Abstract:
1-AMINO-SULFONYL-2-AMINOBENZIMIDAZOLES OF THE FORMULA
IN WHICH X is halogen, lower alkyl or lower alkoxy, N IS 0, 1 OR 2, R and R'' each independently is alkyl with 1 to 6 carbon atoms optionally substituted by at least one of halogen, cyano and lower alkoxy, or R and R'', together with the connecting nitrogen atom, is a heterocyclic ring with 4 to 7 carbon atoms, which possess fungicidal properties.
Abstract:
Fungicidal and bactericidal compositions of and methods of combating fungi and bacteria using dihalocyclopentendiones of the formula
IN WHICH R is a vinyl, aryl or hetero-aromatic radical, which radical may optionally be substituted with lower alkyl, lower haloalkyl, benzyl, phenyl, di-(lower alkyl)amino wherein each alkyl group is independently optionally substituted by halogen, halogen, nitro, nitrile, formyl, carboxyl, alkoxycarbonyl, hydroxyl, alkoxy and azolyl, and Hal is halogen are disclosed.
Abstract:
N-acyl-para-dialkylaminophenyl-hydrazones, i.e., N-(4dialkylamino- and 4- tetra to penta methylene-imino-substituted phenyl)-N-(alkanoyl, chloroalkanoyl, alkenoyl, carboalkoxy, benzoyl and carbophenoxy)-N''-((acetyl and cyano)- (alkanoyl and carboalkoxy)-carbonyl)-hydrazones, or N-(4- dialkylamino-, 4pyrrolidino- and 4-piperidino- substituted phenyl)-N(alkylcarbonyl, chloroalkylcarbonyl, alkenylcarbonyl, alkoxycarbonyl, phenylcarbonyl and phenoxycarbonyl)-N''((methylcarbonyl and cyano)-(alkylcarbonyl and alkoxycarbonyl)carbonyl)-hydrazones, which possess fungicidal properties.
Abstract:
Plant fungicidal compositions are produced which comprise an amount of a compound of the formula:
WHEREIN Y is the anion of an inorganic or organic acid, sufficient to be effective for killing, combatting or controlling plant fungi, in combination with a solid or liquid diluent or carrier. Methods for killing, combatting or controlling fungal diseases in plants comprise applying to the fungi or to the plant to be protected an effective or toxic amount of the above compound.
IN WHICH N IS 0, 1 OR 2, EACH X is halogen, lower alkyl or lower alkoxy, R is lower alkyl, R'' is hydrogen or lower alkyl, R'''' is hydrogen; alkyl optionally substituted by at least one of halogen, nitrile, lower alkoxy, lower alkylmercapto, lower alkoxycarbonyl, phenoxy, halogenophenoxy, alkylphenoxy, alkoxyphenoxy and arylmercapto; cycloalkyl; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or a five- or six-membered heterocyclic radical containing at least one oxygen, sulfur or nitrogen heteroatom, and R'''''' is alkyl; cycloalkyl; alkenyl; or aralkyl optionally substituted in the aryl moiety by at least one of lower alkyl, lower alkoxy and halogen, WHICH POSSESS FUNGICIDAL PROPERTIES.
Abstract:
IN WHICH X is halogen, lower alkyl or lower alkoxy, N IS 0, 1 OR 2, R is hydrogen or lower alkyl, R1 is alkyl of 1-6 carbon atoms, R2 is hydrogen, alkyl with 1-18 carbon atoms optionally substituted by halogen, cyano, lower alkoxy, lower alkoxycarbonyl, phenoxy, halophenoxy, alkylphenoxy or alkoxyphenoxy; cycloalkyl of 5-8 carbon atoms; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or furyl; and R3 is hydrogen, alkyl with 1-18 carbon atoms optionally substituted by halogen, cyano, lower alkoxy, lower alkoxycarbonyl, phenoxy, halophenoxy, alkylphenoxy or alkoxyphenoxy; alkenyl or alkynyl of 2-12 carbon atoms; cycloalkyl of 5-8 carbon atoms; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or furyl, WHICH POSSESS FUNGICIDAL PROPERTIES.
N-alkoxycarbonyl-N''-acyl-N''''-2-acylamidophenyl-guanidines of the formula
Abstract:
Amidophenylisothioureas of the formula IN WHICH N IS 0, 1 OR 2, EACH X is halogen, lower alkyl or lower alkoxy, R is lower alkyl, R'' is hydrogen or lower alkyl, R'''' is hydrogen; alkyl optionally substituted by at least one of halogen, nitrile, lower alkoxy, lower alkylmercapto, lower alkoxycarbonyl, phenoxy, halogenophenoxy; alkylphenoxy, alkoxyphenoxy and arylmercapto; cycloalkyl; aralkyl optionally substituted by halogen, lower alkyl or lower alkoxy; aryl optionally substituted by halogen, lower alkyl or lower alkoxy; or a five- or six-membered heterocyclic radical containing at least one oxygen, sulfur or nitrogen heteroatom, and R'''''' is alkyl; cycloalkyl; alkenyl; or aralkyl optionally substituted in the aryl moiety by at least one of lower alkyl, lower alkoxy and halogen, WHICH POSSESS FUNGICIDAL PROPERTIES.
IN WHICH X IS HALOGEN, LOWER ALKYL OR LOWER ALKOXY, N IS 0, 1 OR 2 R AND R'' EACH INDEPENDENTLY IS ALKYL OF 1 TO 6 CARBON ATOMS, OR R AND R'' TOGETHER WITH THE LINKING NITROGEN ATOM ARE PYRROLIDINO, PIPERIDINO OR MORPHOLINO, OR R" IS ALKYL OF 1 TO 6 CARBON ATOMS OPTIONALLY SUBSTITUTED BY LOWER ALKOXY OR HALOGEN, CYCLOALKYL OF 3 TO 8 CARBON ATOMS, BENZYL OR PHENYL OPTIONALLY SUBSTITUTED BY AT LEAST ONE OF CHKORINE OR METHYL, OR ALKOXY OF 1 TO 6 CARBON ATOMS.
IN WHICH N IS 0, 1 OR 2 X IS HALOGEN, LOWER ALKYL OR ALKOXY, R IS LOWER ALKYL, R'' AND R" ARE EACH HYDROGEN OR LOWER ALKYL, R"'' IS HYDROGEN; ALKYL WITH 1 TO 18 CARBON ATOMS OPTIONALLY SUBSTITUTED BY HALOGEN, NITRILE, LOWER ALKOXY OR LOWER ALKOXYCARBONYL; CYCLOALKYL WITH 5 TO 8 CARBON ATOMS; ARALKYL OPTIONALLY SUBSTITUTED IN THE ARYL MOIETY BY HALOGEN, LOWER ALKYL OR ALKOXY; PHENYL OPTIONALLY SUBSTITUTED BY HALOGEN, LOWER ALKYL OR ALKOXY; ACYL WITH UP TO 18 CARBON ATOMS OPTIONALLY SUBSTITUTED BY HALOGEN OR LOWER ALKOXY; AROYL OPTIONALLY SUBSTITUTED BY HALOGEN, LOWER ALKYL OR ALKOXY; ALKYSULFONYL; ARYLSULFONYL OPTIONALLY SUBSTITUTED BY HALOGEN, AMINO, LOWER ALKYL OR ALKOXY; OR DI-LOWER ALKYLAMINO; OR R" AND R"'', TOGETHER WITH THE BONDING NITROGEN ATOM, FORM A HETEROCYCLIC RING WITH 4 TO 7 CARBON ATOMS, WHICH RING OPTIONALLY CONTAINS OXYGEN OR SULFUR AS FURTHER HETERO-ATOMS, AND R"" IS ALKYL WITH 1 TO 12 CARBON ATOMS, CYCLOALKYL WITH 3 TO 8 CARBON ATOMS, ALKENYL WITH UP TO 12 CARBON ATOMS OR ARALKYL OPTIONALLY SUBSTITUTED IN THE ARYL MOIETY BY HALOGEN, LOWER ALKYL OR ALKOXY, WHICH POSSESS FUNGICIDAL, INSECTICIDAL ACARICIDAL, ANTIBACTERIAL AND GROWTH-REGULATING PROPERTIES.