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    NOVEL IMIDAZOLE DERIVATIVES
    52.
    发明申请
    NOVEL IMIDAZOLE DERIVATIVES 审中-公开
    新咪唑衍生物

    公开(公告)号：US20110311649A1

    公开(公告)日：2011-12-22

    申请号：US12739852

    申请日：2008-10-24

    申请人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah ,  Sebastian Volker Wendeborn

    发明人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah ,  Sebastian Volker Wendeborn

    IPC分类号： A01N43/40 ,  C07D401/14 ,  A01N43/42 ,  A01N57/00 ,  A01N43/54 ,  A01N43/84 ,  A01N59/20 ,  C07D401/04 ,  A01P3/00

    CPC分类号： C07D233/61 ,  C07D233/68 ,  C07D401/04 ,  C07D401/14 ,  C07D409/04 ,  C07D409/14

    摘要： The present invention relates to novel imidazole derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is halogen, C1-C4alkyl or C1-C4haloalkyl; R2 is an optionally substituted aryl or heteroaryl; R3 is halogen; R4 is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, hydroxyl, C1-C4alkoxy, OR6, C1-C4haloalkoxy or cyano; R5 is halogen; R6 is hydrogen, C3-C7 cycloalkyl, C3-C10 alkylcycloalkyl, C1-C6 haloalkyl, C2-C6 alkenyl, C2-C6 haloalkenyl, C3-C7 cycloalkenyl, C2-C6 alkynyl, C2-C6 haloalkynyl or C2-C6 alkyloxyalkyl; X is N or C(R); and R is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; or an agrochemically usable salt form thereof; provided that when X is C(R), R2 cannot be an optionally substituted aryl.

    摘要翻译： 本发明涉及式（I）的新咪唑衍生物作为具有杀微生物活性，特别是杀真菌活性的活性成分：其中R1是卤素，C1-C4烷基或C1-C4卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4是氢，卤素，C1-C4烷基，C1-C4卤代烷基，羟基，C1-C4烷氧基，OR6，C1-C4卤代烷氧基或氰基; R5是卤素; R6是氢，C3-C7环烷基，C3-C10烷基环烷基，C1-C6卤代烷基，C2-C6烯基，C2-C6卤代烯基，C3-C7环烯基，C2-C6炔基，C2-C6卤代炔基或C2-C6烷氧基烷基; X是N或C（R）; 且R为氢，卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基或氰基; 或其农业化学可用的盐形式; 条件是当X是C（R）时，R 2不能是任选取代的芳基。

    NOVEL PYRIDAZINE DERIVATIVES
    53.
    发明申请
    NOVEL PYRIDAZINE DERIVATIVES 审中-公开
    新的吡咯烷酮衍生物

    公开(公告)号：US20100113457A1

    公开(公告)日：2010-05-06

    申请号：US12447025

    申请日：2007-10-23

    申请人： Stephan Trah ,  Clemens Lamberth ,  Sebastian Wendeborn

    发明人： Stephan Trah ,  Clemens Lamberth ,  Sebastian Wendeborn

    IPC分类号： A01N43/58 ,  C07D237/12 ,  C07D237/14 ,  A01P3/00 ,  A01P1/00

    CPC分类号： C07D237/12 ,  A01N43/58 ,  C07D237/14 ,  C07D237/24

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is halogen, nitro, cyano, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy, C1-C4alkylthio or C1-C4haloalkylthio; R3 is an optionally substituted aryl; R4 is fluoro, cyano, C1-C6haloalkyl, C3-C6cycloalkyl, C1-C6haloalkoxy, C1-C6alkylthio or C1-C6haloalkylthio; and n is a whole number from 1 to 4; or an agrochemically usable salt form thereof.

    摘要翻译： 本发明涉及具有杀微生物活性，特别是杀真菌活性的活性成分的式（I）的新哒嗪衍生物，其中R1是氢，C1-C6烷基，C1-C6卤代烷基或C3-C6环烷基; R 2是卤素，硝基，氰基，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基，C 1 -C 4烷硫基或C 1 -C 4卤代烷硫基; R3是任选取代的芳基; R 4是氟，氰基，C 1 -C 6卤代烷基，C 3 -C 6环烷基，C 1 -C 6卤代烷氧基，C 1 -C 6烷硫基或C 1 -C 6卤代烷硫基; n为1〜4的整数; 或其农业化学上可用的盐形式。

    Process for the preparation of pyrazole carboxylic acid amides
    58.
    发明授权
    Process for the preparation of pyrazole carboxylic acid amides 有权
    制备吡唑羧酸酰胺的方法

    公开(公告)号：US08519152B2

    公开(公告)日：2013-08-27

    申请号：US13642406

    申请日：2011-04-14

    申请人： Raphael Dumeunier ,  Florian Schleth ,  Thomas Vettiger ,  Michael Rommel ,  Stephan Trah

    发明人： Raphael Dumeunier ,  Florian Schleth ,  Thomas Vettiger ,  Michael Rommel ,  Stephan Trah

    IPC分类号： C07D231/10 ,  C07D303/02 ,  C07C33/00

    CPC分类号： C07D231/14 ,  C07C17/23 ,  C07C17/30 ,  C07C25/24 ,  C07C29/132 ,  C07C35/52 ,  C07C45/29 ,  C07C209/10 ,  C07C2603/66 ,  C07D303/17 ,  C07C49/697 ,  C07C23/10 ,  C07C25/22 ,  C07C211/61

    摘要： The invention relates to a process for the preparation of the compound of formula (I), which process comprises a) reacting a compound of formula (II), wherein X is chloro or bromo, with an organometallic species in an inert atmosphere to a halobenzyne of formula (X), reacting the halobenzyne of formula X so formed with cyclopentadiene to (III), b) reacting III in the presence of an inert solvent with an oxidant to (IV), c) reacting IV in the presence of a Lewis acid and a hydride source to (V), d) reacting V in the presence of an oxidizing agent, a base and an inert solvent to (VI), e) converting VI in the presence of a phosphane and CCl4 or CHCl3 to (VII), and either f1) reacting VII with NH3 in the presence of a catalyst to the compound of formula (VIII); and g) reacting VIII in the presence of a base with a compound of formula (IX), to the compound of formula (I); or f2) reacting the compound of formula (VII), in the presence of a solvent, a base, a copper catalyst and at least one ligand with the compound of formula (IXa), to the compound of formula (I).

    摘要翻译： 本发明涉及一种制备式（I）化合物的方法，该方法包括：a）使惰性气氛下的有机金属物质使式（II）化合物（其中X为氯或溴）与卤代苯 使式（X）所示的卤代苯与环戊二烯反应，得到（III），b）使III在惰性溶剂存在下与氧化剂反应，得到（Ⅳ），c）使IV在Lewis 酸和氢化物源至（V），d）使V在氧化剂，碱和惰性溶剂的存在下与（VI）反应，e）在磷烷和CCl 4或CHCl 3存在下将VI转化为（VII ），并且f1）使VII与NH 3在催化剂存在下与式（VIII）化合物反应; 和g）在碱存在下使VIII与式（IX）化合物反应，得到式（I）化合物; 或者f2）使式（Ⅶ）化合物在溶剂存在下，碱，铜催化剂和至少一种配体与式（Ⅸa）化合物反应，得到式（I）化合物。

    Pyridazine fungicides
    59.
    发明授权
    Pyridazine fungicides 失效
    哒嗪类杀菌剂

    公开(公告)号：US08410026B2

    公开(公告)日：2013-04-02

    申请号：US12863377

    申请日：2009-01-14

    申请人： Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    发明人： Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    IPC分类号： A01N43/58 ,  A61K31/50 ,  C07D237/00

    CPC分类号： C07D401/04

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is methyl, ethyl or isopropyl; R2 is chloro, fluoro, hydroxy or C1-C2alkoxy; R3 is H, chloro, fluoro, methoxy or C1-C3alkyl; R4 is chloro, fluoro or bromo; and R5 is H, fluoro or methoxy; or an agrochemically usable salt form thereof; with the proviso that when R1 is methyl, R2 is chloro and R3 is H, then R4 or R5 is different from fluoro.

    摘要翻译： 本发明涉及式（I）的新的哒嗪衍生物作为具有杀微生物活性的活性成分，特别是杀真菌活性：其中R1是甲基，乙基或异丙基; R 2是氯，氟，羟基或C 1 -C 2烷氧基; R3是H，氯，氟，甲氧基或C1-C3烷基; R4是氯，氟或溴; R5为H，氟或甲氧基; 或其农业化学可用的盐形式; 条件是当R 1为甲基时，R 2为氯且R 3为H，则R 4或R 5不同于氟。