摘要:
Novel 4-(3-butynyl)aminopyrimidine derivatives represented by general formula [I] are useful as pest control agents. In general formula [I], R1 is a mono- or bi-cyclic ring which may contain 0 to 3 heteroatoms, for example, phenyl or oxazolyl; R2 is a hydrogen atom, —R, —OR, —C(O)OR, —C(O)NHR, —CONR2 (wherein R is straight-chain or branched C1-8 alkyl, or the like), hydroxyalkyl, or the like; R3 is a hydrogen atom, a halogen atom, acyloxy represented by (straight-chain or branched C1-8 aliphatic hydrocarbon group) —CO—O—, or the like; and R4 is a hydrogen atom, a halogen atom, C1-6 alkyl, or the like, or alternatively, R4 and R3 together with the carbon atoms on the pyrimidine ring may form a thiophene ring, a pyrrole ring, an imidazole ring, a benzene ring, a pyrimidine ring, a furan ring, a pyrazine ring, or a pyrrolidine ring.
摘要:
Novel 4-(3-butynyl)aminopyrimidine derivatives represented by general formula [I] are useful as pest control agents. In general formula [I], R1 is a mono- or bi-cyclic ring which may contain 0 to 3 heteroatoms, for example, phenyl or oxazolyl; R2 is a hydrogen atom, —R, —OR, —C(O)OR, —C(O)NHR, —CONR2 (wherein R is straight-chain or branched C1-8 alkyl, or the like), hydroxyalkyl, or the like; R3 is a hydrogen atom, a halogen atom, acyloxy represented by (straight-chain or branched C1-8 aliphatic hydrocarbon group) —CO—O—, or the like; and R4 is a hydrogen atom, a halogen atom, C1-6 alkyl, or the like, or alternatively, R4 and R3 together with the carbon atoms on the pyrimidine ring may form a thiophene ring, a pyrrole ring, an imidazole ring, a benzene ring, a pyrimidine ring, a furan ring, a pyrazine ring, or a pyrrolidine ring.
摘要:
Agri-horticultural pest control compositions having outstanding control effect on pests, in particular, agri-horticultural pests, which comprise as active ingredients one or more 4-(3-butynyl)aminopyrimidine derivatives represented by the general formula [I], namely, where R1 is typically selected from among: a) phenyl c) —SiR5R6R7 (R5, R6, and R7 which may be the same or different represent a linear or branched alkyl having 1-6 carbon atoms, a linear or branched haloalkyl having 1-3 carbon atoms which is substituted by one halogen atom, a linear or branched cyanoalkyl having 1-3 carbon atoms which is substituted by one cyano group, and phenyl); d) hydropgen atom; R2 typically represents a hydrogen atom; R3 typically represents a hydrogen atom; R4 represents a hydrogen atom and one or more agri-horticultural pest control compounds selected from among agri-horticultural antimicrobial compounds, say, multi-site contact active compouns, nucleic acids synthesis inhibitory active compounds, mitosis and cell divesion inhibitory active compounds, and/or agri-horticultural insecticidal, miticidal or nematicidal compounds, say, acetylcholinesterase inhibitors, GABA-gated chloride antagonists, and sodium channel modulators. Since the 4-(3-butynyl)aminopyrimidine derivatives and the existing antimicrobial active compounds and/or insecticidal active compounds are used in admixture, the 4-(3-butynyl)aminopyrimidine derivatives which are useful as pest control agents, particularly as agri-horticultural pest control agents, need be used in smaller amounts and yet their antimicrobial or insecticidal activity can be improved.
摘要翻译:具有对害虫,特别是农业园艺害虫具有突出防治效果的农业园艺害虫防治组合物,其包含作为活性成分的一种或多种由通式[I]表示的4-(3-丁炔基)氨基嘧啶衍生物,即其中 R1通常选自:a)苯基c)-SiR 5 R 6 R 7(可以相同或不同的R 5,R 6和R 7表示具有1-6个碳原子的直链或支链烷基,具有1-3个直链或支链烷基的直链或支链烷基) 被一个卤素原子取代的碳原子,被一个氰基取代的具有1-3个碳原子的直链或支链氰基烷基和苯基); d)氢原子; R2通常表示氢原子; R3通常表示氢原子; R4表示氢原子和一种或多种选自农业园艺抗微生物化合物,例如多位点接触活性化合物,核酸合成抑制活性化合物,有丝分裂和细胞转移抑制活性化合物的农业园艺害虫控制化合物和/ 或农业园艺杀虫,杀螨或杀线虫化合物,例如乙酰胆碱酯酶抑制剂,GABA门控氯化物拮抗剂和钠通道调节剂。 由于4-(3-丁炔基)氨基嘧啶衍生物和现有的抗微生物活性化合物和/或杀虫活性化合物混合使用,可用作害虫防治剂的4-(3-丁炔基)氨基嘧啶衍生物,特别是农业 - 园艺害虫防治剂需要较少量使用,但可以提高其抗微生物或杀虫活性。
摘要:
Agri-horticultural pest control compositions having outstanding control effect on pests, in particular, agri-horticultural pests, which comprise as active ingredients one or more 4-(3-butynyl)aminopyrimidine derivatives represented by the general formula [I], namely, where R1 is typically selected from among: a) phenyl c) —SiR5R6R7 (R5, R6, and R7 which may be the same or different represent a linear or branched alkyl having 1-6 carbon atoms, a linear or branched haloalkyl having 1-3 carbon atoms which is substituted by one halogen atom, a linear or branched cyanoalkyl having 1-3 carbon atoms which is substituted by one cyano group, and phenyl); d) hydropgen atom; R2 typically represents a hydrogen atom; R3 typically represents a hydrogen atom; R4 represents a hydrogen atom and one or more agri-horticultural pest control compounds selected from among agri-horticultural antimicrobial compounds, say, multi-site contact active compounds, nucleic acids synthesis inhibitory active compounds, mitosis and cell division inhibitory active compounds, and/or agri-horticultural insecticidal, miticidal or nematicidal compounds, say, acetylcholinesterase inhibitors, GABA-gated chloride antagonists, and sodium channel modulators. Since the 4-(3-butynyl)aminopyrimidine derivatives and the existing antimicrobial active compounds and/or insecticidal active compounds are used in admixture, the 4-(3-butynyl)aminopyrimidine derivatives which are useful as pest control agents, particularly as agri-horticultural pest control agents, need be used in smaller amounts and yet their antimicrobial or insecticidal activity can be improved.
摘要翻译:具有对害虫,特别是农业园艺害虫具有突出防治效果的农业园艺害虫防治组合物,其包含作为活性成分的一种或多种由通式[I]表示的4-(3-丁炔基)氨基嘧啶衍生物,即其中 R1通常选自:a)苯基c)-SiR 5 R 6 R 7(可以相同或不同的R 5,R 6和R 7表示具有1-6个碳原子的直链或支链烷基,具有1-3个直链或支链烷基的直链或支链烷基) 被一个卤素原子取代的碳原子,被一个氰基取代的具有1-3个碳原子的直链或支链氰基烷基和苯基); d)氢原子; R2通常表示氢原子; R3通常表示氢原子; R4表示氢原子和一种或多种选自农业园艺抗微生物化合物,例如多位点接触活性化合物,核酸合成抑制活性化合物,有丝分裂和细胞分裂抑制活性化合物的农业园艺害虫控制化合物和/ 或农业园艺杀虫,杀螨或杀线虫化合物,例如乙酰胆碱酯酶抑制剂,GABA门控氯化物拮抗剂和钠通道调节剂。 由于4-(3-丁炔基)氨基嘧啶衍生物和现有的抗微生物活性化合物和/或杀虫活性化合物混合使用,可用作害虫防治剂的4-(3-丁炔基)氨基嘧啶衍生物,特别是农业 - 园艺害虫防治剂需要较少量使用,但可以提高其抗微生物或杀虫活性。
摘要:
An individually wrapped absorbent article 1 comprising an absorbent article 2 and a wrapping sheet 3, said absorbent article having a shape being relatively long in a longitudinal direction having a liquid-pervious top-sheet, a liquid-impervious back-sheet and a liquid-retentive absorbent core, on one hand, and said wrapping sheet 3 having a shape being also relatively long in the longitudinal direction arranged to cover the back-sheet of the absorbent article 2, on the other hand, so as to be folded back in the longitudinal direction of the absorbent article 2 by a predetermined fold length dimension L1, respectively, with the top-sheet inside. The wrapping sheet 3 is provided with a first display region 33 having a predetermined length dimension L3 as measured from one end of the wrapping sheet 3 in the longitudinal direction and the length dimension L3 of the first display region 33 is set to be smaller than the fold length dimension L1.
摘要:
A sanitary napkin comprises an absorbing body. The absorbing body includes a fluid-permeable top sheet, a fluid-impermeable back sheet, and an absorber arranged between the top sheet and the back sheet. The napkin comprises a cover sheet for covering the surface of the top sheet. A circumferential edge region of the cover sheet is joined to the absorbing body. A plurality of flaps for fixing the absorbing body to underwear are sectionalized by a sectionalizing line in the central region of the cover sheet. At the time of use, the flaps are folded in the folding regions and are expanded so as to be fixed to the underwear. The flaps include a front flap, a rear flap, a left flap and a right flap. A leakage-preventing region is formed on the cover sheet between the folding regions and the circumferential edge region.
摘要:
Substituted heterocyclic derivatives represented by the formula (I) ##STR1## wherein R, R.sup.1, R.sup.2, R.sup.3, R.sup.4, Q.sup.1, Q.sup.2, Q.sup.3, Q.sup.4, X and Y are as defined, including, specifically, the compound (E)-3-[3-[3-(2-methoxymethyl-8,8-dimethyl-4-nonen-6-ynyl)phenoxymethyl]phenyl]thiophene, exhibit squalene epoxidase inhibiting activity and are useful in the treatment or prophylaxis of hypercholesterolemia, hyperlipidemia and arteriosclerosis.
摘要:
A wiring clip 1 includes: an attaching portion 10 configured to be overlapped with a wiring harness; a locking portion 11 extended vertically from the attaching portion 10 and configured to be locked in a hole provided on a panel; and a pressing portion 12 configured to press the panel in a direction away from the attaching portion 10 when the locking portion 11 is locked in the hole. The pressing portion 12 includes: an inclined portion 19 continued to the attaching portion 10 and inclined with respect to both a vertically extending direction of the locking portion 11 from the attaching portion 10 and a longitudinal direction of the wiring harness overlapped with the attaching portion 10; and a parallel portion 20 continued to the inclined portion 19 and extended parallel to the locking portion 11 from the inclined portion 19. A surface 21a away from the panel of an intersecting portion 21 continued to both the inclined portion 19 and the parallel portion 20 is disposed further away from the panel than a surface 14a nearest the panel of the attaching portion 10.
摘要:
An individually wrapped absorbent article 1 comprising an absorbent article 2 and a wrapping sheet 3, said absorbent article having a shape being relatively long in a longitudinal direction having a liquid-pervious top-sheet, a liquid-impervious back-sheet and a liquid-retentive absorbent core, on one hand, and said wrapping sheet 3 having a shape being also relatively long in the longitudinal direction arranged to cover the back-sheet of the absorbent article 2, on the other hand, so as to be folded back in the longitudinal direction of the absorbent article 2 by a predetermined fold length dimension L1, respectively, with the top-sheet inside. The wrapping sheet 3 is provided with a first display region 33 having a predetermined length dimension L3 as measured from one end of the wrapping sheet 3 in the longitudinal direction and the length dimension L3 of the first display region 33 is set to be smaller than the fold length dimension L1.
摘要:
An absorbent article that realizes favorable erection of gathers and excels in transversal leakage preventing effects. There is disclosed a vertically long absorbent article comprising a surface layer with surface sheet (2), a backside layer with backside sheet (3), an absorbent layer with absorbent body (4) interposed therebetween and a pair of gathers (5,5) formed of a sheetlike member (9) so as to have a hollow on both the side areas of the surface layer in the longitudinal direction thereof. The pair of gathers (5,5) in the state of having a three-dimensional configuration part (10) wherein the sheetlike member (9) makes a convex on the external surface side of the absorbent article in the thickness direction thereof are joined to the surface layer and/or backside layer by a junction portion (11) provided so as to extend in the longitudinal direction of the absorbent article. The three-dimensional configuration part (10) is provided so as to construct a hollow. The junction portion (11) includes a first junction edge portion (10a) defining the edge portion of the three-dimensional configuration part (10) on the inward side in the width direction thereof and a second junction edge portion (10b) defining the edge portion of the three-dimensional configuration part (10) on the outward side in the width direction thereof. Providing that L1 refers to the length of the three-dimensional configuration part (10) from the first junction edge portion (10a) to the second junction edge portion (10b) and L2 refers to the inter-junction-edge-portion distance being the distance between the first junction edge portion (10a) and the second junction edge portion (10b), the ratio thereof, L1/L2 is 2 or greater.