1-amino-sulfonyl-2-aminobenzimidazoles
    1.
    发明授权
    1-amino-sulfonyl-2-aminobenzimidazoles 失效
    1-氨基 - 磺酰基-2-氨基苯并咪唑

    公开(公告)号:US3853908A

    公开(公告)日:1974-12-10

    申请号:US32899873

    申请日:1973-02-02

    Applicant: BAYER AG

    CPC classification number: C07D235/30

    Abstract: 1-AMINO-SULFONYL-2-AMINOBENZIMIDAZOLES OF THE FORMULA

    IN WHICH X is halogen, lower alkyl or lower alkoxy, N IS 0, 1 OR 2, R and R'' each independently is alkyl with 1 to 6 carbon atoms optionally substituted by at least one of halogen, cyano and lower alkoxy, or R and R'', together with the connecting nitrogen atom, is a heterocyclic ring with 4 to 7 carbon atoms, which possess fungicidal properties.

    Abstract translation: 其中X为卤素,低级烷基或低级烷氧基,N为0,1或2,R及R'各自独立地为具有1至6个碳原子的烷基,任选被 卤素,氰基和低级烷氧基中的至少一个,或R和R'连同连接的氮原子是具有4至7个碳原子的杂环,具有杀真菌性质。

    Fungicidal compositions and methods of combating fungi using n-acyl-para-dialkylaminophenyl-hydrazones
    3.
    发明授权
    Fungicidal compositions and methods of combating fungi using n-acyl-para-dialkylaminophenyl-hydrazones 失效
    杀真菌剂组合物及使用N-乙酰 - 对二甲氨基苯丙氨酸的真菌组合方法

    公开(公告)号:US3760078A

    公开(公告)日:1973-09-18

    申请号:US3760078D

    申请日:1972-02-08

    Applicant: BAYER AG

    CPC classification number: A01N37/44

    Abstract: N-acyl-para-dialkylaminophenyl-hydrazones, i.e., N-(4dialkylamino- and 4- tetra to penta methylene-imino-substituted phenyl)-N-(alkanoyl, chloroalkanoyl, alkenoyl, carboalkoxy, benzoyl and carbophenoxy)-N''-((acetyl and cyano)- (alkanoyl and carboalkoxy)-carbonyl)-hydrazones, or N-(4- dialkylamino-, 4pyrrolidino- and 4-piperidino- substituted phenyl)-N(alkylcarbonyl, chloroalkylcarbonyl, alkenylcarbonyl, alkoxycarbonyl, phenylcarbonyl and phenoxycarbonyl)-N''((methylcarbonyl and cyano)-(alkylcarbonyl and alkoxycarbonyl)carbonyl)-hydrazones, which possess fungicidal properties.

    N-trityl-imidazolium salts as a fungicide
    4.
    发明授权
    N-trityl-imidazolium salts as a fungicide 失效
    作为杀真菌剂的N-三嗪咪唑盐

    公开(公告)号:US3719760A

    公开(公告)日:1973-03-06

    申请号:US7363870

    申请日:1970-09-18

    Applicant: BAYER AG

    CPC classification number: C07D231/12 C07D233/56 C07D249/08

    Abstract: Plant fungicidal compositions are produced which comprise an amount of a compound of the formula:

    WHEREIN Y is the anion of an inorganic or organic acid, sufficient to be effective for killing, combatting or controlling plant fungi, in combination with a solid or liquid diluent or carrier. Methods for killing, combatting or controlling fungal diseases in plants comprise applying to the fungi or to the plant to be protected an effective or toxic amount of the above compound.

    Amidophenylisothioureas
    5.
    发明授权
    Amidophenylisothioureas 失效
    AMIDOPHENYLISOTHIOUREAS

    公开(公告)号:US3843715A

    公开(公告)日:1974-10-22

    申请号:US14197871

    申请日:1971-05-10

    Applicant: BAYER AG

    CPC classification number: C07C335/38

    Abstract: Amidophenylisothioureas of the formula

    IN WHICH N IS 0, 1 OR 2, EACH X is halogen, lower alkyl or lower alkoxy, R is lower alkyl, R'' is hydrogen or lower alkyl, R'''' is hydrogen; alkyl optionally substituted by at least one of halogen, nitrile, lower alkoxy, lower alkylmercapto, lower alkoxycarbonyl, phenoxy, halogenophenoxy, alkylphenoxy, alkoxyphenoxy and arylmercapto; cycloalkyl; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or a five- or six-membered heterocyclic radical containing at least one oxygen, sulfur or nitrogen heteroatom, and R'''''' is alkyl; cycloalkyl; alkenyl; or aralkyl optionally substituted in the aryl moiety by at least one of lower alkyl, lower alkoxy and halogen, WHICH POSSESS FUNGICIDAL PROPERTIES.

    N-alkoxycarbonyl-n{40 -acyl-n{41 12-acylamidophenyl-guanidines
    6.
    发明授权
    N-alkoxycarbonyl-n{40 -acyl-n{41 12-acylamidophenyl-guanidines 失效
    N-烷氧羰基-N {40-乙酰基-N- {41,12-氰基戊烯 - 胍

    公开(公告)号:US3835164A

    公开(公告)日:1974-09-10

    申请号:US30330172

    申请日:1972-11-02

    Applicant: BAYER AG

    CPC classification number: C07D307/68

    Abstract: IN WHICH X is halogen, lower alkyl or lower alkoxy, N IS 0, 1 OR 2, R is hydrogen or lower alkyl, R1 is alkyl of 1-6 carbon atoms, R2 is hydrogen, alkyl with 1-18 carbon atoms optionally substituted by halogen, cyano, lower alkoxy, lower alkoxycarbonyl, phenoxy, halophenoxy, alkylphenoxy or alkoxyphenoxy; cycloalkyl of 5-8 carbon atoms; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or furyl; and R3 is hydrogen, alkyl with 1-18 carbon atoms optionally substituted by halogen, cyano, lower alkoxy, lower alkoxycarbonyl, phenoxy, halophenoxy, alkylphenoxy or alkoxyphenoxy; alkenyl or alkynyl of 2-12 carbon atoms; cycloalkyl of 5-8 carbon atoms; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or furyl, WHICH POSSESS FUNGICIDAL PROPERTIES.

    N-alkoxycarbonyl-N''-acyl-N''''-2-acylamidophenyl-guanidines of the formula

    Abstract translation: N-烷氧基羰基-N'-酰基-N“ - 2-酰氨基苯基 - 胍,其中X为卤素,低级烷基或低级烷氧基,N为0,1或2,R为氢或低级烷基,R 1为 氰基,低级烷氧基,低级烷氧基羰基,苯氧基,卤代苯氧基,烷基苯氧基或烷氧基苯氧基;具有1-6个碳原子的烷基, 5-8个碳原子的环烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳基; 或呋喃基; 氰基,低级烷氧基,低级烷氧基羰基,苯氧基,卤代苯氧基,烷基苯氧基或烷氧基苯氧基;具有1-18个碳原子的烷基, 2-12个碳原子的烯基或炔基; 5-8个碳原子的环烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳基; 或呋喃,哪些具有杀真菌性质。

    Combating fungi with amidophenylisothioureas
    8.
    发明授权
    Combating fungi with amidophenylisothioureas 失效
    组合真菌与感染性血友病

    公开(公告)号:US3852463A

    公开(公告)日:1974-12-03

    申请号:US36048473

    申请日:1973-05-15

    Applicant: BAYER AG

    CPC classification number: C07C335/38 Y10S424/08

    Abstract: Amidophenylisothioureas of the formula IN WHICH N IS 0, 1 OR 2, EACH X is halogen, lower alkyl or lower alkoxy, R is lower alkyl, R'' is hydrogen or lower alkyl, R'''' is hydrogen; alkyl optionally substituted by at least one of halogen, nitrile, lower alkoxy, lower alkylmercapto, lower alkoxycarbonyl, phenoxy, halogenophenoxy; alkylphenoxy, alkoxyphenoxy and arylmercapto; cycloalkyl; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or a five- or six-membered heterocyclic radical containing at least one oxygen, sulfur or nitrogen heteroatom, and R'''''' is alkyl; cycloalkyl; alkenyl; or aralkyl optionally substituted in the aryl moiety by at least one of lower alkyl, lower alkoxy and halogen, WHICH POSSESS FUNGICIDAL PROPERTIES.

    Abstract translation: 式I其中N为0,1或2的苯基异硫脲,每个X为卤素,低级烷基或低级烷氧基,R为低级烷基,R'为氢或低级烷基,R“为氢; 任选被卤素,腈,低级烷氧基,低级烷基巯基,低级烷氧基羰基,苯氧基,卤素苯氧基中的至少一种取代的烷基; 烷基苯氧基,烷氧基苯氧基和芳基巯基; 环烷基 任选被卤素,低级烷基或低级烷氧基取代的芳烷基; 任选被卤素,低级烷基或低级烷氧基取代的芳基; 或含有至少一个氧,硫或氮杂原子的五元或六元杂环基,R“是烷基; 环烷基 烯基; 或在芳基部分中被至少一个低级烷基,低级烷氧基和卤素取代的芳烷基,其具有无害的杀真菌性质。

    1-acyl-3-aminosulfonyl-2-imino-benzimidazolines
    9.
    发明授权
    1-acyl-3-aminosulfonyl-2-imino-benzimidazolines 失效
    1-亚氨基-3-氨基磺酰基-2-亚氨基 - 苯并咪唑

    公开(公告)号:US3850954A

    公开(公告)日:1974-11-26

    申请号:US32900073

    申请日:1973-02-02

    Applicant: BAYER AG

    CPC classification number: C07D235/30

    Abstract: 1. A 1-ACYL-3-AMINOSULFONY-2-IMON0-BENZIMIDAZOLINE OF THE FORMULA

    1-(R"-CO-),2-(HN=),3-(R-N(-R'')-SO2-),X(N)-BENZIMIDAZOLINE

    IN WHICH X IS HALOGEN, LOWER ALKYL OR LOWER ALKOXY, N IS 0, 1 OR 2 R AND R'' EACH INDEPENDENTLY IS ALKYL OF 1 TO 6 CARBON ATOMS, OR R AND R'' TOGETHER WITH THE LINKING NITROGEN ATOM ARE PYRROLIDINO, PIPERIDINO OR MORPHOLINO, OR R" IS ALKYL OF 1 TO 6 CARBON ATOMS OPTIONALLY SUBSTITUTED BY LOWER ALKOXY OR HALOGEN, CYCLOALKYL OF 3 TO 8 CARBON ATOMS, BENZYL OR PHENYL OPTIONALLY SUBSTITUTED BY AT LEAST ONE OF CHKORINE OR METHYL, OR ALKOXY OF 1 TO 6 CARBON ATOMS.

    Ureidophenylisothioureas
    10.
    发明授权
    Ureidophenylisothioureas 失效
    UREIDOPHENYLISOTHIOUREAS

    公开(公告)号:US3766243A

    公开(公告)日:1973-10-16

    申请号:US3766243D

    申请日:1971-05-10

    Applicant: BAYER AG

    CPC classification number: C07C335/38 A01N47/42

    Abstract: UREIDOPHENYLISOTHIOUREAS OF THE FORMULA

    1-(R-OOC-NH-C(-S-R"")=N-),2-(R"-N(-R''")-CO-N(-R'')-),(X)N-

    BENZENE

    IN WHICH N IS 0, 1 OR 2 X IS HALOGEN, LOWER ALKYL OR ALKOXY, R IS LOWER ALKYL, R'' AND R" ARE EACH HYDROGEN OR LOWER ALKYL, R"'' IS HYDROGEN; ALKYL WITH 1 TO 18 CARBON ATOMS OPTIONALLY SUBSTITUTED BY HALOGEN, NITRILE, LOWER ALKOXY OR LOWER ALKOXYCARBONYL; CYCLOALKYL WITH 5 TO 8 CARBON ATOMS; ARALKYL OPTIONALLY SUBSTITUTED IN THE ARYL MOIETY BY HALOGEN, LOWER ALKYL OR ALKOXY; PHENYL OPTIONALLY SUBSTITUTED BY HALOGEN, LOWER ALKYL OR ALKOXY; ACYL WITH UP TO 18 CARBON ATOMS OPTIONALLY SUBSTITUTED BY HALOGEN OR LOWER ALKOXY; AROYL OPTIONALLY SUBSTITUTED BY HALOGEN, LOWER ALKYL OR ALKOXY; ALKYSULFONYL; ARYLSULFONYL OPTIONALLY SUBSTITUTED BY HALOGEN, AMINO, LOWER ALKYL OR ALKOXY; OR DI-LOWER ALKYLAMINO; OR R" AND R"'', TOGETHER WITH THE BONDING NITROGEN ATOM, FORM A HETEROCYCLIC RING WITH 4 TO 7 CARBON ATOMS, WHICH RING OPTIONALLY CONTAINS OXYGEN OR SULFUR AS FURTHER HETERO-ATOMS, AND R"" IS ALKYL WITH 1 TO 12 CARBON ATOMS, CYCLOALKYL WITH 3 TO 8 CARBON ATOMS, ALKENYL WITH UP TO 12 CARBON ATOMS OR ARALKYL OPTIONALLY SUBSTITUTED IN THE ARYL MOIETY BY HALOGEN, LOWER ALKYL OR ALKOXY, WHICH POSSESS FUNGICIDAL, INSECTICIDAL ACARICIDAL, ANTIBACTERIAL AND GROWTH-REGULATING PROPERTIES.

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