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1.Compounds useful in the preparation of tryptophan hydroxylase inhibitors 有权
标题翻译: 可用于制备色氨酸羟化酶抑制剂的化合物公开(公告)号:US08450532B2
公开(公告)日:2013-05-28
申请号:US13024469
申请日:2011-02-10
申请人: Hugh Alfred Burgoon , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang , Matthew Mangzhu Zhao
发明人: Hugh Alfred Burgoon , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang , Matthew Mangzhu Zhao
IPC分类号: C07C33/34 , C07C43/205
CPC分类号: A61K31/505 , C07C43/23 , C07D239/42 , C07D239/47 , C07D239/48
摘要: Intermediates and synthetic processes for the preparation of substituted phenylalanine-based compounds (e.g., of Formula I) are disclosed:
摘要翻译: 公开了用于制备取代的苯丙氨酸类化合物(例如式I)的中间体和合成方法:
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公开(公告)号:US20090048280A1
公开(公告)日:2009-02-19
申请号:US11647517
申请日:2006-12-28
申请人: Hugh Alfred Burgoon, JR. , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang
发明人: Hugh Alfred Burgoon, JR. , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang
IPC分类号: A61K31/513 , C07D239/46
CPC分类号: A61K31/505 , C07D239/47
摘要: Intermediates and synthetic processes for the preparation of substituted phenylalanine-based compounds (e.g., of Formula I) are disclosed:
摘要翻译: 公开了用于制备取代的苯丙氨酸类化合物(例如式I)的中间体和合成方法:
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公开(公告)号:US07855291B2
公开(公告)日:2010-12-21
申请号:US11647517
申请日:2006-12-28
申请人: Hugh Alfred Burgoon, Jr. , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang
发明人: Hugh Alfred Burgoon, Jr. , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang
IPC分类号: C07D239/34 , C07D403/12 , A61K31/506 , A61K31/505 , A61P9/02
CPC分类号: A61K31/505 , C07D239/47
摘要: Intermediates and synthetic processes for the preparation of substituted phenylalanine-based compounds (e.g., of Formula I) are disclosed:
摘要翻译: 公开了用于制备取代的苯丙氨酸类化合物(例如式I)的中间体和合成方法:
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4.COMPOUNDS USEFUL IN THE PREPARATION OF TRYPTOPHAN HYDRROXYLASE INHIBITORS 有权
标题翻译: 化合物在制备TRYPTOPHAN HYDRXYLASE抑制剂中有用公开(公告)号:US20110130564A1
公开(公告)日:2011-06-02
申请号:US13024469
申请日:2011-02-10
申请人: Hugh Alfred Burgoon , Ramanaiah Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang , Matthew Mangzhu Zhao
发明人: Hugh Alfred Burgoon , Ramanaiah Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang , Matthew Mangzhu Zhao
IPC分类号: C07D239/47 , C07C43/23
CPC分类号: A61K31/505 , C07C43/23 , C07D239/42 , C07D239/47 , C07D239/48
摘要: Intermediates and synthetic processes for the preparation of substituted phenylalanine-based compounds (e.g., of Formula I) are disclosed:
摘要翻译: 公开了用于制备取代的苯丙氨酸类化合物(例如式I)的中间体和合成方法:
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公开(公告)号:US07897763B2
公开(公告)日:2011-03-01
申请号:US12257558
申请日:2008-10-24
申请人: Hugh Alfred Burgoon , Ramanaiah Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang , Matthew Mangzhu Zhao
发明人: Hugh Alfred Burgoon , Ramanaiah Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang , Matthew Mangzhu Zhao
IPC分类号: C07D239/42 , C07D403/12 , A61K31/506 , A61P9/02
CPC分类号: A61K31/505 , C07C43/23 , C07D239/42 , C07D239/47 , C07D239/48
摘要: Intermediates and synthetic processes for the preparation of substituted phenylalanine-based compounds (e.g., of Formula I) are disclosed:
摘要翻译: 公开了用于制备取代的苯丙氨酸类化合物(例如式I)的中间体和合成方法:
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公开(公告)号:US20090118505A1
公开(公告)日:2009-05-07
申请号:US12257558
申请日:2008-10-24
申请人: Hugh Alfred Burgoon , Ramanaiah Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang , Matthew Mangzhu Zhao
发明人: Hugh Alfred Burgoon , Ramanaiah Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang , Matthew Mangzhu Zhao
IPC分类号: C07D239/47 , C07D239/42 , C07C43/23
CPC分类号: A61K31/505 , C07C43/23 , C07D239/42 , C07D239/47 , C07D239/48
摘要: Intermediates and synthetic processes for the preparation of substituted phenylalanine-based compounds (e.g., of Formula I) are disclosed:
摘要翻译: 公开了用于制备取代的苯丙氨酸类化合物(例如式I)的中间体和合成方法:
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7.METHODS OF PREPARING 4-PHENYL-6-(2,2,2-TRIFLUORO-1-PHENYLETHOXY)PYRIMIDINE-BASED COMPOUNDS 有权
标题翻译: 制备4-苯基-6-(2,2,2-三氟-1-苯基乙基)吡啶基化合物的方法公开(公告)号:US20110301349A1
公开(公告)日:2011-12-08
申请号:US13160678
申请日:2011-06-15
申请人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
发明人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
IPC分类号: C07D239/42 , C07D231/12
CPC分类号: C07D403/12 , C07D231/12
摘要: Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.
摘要翻译: 公开了可用于制备式I化合物及其盐的方法。 还公开了可用于制备这些化合物的中间体。
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公开(公告)号:US07968729B2
公开(公告)日:2011-06-28
申请号:US12732311
申请日:2010-03-26
申请人: Mark S. Bednarz , Hugh Alfred Burgoon, Jr. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
发明人: Mark S. Bednarz , Hugh Alfred Burgoon, Jr. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
IPC分类号: C07D231/10
CPC分类号: C07D403/12 , C07D231/12
摘要: Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.
摘要翻译: 公开了可用于制备式I化合物及其盐的方法。 还公开了可用于制备这些化合物的中间体。
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9.METHODS OF PREPARING 4-PHENYL-6-(2,2,2-TRIFLUORO-1-PHENYLETHOXY)PYRIMIDINE-BASED COMPOUNDS 审中-公开
标题翻译: 制备4-苯基-6-(2,2,2-三氟-1-苯基乙基)吡啶基化合物的方法公开(公告)号:US20090062540A1
公开(公告)日:2009-03-05
申请号:US12196341
申请日:2008-08-22
申请人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
发明人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
IPC分类号: C07D403/12 , C07D231/12
CPC分类号: C07D403/12 , C07D231/12
摘要: Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.
摘要翻译: 公开了可用于制备式I化合物及其盐的方法。 还公开了可用于制备这些化合物的中间体。
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10.Methods of preparing 4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds 有权
标题翻译: 制备4-苯基-6-(2,2,2-三氟-1-苯基乙氧基)嘧啶类化合物的方法公开(公告)号:US08575362B2
公开(公告)日:2013-11-05
申请号:US13160678
申请日:2011-06-15
申请人: Mark S. Bednarz , Hugh Alfred Burgoon, Jr. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
发明人: Mark S. Bednarz , Hugh Alfred Burgoon, Jr. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
IPC分类号: C07D231/12
CPC分类号: C07D403/12 , C07D231/12
摘要: Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.
摘要翻译: 公开了可用于制备式I化合物及其盐的方法。 还公开了可用于制备这些化合物的中间体。
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