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    IMIDAZOLE DERIVATIVES
    61.
    发明申请
    IMIDAZOLE DERIVATIVES 审中-公开
    咪唑衍生物

    公开(公告)号：US20120010195A1

    公开(公告)日：2012-01-12

    申请号：US13256074

    申请日：2010-02-08

    申请人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah

    发明人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah

    IPC分类号： A01N43/46 ,  A01P3/00 ,  C07D403/04

    CPC分类号： C07D233/88

    摘要： The present invention relates to novel imidazole derivatives of formula (I) having microbiocidal, in particular fungicidal, activity, to processes for their preparation and intermediates used in their preparation, to agrochemical compositions comprising them and to the use in agriculture or horticulture for controlling or preventing infestation of plants, harvested food crops, seeds or non-living materials by phytopathogenic microorganisms, preferably fungi.

    摘要翻译： 本发明涉及式（I）的新型咪唑衍生物，其具有杀微生物，特别是杀真菌活性，其制备方法和用于其制备的中间体，包含它们的农用化学组合物以及在农业或园艺中用于控制或 通过植物病原微生物，优选真菌预防植物，收获的食物作物，种子或非生物材料的侵染。

    NOVEL IMIDAZOLE DERIVATIVES
    62.
    发明申请
    NOVEL IMIDAZOLE DERIVATIVES 审中-公开
    新咪唑衍生物

    公开(公告)号：US20110224252A1

    公开(公告)日：2011-09-15

    申请号：US12739863

    申请日：2008-10-24

    申请人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah ,  Sebastian Wendeborn

    发明人： Raphael Dumeunier ,  Clemens Lamberth ,  Stephan Trah ,  Sebastian Wendeborn

    IPC分类号： A01N43/42 ,  C07D233/68 ,  A01N43/50 ,  C07D401/04 ,  A01N43/40 ,  C07D409/04 ,  C07D401/02 ,  A01P3/00

    CPC分类号： C07D401/04 ,  A01N43/50 ,  C07D233/28 ,  C07D401/14 ,  C07D409/14

    摘要： The present invention relates to novel imidazole derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is halogen, C1-C4alkyl or C1-C4haloalkyl; R2 is an optionally substituted aryl or heteroaryl; R3 is halogen; R4 is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; R5 is halogen; X is N or C(R); and R is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; or an agrochemically usable salt form thereof; provided that when X is C(R), R2 cannot be an optionally substituted aryl.

    摘要翻译： 本发明涉及式（I）的新咪唑衍生物作为具有杀微生物活性，特别是杀真菌活性的活性成分：其中R1是卤素，C1-C4烷基或C1-C4卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4是氢，卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或氰基; R5是卤素; X是N或C（R）; 且R为氢，卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基或氰基; 或其农业化学可用的盐形式; 条件是当X是C（R）时，R 2不能是任选取代的芳基。

    FUNGICIDAL COMPOUNDS AND COMPOSITIONS
    65.
    发明申请
    FUNGICIDAL COMPOUNDS AND COMPOSITIONS 审中-公开
    杀真菌化合物和组合物

    公开(公告)号：US20100016339A1

    公开(公告)日：2010-01-21

    申请号：US12375839

    申请日：2007-07-30

    申请人： Jeremy Godwin ,  Stephan Trah ,  Clemens Lamberth ,  Sebastian Volker Wendeborn

    发明人： Jeremy Godwin ,  Stephan Trah ,  Clemens Lamberth ,  Sebastian Volker Wendeborn

    IPC分类号： A01N43/90 ,  C07D237/02 ,  A01N43/58 ,  A01P3/00

    CPC分类号： C07D237/12 ,  A01N43/58

    摘要： The present invention relates, inter alia, to a compound having the formula (I):—wherein (R)n is selected from the group consisting of 4-Br, 4-OCH2CH3, 4-OCH2CF3, 2-CH3-4-Cl, 2-CH3-4-OCH3, 2-CH3-4-OCF3, 2-F-4-Br, 2-F-4-CF3, 3-CH3-4-Br, 3-F-4-Cl, 3-F-4-CH3, 3-F-4-Br, 3-F-4-OCH3 and 3-F-4-F. The present invention further relates to a fungicidal composition comprising a compound having the formula (I)—and also to fungicidal compositions comprising compounds having the formula (II) and/or (III): Furthermore, the present invention relates to methods for controlling pathogenic organisms using the compositions.

    摘要翻译： 本发明特别涉及具有式（I）的化合物：其中（R）n选自4-Br，4-OCH2CH3,4-OCH2CF3,2-CH3-4-Cl ，2-CH3-4-OCH3,2-CH3-4-OCF3,2-F-4-Br，2-F-4-CF3,3-CH3-4-Br，3-F-4-Cl，3 -F-4-CH 3，3-F-4-Br，3-F-4-OCH 3和3-F-4-F。 本发明还涉及包含具有式（I）的化合物的杀真菌组合物，还涉及包含具有式（II）和/或（III）的化合物的杀真菌组合物：此外，本发明涉及控制致病性的方法 使用组合物的生物体。

    Carboxamides as fungicides in agriculture
    67.
    发明授权
    Carboxamides as fungicides in agriculture 失效

    公开(公告)号：US07332518B2

    公开(公告)日：2008-02-19

    申请号：US10470069

    申请日：2002-01-24

    申请人： Harald Walter ,  Stephan Trah

    发明人： Harald Walter ,  Stephan Trah

    IPC分类号： A61K31/415 ,  A61K31/38 ,  C07D231/10 ,  C07D333/22 ,  C07D307/34

    CPC分类号： C07D207/34 ,  C07D231/14 ,  C07D277/56

    摘要： The invention concerns novel carboxamides of formula (I) wherein A is (A1), (A2), (A3), (A4), (A5); Q is (Q1), (Q2), (Q3), (Q4), (Q5), (Q6); R1 is CH2 R2, CH2CH═CHR2, CH═C═CHR2 or COR3; R2 is hydrogen, C1-C6alkyl, C1-C6haloalkyl, C2-C6alkenyl, C2-C6alkynyl, C3-C7cycloalkyl, COOC1-C4alkyl, COOC3-C6alkenyl, COOC3-C6alkynyl or CN; R3 is C1-C6alkyl, C1-C6alkyl substituted by halogen, C1-C6alkoxy or C1-C6haloalkoxy; or is C1-C6alkylthio, C1-C6haloalkylthio, C1-C6alkoxy, C1-C6haloalkoxy; C3-C6alkenyloxy or C3-C6haloalkenyloxy; C3-C6haloalkenyloxy; C3-C6alkynyloxy or C3-C6haloalkynyloxy; R4 is methyl, CF2Cl, CF3, CF2H, CFH2, Cl or Br, R5 is methyl, CF3, CH2OCH3 or CH2OCF3; R6 is hydrogen, fluoro, CF3 or methyl; R7 is hydrogen, methyl or halogen; and Z is phenyl, halophenyl, C5-C7cycloalkyl, C5-C7cycloalkyl substituted by C1-C3alkyl, C1C3haloalkyl or halogen, or a group of the form —CHR8—CH2—CHR9R10 wherein R8, R9 and R10 are independently of each other C1-C3alkyl. The novel compounds have plant-protective properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms, in particular fungi.

    Process for the preparation of pesticides
    70.
    发明授权
    Process for the preparation of pesticides 失效
    农药制备工艺

    公开(公告)号：US06646151B1

    公开(公告)日：2003-11-11

    申请号：US09670147

    申请日：2000-09-26

    申请人： Saleem Farooq ,  Stephan Trah ,  Hugo Ziegler ,  René Zurflüh

    发明人： Saleem Farooq ,  Stephan Trah ,  Hugo Ziegler ,  René Zurflüh

    IPC分类号： C07C24904

    CPC分类号： C07C249/12 ,  C07C251/48 ,  C07C251/60

    摘要： The invention relates to a process for the preparation of compounds of the formula or, if appropriate, a tautomer thereof, in each case in the free form or in salt form, in which A, X, Y, Z, R2, R3, R4, R5, R7, R9 and n are as defined in claim 1 and the C═N double bond marked with E has the E configuration, which comprises a1) reacting either a compound of the formula (II) mentioned above with a compound of the formula (III) mentioned above, in which X1 is a leaving group, or a2) a compound of the formula (IV) mentioned above, if appropriate in the presence of a base, with a compound of the formula (V) mentioned above, or b1) reacting a compound of the formula (VI) mentioned above with a compound of the formula R7—A—X2 (VII), in which X2 is a leaving group, and either further reacting the compound thus obtainable, of the formula (IV), for example according to method a2), or b2) reacting it with hydroxylamine or a salt thereof, if appropriate in the presence of a basic or acid catalyst, and further reacting the compound thus obtainable, of the formula (II), for example according to method a1), or c) reacting a compound of the formula (VIII), mentioned above with a C1-C6alkyl nitrite and further reacting the compound thus obtainable, of the formula (VI), for example according to method b), the E isomers of the compounds of the formulae (II), (IV) and (VI), a process for their preparation and their use for the preparation of compounds of the formula (I).

    摘要翻译： 本发明涉及一种制备式的化合物的方法，如果合适，其合适的是其互变异构体，其各自为游离形式或盐形式，其中A，X，Y，Z，R 2，R 3，R 4， R5，R7，R9和n如权利要求1中所定义，并且用E标记的C = N双键具有E构型，其包括a）使上述式（II）的化合物与式（II） III），其中X1是离去基团，ora2）如果合适的话，在碱的存在下，上述式（Ⅳ）的化合物与上述式（Ⅴ）的化合物相同，反应1）使 上述式（Ⅵ）化合物与式R7-A-X2（Ⅶ）化合物反应，其中X 2为离去基团，并进一步使由此得到的式（Ⅳ）化合物与 根据方法a2）的示例，orb2）如果合适，在碱性或酸性催化剂存在下，使其与羟胺或其盐反应，以及 进一步使由式（II）得到的化合物，例如按照方法a1）进行反应，或者使上述式（Ⅷ）化合物与亚硝酸C 1 -C 6烷基酯反应，并进一步使由此得到的化合物， 式（Ⅵ）化合物的方法，例如根据方法b），式（II），（Ⅳ）和（Ⅵ）化合物的E异构体，其制备方法及其制备方法 式（I）。