1-amino-sulfonyl-2-aminobenzimidazoles
    1.
    发明授权
    1-amino-sulfonyl-2-aminobenzimidazoles 失效
    1-氨基 - 磺酰基-2-氨基苯并咪唑

    公开(公告)号:US3853908A

    公开(公告)日:1974-12-10

    申请号:US32899873

    申请日:1973-02-02

    申请人: BAYER AG

    CPC分类号: C07D235/30

    摘要: 1-AMINO-SULFONYL-2-AMINOBENZIMIDAZOLES OF THE FORMULA

    IN WHICH X is halogen, lower alkyl or lower alkoxy, N IS 0, 1 OR 2, R and R'' each independently is alkyl with 1 to 6 carbon atoms optionally substituted by at least one of halogen, cyano and lower alkoxy, or R and R'', together with the connecting nitrogen atom, is a heterocyclic ring with 4 to 7 carbon atoms, which possess fungicidal properties.

    摘要翻译: 其中X为卤素,低级烷基或低级烷氧基,N为0,1或2,R及R'各自独立地为具有1至6个碳原子的烷基,任选被 卤素,氰基和低级烷氧基中的至少一个,或R和R'连同连接的氮原子是具有4至7个碳原子的杂环,具有杀真菌性质。

    Substituted ureidophenylguanidines
    3.
    发明授权
    Substituted ureidophenylguanidines 失效
    取代的尿嘧啶

    公开(公告)号:US3828094A

    公开(公告)日:1974-08-06

    申请号:US8314770

    申请日:1970-10-22

    申请人: BAYER AG

    CPC分类号: A01N47/44

    摘要: SUBSITUTED UREIDOPHENYLGUANIDINES OF THE FORMULA

    1-(R"''-O-CO-N=C(-NH-CO-O-R"'')-NH-),2-(R''-N(-R")-CO-N(-R)-)

    ,(X)N-BENZENE

    IN WHICH X STANDS FOR HALOGEN, LOWER ALKYL OR LOWER ALKOXY, N STANDS FOR 0, OR 2, R AND R'' STANDS FOR HYROGEN OR LOWER ALKYL, R" STANDS FOR HYDROGEN, CYCLOALKYL, ALKYLSULFONYL WITH UP TO 18 CARBON ATOMS, DI-LOWER ALKYLANINO, OR OPTIONALLY SUBSITUTED ALKYL WITH UP TO 18 CARBON ATOMS, AROYL OR ARYLPHENYL, ACYL WITH UP TO 18 CARBON ATOMS, AROYL OR ARYLSULFONYL, OR R'' AND R" JOINTLY WITH THE CONNECTING NITROGEN ATOMS STAND SOR A HETEROCYCLIC RING WITH 4 TO 7 RING CARBON ATOMS, THE RING POSSIBLY CONTAINING OXYGEN OR SULFUR AS FURTHER HETERO ATOMS, AND R"'' STANDS FOR ALKYL WITH UP TO 12 CARBON ATOMS, WHICH POSSESS FUNGICIDAL PROPERTIES.

    Substituted ureidophenyl thioureas
    4.
    发明授权
    Substituted ureidophenyl thioureas 失效
    替代性尿毒症

    公开(公告)号:US3780089A

    公开(公告)日:1973-12-18

    申请号:US3780089D

    申请日:1970-11-13

    申请人: BAYER AG

    CPC分类号: C07C335/28

    摘要: UREIDOPHENYL THIOUREAS OF THE FORMULA:

    1-(R-OOC-NH-C(=S)-NH-),2-(R"-N(-R''")-CO-N(-R'')-),(X)N-

    BENZENE

    IN WHICH

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

    Amidophenylisothioureas
    6.
    发明授权
    Amidophenylisothioureas 失效
    AMIDOPHENYLISOTHIOUREAS

    公开(公告)号:US3843715A

    公开(公告)日:1974-10-22

    申请号:US14197871

    申请日:1971-05-10

    申请人: BAYER AG

    CPC分类号: C07C335/38

    摘要: Amidophenylisothioureas of the formula

    IN WHICH N IS 0, 1 OR 2, EACH X is halogen, lower alkyl or lower alkoxy, R is lower alkyl, R'' is hydrogen or lower alkyl, R'''' is hydrogen; alkyl optionally substituted by at least one of halogen, nitrile, lower alkoxy, lower alkylmercapto, lower alkoxycarbonyl, phenoxy, halogenophenoxy, alkylphenoxy, alkoxyphenoxy and arylmercapto; cycloalkyl; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or a five- or six-membered heterocyclic radical containing at least one oxygen, sulfur or nitrogen heteroatom, and R'''''' is alkyl; cycloalkyl; alkenyl; or aralkyl optionally substituted in the aryl moiety by at least one of lower alkyl, lower alkoxy and halogen, WHICH POSSESS FUNGICIDAL PROPERTIES.

    N-alkoxycarbonyl-n{40 -acyl-n{41 12-acylamidophenyl-guanidines
    7.
    发明授权
    N-alkoxycarbonyl-n{40 -acyl-n{41 12-acylamidophenyl-guanidines 失效
    N-烷氧羰基-N {40-乙酰基-N- {41,12-氰基戊烯 - 胍

    公开(公告)号:US3835164A

    公开(公告)日:1974-09-10

    申请号:US30330172

    申请日:1972-11-02

    申请人: BAYER AG

    CPC分类号: C07D307/68

    摘要: IN WHICH X is halogen, lower alkyl or lower alkoxy, N IS 0, 1 OR 2, R is hydrogen or lower alkyl, R1 is alkyl of 1-6 carbon atoms, R2 is hydrogen, alkyl with 1-18 carbon atoms optionally substituted by halogen, cyano, lower alkoxy, lower alkoxycarbonyl, phenoxy, halophenoxy, alkylphenoxy or alkoxyphenoxy; cycloalkyl of 5-8 carbon atoms; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or furyl; and R3 is hydrogen, alkyl with 1-18 carbon atoms optionally substituted by halogen, cyano, lower alkoxy, lower alkoxycarbonyl, phenoxy, halophenoxy, alkylphenoxy or alkoxyphenoxy; alkenyl or alkynyl of 2-12 carbon atoms; cycloalkyl of 5-8 carbon atoms; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or furyl, WHICH POSSESS FUNGICIDAL PROPERTIES.

    N-alkoxycarbonyl-N''-acyl-N''''-2-acylamidophenyl-guanidines of the formula

    摘要翻译: N-烷氧基羰基-N'-酰基-N“ - 2-酰氨基苯基 - 胍,其中X为卤素,低级烷基或低级烷氧基,N为0,1或2,R为氢或低级烷基,R 1为 氰基,低级烷氧基,低级烷氧基羰基,苯氧基,卤代苯氧基,烷基苯氧基或烷氧基苯氧基;具有1-6个碳原子的烷基, 5-8个碳原子的环烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳基; 或呋喃基; 氰基,低级烷氧基,低级烷氧基羰基,苯氧基,卤代苯氧基,烷基苯氧基或烷氧基苯氧基;具有1-18个碳原子的烷基, 2-12个碳原子的烯基或炔基; 5-8个碳原子的环烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳基; 或呋喃,哪些具有杀真菌性质。

    Combating fungi with amidophenylisothioureas
    9.
    发明授权
    Combating fungi with amidophenylisothioureas 失效
    组合真菌与感染性血友病

    公开(公告)号:US3852463A

    公开(公告)日:1974-12-03

    申请号:US36048473

    申请日:1973-05-15

    申请人: BAYER AG

    IPC分类号: C07C335/38 A01N9/12 A01N9/20

    CPC分类号: C07C335/38 Y10S424/08

    摘要: Amidophenylisothioureas of the formula IN WHICH N IS 0, 1 OR 2, EACH X is halogen, lower alkyl or lower alkoxy, R is lower alkyl, R'' is hydrogen or lower alkyl, R'''' is hydrogen; alkyl optionally substituted by at least one of halogen, nitrile, lower alkoxy, lower alkylmercapto, lower alkoxycarbonyl, phenoxy, halogenophenoxy; alkylphenoxy, alkoxyphenoxy and arylmercapto; cycloalkyl; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or a five- or six-membered heterocyclic radical containing at least one oxygen, sulfur or nitrogen heteroatom, and R'''''' is alkyl; cycloalkyl; alkenyl; or aralkyl optionally substituted in the aryl moiety by at least one of lower alkyl, lower alkoxy and halogen, WHICH POSSESS FUNGICIDAL PROPERTIES.

    摘要翻译: 式I其中N为0,1或2的苯基异硫脲,每个X为卤素,低级烷基或低级烷氧基,R为低级烷基,R'为氢或低级烷基,R“为氢; 任选被卤素,腈,低级烷氧基,低级烷基巯基,低级烷氧基羰基,苯氧基,卤素苯氧基中的至少一种取代的烷基; 烷基苯氧基,烷氧基苯氧基和芳基巯基; 环烷基 任选被卤素,低级烷基或低级烷氧基取代的芳烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳基; 或含有至少一个氧,硫或氮杂原子的五元或六元杂环基,R“是烷基; 环烷基 烯基; 或在芳基部分中被至少一个低级烷基,低级烷氧基和卤素取代的芳烷基,其具有无害的杀真菌性质。

    1-acyl-3-aminosulfonyl-2-imino-benzimidazolines
    10.
    发明授权
    1-acyl-3-aminosulfonyl-2-imino-benzimidazolines 失效
    1-亚氨基-3-氨基磺酰基-2-亚氨基 - 苯并咪唑

    公开(公告)号:US3850954A

    公开(公告)日:1974-11-26

    申请号:US32900073

    申请日:1973-02-02

    申请人: BAYER AG

    CPC分类号: C07D235/30

    摘要: 1. A 1-ACYL-3-AMINOSULFONY-2-IMON0-BENZIMIDAZOLINE OF THE FORMULA

    1-(R"-CO-),2-(HN=),3-(R-N(-R'')-SO2-),X(N)-BENZIMIDAZOLINE

    IN WHICH X IS HALOGEN, LOWER ALKYL OR LOWER ALKOXY, N IS 0, 1 OR 2 R AND R'' EACH INDEPENDENTLY IS ALKYL OF 1 TO 6 CARBON ATOMS, OR R AND R'' TOGETHER WITH THE LINKING NITROGEN ATOM ARE PYRROLIDINO, PIPERIDINO OR MORPHOLINO, OR R" IS ALKYL OF 1 TO 6 CARBON ATOMS OPTIONALLY SUBSTITUTED BY LOWER ALKOXY OR HALOGEN, CYCLOALKYL OF 3 TO 8 CARBON ATOMS, BENZYL OR PHENYL OPTIONALLY SUBSTITUTED BY AT LEAST ONE OF CHKORINE OR METHYL, OR ALKOXY OF 1 TO 6 CARBON ATOMS.