-
公开(公告)号:US20090318443A1
公开(公告)日:2009-12-24
申请号:US12509886
申请日:2009-07-27
申请人: Rosanne Bonjouklian , Chafiq Hamdouchi Hamdouchi , Chuan Shih , Alfonso De Dios , Miriam Filadelfa Del Prado , Carlos Jaramillo Aguado , Pramila Kotiyan , Mary Margaret Mader , Sheila Pleite Selgas , Concepcion Sanchez-Martinez
发明人: Rosanne Bonjouklian , Chafiq Hamdouchi Hamdouchi , Chuan Shih , Alfonso De Dios , Miriam Filadelfa Del Prado , Carlos Jaramillo Aguado , Pramila Kotiyan , Mary Margaret Mader , Sheila Pleite Selgas , Concepcion Sanchez-Martinez
IPC分类号: A61K31/5377 , A61K31/437 , A61P35/00
CPC分类号: C07D471/04
摘要: The present invention provides kinase inhibitors of Formula I.
-
公开(公告)号:US07582652B2
公开(公告)日:2009-09-01
申请号:US10597283
申请日:2005-01-25
申请人: Rosanne Bonjouklian , Chafiq Hamdouchi , Chuan Shih , Alfonso De Dios , Miriam Filadelfa del Prado , Carlos Jaramillo Aguado , Pramila Kotiyan , Mary Margaret Mader , Sheila Pleite Selgas , Concepcion Sanchez-Martinez
发明人: Rosanne Bonjouklian , Chafiq Hamdouchi , Chuan Shih , Alfonso De Dios , Miriam Filadelfa del Prado , Carlos Jaramillo Aguado , Pramila Kotiyan , Mary Margaret Mader , Sheila Pleite Selgas , Concepcion Sanchez-Martinez
IPC分类号: A01N43/42 , A61K31/44 , C07D513/02 , C07D515/02
CPC分类号: C07D471/04
摘要: The present invention provides kinase inhibitors of Formula I.
摘要翻译: 本发明提供式I的激酶抑制剂。
-
公开(公告)号:US20090036445A1
公开(公告)日:2009-02-05
申请号:US10597283
申请日:2005-01-25
申请人: Rosanne Bonjouklian , Chafiq Hamdouchi , Chuan Shih , Alfonso De Dios , Miriam Filadelfa del Prado , Carlos Jaramillo Aguado , Pramila Kotiyan , Mary Margaret Mader , Sheila Pleite Selgas , Concepcion Sanchez-Martinez
发明人: Rosanne Bonjouklian , Chafiq Hamdouchi , Chuan Shih , Alfonso De Dios , Miriam Filadelfa del Prado , Carlos Jaramillo Aguado , Pramila Kotiyan , Mary Margaret Mader , Sheila Pleite Selgas , Concepcion Sanchez-Martinez
IPC分类号: A61K31/437 , A61P35/00 , A61K31/5377 , C07D471/04
CPC分类号: C07D471/04
摘要: The present invention provides kinase inhibitors of Formula I.
摘要翻译: 本发明提供式I的激酶抑制剂。
-
公开(公告)号:US07320995B2
公开(公告)日:2008-01-22
申请号:US10522227
申请日:2003-07-31
申请人: Rosanne Bonjouklian , Jose Eugenio De Diego Gomez , Alfonso De Dios , Chafiq Hamdouchi Hamdouchi , Tiecho Li , Beatriz Lopez De Uralde Garmendia , Michal Vieth , Jeremy Schulenberg York , Robert Dean Dally , Miriam Filadelfa Del Prado Catalina , Carlos Jaramillo Aguado , Luisa Maria Martin-Cabrejas , Carlos Montero Salgado , Sheila Pleite Selgas , Concepcion Sanchez-Martinez , Timothy Alan Shepherd , James Howard Wikel
发明人: Rosanne Bonjouklian , Jose Eugenio De Diego Gomez , Alfonso De Dios , Chafiq Hamdouchi Hamdouchi , Tiecho Li , Beatriz Lopez De Uralde Garmendia , Michal Vieth , Jeremy Schulenberg York , Robert Dean Dally , Miriam Filadelfa Del Prado Catalina , Carlos Jaramillo Aguado , Luisa Maria Martin-Cabrejas , Carlos Montero Salgado , Sheila Pleite Selgas , Concepcion Sanchez-Martinez , Timothy Alan Shepherd , James Howard Wikel
IPC分类号: A61K31/4184 , A61K31/428 , C07D277/68 , C07D235/10
CPC分类号: C07D403/04 , C07D413/04 , C07D413/14 , C07D417/04 , C07D513/04
摘要: The present invention provides kinase inhibitors of Formula I: wherein W represents inter alia imidazol, oxazol, pyrazol, thiazol as triazol, which are substituted by phenyl or thienyl. The disclosed compounds inhibit p-38 kinase and are useful in the treatment of metastasis or rheumatoid arthritis
摘要翻译: 本发明提供式I的激酶抑制剂:其中W代表由苯基或噻吩取代的咪唑,恶唑,吡唑,噻唑三唑。 所公开的化合物抑制p-38激酶,并且可用于治疗转移或类风湿性关节炎
-
公开(公告)号:US20050272791A1
公开(公告)日:2005-12-08
申请号:US10522227
申请日:2003-07-31
申请人: Rosanne Bonjouklian , Jose De Diego Gomez , Alfonso De Dios , Chafiq Hamdouchi , Tiecho Li , Beatriz De Uralde Garmendia , Michal Vieth , Jeremy York , Robert Dally , Miriam Del Prado Catalina , Carlos Jaramillo Aguado , Luisa Martin-Cabrejas , Carlos Montero Salgado , Sheila Pleite Selgas , Concepcion Sanchez-Martinez , Timothy Shepherd , James Wikel
发明人: Rosanne Bonjouklian , Jose De Diego Gomez , Alfonso De Dios , Chafiq Hamdouchi , Tiecho Li , Beatriz De Uralde Garmendia , Michal Vieth , Jeremy York , Robert Dally , Miriam Del Prado Catalina , Carlos Jaramillo Aguado , Luisa Martin-Cabrejas , Carlos Montero Salgado , Sheila Pleite Selgas , Concepcion Sanchez-Martinez , Timothy Shepherd , James Wikel
IPC分类号: A61K31/41 , A61K31/4184 , A61P35/04 , C07D401/14 , C07D403/04 , C07D403/14 , C07D405/14 , C07D409/04 , C07D409/14 , C07D413/04 , C07D413/14 , C07D417/04 , C07D471/04 , C07D487/04 , C07D513/04 , C07D43/02
CPC分类号: C07D403/04 , C07D413/04 , C07D413/14 , C07D417/04 , C07D513/04
摘要: The present invention provides kinase inhibitors of Formula I: wherein W represents inter alia imidazol, oxazol, pyrazol, thiazol as triazol, which are substituted by phenyl or thienyl. The disclosed compounds inhibit p-38 kinase and are useful in the treatment of metastasis or rheumatoid arthritis.
摘要翻译: 本发明提供式I的激酶抑制剂:其中W代表由苯基或噻吩取代的咪唑,恶唑,吡唑,噻唑三唑。 所公开的化合物抑制p-38激酶,并且可用于治疗转移或类风湿性关节炎。
-
6.
公开(公告)号:US20080275056A1
公开(公告)日:2008-11-06
申请号:US12089420
申请日:2006-10-23
申请人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz Lopez Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz Lopez Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/496 , C07D401/14 , A61K31/4725
CPC分类号: C07D403/12 , C07D403/14
摘要: The present invention provides kinase inhibitors of Formula (I) wherein R1, R2, and X are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供其中R1,R2和X如本文所述的式(I)的激酶抑制剂或其药学上可接受的盐。
-
公开(公告)号:US07084170B2
公开(公告)日:2006-08-01
申请号:US10490935
申请日:2002-10-15
申请人: Cora Sue Grossman , Philip Arthur Hipskind , Ho-Shen Lin , Karen Lynn Lobb , Beatriz Lopez de Uralde Garmendia , Jose Eduardo Lopez , Mary Margaret Mader , Michael Enrico Richett , Chuan Shih , Alfonso De Dios
发明人: Cora Sue Grossman , Philip Arthur Hipskind , Ho-Shen Lin , Karen Lynn Lobb , Beatriz Lopez de Uralde Garmendia , Jose Eduardo Lopez , Mary Margaret Mader , Michael Enrico Richett , Chuan Shih , Alfonso De Dios
IPC分类号: A61K31/381 , C07D333/34
CPC分类号: C07D277/36 , C07D333/34 , C07D333/38
摘要: The present invention provides antineoplastic compounds of the formula: and antineoplastic methods.
摘要翻译: 本发明提供下式的抗肿瘤化合物和抗肿瘤方法。
-
公开(公告)号:US07250430B2
公开(公告)日:2007-07-31
申请号:US11447457
申请日:2006-06-06
申请人: Cora Sue Grossman , Philip Arthur Hipskind , Ho-Shen Lin , Karen Lynn Lobb , Beatriz Lopez de Uralde Garmendia , Jose Eduardo Lopez , Mary Margaret Mader , Michael Enrico Richett , Chuan Shih , Alfonso De Dios
发明人: Cora Sue Grossman , Philip Arthur Hipskind , Ho-Shen Lin , Karen Lynn Lobb , Beatriz Lopez de Uralde Garmendia , Jose Eduardo Lopez , Mary Margaret Mader , Michael Enrico Richett , Chuan Shih , Alfonso De Dios
IPC分类号: A61K31/381 , A61K31/426
CPC分类号: C07D277/36 , C07D333/34 , C07D333/38
摘要: The present invention provides antineoplastic compounds of the formula: and antineoplastic methods.
摘要翻译: 本发明提供下式的抗肿瘤化合物和抗肿瘤方法。
-
公开(公告)号:US07652015B2
公开(公告)日:2010-01-26
申请号:US12088526
申请日:2006-10-25
申请人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz López De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz López De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/4439 , A61K31/454 , C07D401/12 , C07D401/14 , C07D409/14
CPC分类号: C07D401/12 , C07D401/14
摘要: The present invention provides kinase inhibitors of Formula (I). Wherein R1, R2, X and Z are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供式(I)的激酶抑制剂。 其中R1,R2,X和Z如本文所述,或其药学上可接受的盐。
-
10.
公开(公告)号:US07582638B2
公开(公告)日:2009-09-01
申请号:US12089420
申请日:2006-10-23
申请人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz López de Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz López de Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/4725 , A61K31/496 , C07D403/141
CPC分类号: C07D403/12 , C07D403/14
摘要: The present invention provides kinase inhibitors of Formula (I) wherein R1, R2, and X are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供其中R1,R2和X如本文所述的式(I)的激酶抑制剂或其药学上可接受的盐。
-
-
-
-
-
-
-
-
-