摘要:
1-AMINO-SULFONYL-2-AMINOBENZIMIDAZOLES OF THE FORMULA
IN WHICH X is halogen, lower alkyl or lower alkoxy, N IS 0, 1 OR 2, R and R'' each independently is alkyl with 1 to 6 carbon atoms optionally substituted by at least one of halogen, cyano and lower alkoxy, or R and R'', together with the connecting nitrogen atom, is a heterocyclic ring with 4 to 7 carbon atoms, which possess fungicidal properties.
摘要:
1-(2''-CYCLOHEXYLIDENIMINOPHENYL) - 3 - ALKOXYCARBONYL2-THIOUREAS OF THE GENERAL FORMULA IN WHICH X IS HYDROGEN OR ALKYL WITH 1 TO 6 CARBON ATOMS, N IS 0, 1, 2 OR 3, R IS LOWER ALKYL, AND R'' IS ALKYL WITH 1 TO 6 CARBON ATOMS, WHICH POSSESS FUNGICIDAL, BACTERICIDAL, INSECTICIDAL AND ACARICIDAL PROPERTIES.
IN WHICH X STANDS FOR HALOGEN, LOWER ALKYL OR LOWER ALKOXY, N STANDS FOR 0, OR 2, R AND R'' STANDS FOR HYROGEN OR LOWER ALKYL, R" STANDS FOR HYDROGEN, CYCLOALKYL, ALKYLSULFONYL WITH UP TO 18 CARBON ATOMS, DI-LOWER ALKYLANINO, OR OPTIONALLY SUBSITUTED ALKYL WITH UP TO 18 CARBON ATOMS, AROYL OR ARYLPHENYL, ACYL WITH UP TO 18 CARBON ATOMS, AROYL OR ARYLSULFONYL, OR R'' AND R" JOINTLY WITH THE CONNECTING NITROGEN ATOMS STAND SOR A HETEROCYCLIC RING WITH 4 TO 7 RING CARBON ATOMS, THE RING POSSIBLY CONTAINING OXYGEN OR SULFUR AS FURTHER HETERO ATOMS, AND R"'' STANDS FOR ALKYL WITH UP TO 12 CARBON ATOMS, WHICH POSSESS FUNGICIDAL PROPERTIES.
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
摘要:
1-(N-(ALKYL, CYCLOALKYL, PHENYL OR SUBSTITUTED PHENYL)-SOR -O-CARBONYL-CARBAMIDYL)-BENZIMIDAZOLE-2-YL-CARBAMIC ACID ALKYL ESTERS, WHICH POSSESS FUNGICIDAL PROPERTIES AND WHICH MAY BE PRODUCED BY CONVENTIONAL METHODS.
IN WHICH N IS 0, 1 OR 2, EACH X is halogen, lower alkyl or lower alkoxy, R is lower alkyl, R'' is hydrogen or lower alkyl, R'''' is hydrogen; alkyl optionally substituted by at least one of halogen, nitrile, lower alkoxy, lower alkylmercapto, lower alkoxycarbonyl, phenoxy, halogenophenoxy, alkylphenoxy, alkoxyphenoxy and arylmercapto; cycloalkyl; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or a five- or six-membered heterocyclic radical containing at least one oxygen, sulfur or nitrogen heteroatom, and R'''''' is alkyl; cycloalkyl; alkenyl; or aralkyl optionally substituted in the aryl moiety by at least one of lower alkyl, lower alkoxy and halogen, WHICH POSSESS FUNGICIDAL PROPERTIES.
摘要:
IN WHICH X is halogen, lower alkyl or lower alkoxy, N IS 0, 1 OR 2, R is hydrogen or lower alkyl, R1 is alkyl of 1-6 carbon atoms, R2 is hydrogen, alkyl with 1-18 carbon atoms optionally substituted by halogen, cyano, lower alkoxy, lower alkoxycarbonyl, phenoxy, halophenoxy, alkylphenoxy or alkoxyphenoxy; cycloalkyl of 5-8 carbon atoms; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or furyl; and R3 is hydrogen, alkyl with 1-18 carbon atoms optionally substituted by halogen, cyano, lower alkoxy, lower alkoxycarbonyl, phenoxy, halophenoxy, alkylphenoxy or alkoxyphenoxy; alkenyl or alkynyl of 2-12 carbon atoms; cycloalkyl of 5-8 carbon atoms; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or furyl, WHICH POSSESS FUNGICIDAL PROPERTIES.
N-alkoxycarbonyl-N''-acyl-N''''-2-acylamidophenyl-guanidines of the formula
摘要:
Amidophenylisothioureas of the formula IN WHICH N IS 0, 1 OR 2, EACH X is halogen, lower alkyl or lower alkoxy, R is lower alkyl, R'' is hydrogen or lower alkyl, R'''' is hydrogen; alkyl optionally substituted by at least one of halogen, nitrile, lower alkoxy, lower alkylmercapto, lower alkoxycarbonyl, phenoxy, halogenophenoxy; alkylphenoxy, alkoxyphenoxy and arylmercapto; cycloalkyl; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or a five- or six-membered heterocyclic radical containing at least one oxygen, sulfur or nitrogen heteroatom, and R'''''' is alkyl; cycloalkyl; alkenyl; or aralkyl optionally substituted in the aryl moiety by at least one of lower alkyl, lower alkoxy and halogen, WHICH POSSESS FUNGICIDAL PROPERTIES.
IN WHICH X IS HALOGEN, LOWER ALKYL OR LOWER ALKOXY, N IS 0, 1 OR 2 R AND R'' EACH INDEPENDENTLY IS ALKYL OF 1 TO 6 CARBON ATOMS, OR R AND R'' TOGETHER WITH THE LINKING NITROGEN ATOM ARE PYRROLIDINO, PIPERIDINO OR MORPHOLINO, OR R" IS ALKYL OF 1 TO 6 CARBON ATOMS OPTIONALLY SUBSTITUTED BY LOWER ALKOXY OR HALOGEN, CYCLOALKYL OF 3 TO 8 CARBON ATOMS, BENZYL OR PHENYL OPTIONALLY SUBSTITUTED BY AT LEAST ONE OF CHKORINE OR METHYL, OR ALKOXY OF 1 TO 6 CARBON ATOMS.