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公开(公告)号：US20170226102A1
公开(公告)日：2017-08-10
申请号：US15501730
申请日：2015-08-07
Applicant: Janssen Sciences Ireland UC
Inventor： Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Jérôme Émile Georges Guillemont , David Craig Mc Gowan , Werner Constant Johan Embrechts , Ludwig Paul Cooymans , Antoine Benjamin Michaut
IPC: C07D417/14 , C07D403/04 , A61K31/506 , C07D413/14 , C07D401/14 , C07D401/04 , C07D403/14 , C07D405/14 , A61K45/06 , A61K31/4439
Abstract: The invention relates to compounds having the structure of formula (I) which can be used for the treatment of or against influenza infections.
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2.发明申请公开(公告)号：US20150336955A1
公开(公告)日：2015-11-26
申请号：US14818094
申请日：2015-08-04
Applicant: Janssen Sciences Ireland UC
Inventor： David Craig Mc Gowan , Pierre Jean-Marie Bernard RABOISSON , Tim Hugo Maria JONCKERS , Mourad DAOUBI KHAMLICHI
IPC: C07D471/04
CPC classification number: C07D471/04 , A61K31/519
Abstract: This invention relates to piperidino-pyrimidine derivatives, processes for their preparation, pharmaceutical compositions, and their use in treating viral infections.
Abstract translation: 本发明涉及哌啶子基 - 嘧啶衍生物，其制备方法，药物组合物及其在治疗病毒感染中的用途。
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3.发明申请HETEROCYCLIC SUBSTITUTED 2-AMINO QUINAZOLINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS 有权用于治疗病毒感染的杂环取代的2-氨基喹唑啉衍生物公开(公告)号：US20150284339A1
公开(公告)日：2015-10-08
申请号：US14443305
申请日：2013-11-15
Applicant: JANSSEN SCIENCES IRELAND UC
Inventor： Stefaan Julien Last , David Craig Mc Gowan , Werner Embrechts , Serge Maria Aloysius Pieters , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson
IPC: C07D239/84 , C07D403/12 , C07D413/12 , C07D401/12 , C07D417/12
CPC classification number: C07D239/84 , C07D239/95 , C07D401/12 , C07D403/12 , C07D413/12 , C07D417/12
Abstract: This invention relates to heterocyclic substituted 2-amino-quinazoline derivatives, processes for their preparation, pharmaceutical compositions, and their use in treating viral infections.
Abstract translation: 本发明涉及杂环取代的2-氨基 - 喹唑啉衍生物，其制备方法，药物组合物及其在治疗病毒感染中的用途。
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4.发明申请ALKYLPYRIMIDINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS AND FURTHER DISEASES 有权用于治疗病毒感染和进一步疾病的亚胺嘧啶衍生物公开(公告)号：US20150239872A1
公开(公告)日：2015-08-27
申请号：US14420066
申请日：2013-08-09
Applicant: JANSSEN SCIENCES IRELAND UC
IPC: C07D409/06 , C07D401/06 , C07D239/49 , C07D239/48
CPC classification number: C07D409/06 , C07D239/48 , C07D239/49 , C07D401/06
Abstract: This invention relates to alkylpyrimidine derivatives, processes for their preparation, pharmaceutical compositions, and their use in therapy.
Abstract translation: 本发明涉及烷基嘧啶衍生物，其制备方法，药物组合物及其在治疗中的应用。
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![Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases](/abs-image/US/2017/02/16/US20170044169A1/abs.jpg.150x150.jpg)
5.发明申请Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases 审中-公开吡咯并[3,2-d]嘧啶衍生物，用于治疗病毒感染等疾病公开(公告)号：US20170044169A1
公开(公告)日：2017-02-16
申请号：US15333947
申请日：2016-10-25
Applicant: JANSSEN SCIENCES IRELAND UC
Inventor： David Craig Mc Gowan , Stefaan Julien Last , Serge Maria Aloysius Pieters , Werner Embrechts , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson
IPC: C07D487/04 , C07D519/00
CPC classification number: C07D487/04 , A61K31/407 , A61K31/519 , A61P31/12 , C07D519/00
Abstract: This invention concerns pyrrolo[3,2-d]pyrimidine derivatives, processes for their preparation, pharmaceutical compositions, and their use in treatment and/or therapy of diseases.
Abstract translation: 本发明涉及吡咯并[3,2-d]嘧啶衍生物，其制备方法，药物组合物及其在治疗和/或治疗疾病中的用途。
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Patent Agency Ranking
公开(公告)号：US20150210719A1
公开(公告)日：2015-07-30
申请号：US14417511
申请日：2013-08-09
Applicant: JANSSEN SCIENCES IRELAND UC
Inventor： Jerôme Emile Georges Guillemont , David Francis Alain Lançois , Magali Madeleine Simone Motte , Wendy Mia Albert Balemans , Steffen Friedrich Walter Weidner , David Craig Mc Gowan , Anil Koul
IPC: C07D519/00 , C07D405/14 , C07D409/14 , C07D417/14 , C07D513/14 , C07D498/04 , C07D471/04 , C07D498/14 , C07D471/14 , C07D401/14 , C07D401/06
CPC classification number: C07D519/00 , C07D401/06 , C07D401/12 , C07D401/14 , C07D405/12 , C07D405/14 , C07D409/14 , C07D417/14 , C07D471/04 , C07D471/14 , C07D498/04 , C07D498/14 , C07D513/14
Abstract: The present invention is related to novel compounds of formula (I) that may inhibit the activity of the FabI enzyme, and which are useful in the treatment of bacterial infections. It further relates to pharmaceutical compositions comprising these compounds, and chemical processes for preparing these compounds.
Abstract translation: 本发明涉及可抑制FabI酶的活性的新型式（I）化合物，其可用于治疗细菌感染。 它还涉及包含这些化合物的药物组合物和用于制备这些化合物的化学方法。
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公开(公告)号：US09884818B2
公开(公告)日：2018-02-06
申请号：US14891864
申请日：2014-05-16
Applicant: Janssen Sciences Ireland UC
Inventor： Koen Vandyck , Geerwin Yvonne Paul Haché , Stefaan Julien Last , David Craig Mc Gowan , Geert Rombouts , Wim Gaston Verschueren , Pierre Jean-Marie Bernard Raboisson
IPC: C07D207/36 , C07D403/12 , C07D405/12 , A61K31/401 , C07D207/40 , A61K45/06
CPC classification number: C07D207/36 , A61K31/401 , A61K45/06 , C07D207/40 , C07D403/12 , C07D405/12 , A61K2300/00
Abstract: Inhibitors of HBV replication of Formula (ID) including stereochemically isomeric forms, and salts, hydrates, solvates thereof, wherein X, Ra to Rd and R4 to R6 have the meaning as defined herein. The present invention also relates to processes for preparing compounds of Formula (ID), pharmaceutical compositions containing them and their use, alone or in combination with other HBV inhibitors, in HBV therapy.
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公开(公告)号：US09790191B2
公开(公告)日：2017-10-17
申请号：US14431973
申请日：2013-10-03
Applicant: JANSSEN SCIENCES IRELAND UC
Inventor： David Craig Mc Gowan , Serge Marie Aloysius Pieters , Werner Embrechts , Stefaan Julien Last , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson
IPC: C07D239/47 , C07D401/12 , C07D213/75 , C07D239/48
CPC classification number: C07D239/47 , C07D213/75 , C07D239/48
Abstract: This invention relates to acylaminopyrimidine derivatives, processes for their preparation, pharmaceutical compositions, and their use in therapy.
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公开(公告)号：US20150376140A1
公开(公告)日：2015-12-31
申请号：US14769773
申请日：2014-02-20
Applicant: JANSSEN SCIENCES IRELAND UC
IPC: C07D239/47
CPC classification number: C07D239/47 , A61K31/505 , C07D239/48
Abstract: This invention relates to 2-aminopyrimidine derivatives, processes for their preparation, pharmaceutical compositions, and their use in treating viral infections.
Abstract translation: 本发明涉及2-氨基嘧啶衍生物，其制备方法，药物组合物及其在治疗病毒感染中的用途。
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10.发明申请ACYLAMINOPYRIMIDINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS AND FURTHER DISEASES 有权用于治疗病毒性感染和进一步疾病的氨基亚氨基嘧啶衍生物公开(公告)号：US20150274676A1
公开(公告)日：2015-10-01
申请号：US14431973
申请日：2013-10-03
Applicant: JANSSEN SCIENCES IRELAND UC
Inventor： David Craig Mc Gowan , Serge Marie Aloysius Pieters , Werner Embrechts , Stefaan Julien Last , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson
IPC: C07D239/47
CPC classification number: C07D239/47 , C07D213/75 , C07D239/48
Abstract: This invention relates to acylaminopyrimidine derivatives, processes for their preparation, pharmaceutical compositions, and their use in therapy.
Abstract translation: 本发明涉及酰氨基嘧啶衍生物，其制备方法，药物组合物及其在治疗中的应用。
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