Resorcine Derivatives and Their Use as Pesticides

    公开(公告)号:US20090209598A1

    公开(公告)日:2009-08-20

    申请号:US12093543

    申请日:2006-11-10

    摘要: This invention relates to resorcine derivatives of formula (I) wherein R1 is phenyl or a 5- to 6-membered heteroaromatic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the heteroaromatic ring may be fused to a ring selected from phenyl and a 5- to 6-membered saturated, partially unsaturated or aromatic heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the 5- to 6-membered heteroaromatic ring or the respective fused ring systems may be unsubstituted or substituted by any combination of 1 to 6 optionally substituted groups R3, wherein R3 is halogen, cyano, nitro, hydroxy, mercapto, amino, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, halocycloalkyl, halocycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, haloalkenyloxy, haloalkynyloxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, haloalkenylthio, haloalkynylthio, alkylamino, alkenylamino, alkynylamino, dialkylamino, dialkenylamino, dialkynylamino, alkyl-alkenylamino, alkyl-alkynylamino, alkenyl-alkynylamino, trialkylsilyl, or phenyl or a 5- to 7-membered saturated or partially unsaturated heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, sulfur and nitrogen or a 5- to 6-membered heteraromatic ring system which may contain 1 to 4 heteroatoms selected from oxygen, nitrogen and sulfur, which phenyl and which heteroaromatic ring may be bonded via an oxygen or a sulfur atom, or —C(=G)Ra, —C(=G)ORa, —C(=G)NRa2, —C(=G)[N═SRa2], —C(═NORa)Ra, —C(═NORa)NRa2, —C(═NNRa2)Ra, —OC(=G)-OC(=G)ORa, N═SRa2, —NRaC(=G)Ra, —N[C(=G)Ra]2, —NRaC(=G)ORa, —C(=G)NRa—NRa2, —C(=G)NRa—NRa[C(=G)Ra], —NRa—C(=G)NRa2, —NRa—NRaC(=G)Ra, —NRa—N[C(=G)Ra]2, —N[(C=G)Ra]—NRa2, —NRa—NRa[(C=G)GRa], —NRa[(C=G)NRa2, —NRa[C═NRa]Ra, —NRa(C═NRa)NRa2, —O—NRa2, —O—NRa(C=G)Ra, —SO2NRa2, —NRaSO2Ra, —S(═O)Ra, —S(═O)2Ra, —SO2ORa, or —OSO2Ra, wherein G is oxygen or sulfur and Ra is as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, alkoxy, or haloalkoxy, x is 2, 3, 4, 5, 6, or 7, or the diastereomers, enantiomers, salts or N-oxides thereof, with the proviso that R1 is not 5-chloro-2,2,-dimethyl-2,3-dihydrobenzo[b]furan-7-yl when R2 is hydrogen and x is 3 or 4, processes and intermediates for the preparation of compounds I, use of compounds I for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds I.

    2-cyano-3(halo)alkoxy-benzenesulfonamide compounds for combating animal pests
    72.
    发明授权
    2-cyano-3(halo)alkoxy-benzenesulfonamide compounds for combating animal pests 失效
    用于对抗动物害虫的2-氰基-3-(卤代)烷氧基 - 苯磺酰胺化合物

    公开(公告)号:US07544637B2

    公开(公告)日:2009-06-09

    申请号:US11791398

    申请日:2005-11-24

    摘要: The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds I where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to the use of compounds I and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula I and/or at least one agriculturally acceptable salt thereof. a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula I

    摘要翻译: 本发明涉及2-氰基-3-(卤代)烷氧基 - 苯磺酰胺化合物I,其中变量Alk和R1至R5如权利要求1所定义,和/或其农业上有用的盐。 此外,本发明涉及化合物I和/或其盐对抗动物害虫的用途; 包含至少一种式I化合物和/或至少一种农业上可用的I盐和至少一种惰性液体和/或其农业上可接受的载体的农药组合物,其具有杀虫作用,如果需要 ,至少一种表面活性剂; 以及一种对抗动物害虫的方法,包括使动物有害生物,其习惯,繁殖地,食物供应,植物,种子,土壤,区域,动物害虫生长或可能生长的区域,材料或环境,或材料,植物 ,防止动物攻击或侵染的种子,土壤,表面或空间与杀虫有效量的式I的至少一个2-氰基-3-(卤代)烷氧基 - 苯磺酰胺化合物和/或至少一种农业上可接受的盐 其中。 包括从土壤和叶面昆虫中保护种子免受土壤昆虫和所得植物的根和芽的方法,包括在种子播种前和/或后发芽后将种子与2-氰基-3-(卤代)烷氧基 - 苯磺酰胺 通式I的化合物

    1-(1,2 Diphenyl-Ethyl)-3-(2-Hydroxyethyl)-Thiourea Compounds For Combating Animal Pests
    74.
    发明申请
    1-(1,2 Diphenyl-Ethyl)-3-(2-Hydroxyethyl)-Thiourea Compounds For Combating Animal Pests 审中-公开
    1-(1,2二苯基 - 乙基)-3-(2-羟乙基) - 硫脲化合物用于防治动物害虫

    公开(公告)号:US20080161403A1

    公开(公告)日:2008-07-03

    申请号:US11914959

    申请日:2006-05-18

    IPC分类号: A01N47/28 A01P15/00

    CPC分类号: C07C335/12 A01N47/28

    摘要: The present invention relates to a method of combating animal pests which comprises contacting the animal pest, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation, with a pesticidally effective amount of at least one 1-(1,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compound I or an agriculturally acceptable salt thereof, wherein m is 0 to 5, n is 0 to 5, R3 and R4 are H or optionally substituted alkyl, haloalkyl, cycloalkyl, phenyl or benzyl, R7, R8, R9 and R10 are H or optionally substituted C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkylamino, C1-C6-alkoxy, C3-C6-cycloalkyl, phenyl or benzyl and the variables R1, R2, R5 and R6 are as defined in the claims. The invention relates also to a method for protecting crops from attack or infestation by animal pests, a method for protecting non-living materials from attack or infestation by animal pests, novel 1-(1,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compounds I and their agriculturally acceptable salts as well as to an agricultural composition comprising a 1-(1,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compound I or a salt thereof.

    摘要翻译: 本发明涉及一种防治动物害虫的方法,包括使动物害虫,其习惯,繁殖地,食物供应,植物,种子,土壤,区域,动物害虫生长或可能生长的物质或环境接触,或 具有杀虫有效量的至少一种1-(1,2-二苯基 - 乙基)-3-(2-羟基乙基)-3-甲基苯酚的物质,植物,种子,土壤,表面或空间,以免受动物攻击或侵染, 硫脲化合物I或其农业上可接受的盐,其中m为0至5,n为0至5,R 3和R 4为H或任选取代的烷基,卤代烷基 ,环烷基,苯基或苄基,R 7,R 8,R 9和R 10是H或任选地 取代的C 1 -C 6 - 烷基,C 1 -C 6 - 卤代烷基,C 1 C 1 -C 6 - 烷基氨基,C 1 -C 6 - 烷氧基,C 3 -C C 6 - 环烷基,苯基或苄基和变量R 1 R 2,R 5,R 6和R 6如权利要求中所定义。 本发明还涉及一种保护作物免受动物害虫攻击或侵染的方法,一种保护非生物材料免受动物害虫侵袭或侵染的方法,新的1-(1,2-二苯基 - 乙基)-3-( 2-羟乙基) - 硫脲化合物I及其农业上可接受的盐,以及包含1-(1,2-二苯基 - 乙基)-3-(2-羟乙基) - 硫脲化合物I或其盐的农业组合物。