公开(公告)号：US20100311974A1

公开(公告)日：2010-12-09

申请号：US12846235

申请日：2010-07-29

申请人： Takashi FURUYA ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

发明人： Takashi FURUYA ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

IPC分类号： C07D241/12 ,  C07C211/52

CPC分类号： A01N43/60 ,  C07C211/52 ,  C07C217/08 ,  C07C217/10 ,  C07C217/76 ,  C07C233/25 ,  C07C255/25 ,  C07C271/28 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14 ,  C07D241/24

摘要： Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: wherein R1 is H, C1-6 alkyl, halo C1-6 alkyl, or the like; R2 is halogeno, C1-6 alkyl, or the like; G is C2-10 alkyl or the like; Z is oxygen or sulfur; X's are each independently H, halogeno, or the like; Y's are each independently H, halogeno, cyano, or the like; and m and n are each an integer of 1 to 3.

摘要翻译： 由通式（I）表示的取代吡嗪羧酰苯胺衍生物或其盐; 它们的中间体; 用于农业和园艺用途的农药（如杀虫剂和杀螨剂），含有化合物作为活性成分; 及其用途：其中R 1为H，C 1-6烷基，卤代C 1-6烷基等; R2是卤代，C1-6烷基等; G为C 2-10烷基等; Z是氧或硫; X各自独立地为H，卤素等; Y各自独立地为H，卤代，氰基等; m和n分别为1〜3的整数。

公开(公告)号：US08269045B2

公开(公告)日：2012-09-18

申请号：US12846235

申请日：2010-07-29

申请人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

IPC分类号： C07C211/45 ,  C07C211/52 ,  C07D241/24 ,  A01N43/60

CPC分类号： A01N43/60 ,  C07C211/52 ,  C07C217/08 ,  C07C217/10 ,  C07C217/76 ,  C07C233/25 ,  C07C255/25 ,  C07C271/28 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14 ,  C07D241/24

摘要： Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: wherein R1 is H, C1-6 alkyl, halo C1-6 alkyl, or the like; R2 is halogeno, C1-6 alkyl, or the like; G is C2-10 alkyl or the like; Z is oxygen or sulfur; X's are each independently H, halogeno, or the like; Y's are each independently H, halogeno, cyano, or the like; and m and n are each an integer of 1 to 3.

摘要翻译： 由通式（I）表示的取代吡嗪羧酰苯胺衍生物或其盐; 它们的中间体; 用于农业和园艺用途的农药（如杀虫剂和杀螨剂），含有化合物作为活性成分; 及其用途：其中R 1为H，C 1-6烷基，卤代C 1-6烷基等; R2是卤代，C1-6烷基等; G为C 2-10烷基等; Z是氧或硫; X各自独立地为H，卤素等; Y各自独立地为H，卤代，氰基等; m和n分别为1〜3的整数。

公开(公告)号：US07910735B2

公开(公告)日：2011-03-22

申请号：US11597185

申请日：2005-05-26

申请人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

IPC分类号： C07D241/02

CPC分类号： A01N43/60 ,  C07C211/52 ,  C07C217/08 ,  C07C217/10 ,  C07C217/76 ,  C07C233/25 ,  C07C255/25 ,  C07C271/28 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14 ,  C07D241/24

摘要： Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: wherein R1 is H, C1-6 alkyl, halo C1-6 alkyl, or the like; R2 is halogeno, C1-6 alkyl, or the like; G is C2-10 alkyl or the like; Z is oxygen or sulfur; X's are each independently H, halogeno, or the like; Y's are each independently H, halogeno, cyano, or the like; and m and n are each an integer of 1 to 3.

摘要翻译： 由通式（I）表示的取代吡嗪羧酰苯胺衍生物或其盐; 它们的中间体; 用于农业和园艺用途的农药（如杀虫剂和杀螨剂），含有化合物作为活性成分; 及其用途：其中R 1为H，C 1-6烷基，卤代C 1-6烷基等; R2是卤代，C1-6烷基等; G为C 2-10烷基等; Z是氧或硫; X各自独立地为H，卤素等; Y各自独立地为H，卤代，氰基等; m和n分别为1〜3的整数。

公开(公告)号：US20090105325A1

公开(公告)日：2009-04-23

申请号：US11990282

申请日：2006-08-11

申请人： Takashi Furuya ,  Hideo Kanno ,  Kozo Machiya ,  Akiyuki Suwa ,  Noriaki Yasokawa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Hideo Kanno ,  Kozo Machiya ,  Akiyuki Suwa ,  Noriaki Yasokawa ,  Shinsuke Fujioka

IPC分类号： A01N43/56 ,  C07D231/14 ,  C07C215/68

CPC分类号： C07D231/14 ,  A01N43/56 ,  A01N43/78 ,  C07C211/52 ,  C07C217/76 ,  C07D403/12 ,  C07D409/12 ,  C07D417/12

摘要： The substituted pyrazolecarboxanilide derivatives represented by of the formula (I) wherein R1 is H, alkyl, alkylcarbonyl, alkenylcarbonyl, cycloalkyl, phenylalkyl, phenylcarbonyl and the like; R2 is H, halogen, alkyl, CN, OH, alkoxy, phenoxy, phenylthio, phenylsulfonyl and the like; G is alkyl, alkenyl, alkynyl, cycloalkyl, C3-C10 cycloalkenyl and the like; Z is O or S; X is H, halogen, CN, NO2, alkyl and the like; Y1 is H, alkyl, alkenyl, phenyl, alkoxyalkyl and the like; Y2 is H, halogen, CN, NO2, OH, mercapto, amino, carboxyl, C1-C6 alkyl, phenyl, phenoxy, heterocycle and the like, m is 1 or 2; and n is 1-3, and salts thereof exhibit a superior effect as agrohorticultural insecticides or acaricides.

摘要翻译： 由式（I）表示的取代的吡唑并苯甲酰胺衍生物，其中R1是H，烷基，烷基羰基，烯基羰基，环烷基，苯基烷基，苯基羰基等; R2是H，卤素，烷基，CN，OH，烷氧基，苯氧基，苯硫基，苯基磺酰基等; G是烷基，烯基，炔基，环烷基，C 3 -C 10环烯基等; Z是O或S; X是H，卤素，CN，NO 2，烷基等; Y1是H，烷基，烯基，苯基，烷氧基烷基等; Y2是H，卤素，CN，NO2，OH，巯基，氨基，羧基，C1-C6烷基，苯基，苯氧基，杂环等，m是1或2; n为1-3，其盐作为农业杀虫剂或杀螨剂具有优异的效果。

公开(公告)号：US08404861B2

公开(公告)日：2013-03-26

申请号：US11990282

申请日：2006-08-11

申请人： Takashi Furuya ,  Hideo Kanno ,  Kozo Machiya ,  Akiyuki Suwa ,  Noriaki Yasokawa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Hideo Kanno ,  Kozo Machiya ,  Akiyuki Suwa ,  Noriaki Yasokawa ,  Shinsuke Fujioka

IPC分类号： C07D231/14

CPC分类号： C07D231/14 ,  A01N43/56 ,  A01N43/78 ,  C07C211/52 ,  C07C217/76 ,  C07D403/12 ,  C07D409/12 ,  C07D417/12

摘要： The substituted pyrazolecarboxanilide derivatives represented by of the formula (I) wherein R1 is H, alkyl, alkylcarbonyl, alkenylcarbonyl, cycloalkyl, phenylalkyl, phenylcarbonyl and the like; R2 is H, halogen, alkyl, CN, OH, alkoxy, phenoxy, phenylthio, phenylsulfonyl and the like; G is alkyl, alkenyl, alkynyl, cycloalkyl, C3-C10 cycloalkenyl and the like; Z is O or S; X is H, halogen, CN, NO2, alkyl and the like; Y1 is H, alkyl, alkenyl, phenyl, alkoxyalkyl and the like; Y2 is H, halogen, CN, NO2, OH, mercapto, amino, carboxyl, C1-C6 alkyl, phenyl, phenoxy, heterocycle and the like, m is 1 or 2; and n is 1-3, and salts thereof exhibit a superior effect as agrohorticultural insecticides or acaricides.

摘要翻译： 由式（I）表示的取代的吡唑并苯甲酰胺衍生物，其中R1是H，烷基，烷基羰基，烯基羰基，环烷基，苯基烷基，苯基羰基等; R2是H，卤素，烷基，CN，OH，烷氧基，苯氧基，苯硫基，苯基磺酰基等; G是烷基，烯基，炔基，环烷基，C 3 -C 10环烯基等; Z是O或S; X是H，卤素，CN，NO 2，烷基等; Y1是H，烷基，烯基，苯基，烷氧基烷基等; Y2是H，卤素，CN，NO2，OH，巯基，氨基，羧基，C1-C6烷基，苯基，苯氧基，杂环等，m是1或2; n为1-3，其盐作为农业杀虫剂或杀螨剂具有优异的效果。

公开(公告)号：US20080064708A1

公开(公告)日：2008-03-13

申请号：US11597185

申请日：2005-05-26

申请人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

IPC分类号： A61K31/4965 ,  C07D241/02

CPC分类号： A01N43/60 ,  C07C211/52 ,  C07C217/08 ,  C07C217/10 ,  C07C217/76 ,  C07C233/25 ,  C07C255/25 ,  C07C271/28 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14 ,  C07D241/24

摘要： Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: wherein R1 is H, C1-6 alkyl, halo C1-6 alkyl, or the like; R2 is halogeno, C1-6 alkyl, or the like; G is C2-10 alkyl or the like; Z is oxygen or sulfur; X's are each independently H, halogeno, or the like; Y's are each independently H, halogeno, cyano, or the like; and m and n are each an integer of 1 to 3.

摘要翻译： 由通式（I）表示的取代吡嗪羧酰苯胺衍生物或其盐; 它们的中间体; 用于农业和园艺用途的农药（如杀虫剂和杀螨剂），含有化合物作为活性成分; 及其用途：其中R 1是H，C 1-6烷基，卤代C 1-6烷基等; R 2是卤代，C 1-6烷基等; G是C 2〜C 10烷基等; Z是氧或硫; X各自独立地为H，卤素等; Y各自独立地为H，卤代，氰基等; m和n分别为1〜3的整数。

公开(公告)号：US07994339B2

公开(公告)日：2011-08-09

申请号：US12086433

申请日：2006-12-14

申请人： Hiroto Harayama ,  Masanori Tohnishi ,  Shinsuke Fujioka ,  Akiyuki Suwa

发明人： Hiroto Harayama ,  Masanori Tohnishi ,  Shinsuke Fujioka ,  Akiyuki Suwa

IPC分类号： C07D257/04

CPC分类号： A01N43/713 ,  C07D257/04

摘要： Disclosed is a phthalamide derivative represented by the general formula (I) or a salt thereof, which shows an excellent controlling effect for use as an agricultural or horticultural insecticide alone or in combination with other agricultural or horticultural insecticide, acaricide, nematicide, fungicide, herbicide, plant growth regulator, biopesticide or the like.

摘要翻译： 公开了由通式（I）表示的邻苯二甲酰胺衍生物或其盐，其单独或与其他农业或园艺杀虫剂，杀螨剂，杀线虫剂，杀真菌剂，除草剂组合使用，作为农业或园艺杀虫剂具有优异的防治效果 ，植物生长调节剂，生物农药等。

公开(公告)号：US20090111861A1

公开(公告)日：2009-04-30

申请号：US12086433

申请日：2006-12-14

申请人： Hiroto Harayama ,  Masanori Tohnishi ,  Shinsuke Fujioka ,  Akiyuki Suwa

发明人： Hiroto Harayama ,  Masanori Tohnishi ,  Shinsuke Fujioka ,  Akiyuki Suwa

IPC分类号： A01N43/713 ,  C07D257/04 ,  A01P7/04

CPC分类号： A01N43/713 ,  C07D257/04

摘要： Disclosed is a phthalamide derivative represented by the general formula (I) or a salt thereof, which shows an excellent controlling effect for use as an agricultural or horticultural insecticide alone or in combination with other agricultural or horticultural insecticide, acaricide, nematicide, fungicide, herbicide, plant growth regulator, biopesticide or the like.

摘要翻译： 公开了由通式（I）表示的邻苯二甲酰胺衍生物或其盐，其单独或与其他农业或园艺杀虫剂，杀螨剂，杀线虫剂，杀真菌剂，除草剂组合使用，作为农业或园艺杀虫剂具有优异的防治效果 ，植物生长调节剂，生物农药等。

公开(公告)号：US07256192B2

公开(公告)日：2007-08-14

申请号：US10168334

申请日：2000-12-22

申请人： Masanori Tohnishi ,  Eiji Kohno ,  Hayami Nakao ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka

发明人： Masanori Tohnishi ,  Eiji Kohno ,  Hayami Nakao ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka

IPC分类号： A01N43/58 ,  A61K31/50

CPC分类号： C07D295/205 ,  A01N37/30 ,  A01N41/06 ,  A01N43/16 ,  A01N43/28 ,  A01N43/40 ,  A01N47/12 ,  A01N47/28 ,  A01N57/14 ,  C07C233/66 ,  C07C233/69 ,  C07C233/75 ,  C07C233/78 ,  C07C239/16 ,  C07C271/12 ,  C07C271/20 ,  C07C271/28 ,  C07C275/14 ,  C07C307/06 ,  C07C311/05 ,  C07C311/18 ,  C07C323/12 ,  C07C323/43 ,  C07C335/08 ,  C07C2601/02 ,  C07F9/2458

摘要： The present invention relates to an aromatic diamide derivative represented by the general formula (I): [A1 is optionally substituted (C1-C8)alkylene group, (C3-C8)alkenylene group or the like, B is —O— or —N(R4)— (wherein R4 is H, (C1-C6)alkyl, halo(C1-C6)alkyl or the like), R1 is H, (C1-C6)alkyl, optionally substituted phenyl, optionally substituted heterocyclic group, or the like, R2 and R3 are each H, (C3-C6)cycloalkyl or —A2—R8 (A2 is —C(═O)—, —C(═S)— or —C(═NR9)—, R8 and R9 are each H, (C1-C6)alkyl or the like), Q1 to Q5 are each carbon or nitrogen, X and Y are each halogen, cyano, nitro, (C3-C6)cycloalkyl, optionally substituted phenyl, optionally substituted heterocyclic group, or the like, n is 0 to 4, m is 1 to 5, and Z1 and Z2 are each O or S] or a salt thereof, an agricultural and horticultural chemical, and a usage of the chemical. The agricultural and horticultural chemicals of the present invention exhibit remarkable controlling effects against various insect pests such as agricultural, forest and horticultural insect pests, and stored grain insect pests, etc., which injure paddy rice, fruit trees, vegetables, other crop plants, flowers and ornamental plants, and the like.

公开(公告)号：US06559341B2

公开(公告)日：2003-05-06

申请号：US10035132

申请日：2002-01-04

申请人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

发明人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

IPC分类号： C07C2146

CPC分类号： C07D213/40 ,  C07C211/52 ,  C07C233/65 ,  C07C233/66 ,  C07C233/75 ,  C07C233/81 ,  C07C233/91 ,  C07C233/92 ,  C07C235/64 ,  C07C235/84 ,  C07C237/22 ,  C07C251/48 ,  C07C255/57 ,  C07C261/04 ,  C07C271/20 ,  C07C271/64 ,  C07D213/70 ,  C07D263/32 ,  C07D277/30 ,  C07D295/192 ,  C07D307/52 ,  C07D333/20 ,  C07F9/18 ,  C07F9/4021

摘要： The present invention provides a phthalic acid diamide derivative represented by the general formula (I) (wherein R1, R2 and R3 are each H, C3-C6 cycloalkyl group, group of the formula —A1—Ql or the like; X may be the same or different and are each halogen atom, nitro group, phenyl group, group of the formula —A2—R7 or the like; n is 1 to 4; Y may be same or different and are each halogen atom, cyano group, phenyl group, group of the formula —A2—R7 or the like; m is 1 to 5; Z1 and Z2 are each O or S), fluorine-containing aniline compound represented by the general formula (ST-I) as starting material for said phthalic acid diamide derivative (wherein Ra is halogen atom, C1-C6 alkyl group or the like and Rb, Rc and Rd is H or C2-C6 perfluoroalkyl group), and an agricultural and horticultural insecticide containing said phthaldiamide derivative, as well as to provide a method for use of said insecticide. The agricultural and horticultural insecticides of the present invention show excellent activities for controlling injurious insects.

摘要翻译： 本发明提供由通式（I）表示的邻苯二甲酸二酰胺衍生物（其中R1，R2和R3分别为H，C3-C6环烷基，式-A1-Q1等基团等; X可以是 相同或不同，各自为卤原子，硝基，苯基，式-A2-R7等基团; n为1至4; Y可以相同或不同，各自为卤素原子，氰基，苯基 式-A2-R7等基团; m为1〜5; Z 1和Z 2各自为O或S），由通式（ST-I）表示的含氟苯胺化合物作为所述邻苯二甲酸 酸式二酰胺衍生物（其中Ra为卤素原子，C1-C6烷基等，Rb，Rc和Rd为H或C2-C6全氟烷基），以及含有所述邻苯二甲酰胺衍生物的农业和园艺杀虫剂， 一种使用所述杀虫剂的方法。 本发明的农业和园艺杀虫剂显示出控制有害昆虫的优良活性。