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    Percyquinnin, a process for its production and its use as a pharmaceutical
    4.
    发明授权
    Percyquinnin, a process for its production and its use as a pharmaceutical 有权
    Percyquinnin，其生产过程及其作为药物的使用

    公开(公告)号：US06596518B2

    公开(公告)日：2003-07-22

    申请号：US09826866

    申请日：2001-04-06

    申请人： Cordula Hopmann ,  Michael Kurz ,  Guenter Mueller ,  Luigi Toti

    发明人： Cordula Hopmann ,  Michael Kurz ,  Guenter Mueller ,  Luigi Toti

    IPC分类号： C12P1702

    CPC分类号： C12R1/645 ,  C07D305/14 ,  C12P17/02

    摘要： The present invention relates to a compound named Percyquinnin that is obtainable by cultivating a basidiomycetes Stereum complicatum (DSM 13303), and to its pharmaceutically acceptable salts. The present invention further relates to a process for the production of Percyquinnin and to the use of Percyquinnin and its pharmaceutically acceptable salts as pharmaceuticals, in particular to their use as inhibitors of lipase.

    摘要翻译： 本发明涉及可通过培养担子菌（Stereum complicatum）（DSM 13303）获得的称为Percyquinnin的化合物及其药学上可接受的盐。 本发明进一步涉及一种生产珀金喹素的方法，以及使用过氧喹啉及其药学上可接受的盐作为药物，特别是其作为脂肪酶抑制剂的用途。

    Optical media protection driver
    6.
    发明授权
    Optical media protection driver 有权
    光媒体保护驱动

    公开(公告)号：US08875241B2

    公开(公告)日：2014-10-28

    申请号：US10552288

    申请日：2004-03-25

    申请人： Andreas Winter ,  Michael Kurz

    发明人： Andreas Winter ,  Michael Kurz

    IPC分类号： G06F17/30 ,  G11B20/00 ,  G06F21/10

    CPC分类号： G06F21/10 ,  G06F2221/0744 ,  G06F2221/2153 ,  G11B20/00086 ,  G11B20/00173 ,  G11B20/00202 ,  G11B20/00659 ,  G11B20/00688 ,  G11B20/00695 ,  G11B20/00884 ,  G11B20/00927

    摘要： A method to protect content within protected data areas on a target optical record carrier against unauthorized reading and/or copying with a computer, comprises the steps of—determining whether a target optical record carrier or a non-target optical record carrier is inserted into a drive of the computer, and—in case a target optical record carrier is inserted into the drive of the computer—modifying read requests to the protected data areas so that no data is read or the read data is useless, and/or—modifying write commands in respect to the data within the protected data areas to a recordable record carrier or other storage so that the written data is useless.

    摘要翻译： 一种用于保护目标光学记录载体上的受保护数据区域内的内容以防止未经授权的读取和/或与计算机复制的方法包括以下步骤：确定目标光学记录载体或非目标光学记录载体是否被插入到 并且在目标光学记录载体被插入计算机修改读取请求的驱动器到受保护数据区域的情况下，使得没有数据被读取或读取数据是无用的，和/或修改写入 关于受保护数据区域内的数据到可记录记录载体或其他存储器的命令，使得写入的数据是无用的。

    Cephaibols: novel antiparasitics from Acremonium tubakii, process for their production, and use thereof
    9.
    发明授权
    Cephaibols: novel antiparasitics from Acremonium tubakii, process for their production, and use thereof 有权
    头孢唑醇：来自Acremonium tubakii的新型抗寄生虫药，其生产方法及其用途

    公开(公告)号：US07067112B2

    公开(公告)日：2006-06-27

    申请号：US10411144

    申请日：2003-04-11

    申请人： Laszlo Vertesy ,  Michael Kurz ,  Matthias Schiell ,  Joachim Hofmann

    发明人： Laszlo Vertesy ,  Michael Kurz ,  Matthias Schiell ,  Joachim Hofmann

    IPC分类号： A61K49/00 ,  A61K38/10 ,  C07K7/08

    CPC分类号： C07K7/08 ,  A61K38/00

    摘要： The invention relates to compounds of the formula I AcPhe-Aib-Aib-Aib-x-w-Leu-y-Aib-Hyp-Gln-z-Hyp-Aib-Pro-R   (I) in which R is Phe-ol or Phe-al and w, x, y, and z have the following meanings: a) w is Gly or Ala; x is Aib and y and z are Iva; b) w is Gly; x, y and z are Iva; c) w is Gly; x and z are Aib and y is Iva; d) w is Gly; x, y and z are Aib; or e) w is Gly; x and y are Aib and z is Iva; or of the formula II AcPhe-Iva-Gln-Aib-lle-Thr-Aib-Leu-Aib-x-Gln-Aib-Hyp-Aib-Pro-Phe-Ser,   (II) wherein x is Hyp or Pro, which are synthesized by Acremonium tubakii FH 1685 DSM 12774 during fermentation and released into the culture medium, a process for the isolation of the cephaibols from the culture medium, and their purification, and the use of the cephaibols as pharmacologically active compounds, in particular for the control of parasites.

    摘要翻译： 本发明涉及式I化合物<？in-line-formula description =“In-line Formulas”end =“lead”→AcPhe-Aib-Aib-Aib-xw-Leu-y-Aib-Hyp-Gln -z-Hyp-Aib-Pro-R（I）<？in-line-formula description =“In-line Formulas”end =“tail”？>其中R是Phe-ol或Phe-al，w，x ，y和z具有以下含义：a）w是Gly或Ala; x是Aib，y和z是Iva; b）w是Gly; x，y和z是Iva; c）w是Gly; x和z是Aib，y是Iva; d）w是Gly; x，y和z是Aib; 或e）w是Gly; x和y是Aib，z是Iva; AcPhe-Iva-Gln-Aib-Lle-Thr-Aib-Leu-Aib-x-Gln-Aib，或者式II <？in-line-formula description =“In-line Formulas”end =“lead” -Hyp-Aib-Pro-Phe-Ser，（II）<？在线公式描述=“在线公式”end =“tail”？>其中x是Hyp或Pro，它们是由Acremonium tubakii FH 1685 DSM 12774在发酵过程中释放到培养基中，从培养基中分离头孢胆素的方法及其纯化，以及将头孢唑醇用作药物活性化合物，特别是用于控制寄生虫的方法。

    Fuel injection device for internal combustion engines
    10.
    发明授权
    Fuel injection device for internal combustion engines 失效
    内燃机燃油喷射装置

    公开(公告)号：US06994280B2

    公开(公告)日：2006-02-07

    申请号：US10296705

    申请日：2002-03-22

    申请人： Michael Kurz ,  Gerd Wahr

    发明人： Michael Kurz ,  Gerd Wahr

    IPC分类号： F02M59/00 ,  F02M61/00 ,  F02M63/00 ,  F02M47/02 ,  B05B1/00

    CPC分类号： F02M61/168 ,  F02M61/16

    摘要： A fuel injector for internal combustion engines, includes a base body, an injection housing and a fastening device. The fastening device includes at least one lock nut with an annular land and an annular shoulder on the injection housing. By means of the fastening device, the injection housing is braced axially against the base body. A fuel inlet and at least one valve element are also provided. To improve the seal between the base body and the injection housing, the fastening device has at least one annular face which is oriented toward the annular land of the lock nut and is curved convexly in the manner of a spherical-segmental face.

    摘要翻译： 一种用于内燃机的燃料喷射器，包括基体，注射壳体和紧固装置。 紧固装置包括至少一个具有环形接合面的锁紧螺母和注射壳体上的环形肩部。 通过紧固装置，注射壳体轴向地支撑在基体上。 还提供燃料入口和至少一个阀元件。 为了改善基体和注射壳体之间的密封，紧固装置具有至少一个朝向锁定螺母的环形平台的环形面，并且以球形节面的方式凸出地弯曲。