N-cycloalkyl-3-alkenybenzoyl-pyrazole derivatives
    74.
    发明授权
    N-cycloalkyl-3-alkenybenzoyl-pyrazole derivatives 失效
    N-环烷基-3-烯基苯甲酰基 - 吡唑衍生物

    公开(公告)号:US06475957B1

    公开(公告)日:2002-11-05

    申请号:US10019047

    申请日:2001-12-27

    IPC分类号: A01N4356

    CPC分类号: A01N43/56 C07D231/20

    摘要: Cycloalkyl-substituted benzoylpyrazoles of the formula I where the variables have, for example, the following meanings: R1 is hydrogen, nitro, halogen, cyano, thiocyanato, or an unsubstituted or substituted aliphatic radical; R2 is an unsubstituted or substituted aliphatic radical, halogen, nitro, or substituted sulfonyl or amino groups, R3 is hydrogen, halogen, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C2-C6-alkenyl or C2-C6-alkynyl; R4, R5 are hydrogen, nitro, halogen, cyano, thiocyanato, an unsubstituted or substituted aliphatic radical or substituted sulfonyl or amino groups; R6 is hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C3-C8-cycloalkyl; R7 is a cyclic ring system having 3-14 ring atoms; R16 is hydroxyl or a substituted hydroxyl group; and their tautomers or agriculturally useful salts are described. Moreover, the invention describes processes for preparing compounds of the formula I, compositions comprising them, and the use of the compounds of the formula I and of the compositions comprising them for controlling harmful plants.

    摘要翻译: 式I的环烷基取代的苯甲酰基吡唑,其中变量具有例如以下含义:R 1是氢,硝基,卤素,氰基,氰硫基或未取代或取代的脂族基; R 2是未取代或取代的脂族基,卤素, 硝基或取代的磺酰基或氨基,R 3是氢,卤素,C 1 -C 6烷基,C 1 -C 6卤代烷基,C 1 -C 6 - 烷氧基,C 2 -C 6 - 烯基或C 2 -C 6 - 炔基; R 4,R 5是氢 硝基,卤素,氰基,氰硫基,未取代或取代的脂族基团或取代的磺酰基或氨基; R 6是氢,卤素,C 1 -C 6烷基,C 1 -C 6 - 烷氧基,C 3 -C 8环烷基; 具有3-14个环原子的环系; R 16是羟基或取代的羟基;并且描述了它们的互变异构体或农业上有用的盐。此外,本发明描述了制备式I化合物的方法,包含它们的组合物,以及使用 式I化合物和组合物的化合物 包括它们用于控制有害植物。

    2-benzoylcyclohexane-1,3-dione as herbicides
    75.
    发明授权
    2-benzoylcyclohexane-1,3-dione as herbicides 有权
    2-苯甲酰基环己烷-1,3-二酮作为除草剂

    公开(公告)号:US06432881B1

    公开(公告)日:2002-08-13

    申请号:US09485231

    申请日:2000-02-07

    IPC分类号: C07D23112

    摘要: 2-Benzoylcyclohexane-1,3-diones of formula I : where: R1 and R2 are each hydrogen, mercapto, nitro, halogen, cyano, thiocyanato, alkyl, haloalkyl, alkoxy, alkenyl, alkynyl, —OR3, —OCOR3, —OSO2R3, —S(O)nR3 (n=0, 1, 2), —SO2OR3, —SO2N(R3)2, —NR3SO2R3 or —NR3COR3; R3 is hydrogen or optionally substituted alkyl, haloalkyl, alkenyl, alkynyl, phenyl or phenylalkyl; Q is optionally substituted cyclohexane-2-yl-1,3-dione; X1 is optionally substituted alkylene, propenylene, alkenylene or alkynylene; R4 is hydrogen or optionally substituted alkyl, alkenyl, alkynyl, phenyl, phenylalkyl; Het is a three- to six-membered, optionally substituted heterocyclic or heteroaromatic group; and agriculturally useful salts thereof, processes and intermediates for preparing compounds of formula I, compositions comprising them, and the use of the compounds of formula I and the compositions comprising them for controlling harmful plants are described.

    摘要翻译: 式I的2-苯甲酰基环己烷-1,3-二酮其中:R1和R2各自为氢,巯基,硝基,卤素,氰基,氰硫基,烷基,卤代烷基,烷氧基,烯基,炔基,-OR3,-OCOR3,-OSO2R3 ,-S(O)n R 3(n = 0,1,2),-SO 2 OR 3,-SO 2 N(R 3)2,-NR 3 SO 2 R 3或-NR 3 COR 3; R 3是氢或任选取代的烷基,卤代烷基,烯基,炔基,苯基或苯基 Q是任选取代的环己烷-2-基-1,3-二酮; X 1是任选取代的亚烷基,亚丙烯基,亚烯基或亚炔基; R 4是氢或任选取代的烷基,烯基,炔基,苯基,苯基烷基; 至六元,任选取代的杂环或杂芳族基团;及其农业上有用的盐,制备式I化合物的方法和中间体,包含它们的组合物,以及式I化合物及其组合物用于控制有害植物的用途 被描述。

    3-(heterocyclyl)-substituted benzolpyrazols
    77.
    发明授权
    3-(heterocyclyl)-substituted benzolpyrazols 失效
    3-(杂环基)取代的苯并吡唑

    公开(公告)号:US06831039B1

    公开(公告)日:2004-12-14

    申请号:US09857067

    申请日:2001-05-21

    IPC分类号: A01N4356

    CPC分类号: C07D413/10 C07D231/20

    摘要: The invention relates to 3-(heterocyclyl)-substituted benzoylpyrazois of formula (I), wherein the variables have the following meanings: X is O, NH or N-alkyl; R1 is alkyl; R2, R3, R4, R5 are hydrogen, alkyl or alkyl halide; R6 is halogen, nitro, alkyl halide, alkoxy, halogenalkoxy, alkylthio, halogenalkylthio, alkylsulfonyl or halogenalkylsulfonyl; R7 is hydroxy, alkoxy, alkenyloxy, alkylsulfonyloxy, alkylcarboyloxy, alkylthiocarbonyloxy, phenylsulfonyloxy or phenylcarbonyloxy, and the phenyl radical can be substituted; R8, R9 are alkyl; R10 is hydrogen or alkyl; and R11 is hydrogen or alkyl; and to their agriculturally useable salts. The invention also relates to intermediate products and methods for producing the inventive compounds and to the use of these compounds or products containing them for combating undesirable plants.

    摘要翻译: 本发明涉及式(I)的3-(杂环基)取代的苯甲酰基吡啶,其中变量具有以下含义:X是O,NH或N-烷基; R 1是烷基; R 2,R 3,R 4,R 5是氢,烷基或烷基卤; R 6是卤素,硝基,烷基卤,烷氧基,卤代烷氧基,烷硫基,卤代烷硫基,烷基磺酰基或卤代烷基磺酰基; R 7是羟基,烷氧基,烯氧基,烷基磺酰氧基,烷基羰氧基,烷硫基羰基氧基,苯基磺酰氧基或苯基羰基氧基,苯基可以被取代; R 8,R 9是烷基; R 10是氢或烷基; 和R 11是氢或烷基; 以及其农业上可用的盐类。 本发明还涉及用于生产本发明化合物的中间产物和方法以及含有它们的这些化合物或产品用于对抗不期望的植物的用途。

    2-benzoyl-cyclohexane-1,3-diones
    80.
    发明授权

    公开(公告)号:US06559100B1

    公开(公告)日:2003-05-06

    申请号:US09485223

    申请日:2000-02-07

    IPC分类号: C07D2604

    摘要: Substituted 2-benzoylcyclohexane-1,3-diones of the formula I where: R1 and R2 are each hydrogen, mercapto, nitro, halogen, cyano, thiocyanato, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C2-C6-alkenyl, C2-C6-alkynyl, —OR3, —OCOR3, —OSO2R3, —S(O)nR3, —SO2OR3, —SO2N(R3)2, —NR3SO2R3 or —NR3COR3; R3 is hydrogen, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-alkynyl, phenyl or phenyl-C1-C6-alkyl; where the abovementioned alkyl radicals may be partially or fully halogenated and/or may carry one to three of the following groups: hydroxyl, mercapto, amino, cyano, R3, —OR3, —SR3, —N(R3)2, ═NOR3, —OCOR3, —SCOR3, —NR3COR3, —CO2R3, —COSR3, —CON(R3)2, C1-C4-alkyliminooxy, C1-C4-alkoxyamino, C1-C4-alkylcarbonyl, C1-C4-alkoxy-C2-C6-alkoxycarbonyl, C1-C4-alkylsulfonyl, heterocyclyl, heterocyclyloxy, phenyl, benzyl, hetaryl, phenoxy, benzyloxy and hetaryloxy, where the eight last mentioned radicals may in turn be substituted; n is 0, 1 or 2; Q is a cyclohexane-1,3-dione ring with or without substitution which is attached in position 2; X1 is a straight-chain or branched C1-C6-alkylene, a C2-C6-alkenylene or a C2-C6-alkynylene chain, where the abovementioned alkylene, alkenylene or alkynylene radicals may be partially halogenated and/or may carry one to three of the following groups: —OR4, —OCOR4, —OCONHR4 or —OSO2R4; except for those of the abovementioned alkenylene radicals where the double bond is &agr;,&bgr; to the phenyl ring and where Het is linked to the double bond via the &bgr; position; R4 is hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, phenyl, phenyl-C1-C6-alkyl, where the abovementioned alkyl, alkenyl or alkynyl radicals may be partially or fully halogenated and/or may be substituted by one or more of the following radicals: hydroxyl, mercapto, amino, cyano, nitro, formyl, C1-C4-alkylamino, C1-C4-dialkylamino, C1-C4-alkoxycarbonyl, C1-C4-alkylcarbonyl, C1-C4-alkylcarbonyloxy, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkylthio, C1-C4-haloalkylthio, C1-C4-alkoxy, C1-C4-haloalkoxy; Het is a three- to six-membered partially or fully saturated heterocyclic group or a three- to six-membered heteroaromatic group having up to three hetero atoms selected from the group consisting of: nitrogen, oxygen or sulfur, where the abovementioned heterocyclic or heteroaromatic group may be partially or fully halogenated and/or may be substituted by R5; R5 is hydrogen, hydroxyl, mercapto, amino, cyano, nitro, formyl, C1-C4-alkylamino, C1-C4-dialkylamino, C1-C4-alkoxycarbonyl, C1-C4-alkylcarbonyl, C1-C4-alkylcarbonyloxy, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkylthio, C1-C4-haloalkylthio, C1-C4-alkoxy, C1-C4-haloalkoxy, where the alkyl radicals may in each case be substituted by in each case one or more of the following radicals: cyano, formyl, C1-C4-alkylamino, C1-C4-dialkylamino, C1-C4-alkoxycarbonyl, C1-C4-alkylcarbonyl, C1-C4-alkylcarbonyloxy, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkylthio, C1-C4-haloalkylthio, C1-C4-alkoxy, C1-C4-haloalkoxy; and agriculturally useful salts thereof, processes and intermediates for preparing compounds of the formula I, compositions comprising them, and the use of the compounds of the formula I and compositions comprising them for controlling harmful plants are described.