公开(公告)号：US4666933A

公开(公告)日：1987-05-19

申请号：US875129

申请日：1986-06-17

申请人： Klaus Jelich ,  Wolfgang Kramer ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

发明人： Klaus Jelich ,  Wolfgang Kramer ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC分类号： A01N43/56 ,  C07D231/46 ,  C07D405/06 ,  C07D405/12

CPC分类号： C07D405/06 ,  A01N43/56 ,  C07D231/46 ,  C07D405/12

摘要： Fungicidally active substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 is hydrogen or alkyl,R.sup.2 is hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, hydroxycarbonylalkyl or alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or in each case optionally substituted oxiranylmethyl, aralkyl or aryl, andR.sup.3 is alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, cycloalkyl or cycloalkylalkyl, or in each case optionally substituted aralkyl, aryloxyalkyl or arylthioalkyl, but wherein R.sup.3 is methyl or ethyl only if R.sup.1 and/or R.sup.2 is not hydrogen or methyl.

摘要翻译： R 1为氢或烷基，R 2为氢，烷基，烯基，炔基，氰基烷基，羟基烷基，烷氧基烷基，羟基羰基烷基或烷氧基羰基烷基，氨基羰基烷基，烷基氨基羰基烷基或二烷基氨基羰基烷基的芳香族活性取代的吡唑啉-5-酮 每种情况下任选取代的环氧乙烷基甲基，芳烷基或芳基，R 3是烷基，烯基，炔基，氰基烷基，羟基烷基，烷氧基烷基，羟基羰基烷基，烷氧基羰基烷基，环烷基或环烷基烷基，或在每种情况下任选取代的芳烷基，芳氧基烷基或芳硫基烷基， 或仅在R 1和/或R 2不是氢或甲基时为乙基。

公开(公告)号：US4743615A

公开(公告)日：1988-05-10

申请号：US925184

申请日：1986-10-31

申请人： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

发明人： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC分类号： C07D231/46 ,  A01N43/56 ,  C07D239/48 ,  C07D405/06

CPC分类号： C07D405/06 ,  A01N43/56 ,  C07D239/48

摘要： Fungicidally active substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represents hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represents in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl, andR.sup.3 represents halogenoalkyl, halogenoalkenyl or halogenoalkinyl, or represents substituted cycloalkyl, or represents substituted cycloalkylalkyl.

摘要翻译： R1和R2各自独立地表示氢，烷基，烯基，炔基，氰基烷基，羟基烷基，烷氧基烷基，烷硫基烷基，烷氧基羰基，羟基羰基烷基，烷氧基羰基烷基，氨基羰基烷基，烷基氨基羰基烷基，烷基氨基羰基烷基 或二烷基氨基羰基烷基，或在每种情况下表示任选取代的环氧烷基烷基，芳烷基，杂环基或芳基，并且R 3表示卤代烷基，卤代烯基或卤代链烯基，或表示取代的环烷基，或表示取代的环烷基烷基。

公开(公告)号：US4929738A

公开(公告)日：1990-05-29

申请号：US350064

申请日：1989-05-10

申请人： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

发明人： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC分类号： A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  A01N43/824 ,  C07D231/46 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D417/12 ,  C07D417/14 ,  C07D307/16 ,  C07D307/46 ,  C07D333/24

CPC分类号： C07D401/12 ,  A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

摘要： Microbicidal substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an optionally substituted heterocyclic radial.Intermediates therefor of the formula ##STR2## in which R is alkyl, are also new.

公开(公告)号：US4864029A

公开(公告)日：1989-09-05

申请号：US192799

申请日：1988-05-11

申请人： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

发明人： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC分类号： A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  A01N43/824 ,  C07D231/46 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D417/12 ,  C07D417/14

CPC分类号： C07D401/12 ,  A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

摘要： Microbicidal substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkyllaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an optionally substituted heterocyclic radical.Intermediates therefor of the formula ##STR2## in which R is alkyl, are also new.

摘要翻译： 其中R1和R2彼此独立地表示氢，烷基，烯基，炔基，氰基烷基，羟基烷基，烷氧基烷基，烷硫基烷基，烷氧基羰基，羟基羰基烷基，烷氧基羰基烷基，氨基羰基烷基，烷基氨基羰基烷基或氨基羰基烷基， 二烷基氨基羰基烷基，或在每种情况下表示任选取代的环氧烷基烷基，芳烷基，杂环基或芳基，Het表示任选取代的杂环基。 其中R为烷基的式“IMAGE”的中间体也是新的。

公开(公告)号：US4767775A

公开(公告)日：1988-08-30

申请号：US890245

申请日：1986-07-24

申请人： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

发明人： Klaus Jelich ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC分类号： A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  A01N43/824 ,  C07D231/46 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D417/12 ,  C07D417/14 ,  C07D419/12

CPC分类号： C07D401/12 ,  A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  A01N43/82 ,  C07D231/48 ,  C07D261/08 ,  C07D333/28 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

摘要： Microbicidal substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an optionally substituted heterocyclic radical.Intermediates therefor of the formula ##STR2## in which R is alkyl, are also disclosed.

摘要翻译： 其中R1和R2各自独立地表示氢，烷基，烯基，炔基，氰基烷基，羟基烷基，烷氧基烷基，烷硫基烷基，烷氧基羰基，羟基羰基烷基，烷氧基羰基烷基，氨基羰基烷基，烷基氨基羰基烷基或氨基羰基烷基的杀微生物取代的吡唑啉-5-酮 二烷基氨基羰基烷基，或在每种情况下表示任选取代的环氧烷基烷基，芳烷基，杂环基或芳基，Het表示任选取代的杂环基。 还公开了其中R为烷基的式“IMAGE”的中间体。

公开(公告)号：US4988729A

公开(公告)日：1991-01-29

申请号：US423607

申请日：1989-10-17

申请人： Wolfgang Kramer ,  Joachim Weissmuller ,  Graham Holmwood ,  Dieter Berg ,  Stefan Dutzmann ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

发明人： Wolfgang Kramer ,  Joachim Weissmuller ,  Graham Holmwood ,  Dieter Berg ,  Stefan Dutzmann ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC分类号： A01N43/08 ,  A01N43/28 ,  C07D307/14 ,  C07D307/22 ,  C07D317/28 ,  C07D327/04 ,  C07D407/12 ,  C07D417/12

CPC分类号： C07D407/12 ,  A01N43/08 ,  A01N43/28 ,  C07D307/14 ,  C07D317/28 ,  C07D327/04

摘要： Combattting fungi and bacteria with aminomethylheterocyclic compounds of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, in each case optionally substituted tetrahydronaphthyl, decahydronaphthyl, cycloalkyl or cycloalkenyl, furthermore alkyl which is substituted by cycloalkyl, cycloalkenyl, cycloalkyloxy or cycloalkylthio, where the cyclic radicals may optionally be substituted, furthermore optionally substituted aryl, in addition alkyl which is substituted by aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl, or alkenyl which is substituted by aryl, where the aryl radicals may in each case optionally be substituted;R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl, alkenyl, alkinyl, alkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dialkoxyalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, aralkyl, aralkenyl, furanylalkyl, tetrahydrofuranylalkyl, tetrahydropyranylalkyl, dioxolanylalkyl or dioxanylalkyl, andX represents oxygen, sulphur or a CH.sub.2 group,or acid additon salts thereof. Many of the compounds wherein R.sup.1 has a narrower meaning are new.

摘要翻译： 用下式（Ⅰ）的氨基甲基杂环化合物与R1代表氢，烷基，烯基，各取代四氢萘基，十氢萘基，环烷基或环烯基，以及被环烷基，环烯基，环烷氧基 或环烷硫基，其中环状基团可任选被取代，此外任选取代的芳基，另外被芳基，芳氧基，芳硫基，芳基亚磺酰基或芳基磺酰基取代的烷基或被芳基取代的烯基，其中芳基可以在每种情况下 任选被取代; R 2表示氢或甲基，R 3表示烷基，烯基，炔基，烷氧基烷基，羟基烷基，羟基烷氧基烷基，二烷氧基烷基，或在每种情况下任选取代的环烷基，环烷基烷基，芳基，芳烷基，芳烯基，呋喃基烷基，四氢呋喃基烷基，四氢吡喃基烷基，二氧戊环烷基或二烷基烷基，X 代表氧，硫或CH2基，或其酸加成盐。 其中R1具有较窄含义的许多化合物是新的。

公开(公告)号：US4917720A

公开(公告)日：1990-04-17

申请号：US256808

申请日：1988-10-12

申请人： Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

发明人： Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

IPC分类号： C07C43/225 ,  A01N43/50 ,  A01N43/653 ,  C07C41/00 ,  C07C45/00 ,  C07C49/167 ,  C07C49/175 ,  C07C67/00 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00

CPC分类号： C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

摘要： Azolyl ether ketones and alcohols of the formula ##STR1## in which R.sup.1 and R.sup.2 each independently represents alkyl with more than one carbon atom, orR.sup.1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlorovinyl, andR.sup.2 represents alkyl,R.sup.3 represents alkyl,A represents the keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group,X represents oxygen or sulfur andAr represents optionally substituted phenyl,or addition products thereof with acids and metal salts, are active against fungi and in regulating the growth of plants. New intermediates therefor are also shown.

公开(公告)号：US4878939A

公开(公告)日：1989-11-07

申请号：US258108

申请日：1988-10-13

申请人： Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

发明人： Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

IPC分类号： C07C43/225 ,  A01N43/50 ,  A01N43/653 ,  C07C41/00 ,  C07C45/00 ,  C07C49/167 ,  C07C49/175 ,  C07C67/00 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00

CPC分类号： C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

摘要： Azolyl ether ketones and alcohols of the formula ##STR1## in which R.sup.1 and R.sup.2 each independently represents alkyl with more than one carbon atom, orR.sup.1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlorovinyl, andR.sup.2 represents alkyl,R.sup.3 represents alkyl,A represents the keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group,X represents oxygen or sulphur andAr represents optionally substituted phenyl,or addition products thereof with acids and metal salts, are active against fungi and in regulating the growth of plants. New intermediates therefor are also shown.

摘要翻译： 其中R 1和R 2各自独立地表示具有多于一个碳原子的烷基，或者R 1表示二氯甲基，三氯甲基，氯乙烯基或二氯乙烯基，并且R 2表示烷基，R 3表示烷基， 酮基或CH（OH）基，Z表示氮原子或CH基，X表示氧或硫，Ar表示任选取代的苯基，或其与酸和金属盐的加成产物对真菌有活性， 植物生长。 还显示了其新的中间体。

公开(公告)号：US4615725A

公开(公告)日：1986-10-07

申请号：US720827

申请日：1985-04-08

申请人： Joachim Weissmuller ,  Wolfgang Kramer ,  Dieter Berg ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

发明人： Joachim Weissmuller ,  Wolfgang Kramer ,  Dieter Berg ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

IPC分类号： C07D317/28 ,  A01N43/08 ,  C07C17/26 ,  C07C33/48 ,  C07C43/23 ,  C07D303/22 ,  C07D307/10 ,  C07D307/12 ,  C07D307/14 ,  C07D405/06 ,  C07D413/06 ,  A01N43/40

CPC分类号： C07D303/22 ,  A01N43/08 ,  C07C17/2632 ,  C07C33/483 ,  C07C43/23 ,  C07D307/10 ,  C07D307/12 ,  C07D307/14 ,  C07D405/06 ,  C07D413/06

摘要： Tetrahydrofuran-2-ylmethylamines of the formula ##STR1## in which R.sup.1 represents optionally substituted naphthyl, optionally substituted cycloalkyl or cycloalkenyl, optionally substituted phenyl, or alkyl which is substituted by in each case optionally substituted phenyl, phenoxy or phenylthio,R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl andR.sup.4 represents alkyl, alkenyl, alkinyl or optionally substituted aralkyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical, which can contain further hetero-atoms,excluding the compounds in which R.sup.3 and R.sup.4 both represent methyl, R.sup.1 represents unsubstituted phenyl and R.sup.2 at the same time represents hydrogen, or plant-tolerated addition products thereof with acids or metal salts, which possess fungicidal and plant growth regulating activities.

摘要翻译： 式“IMAGE”的四氢呋喃-2-基甲胺，其中R 1表示任选取代的萘基，任选取代的环烷基或环烯基，任选取代的苯基或被各种情况下被任意取代的苯基，苯氧基或苯硫基取代的烷基，R 2表示氢或 甲基，R 3表示烷基，R 4表示烷基，烯基，炔基或任选取代的芳烷基，或者R 3和R 4与它们所键合的氮原子一起代表任选取代的杂环基，其可含有其它杂原子，不包括 其中R3和R4都表示甲基，R1代表未取代的苯基和R2同时表示具有杀真菌和植物生长调节活性的氢或其与酸或金属盐的植物耐受加成产物。

公开(公告)号：US5128368A

公开(公告)日：1992-07-07

申请号：US595143

申请日：1990-10-10

申请人： Wolfgang Kramer ,  Joachim Weissmuller ,  Graham Holmwood ,  Dieter Berg ,  Stefan Dutzmann ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

发明人： Wolfgang Kramer ,  Joachim Weissmuller ,  Graham Holmwood ,  Dieter Berg ,  Stefan Dutzmann ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC分类号： A01N43/08 ,  A01N43/28 ,  C07D307/14 ,  C07D307/22 ,  C07D317/28 ,  C07D327/04 ,  C07D407/12 ,  C07D417/12

CPC分类号： C07D407/12 ,  A01N43/08 ,  A01N43/28 ,  C07D307/14 ,  C07D317/28 ,  C07D327/04

摘要： Combatting fungi and bacteria with aminomethylheterocyclic compounds of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, in each case optionally substituted tetrahydronaphthyl, decahydronaphthyl, cycloalkyl or cycloalkenyl, furthermore alkyl which is substituted by cycloalkyl, cycloalkenyl, cycloalkyloxy or cycloalkylthio, where the cyclic radicals may optionally be substituted, furthermore optionally substituted aryl, in addition alkyl which is substituted by aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl, or alkenyl which is substituted by aryl, where the aryl radicals may in each case optionally be substituted;R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl, alkenyl, alkinyl, alkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dialkoxyalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, aralkyl, aralkenyl, furanylalkyl, tetrahydrofuranylalkyl, tetrahydropyranylalkyl, dioxolanylalkyl or dioxanylalkyl, andX represents oxygen, sulphur or a CH.sub.2 group,or acid addition salts thereof.Many of the compounds wherein R.sup.1 has a narrower meaning are new.

摘要翻译： 用下式（Ⅰ）的氨基甲基杂环化合物与R1代表氢，烷基，烯基，各取代四氢萘基，十氢萘基，环烷基或环烯基，以及被环烷基，环烯基，环烷基 或环烷硫基，其中环状基团可任选被取代，此外任选取代的芳基，另外被芳基，芳氧基，芳硫基，芳基亚磺酰基或芳基磺酰基取代的烷基或被芳基取代的烯基，其中芳基可以在每种情况下 任选被取代; R 2表示氢或甲基，R 3表示烷基，烯基，炔基，烷氧基烷基，羟基烷基，羟基烷氧基烷基，二烷氧基烷基，或在每种情况下任选取代的环烷基，环烷基烷基，芳基，芳烷基，芳烯基，呋喃基烷基，四氢呋喃基烷基，四氢吡喃基烷基，二氧戊环烷基或二烷基烷基，X 代表氧，硫或CH2基，或其酸加成盐。 其中R1具有较窄含义的许多化合物是新的。