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公开(公告)号:US09604938B2
公开(公告)日:2017-03-28
申请号:US14239193
申请日:2012-08-17
申请人: Michael Jonathan Bury , Linda N. Casillas , Adam K. Charnley , Michael P. Demartino , Xiaoyang Dong , Patrick M. Eidam , Pamela A. Haile , Robert W. Marquis, Jr. , Joshi M. Ramanjulu , Joseph J. Romano , Ami Lakdawala Shah , Robert R. Singhaus, Jr. , Gren Wang
发明人: Michael Jonathan Bury , Linda N. Casillas , Adam K. Charnley , Michael P. Demartino , Xiaoyang Dong , Patrick M. Eidam , Pamela A. Haile , Robert W. Marquis, Jr. , Joshi M. Ramanjulu , Joseph J. Romano , Ami Lakdawala Shah , Robert R. Singhaus, Jr. , Gren Wang
IPC分类号: C07D239/94 , C07D403/12 , C07D417/12 , C07D417/14 , C07D471/04
CPC分类号: C07D239/94 , C07D403/12 , C07D417/12 , C07D417/14 , C07D471/04
摘要: Disclosed are compounds having the formula (Formula I)): wherein R1, R2, R3 and Z are as defined herein, and methods of making and using the same.
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公开(公告)号:US20140206688A1
公开(公告)日:2014-07-24
申请号:US14239193
申请日:2012-08-17
申请人: Michael Jonathan Bury , Linda N. Casillas , Adam K. Charnley , Michael P. Demartino , Xiaoyang Dong , Patrick M. Eidam , Pamela A. Haile , Robert W. Marquis, JR. , Joshi M. Ramanjulu , Joseph J. Romano , Ami Lakdawala Shah , Robert R. Singhaus, JR. , Gren Wang
发明人: Michael Jonathan Bury , Linda N. Casillas , Adam K. Charnley , Michael P. Demartino , Xiaoyang Dong , Patrick M. Eidam , Pamela A. Haile , Robert W. Marquis, JR. , Joshi M. Ramanjulu , Joseph J. Romano , Ami Lakdawala Shah , Robert R. Singhaus, JR. , Gren Wang
IPC分类号: C07D239/94 , C07D471/04 , C07D417/14 , C07D417/12 , C07D403/12
CPC分类号: C07D239/94 , C07D403/12 , C07D417/12 , C07D417/14 , C07D471/04
摘要: Disclosed are compounds having the formula (Formula I)): wherein R1, R2, R3 and Z are as defined herein, and methods of making and using the same.
摘要翻译: 公开了具有式(式I))的化合物:其中R 1,R 2,R 3和Z如本文所定义,及其制备和使用方法。
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公开(公告)号:US20130018039A1
公开(公告)日:2013-01-17
申请号:US13637443
申请日:2011-03-31
申请人: Vera Q. Bodmer , Linda N. Casillas , Michael P. DeMartino , Philip A. Harris , Bryan W. King , Ami Lakdawala Shah , Lara Kathryn Leister , Joshi M. Ramanjulu , Joseph J. Romano , Gren Z. Wang , Matthew A. Wilson , David Duff Wisnoski
发明人: Vera Q. Bodmer , Linda N. Casillas , Michael P. DeMartino , Philip A. Harris , Bryan W. King , Ami Lakdawala Shah , Lara Kathryn Leister , Joshi M. Ramanjulu , Joseph J. Romano , Gren Z. Wang , Matthew A. Wilson , David Duff Wisnoski
IPC分类号: A61K31/4184 , C07D401/14 , C07D405/14 , C07D235/14 , C07D417/14 , C07D403/14 , C07D471/04 , A61K31/5377 , A61K31/4439 , A61K31/428 , A61K31/4245 , A61K31/437 , A61K31/496 , A61P17/00 , A61P3/10 , A61P19/02 , A61P1/04 , A61P1/16 , A61P11/06 , A61P37/06 , C07D413/14
CPC分类号: C07D417/14 , C07D401/14 , C07D403/04 , C07D403/14 , C07D405/14 , C07D413/14 , C07D471/04
摘要: Disclosed are compounds having the formula: wherein R1A, R1B, R2 and R3 are defined herein, and methods of making and using the same.
摘要翻译: 公开了具有下式的化合物:其中R1A,R1B,R2和R3如本文所定义,以及制备和使用该化合物的方法。
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公开(公告)号:US08399517B2
公开(公告)日:2013-03-19
申请号:US12894644
申请日:2010-09-30
IPC分类号: A61K31/195 , C07C229/00
CPC分类号: C07C217/54 , C07C217/30 , C07C217/32 , C07C217/34 , C07C229/34 , C07C2602/08
摘要: Novel calcilytic compounds and methods of using them are provided.
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公开(公告)号:US07829594B2
公开(公告)日:2010-11-09
申请号:US12393284
申请日:2009-02-26
IPC分类号: A61K31/195 , C07C229/00
CPC分类号: C07C217/54 , C07C217/30 , C07C217/32 , C07C217/34 , C07C229/34 , C07C2602/08
摘要: Novel calcilytic compounds and methods of using them are provided.
摘要翻译: 提供新的钙质化合物及其使用方法。
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公开(公告)号:US20090163589A1
公开(公告)日:2009-06-25
申请号:US12393284
申请日:2009-02-26
IPC分类号: A61K31/216 , A61K31/195
CPC分类号: C07C217/54 , C07C217/30 , C07C217/32 , C07C217/34 , C07C229/34 , C07C2602/08
摘要: Novel calcilytic compounds and methods of using them are provided.
摘要翻译: 提供新的钙质化合物及其使用方法。
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公开(公告)号:US07514473B2
公开(公告)日:2009-04-07
申请号:US10536416
申请日:2003-11-25
IPC分类号: C07C229/00 , A61K31/195
CPC分类号: C07C217/54 , C07C217/30 , C07C217/32 , C07C217/34 , C07C229/34 , C07C2602/08
摘要: Novel Calcilytic compounds and methods of using them are provided.
摘要翻译: 提供了新的钙质化合物及其使用方法。
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公开(公告)号:US07902394B2
公开(公告)日:2011-03-08
申请号:US12518482
申请日:2007-12-18
IPC分类号: C07C229/00 , C07D333/12 , A01N37/10
CPC分类号: C07C229/34 , C07C323/32 , C07C2602/08 , C07D333/20
摘要: Novel calcilytic compounds of Formula (I), pharmaceutical compositions, methods of synthesis, and methods of using them are provided.
摘要翻译: 提供式(I)的新型钙质化合物,药物组合物,合成方法及其使用方法。
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公开(公告)号:US20100029782A1
公开(公告)日:2010-02-04
申请号:US12518482
申请日:2007-12-18
IPC分类号: A61K31/135 , C07C215/00 , A61P19/00
CPC分类号: C07C229/34 , C07C323/32 , C07C2602/08 , C07D333/20
摘要: Novel calcilytic compounds of Formula (I), pharmaceutical compositions, methods of synthesis, and methods of using them are provided.
摘要翻译: 提供式(I)的新型钙质化合物,药物组合物,合成方法及其使用方法。
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公开(公告)号:US20090137557A1
公开(公告)日:2009-05-28
申请号:US12094665
申请日:2006-11-21
申请人: Thomas Wen Fu Ku , Hong Lin , Juan I. Luengo , Robert W. Marquis Jr. , Joshi M. Ramanjulu , Robert Trout , Dennis S. Yamashita
发明人: Thomas Wen Fu Ku , Hong Lin , Juan I. Luengo , Robert W. Marquis Jr. , Joshi M. Ramanjulu , Robert Trout , Dennis S. Yamashita
IPC分类号: A61K31/513 , C07D239/22 , C07D413/04 , A61K31/55 , A61P19/10 , A61K31/5377 , C07D487/04
CPC分类号: C07D239/36 , C07D239/40 , C07D239/47 , C07D239/72 , C07D239/91 , C07D401/04 , C07D403/04 , C07D405/04 , C07D409/04 , C07D409/06 , C07D409/14 , C07D413/14 , C07D417/04 , C07D417/14 , C07D487/04 , C07D491/044
摘要: Novel calcilytic compounds, pharmaceutical compositions, methods of synthesis and methods of using them are provided.
摘要翻译: 提供了新的钙化合物,药物组合物,合成方法和使用它们的方法。
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