Oxime derivatives, hydrazone derivatives and use thereof
    1.
    发明授权
    Oxime derivatives, hydrazone derivatives and use thereof 失效
    肟衍生物,腙衍生物及其用途

    公开(公告)号:US06251949B1

    公开(公告)日:2001-06-26

    申请号:US09457672

    申请日:1999-12-09

    IPC分类号: A61K3115

    摘要: Compounds having fungicidal activities and represented by general formula (I) and salts and hydrates thereof wherein R1 represents an optionally substituted aryl, an optionally substituted alkyl or the like; R2 represents an optionally substituted alkyl, an optionally substituted alkenyl, an optionally substituted alkynyl, an optionally substituted aryl, an optionally substituted heterocyclic group or the like; R3 represents an optionally substituted alkyl, an optionally substituted alkenyl, an optionally substituted alkynyl, an optionally substituted arylsulfonyl, an optionally substituted heterocyclic group or the like; R4 and R5, which may be the same or different, represent each a hydrogen atom, an optionally substituted alkyl, or an optionally substituted alkoxy, or R4 and R5 may form together with the adjacent nitrogen atom an optionally substituted monocycle or polycycle; X and Y, which may be the same or different, represents each an oxygen atom or NR6 wherein R6 represents a hydrogen atom, an optionally substituted alkyl, an optionally substituted aryl, an optionally substituted alkanoyl, or an optionally substituted aroyl; Z represents an oxygen atom or a sulfur atom; and a wavy line (˜) represents the configuration of an E isomer, a Z isomer, or a mixture thereof.

    摘要翻译: 具有杀真菌活性并由通式(I)表示的化合物及其盐和水合物,其中R 1表示任选取代的芳基,任选取代的烷基等; R 2表示任选取代的烷基,任选取代的烯基,任选取代的炔基,任选取代的芳基,任选取代的杂环基等; R 3表示任选取代的烷基,任选取代的烯基,任选取代的炔基,任选取代的芳基磺酰基,任选取代的杂环基团等; R 4和R 5可以相同或不同,表示氢原子,任选取代的烷基或任选取代的烷氧基,或者R 4和R 5可以与相邻的氮原子一起形成任选取代的单环或多环; X和Y可以相同或不同,表示每个氧原子或NR 6,其中R 6表示氢原子,任选取代的烷基,任选取代的芳基,任选取代的烷酰基或任选取代的芳酰基; Z表示氧原子或硫原子; 波浪线(〜)表示E异构体,Z异构体或其混合物的构型。

    Oxime derivative and bactericide containing the same as active ingredient
    9.
    发明授权
    Oxime derivative and bactericide containing the same as active ingredient 失效
    含有与活性成分相同的肟衍生物和杀菌剂

    公开(公告)号:US06268312B1

    公开(公告)日:2001-07-31

    申请号:US09370255

    申请日:1999-08-09

    IPC分类号: A01N4348

    摘要: A compound represented by general formula (I) or a salt thereof, a process for producing the same, an intermediate for the production thereof, and a bactericide (fungicide) containing the same as the active ingredient wherein R1 represent optionally substituted aryl, optionally substituted heterocycle, mono- or di-substituted methyleneamino, optionally substituted (substituted imino)methyl, optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkynyl, substituted carbonyl or substituted sulfonyl; R2 represents alkyl, alkenyl, alkynyl or cycloalkyl; R3 represents optionally substituted heterocycle; R4 represents hydrogen, alkyl, alkoxy, halogen, nitro, cyano or haloalkyl; M represents oxygen, S(O)i (i being 0, 1 or 2), NR16 (R16 being hydrogen, alkyl or acyl) or a single bond; n represents 0 or 1, provided n represent 1 when R3 represents imidazol-1-yl or 1H-1,2,4-triazol-1-yl; and the symbol˜represents the E form, Z form or a mixture thereof.

    摘要翻译: 由通式(I)表示的化合物或其盐,其制备方法,其制备中间体和含有该活性成分的杀菌剂(杀真菌剂),其中R 1表示任选取代的芳基,任选取代的 取代的亚氨基甲基,任选取代的烷基,任选取代的烯基,任选取代的炔基,取代的羰基或取代的磺酰基; R2代表烷基,烯基,炔基或环烷基; R3表示任选取代的杂环; R4代表氢,烷基,烷氧基,卤素,硝基,氰基或卤代烷基; M表示氧,S(O)i(i为0,1或2),NR 16(R 16为氢,烷基或酰基)或单键; 当R 3表示咪唑-1-基或1H-1,2,4-三唑-1-基时,n表示0或1,条件是n表示1。 符号〜表示E形式,Z形式或其混合物。