫的方法以及用于对抗动物害虫的农业组合物。 此外，本发明涉及用于对抗动物害虫的兽用组合物。

公开(公告)号：US07989394B2

公开(公告)日：2011-08-02

申请号：US12305419

申请日：2007-06-29

申请人： Markus Kordes ,  Delphine Breuninger ,  Ronan Le Vezouet ,  Christopher Koradin ,  Livio Tedeschi ,  Michael Puhl ,  Deborah L. Culbertson

发明人： Markus Kordes ,  Delphine Breuninger ,  Ronan Le Vezouet ,  Christopher Koradin ,  Livio Tedeschi ,  Michael Puhl ,  Deborah L. Culbertson

IPC分类号： A01N43/76 ,  A01N43/78 ,  C07D277/04 ,  C07D277/08

CPC分类号： C07D333/20 ,  C07D213/40 ,  C07D231/12 ,  C07D307/52 ,  C07D413/12 ,  C07D417/12

摘要： The present invention relates to 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane compounds (I) and 1-(aminothiocarbonylamino)-2-aryl-1-hetaryl-ethane compounds (II) and their salts which are useful for combating animal pest, in particular insects, arachnids and nematodes. Furthermore, the present invention relates to a method for combating animal pests selected from insects, arachnids and nematodes, and to agricultural compositions for combating animal pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests.

摘要翻译： 本发明涉及1-（吡唑啉-2-基） - 氨基-2-芳基-1-杂芳基 - 乙烷化合物（I）和1-（氨基硫代羰基氨基）-2-芳基-1-杂芳基 - 乙烷化合物（II） 和它们的盐可用于对抗动物害虫，特别是昆虫，蜘蛛和线虫。 此外，本发明涉及一种防治选自昆虫，蜘蛛和线虫的动物害虫的方法以及用于对抗动物害虫的农业组合物。 此外，本发明涉及用于对抗动物害虫的兽用组合物。

公开(公告)号：US20100298138A1

公开(公告)日：2010-11-25

申请号：US12600852

申请日：2008-05-23

申请人： Christopher Koradin ,  Markus Kordes ,  Ernst Baumann ,  Ronan Le Vezouet ,  Deborah L. Culbertson

发明人： Christopher Koradin ,  Markus Kordes ,  Ernst Baumann ,  Ronan Le Vezouet ,  Deborah L. Culbertson

IPC分类号： A01C1/06 ,  A01P7/04 ,  A01P7/02 ,  A01P5/00 ,  A01N43/78 ,  A61K31/426 ,  C07D277/18 ,  A61P33/00 ,  C07C335/12 ,  A61K31/17 ,  A01N47/28 ,  C07C69/347 ,  C07C69/708 ,  C07D261/18 ,  A61K31/42 ,  A01N43/80 ,  C07D213/80 ,  A61K31/44 ,  A01N43/40 ,  C07C69/736 ,  A61K31/216 ,  C07C69/78 ,  C07D307/68 ,  A61K31/341 ,  A01N43/08

CPC分类号： C07D261/18 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N47/32 ,  C07C275/26 ,  C07C279/16 ,  C07C335/14 ,  C07C2602/08 ,  C07C2602/10 ,  C07D213/80 ,  C07D233/50 ,  C07D263/28 ,  C07D277/18 ,  C07D317/60

摘要： The present invention relates to the use of aminoazoline and urea derivatives for com-bating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds and to specific azoline and urea derivatives.

摘要翻译： 本发明涉及氨基唑啉和脲衍生物在动物害虫中的应用。 本发明还涉及通过使用这些化合物，种子和包含所述化合物的农业和兽用组合物以及特定的唑啉和脲衍生物来控制动物害虫的方法。