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    Pesticidal triazine-derivatives
    52.
    发明授权
    Pesticidal triazine-derivatives 失效
    杀虫三嗪衍生物

    公开(公告)号：US06723720B2

    公开(公告)日：2004-04-20

    申请号：US10006954

    申请日：2001-11-05

    Applicant: Arthur Steiger ,  Werner Zambach ,  André Jeanguenat ,  Martin Eberle ,  Stephan Trah ,  Saleem Farooq

    Inventor： Arthur Steiger ,  Werner Zambach ,  André Jeanguenat ,  Martin Eberle ,  Stephan Trah ,  Saleem Farooq

    IPC: C07D253065

    CPC classification number: A01N57/22 ,  A01N43/707 ,  C07D253/07

    Abstract: A compound of formula wherein R1 is unsubstituted or substituted aryl or heteroaryl, the substituents of the aryl and heteroaryl rings being selected, for example, from the group consisting of OH, halogen, CN, NO2, C1-C6alkyl, C3-C8cycloalkyl, C1-C6alkyl-C3-C8cycloalkyl, C3-C8cycloalkyl-C1-C6alkyl, C1-C6haloalkyl, C3-C8halocycloalkyl, C1-C6alkoxy and phenyl; phenoxy; phenylthio; phenylamino; and phenyl-(C1-C6alkyl)-amino; the substituents of the phenoxy, phenylthio, phenylamino and phenyl-(C1-C6alkyl)-amino groups being selected from the group consisting of halogen, CN, NO2, C1-C6alkyl, C3-C8cycloalkyl, C1-C6haloalkyl, C3-C8halocycloalkyl, C1-C6alkoxy, C3-C8cycloalkoxy, C1-C6alkylthio, C3-C8cycloalkylthio, C1-C6haloalkylthio and C3-C8halocycloalkylthio; R2 is, for example, H, OH, halogen, CN, NO2, C1-C6alkyl or C1-C6alkoxy; A is, for example, a single bond, C1-C12alkylene, O or O(C1-C12alkylene); R4 is H, C1-C6alkyl, C3-C8cycloalkyl, C1-C6haloalkyl, C1-C6alkoxy, N(R5)2 or C1-C6alkoxy-C2-C6alkyl; R5 is H, C1-C6alkyl, C3-C8cycloalkyl, C1-C6haloalkyl or aryl-C1-C6alkyl; X1 is R10; X2 and X3 are each independently of the other H or R10; R10 is, for example, halogen, CN, NO2, C1-C6alkyl or C3-C8cycloalkyl; and n is 0, 1 or 2, and to their physiologically tolerable and agrochemically acceptable addition compounds, and where appropriate to E/Z isomers, to mixtures of E/Z isomers and/or to tautomers, in each case in free form or in salt form. The compounds, in free form or in agrochemically acceptable salt form, exhibit advantageous pesticidal properties. They are suitable especially in the control of pests in agriculture and stored goods and also in the keeping of domestic animals.

    Abstract translation: 化合物R1是未取代或取代的芳基或杂芳基，芳基和杂芳基环的取代基选自例如由OH，卤素，CN，NO 2，C 1 -C 6烷基，C 3 -C 8环烷基，C 1 -C 6烷基 - C 3 -C 8环烷基，C 3 -C 8环烷基-C 1 -C 6烷基，C 1 -C 6卤代烷基，C 3 -C 8卤代环烷基，C 1 -C 6烷氧基和苯基; 苯氧基 苯硫基 苯基氨基; 苯基 - （C 1 -C 6烷基） - 氨基;苯氧基，苯硫基，苯基氨基和苯基 - （C 1 -C 6烷基） - 氨基的取代基选自卤素，CN，NO 2，C 1 -C 6烷基， C 3 -C 8卤代烷基，C 1 -C 6卤代烷基，C 3 -C 8卤代环烷基，C 1 -C 6烷氧基，C 3 -C 8环烷氧基，C 1 -C 6烷硫基，C 3 -C 8环烷硫基，C 1 -C 6卤代烷硫基和C 3 -C 8卤代环烷硫基; R 2为例如H，OH，卤素，CN， C1-C6烷基或C1-C6烷氧基; A是例如单键，C1-C12亚烷基，O或O（C1-C12亚烷基）; R4是H，C1-C6烷基，C3-C8环烷基，C1-C6卤代烷基，C1-C6烷氧基 ，N（R 5）2或C 1 -C 6烷氧基-C 2 -C 6烷基; R 5是H，C 1 -C 6烷基，C 3 -C 8环烷基，C 1 -C 6卤代烷基或芳基-C 1 -C 6烷基; X 1是R 10; X 2和X 3各自独立地为H或R 10; R 10为例如卤素，CN，NO 2，C 1 -C 6烷基或C 3 -C 8环烷基; 和n为0,1或2，以及其生理上可耐受和农业化学上可接受的加成化合物，以及适用于E / Z异构体的E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或 游离形式或农业化学上可接受的盐形式的化合物表现出有利的杀虫性质。 它们特别适用于控制农业和储存物中的害虫以及保存家畜。

    Process for the preparation of pyrazole carboxylic acid amides
    56.
    发明授权
    Process for the preparation of pyrazole carboxylic acid amides 有权
    制备吡唑羧酸酰胺的方法

    公开(公告)号：US08519152B2

    公开(公告)日：2013-08-27

    申请号：US13642406

    申请日：2011-04-14

    Applicant: Raphael Dumeunier ,  Florian Schleth ,  Thomas Vettiger ,  Michael Rommel ,  Stephan Trah

    Inventor： Raphael Dumeunier ,  Florian Schleth ,  Thomas Vettiger ,  Michael Rommel ,  Stephan Trah

    IPC: C07D231/10 ,  C07D303/02 ,  C07C33/00

    CPC classification number: C07D231/14 ,  C07C17/23 ,  C07C17/30 ,  C07C25/24 ,  C07C29/132 ,  C07C35/52 ,  C07C45/29 ,  C07C209/10 ,  C07C2603/66 ,  C07D303/17 ,  C07C49/697 ,  C07C23/10 ,  C07C25/22 ,  C07C211/61

    Abstract: The invention relates to a process for the preparation of the compound of formula (I), which process comprises a) reacting a compound of formula (II), wherein X is chloro or bromo, with an organometallic species in an inert atmosphere to a halobenzyne of formula (X), reacting the halobenzyne of formula X so formed with cyclopentadiene to (III), b) reacting III in the presence of an inert solvent with an oxidant to (IV), c) reacting IV in the presence of a Lewis acid and a hydride source to (V), d) reacting V in the presence of an oxidizing agent, a base and an inert solvent to (VI), e) converting VI in the presence of a phosphane and CCl4 or CHCl3 to (VII), and either f1) reacting VII with NH3 in the presence of a catalyst to the compound of formula (VIII); and g) reacting VIII in the presence of a base with a compound of formula (IX), to the compound of formula (I); or f2) reacting the compound of formula (VII), in the presence of a solvent, a base, a copper catalyst and at least one ligand with the compound of formula (IXa), to the compound of formula (I).

    Abstract translation: 本发明涉及一种制备式（I）化合物的方法，该方法包括：a）使惰性气氛下的有机金属物质使式（II）化合物（其中X为氯或溴）与卤代苯 使式（X）所示的卤代苯与环戊二烯反应，得到（III），b）使III在惰性溶剂存在下与氧化剂反应，得到（Ⅳ），c）使IV在Lewis 酸和氢化物源至（V），d）使V在氧化剂，碱和惰性溶剂的存在下与（VI）反应，e）在磷烷和CCl 4或CHCl 3存在下将VI转化为（VII ），并且f1）使VII与NH 3在催化剂存在下与式（VIII）化合物反应; 和g）在碱存在下使VIII与式（IX）化合物反应，得到式（I）化合物; 或者f2）使式（Ⅶ）化合物在溶剂存在下，碱，铜催化剂和至少一种配体与式（Ⅸa）化合物反应，得到式（I）化合物。

    Pyridazine fungicides
    57.
    发明授权
    Pyridazine fungicides 失效
    哒嗪类杀菌剂

    公开(公告)号：US08410026B2

    公开(公告)日：2013-04-02

    申请号：US12863377

    申请日：2009-01-14

    Applicant: Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    Inventor： Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    IPC: A01N43/58 ,  A61K31/50 ,  C07D237/00

    CPC classification number: C07D401/04

    Abstract: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is methyl, ethyl or isopropyl; R2 is chloro, fluoro, hydroxy or C1-C2alkoxy; R3 is H, chloro, fluoro, methoxy or C1-C3alkyl; R4 is chloro, fluoro or bromo; and R5 is H, fluoro or methoxy; or an agrochemically usable salt form thereof; with the proviso that when R1 is methyl, R2 is chloro and R3 is H, then R4 or R5 is different from fluoro.

    Abstract translation: 本发明涉及式（I）的新的哒嗪衍生物作为具有杀微生物活性的活性成分，特别是杀真菌活性：其中R1是甲基，乙基或异丙基; R 2是氯，氟，羟基或C 1 -C 2烷氧基; R3是H，氯，氟，甲氧基或C1-C3烷基; R4是氯，氟或溴; R5为H，氟或甲氧基; 或其农业化学可用的盐形式; 条件是当R 1为甲基时，R 2为氯且R 3为H，则R 4或R 5不同于氟。

    IMIDAZOLE DERIVATIVES
    59.
    发明申请
    IMIDAZOLE DERIVATIVES 审中-公开
    咪唑衍生物

    公开(公告)号：US20120010195A1

    公开(公告)日：2012-01-12

    申请号：US13256074

    申请日：2010-02-08

    Applicant: Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah

    Inventor： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah

    IPC: A01N43/46 ,  A01P3/00 ,  C07D403/04

    CPC classification number: C07D233/88

    Abstract: The present invention relates to novel imidazole derivatives of formula (I) having microbiocidal, in particular fungicidal, activity, to processes for their preparation and intermediates used in their preparation, to agrochemical compositions comprising them and to the use in agriculture or horticulture for controlling or preventing infestation of plants, harvested food crops, seeds or non-living materials by phytopathogenic microorganisms, preferably fungi.

    Abstract translation: 本发明涉及式（I）的新型咪唑衍生物，其具有杀微生物，特别是杀真菌活性，其制备方法和用于其制备的中间体，包含它们的农用化学组合物以及在农业或园艺中用于控制或 通过植物病原微生物，优选真菌预防植物，收获的食物作物，种子或非生物材料的侵染。

    NOVEL IMIDAZOLE DERIVATIVES
    60.
    发明申请
    NOVEL IMIDAZOLE DERIVATIVES 审中-公开
    新咪唑衍生物

    公开(公告)号：US20110224252A1

    公开(公告)日：2011-09-15

    申请号：US12739863

    申请日：2008-10-24

    Applicant: Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah ,  Sebastian Wendeborn

    Inventor： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah ,  Sebastian Wendeborn

    IPC: A01N43/42 ,  C07D233/68 ,  A01N43/50 ,  C07D401/04 ,  A01N43/40 ,  C07D409/04 ,  C07D401/02 ,  A01P3/00

    CPC classification number: C07D401/04 ,  A01N43/50 ,  C07D233/28 ,  C07D401/14 ,  C07D409/14

    Abstract: The present invention relates to novel imidazole derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is halogen, C1-C4alkyl or C1-C4haloalkyl; R2 is an optionally substituted aryl or heteroaryl; R3 is halogen; R4 is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; R5 is halogen; X is N or C(R); and R is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; or an agrochemically usable salt form thereof; provided that when X is C(R), R2 cannot be an optionally substituted aryl.

    Abstract translation: 本发明涉及式（I）的新咪唑衍生物作为具有杀微生物活性，特别是杀真菌活性的活性成分：其中R1是卤素，C1-C4烷基或C1-C4卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4是氢，卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或氰基; R5是卤素; X是N或C（R）; 且R为氢，卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基或氰基; 或其农业化学可用的盐形式; 条件是当X是C（R）时，R 2不能是任选取代的芳基。

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