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1.
公开(公告)号:US20150272120A1
公开(公告)日:2015-10-01
申请号:US14441304
申请日:2013-11-08
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: Myriem El Qacemi , Jerome Yves Cassayre , Guillaume Berthon , Girish Rawal , Rupesh Patre
IPC: A01N43/10 , C07D333/24 , C07D409/12 , A01N43/20 , A01N43/653 , A01N43/80 , A01N43/40 , C07D333/32 , C07D333/48 , C07D409/10 , C07D333/40 , C07D413/12
CPC classification number: A01N43/10 , A01N37/10 , A01N43/20 , A01N43/40 , A01N43/653 , A01N43/80 , C07D333/24 , C07D333/32 , C07D333/38 , C07D333/40 , C07D333/48 , C07D409/10 , C07D409/12 , C07D413/12
Abstract: The present invention provides compounds of formula (I) wherein Q is Q1 or Q2 P is P0, heterocyclyl or heterocyclyl substituted by one to five Z; Y1, Y2, Y3 and Y4 are independently of each other C—H, C—R5, or nitrogen; G1 is oxygen or sulfur; R1 is hydrogen, C1-C8alkyl, C1-C8alkoxy-, C1-C8alkylcarbonyl-, or C1-C8alkoxycarbonyl-; X4 is C1-C8haloalkyl; R4 is aryl or aryl substituted by one to five R9, or heteroaryl or heteroaryl substituted by one to five R9; n is 0, 1 or 2; and Z, R2, R5 and R9 are as defined in the claims. The invention also provides methods of controlling insects, acarines, nematodes or molluscs comprising applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, nematicidally or molluscicidally effective amount of a compound of formula (I).
Abstract translation: 本发明提供式(I)化合物,其中Q为Q 1或Q 2为PO,杂环基或被1至5个Z取代的杂环基; Y1,Y2,Y3和Y4彼此独立地为C-H,C-R5或氮; G1是氧或硫; R 1是氢,C 1 -C 8烷基,C 1 -C 8烷氧基 - ,C 1 -C 8烷基羰基 - 或C 1 -C 8烷氧基羰基 - X4是C1-C8卤代烷基; R4是被1至5个R9取代的芳基或芳基,或被1至5个R9取代的杂芳基或杂芳基; n为0,1或2; 并且Z,R2,R5和R9如权利要求中所定义。 本发明还提供了控制昆虫,螨虫,线虫或软体动物的方法,其包括将有害生物施用于有害生物的场所或易受害虫攻击的植物,杀虫剂,杀螨剂,杀线虫剂或杀软体动物剂有效量的化合物 的式(I)化合物。
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公开(公告)号:US09598389B2
公开(公告)日:2017-03-21
申请号:US14771600
申请日:2014-03-06
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: Long Lu , Jerome Yves Cassayre , Torsten Luksch , Myriem El Qacemi , Guillaume Berthon , Yaming Wu
IPC: C07D307/79 , C07C233/33 , A01N43/10 , C07D405/12 , C07D413/12 , A01N43/80 , C07D409/12 , A01N43/40 , A01N43/60 , C07C233/25 , C07D405/10 , A01N43/90 , A01N43/12 , C07D333/54 , C07D405/04 , A01N37/22 , A01N43/20 , A01N43/54 , A01N43/713
CPC classification number: C07D307/79 , A01N37/22 , A01N43/10 , A01N43/12 , A01N43/20 , A01N43/40 , A01N43/54 , A01N43/60 , A01N43/713 , A01N43/80 , A01N43/90 , C07C233/25 , C07C233/33 , C07D333/54 , C07D405/04 , C07D405/10 , C07D405/12 , C07D409/12 , C07D413/12
Abstract: Provided are compounds of formula (I) and methods of controlling insects, acarines, nematodes or molluscs, which comprises applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, nematicidally or molluscicidally effective amount of a compound of formula (I).
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公开(公告)号:US20140128358A1
公开(公告)日:2014-05-08
申请号:US13878118
申请日:2011-10-03
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: Jerome Yves Cassayre , Peter Renold , Myriem El Qacemi , Guillaume Berthon
CPC classification number: A01N43/78 , A01N43/36 , A01N43/40 , A01N43/50 , A01N43/60 , C07D207/08 , C07D401/04 , C07D409/10 , C07D409/14
Abstract: The invention relates to compounds of formula (I): where A1, A2, A3, A4, G1, R1, R2, R3 and R4 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.
Abstract translation: 本发明涉及式(I)化合物:其中A1,A2,A3,A4,G1,R1,R2,R3和R4如权利要求1所定义; 或其盐或N-氧化物。 此外,本发明涉及制备式(I)化合物的方法和中间体,其包含式(I)化合物的杀虫,杀螨,杀线虫和杀软体动物的组合物和使用式(I)化合物控制的方法 昆虫,螨虫,线虫和软体动物害虫。
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公开(公告)号:US09686988B2
公开(公告)日:2017-06-27
申请号:US14442699
申请日:2013-11-21
Applicant: Syngenta Participations AG
Inventor: Girish Rawal , Rupesh Patre , Guillaume Berthon , Jerome Yves Cassayre , Myriem El Qacemi
IPC: A01N43/80 , A01N43/10 , C07D261/04 , C07D333/18 , C07D413/12 , C07D333/38
CPC classification number: A01N43/80 , A01N43/10 , C07D261/04 , C07D333/18 , C07D333/38 , C07D413/12
Abstract: The present invention provides compounds of formula (I) wherein R1, R2, R3, R4, n, A1, A2, A3, Y1, Y2, and Y3 are as defined in the claims. The invention also relates to processes and intermediates for preparing these compounds, to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising these compounds and to methods of using these compounds to control insect, acarine, nematode and mollusc pests.
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公开(公告)号:US10517294B2
公开(公告)日:2019-12-31
申请号:US14441304
申请日:2013-11-08
Applicant: Syngenta Participations AG
Inventor: Myriem El Qacemi , Jerome Yves Cassayre , Guillaume Berthon , Girish Rawal , Rupesh Patre
IPC: A01N43/10 , C07D333/40 , C07D333/24 , C07D409/12 , A01N43/20 , C07D413/12 , A01N43/80 , A01N43/40 , C07D333/32 , C07D333/48 , C07D409/10 , A01N43/653 , A01N37/10 , C07D333/38
Abstract: The present invention provides compounds of formula (I) wherein Q is Q1 or Q2 P is P0, heterocyclyl or heterocyclyl substituted by one to five Z; Y1, Y2, Y3 and Y4 are independently of each other C—H, C—R5, or nitrogen; G1 is oxygen or sulfur; R1 is hydrogen, C1-C8alkyl, C1-C8alkoxy-, C1-C8alkylcarbonyl-, or C1-C8alkoxycarbonyl-; X4 is C1-C8haloalkyl; R4 is aryl or aryl substituted by one to five R9, or heteroaryl or heteroaryl substituted by one to five R9; n is 0, 1 or 2; and Z, R2, R5 and R9 are as defined in the claims. The invention also provides methods of controlling insects, acarines, nematodes or molluscs comprising applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, nematicidally or molluscicidally effective amount of a compound of formula (I).
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公开(公告)号:US20170283405A1
公开(公告)日:2017-10-05
申请号:US15628804
申请日:2017-06-21
Applicant: Syngenta Participations AG
Inventor: Long Lu , Jerome Yves Cassayre , Guillaume Berthon , Myriem El Qacemi , Yaming Wu
IPC: C07D413/12 , C07D231/06 , A01N43/78 , A01N43/80 , C07D409/12 , A01N53/00 , A01N43/60 , A01N43/90 , A01N43/16 , A01N43/56 , A01N43/58
CPC classification number: C07D413/12 , A01N43/16 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/78 , A01N43/80 , A01N43/90 , A01N53/00 , C07D231/06 , C07D409/12
Abstract: The present invention relates to compounds of formula I wherein P is selected from P1 and P2, or P and R5 together are P3 or P is a heterocycle H, selected from H1 to H9 wherein Y1, Y2, and Y3 are independently of each other C—H, C—R5, or nitrogen; and G1, G2, G3, Z, R1, R2, R3, R4, R5, R6a, R6b, R7, R8, R9, R10, R11, p, n and k are as defined in the claims. The invention also relates to methods of controlling insects, acarines, nematodes or molluscs which comprises applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, nematicidally or molluscicidally effective amount of a compound of formula I.
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公开(公告)号:US10287281B2
公开(公告)日:2019-05-14
申请号:US15628804
申请日:2017-06-21
Applicant: Syngenta Participations AG
Inventor: Long Lu , Jerome Yves Cassayre , Guillaume Berthon , Myriem El Qacemi , Yaming Wu
IPC: C07D413/12 , C07D231/36 , C07D409/12 , A01N43/78 , A01N53/00 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/90 , A01N43/16 , C07D231/06 , A01N43/80
Abstract: The present invention relates to compounds of formula I wherein P is selected from P1 and P2, or P and R5 together are P3 or P is a heterocycle H, selected from H1 to H9 wherein Y1, Y2, and Y3 are independently of each other C—H, C—R5, or nitrogen; and G1, G2, G3, Z, R1, R2, R3, R4, R5, R6a, R6b, R7, R8, R9, R10, R11, p, n and k are as defined in the claims. The invention also relates to methods of controlling insects, acarines, nematodes or molluscs which comprises applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, nematicidally or molluscicidally effective amount of a compound of formula I.
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公开(公告)号:US09776994B2
公开(公告)日:2017-10-03
申请号:US14762319
申请日:2014-01-23
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: Long Lu , Jerome Yves Cassayre , Guillaume Berthon , Myriem El Qacemi , Yaming Wu
IPC: C07D413/12 , C07D231/06 , C07D409/12 , A01N43/56 , A01N43/80 , A01N43/58 , A01N43/60 , A01N43/90 , A01N53/00 , A01N43/16 , A01N43/78
CPC classification number: C07D413/12 , A01N43/16 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/78 , A01N43/80 , A01N43/90 , A01N53/00 , C07D231/06 , C07D409/12
Abstract: The present invention relates to compounds of formula (I) wherein P is selected from P1 and P2, or P and R5 together are P3 or P is a heterocycle H, selected from H1 to H9 wherein Y1, Y2 and Y3 are independently of each other C—H, C—R5, or nitrogen; and G1, G2, G3, Z, R1, R2, R3, R4, R5, R6a, R6b, R7, R8, R9, R10, R11, p, n and k are as defined in the claims. The invention also relates to methods of controlling insects, acarines, nematodes or molluscs which comprises applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, nematicidally or molluscicidally effective amount of a compound of formula (I).
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9.
公开(公告)号:US09675073B2
公开(公告)日:2017-06-13
申请号:US14442952
申请日:2013-11-21
Applicant: Syngenta Participations AG
Inventor: Girish Rawal , Rupesh Patre , Guillaume Berthon , Jerome Yves Cassayre , Myriem El Qacemi
IPC: A01N43/80 , A01N43/10 , C07D333/24 , C07D261/04 , C07D413/12 , C07C317/32 , A01N43/36 , C07D333/18 , A01N43/08
CPC classification number: A01N43/80 , A01N43/08 , A01N43/10 , A01N43/36 , C07C317/32 , C07D261/04 , C07D333/18 , C07D333/24 , C07D413/12
Abstract: The present invention provides compounds of formula (I) wherein R1, R2, R3, R4, n, A1, A2, A3, A4, Y1, Y2 and Y3 are as defined in the claims. The invention also relates to processes and intermediates for preparing these compounds, to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising these compounds and to methods of using these compounds to control insect, acarine, nematode and mollusc pests.
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10.
公开(公告)号:US09469633B2
公开(公告)日:2016-10-18
申请号:US14346773
申请日:2012-09-28
Applicant: SYNGENTA PARTICIPATIONS AG
Inventor: Tomas Smejkal , Helmars Smits , Sebastian Volker Wendeborn , Guillaume Berthon , Jerome Yves Cassayre , Myriem El Qacemi
IPC: C07D207/408 , C07D207/40 , C07D207/404 , C08F8/32 , C07D207/412 , C07D207/325 , C07C255/41 , C07C253/10 , C07C253/30 , C07D453/04 , C07D409/12 , C07D207/08 , C07D207/267 , C07D207/333 , C07D307/46 , C07C255/40 , C07D207/12
CPC classification number: C07D453/04 , C07C253/10 , C07C253/30 , C07C255/40 , C07C255/41 , C07D207/08 , C07D207/12 , C07D207/267 , C07D207/325 , C07D207/333 , C07D207/40 , C07D307/46 , C07D409/12
Abstract: The present invention relates to processes for the enantio-selective preparation of spyrrolidine derivatives useful in the manufacture of pesticidally active compounds, as well as to intermediates in the processes. The processes include those comprising(a-i) reacting a compound of formula Ia wherein P is alkyl, aryl or heteroaryl, each optionally substituted, wherein the heteroaryl is connected at P via a ring carbon atom; R1 is chlorodifluoromethyl or trifluoromethyl; R2 is aryl or heteroaryl, each optionally substituted; with a source of cyanide in the presence a chiral catalyst to give a compound of formula IIa wherein P, R1 and R2 are as defined for the compound of formula Ia; and (a-ii) oxidizing the compound of formula IIa with a peroxy acid, or peroxide in the presence of an acid to give a compound of formula VI wherein R1 and R2 are as defined for the compound of formula Ia.
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