"> AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4
    4.
    发明申请
    AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4"-OR 4'-POSITION 有权
    在4“-OR 4'-位置具有烷氧基取代基的AVERMECTIN B1和AVERMECTIN B1单糖衍生物

    公开(公告)号:US20110230429A1

    公开(公告)日:2011-09-22

    申请号:US13117292

    申请日:2011-05-27

    IPC分类号: A01N43/22 C07H17/08 A01P7/00

    CPC分类号: C07H17/08 A61K31/7042

    摘要: What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

    摘要翻译: 描述的是下式的化合物,其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基,C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基,C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH,卤素,CN,-N 3,-NO 2,C 3 -C 8 - 环烷基,降冰片基 - ,C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基,C 1 -C 12烷氧基,C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基,C 3 -C 8环烷氧基,C 1 -C 12卤代烷氧基,C 1 -C 12烷硫基,C 3 -C 8环烷硫基, C 1 -C 12烷基亚磺酰基,C 3 -C 8环烷基亚磺酰基,C 1 -C 12卤代烷基亚磺酰基,C 3 -C 8卤代环烷基亚磺酰基,C 1 -C 12烷基磺酰基,C 3 -C 8环烷基磺酰基,C 1 -C 12卤代烷基磺酰基, 卤代环烷基磺酰基,-NR4R6,-X-C(= Y)-R4,-X-C(= Y)-Z-R4,-P(= O)(OC1-C6-烷基)2,芳基,杂环基,芳氧基, 芳硫基和杂环氧基; R3是例如任选取代的H,C 1 -C 12 - 烷基或C 1 -C 12 - 烷基,并且在适用的情况下,E / Z异构体,E / Z异构体和/或互变异构体的混合物,在每种情况下为游离形式或 盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法,以及这些化合物和组合物的用途。

    3-AMINO-BENZO [D] ISOTHIAZOLE DIOXIDE DERIVATIVES AND THEIR USE AS PESTICIDES
    5.
    发明申请
    3-AMINO-BENZO [D] ISOTHIAZOLE DIOXIDE DERIVATIVES AND THEIR USE AS PESTICIDES 失效
    3-氨基苯并[D]异噻唑二酮衍生物及其作为杀虫剂的用途

    公开(公告)号:US20110071200A1

    公开(公告)日:2011-03-24

    申请号:US12993983

    申请日:2009-05-18

    CPC分类号: C07D275/06

    摘要: A compound of Formula (I) or Formula (II) where W is C—R3; X is C—R4; Y is C—R5; R1 and R6, independently of each other, is, for example, H, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl or C1-C6-alkyl-C(═O); R2 is H; and R3, R4 and R5, independently of each other, are, for example, H, halogen, cyano, nitro, C1-C6-alkyl, or C1-C6-haloalkyl; provided that in formula II R1 is H and R6 is as defined above; and in formula I that (a) at least one of R1 and R3 to R6 is other than hydrogen, (b) R3 or R4 is other than C1 when in each instance the remaining five groups of R1 to R6 are hydrogen, and (c) (i) R3 is other than methyl, (ii) R4 is other than C1, (iii) R5 is other than C1 and (iv) R3 is not C1 when R5 is methoxy, when in each instance (i) to (iv) R1 is H, R6 is MeC(═O), and remaining groups of R2 to R5 are hydrogen; and/or salts thereof; and their use as as pesticidal agents.

    摘要翻译: 式(I)或式(II)的化合物,其中W是C-R 3; X是C-R4; Y为C-R5; R 1和R 6彼此独立地是例如H,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基,C 2 -C 6 - 炔基,C 3 -C 8 - 环烷基或C 1 -C 6 - 烷基-C(= O ); R2为H; 和R 3,R 4和R 5彼此独立地是例如H,卤素,氰基,硝基,C 1 -C 6烷基或C 1 -C 6卤代烷基; 条件是式Ⅱ中R 1为H且R 6如上定义; (a)R1和R3至R6中的至少一个不是氢,(b)R 3或R 4不同于C 1,当R 5至R 6的剩余五个基团为氢时,和(c )(i)R 3不是甲基,(ⅱ)R 4不是C 1,(ⅲ)R 5不是C 1,(ⅳ)当R 5是甲氧基时,R 3不是C 1,当(i)〜 )R1为H,R6为MeC(= O),R2至R5的其余基团为氢; 和/或其盐; 以及其作为杀虫剂的用途。

    Chemical compounds
    6.
    发明授权
    Chemical compounds 失效
    化合物

    公开(公告)号:US08629284B2

    公开(公告)日:2014-01-14

    申请号:US13129063

    申请日:2009-10-27

    摘要: A compound of the formula I or where W, X and Y are for example each CH; R1 is H; R2 is halogen; and R6 is, for formula I, for example, OH, CN, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C6-alkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkenyloxy, C2-C6-alkynyl, C2-C6-haloalkynyl, C2-C6-alkynyloxy, optionally substituted C1 to C3-alkyl, or optionally substituted C1-C6-alkoxy, or R6 is, for formula II, for example, CN, C3-C8-cycloalkyl, or optionally substituted C3-C6-alkyl; and/or salts thereof; and their use as as pesticidal agents.

    摘要翻译: 式I化合物或其中W,X和Y为例如CH; R1是H; R2是卤素; 对于式I,R 6为例如OH,CN,C 3 -C 8 - 环烷基,C 3 -C 8 - 环烷基-C 1 -C 6烷基,C 2 -C 6 - 烯基,C 2 -C 6 - 卤代烯基,C 2 -C 6 - 烯氧基 ,C 2 -C 6炔基,C 2 -C 6 - 卤代炔基,C 2 -C 6 - 炔氧基,任选取代的C 1至C 3 - 烷基或任选取代的C 1 -C 6 - 烷氧基,或R 6为式II,例如CN,C 3 -C 8 - 环烷基或任选取代的C 3 -C 6 - 烷基; 和/或其盐; 以及其作为杀虫剂的用途。

    3-amino-benzo [D] isothiazole dioxide derivatives and their use as pesticides
    7.
    发明授权
    3-amino-benzo [D] isothiazole dioxide derivatives and their use as pesticides 失效
    3-氨基 - 苯并[D]异噻唑二氧化物衍生物及其作为农药的用途

    公开(公告)号:US08563744B2

    公开(公告)日:2013-10-22

    申请号:US12993983

    申请日:2009-05-18

    IPC分类号: C07D275/06 A61K31/425

    CPC分类号: C07D275/06

    摘要: A compound of Formula (I) or Formula (II) where W is C—R3; X is C—R4; Y is C—R5; R1 and R6, independently of each other, is, for example, H, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl or C1-C6-alkyl-C(═O); R2 is H; and R3, R4 and R5, independently of each other, are, for example, H, halogen, cyano, nitro, C1-C6-alkyl, or C1-C6-haloalkyl; provided that in formula II R1 is H and R6 is as defined above; and in formula I that (a) at least one of R1 and R3 to R6 is other than hydrogen, (b) R3 or R4 is other than C1 when in each instance the remaining five groups of R1 to R6 are hydrogen, and (c) (i) R3 is other than methyl, (ii) R4 is other than C1, (iii) R5 is other than C1 and (iv) R3 is not C1 when R5 is methoxy, when in each instance (i) to (iv) R1 is H, R6 is MeC(═O), and remaining groups of R2 to R5 are hydrogen; and/or salts thereof; and their use as as pesticidal agents.

    摘要翻译: 式(I)或式(II)的化合物,其中W是C-R 3; X是C-R4; Y为C-R5; R 1和R 6彼此独立地是例如H,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基,C 2 -C 6 - 炔基,C 3 -C 8 - 环烷基或C 1 -C 6 - 烷基-C(= O ); R2为H; 和R 3,R 4和R 5彼此独立地是例如H,卤素,氰基,硝基,C 1 -C 6烷基或C 1 -C 6卤代烷基; 条件是式Ⅱ中R 1为H且R 6如上定义; (a)R1和R3至R6中的至少一个不是氢,(b)R 3或R 4不同于C 1,当R 5至R 6的剩余五个基团为氢时,和(c )(i)R 3不是甲基,(ⅱ)R 4不是C 1,(ⅲ)R 5不是C 1,(ⅳ)当R 5是甲氧基时,R 3不是C 1,当(i)〜 )R1为H,R6为MeC(= O),R2至R5的其余基团为氢; 和/或其盐; 以及其作为杀虫剂的用途。

    "> Avermectins and Avermectin Monosacharides Substituted in the 4'-and 4
    8.
    发明申请
    Avermectins and Avermectin Monosacharides Substituted in the 4'-and 4" Position Having Pesticidal Properties 有权
    在4'和4“位置具有农药性质的阿维菌素和阿维菌素单糖

    公开(公告)号:US20080194498A1

    公开(公告)日:2008-08-14

    申请号:US10568715

    申请日:2004-08-27

    IPC分类号: A01N43/90 C07H17/08 A01P17/00

    CPC分类号: A01N43/90 C07H19/01

    摘要: Described is a compound of the formula (1) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and either (A) R2 is —N(R3)R4, and (1) X is 0, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl; or (2) X is S, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl; or (3) X is 0 or S, wherein R3 and R4 together are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) R2 is OR5, X is 0 or S, wherein R5 is, for instance, C1-C12alkyl, mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity.

    摘要翻译: 描述了式(1)的化合物,其中碳原子22和23之间的键是单键或双键; m为0或1; R 1是C 1 -C 12烷基,C 3 -C 8烷基,C 3 -C 12烷基,C 3 -C 12烷基,C 3 -C 12烷基, >环烷基或C 2 -C 12 - 烯基; (A)R 2是-N(R 3)R 4,和(1)X是0,其中R 3是例如氢,未取代的或一至五取代的C 1 -C 12烷基,R 4是氢, 是例如一至五取代的C 1 -C 12烷基,未取代或单取代或五取代的C 3 -C 12烷基, 12环烷基; 或(2)X是S,其中R 3是例如氢,未取代的或一至五取代的C 1 -C 12 - 烷基和R 4是例如氢,未取代的或一至五取代的C 1 -C 12烷基; 或(3)X为0或S,其中R 3和R 4一起为例如三至七元亚烷基或四至七元亚烷基, 多元亚烯基桥; 或(B)R 2是OR 5,X是0或S,其中R 5是例如C 1 C 1 -C 12烷基,一至五取代C 1 -C 12烷基; 或者如果合适的话,E / Z异构体,E / Z异构体混合物和/或其互变异构体在每种情况下都是游离形式或盐形式; 这种化合物显示出杀虫活性。