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15 条记录 (耗时 0.028 秒)

    Novel cyclic phosphate diesters of 1,3-propane-1-aryl diols and their use in preparing prodrugs
    1.
    发明申请
    Novel cyclic phosphate diesters of 1,3-propane-1-aryl diols and their use in preparing prodrugs 有权
    1,3-丙烷-1-芳基二醇的新型环状磷酸二酯及其在制备前药中的用途

    公开(公告)号：US20070021388A1

    公开(公告)日：2007-01-25

    申请号：US11528283

    申请日：2006-09-28

    申请人： K. Reddy ,  William Craigo ,  Zhili Sun ,  Serge Boyer ,  Bheemarao Ugarkar

    发明人： K. Reddy ,  William Craigo ,  Zhili Sun ,  Serge Boyer ,  Bheemarao Ugarkar

    IPC分类号： A61K31/675 ,  C07F9/6512 ,  C07F9/6509

    CPC分类号： C07F9/65742 ,  C07H19/04

    摘要： Compounds of Formula I, their preparation and synthetic intermediates, and their use in the synthesis of prodrugs: wherein: V and L are trans relative to one another; V is selected from group consisting of carbocyclic aryl, substituted carbocyclic aryl, heteroaryl, and substituted heteroaryl; and L is a leaving group selected from the group consisting of halogen, alkyl sulfonate, aryloxy optionally substituted with 1-2 substituents, N-containing heteroaryl, and N-hydroxy-nitrogen containing heteroaryl; and salts thereof.

    摘要翻译： 式I化合物，其制备方法和合成中间体及其在前体药物合成中的应用：其中：V和L相对于彼此是反式的; V选自碳环芳基，取代的碳环芳基，杂芳基和取代的杂芳基; 并且L是选自卤素，烷基磺酸酯，任选被1-2个取代基取代的芳氧基，含N杂芳基和N-羟基 - 含氮杂芳基的离去基团; 及其盐。

    Cyclic phosphate diesters of 1,3-propane-1-aryl diols and their use in preparing prodrugs
    3.
    发明授权
    Cyclic phosphate diesters of 1,3-propane-1-aryl diols and their use in preparing prodrugs 有权
    1,3-丙烷-1-芳基二醇的环磷酸二酯及其在制备前药中的用途

    公开(公告)号：US07498320B2

    公开(公告)日：2009-03-03

    申请号：US11528283

    申请日：2006-09-28

    申请人： K. Raja Reddy ,  William Craigo ,  Zhili Sun ,  Serge Boyer ,  Bheemarao G. Ugarkar

    发明人： K. Raja Reddy ,  William Craigo ,  Zhili Sun ,  Serge Boyer ,  Bheemarao G. Ugarkar

    IPC分类号： A61K31/665 ,  C07F9/02

    CPC分类号： C07F9/65742 ,  C07H19/04

    摘要： Compounds of Formula I, their preparation and synthetic intermediates, and their use in the synthesis of prodrugs: wherein: V and L are trans relative to one another; V is selected from group consisting of carbocyclic aryl, substituted carbocyclic aryl, heteroaryl, and substituted heteroaryl; and L is a leaving group selected from the group consisting of halogen, alkyl sulfonate, aryloxy optionally substituted with 1-2 substituents, N-containing heteroaryl, and N-hydroxy-nitrogen containing heteroaryl; and salts thereof.

    摘要翻译： 式I化合物，其制备方法和合成中间体及其在前体药物合成中的应用：其中：V和L相对于彼此是反式的; V选自碳环芳基，取代的碳环芳基，杂芳基和取代的杂芳基; 并且L是选自卤素，烷基磺酸酯，任选被1-2个取代基取代的芳氧基，含N杂芳基和N-羟基 - 含氮杂芳基的离去基团; 及其盐。

    Device and method for regulation the temperature and/or power of a cooking apparatus
    5.
    发明授权
    Device and method for regulation the temperature and/or power of a cooking apparatus 失效
    用于调节烹饪设备的温度和/或功率的装置和方法

    公开(公告)号：US5324917A

    公开(公告)日：1994-06-28

    申请号：US836264

    申请日：1992-02-28

    申请人： Serge Boyer ,  Didier Gouardo ,  Pierre Pitot

    发明人： Serge Boyer ,  Didier Gouardo ,  Pierre Pitot

    IPC分类号： A47J27/62 ,  G05D23/19 ,  H05B6/06 ,  H05B1/02

    CPC分类号： H05B6/062 ,  A47J27/62 ,  G05D23/1906 ,  G05D23/1951

    摘要： A device and method for regulating a cooking apparatus. In order to obtain an effective servocontrol of the desired temperature with a cooking surface, when cooking for example by induction, a servocontrol curve is used in the plane (i.e., temperature, variation of the temperature as a function of time). Each time the curve is crossed the heating power is cut off or reduced. The device and method applies principally to monitoring of the heating device. The device according to the present invention is particularly well adapted to cooking surfaces and especially to cooking surfaces wherein cooking is done by induction.

    摘要翻译： PCT No.PCT / FR90 / 00660 Sec。 一九九二年二月二十八日 102（e）日期1992年2月28日PCT提交1990年9月14日PCT公布。 第WO91 / 04524号公报 日期1994年4月4日。一种用于调节烹饪设备的装置和方法。 为了通过烹饪表面获得期望温度的有效伺服控制，当例如通过感应进行烹饪时，在平面中使用伺服控制曲线（即，温度，作为时间的函数的温度变化）。 每当曲线过渡时，加热功率被切断或减小。 该装置和方法主要适用于监测加热装置。 根据本发明的装置特别适用于烹饪表面，特别适用于通过感应进行烹饪的烹饪表面。

    Method for checking takeoff or landing parameters, and associated device
    6.
    发明申请
    Method for checking takeoff or landing parameters, and associated device 有权
    检查起飞或着陆参数的方法及相关设备

    公开(公告)号：US20070124034A1

    公开(公告)日：2007-05-31

    申请号：US11563743

    申请日：2006-11-28

    申请人： Fabien Pitard ,  Jean-Pierre Demortier ,  Serge Laporte ,  Serge Boyer ,  Bernard Deret ,  Laurent Fonteneau

    发明人： Fabien Pitard ,  Jean-Pierre Demortier ,  Serge Laporte ,  Serge Boyer ,  Bernard Deret ,  Laurent Fonteneau

    IPC分类号： G06F19/00

    CPC分类号： G05D1/0083

    摘要： A method for checking takeoff or landing parameters of an aircraft comprises a step (E101) of determining takeoff or landing parameters on the basis of a series of input conditions. It additionally comprises the following steps: calculation (E103) of regulatory data on the basis of determined takeoff or landing parameters; and comparison (E104) of the calculated regulatory data with predefined threshold values, with a view to establishing whether the determined takeoff or landing parameters are valid or invalid. Use to ensure reliability of the determination of optimized takeoff or landing parameters.

    摘要翻译： 用于检查飞行器起飞或着陆参数的方法包括基于一系列输入条件来确定起飞或着陆参数的步骤（E 101）。 它还包括以下步骤：根据确定的起飞或着陆参数来计算（E 103）监管数据; 以及计算的调节数据与预定阈值的比较（E 104），以便确定所确定的起飞或着陆参数是有效还是无效。 用于确定优化起飞或着陆参数的可靠性。

    Novel cytarabine monophosphate prodrugs
    7.
    发明申请
    Novel cytarabine monophosphate prodrugs 有权
    新型阿糖胞苷单磷酸前药

    公开(公告)号：US20070037774A1

    公开(公告)日：2007-02-15

    申请号：US11582383

    申请日：2006-10-18

    申请人： Serge Boyer ,  Mark Erion

    发明人： Serge Boyer ,  Mark Erion

    IPC分类号： A61K31/7072 ,  C07H19/00

    CPC分类号： C07F9/65742 ,  C07H19/04

    摘要： Compounds of Formula I, their preparation and uses are described: wherein: M and V are cis to one another and MH is cytarabine; the 5′ oxygen of said cytarabine is attached to the phosphorus; V is 4-pyridyl; and pharmaceutically acceptable prodrugs and salts thereof.

    摘要翻译： 描述式I化合物及其制备和用途：其中：M和V彼此是顺式的，MH是阿糖胞苷; 所述阿糖胞苷的5'氧与磷结合; V是4-吡啶基; 及其药学上可接受的前药及其盐。

    Temperature-measuring device for an induction-type cooking appliance and appliance having such a device
    8.
    发明授权
    Temperature-measuring device for an induction-type cooking appliance and appliance having such a device 失效
    具有这种装置的感应式烹饪器具和器具的温度测量装置

    公开(公告)号：US5283412A

    公开(公告)日：1994-02-01

    申请号：US552097

    申请日：1990-07-13

    申请人： Didier Gouardo ,  Serge Boyer ,  Pierre Pitot

    发明人： Didier Gouardo ,  Serge Boyer ,  Pierre Pitot

    IPC分类号： G01K1/16 ,  A47J29/00 ,  G01K13/00 ,  H05B6/12 ,  H05B5/04

    CPC分类号： H05B6/062 ,  H05B2213/07

    摘要： A temperature-measuring device for an induction-type cooking appliance is disclosed with a heat measuring device for an induction-type cooking hob including a heat conductor for measuring the temperature of a sauce pan or its contents independently of its diameter or its bottom surface configuration. A heat conductor includes modifications which minimize the effects of currents provided by the induction heating. The device allows for the measurement of temperature during induction heating.

    摘要翻译： 公开了一种用于感应式烹饪器具的温度测量装置，该测量装置包括用于独立于其直径或其底部表面构造测量酱汁盘或其内容物的温度的热导体的感应型烹饪灶台 。 热导体包括使感应加热提供的电流的影响最小化的修改。 该装置允许感应加热期间的温度测量。

    Cytarabine monophosphate prodrugs
    10.
    发明授权
    Cytarabine monophosphate prodrugs 有权
    阿糖胞苷单磷酸前药

    公开(公告)号：US07553826B2

    公开(公告)日：2009-06-30

    申请号：US11582383

    申请日：2006-10-18

    申请人： Serge Boyer ,  Mark D. Erion

    发明人： Serge Boyer ,  Mark D. Erion

    IPC分类号： A61K31/661 ,  C07D239/20 ,  C07F9/6558

    CPC分类号： C07F9/65742 ,  C07H19/04

    摘要： Compounds of Formula I, their preparation and uses are described: wherein: M and V are cis to one another and MH is cytarabine; the 5′ oxygen of said cytarabine is attached to the phosphorus; V is 4-pyridyl; and pharmaceutically acceptable prodrugs and salts thereof.

    摘要翻译： 描述式I化合物及其制备和用途：其中：M和V彼此是顺式的，MH是阿糖胞苷; 所述阿糖胞苷的5'氧与磷结合; V是4-吡啶基; 及其药学上可接受的前药及其盐。