公开(公告)号：US20090105325A1

公开(公告)日：2009-04-23

申请号：US11990282

申请日：2006-08-11

申请人： Takashi Furuya ,  Hideo Kanno ,  Kozo Machiya ,  Akiyuki Suwa ,  Noriaki Yasokawa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Hideo Kanno ,  Kozo Machiya ,  Akiyuki Suwa ,  Noriaki Yasokawa ,  Shinsuke Fujioka

IPC分类号： A01N43/56 ,  C07D231/14 ,  C07C215/68

CPC分类号： C07D231/14 ,  A01N43/56 ,  A01N43/78 ,  C07C211/52 ,  C07C217/76 ,  C07D403/12 ,  C07D409/12 ,  C07D417/12

摘要： The substituted pyrazolecarboxanilide derivatives represented by of the formula (I) wherein R1 is H, alkyl, alkylcarbonyl, alkenylcarbonyl, cycloalkyl, phenylalkyl, phenylcarbonyl and the like; R2 is H, halogen, alkyl, CN, OH, alkoxy, phenoxy, phenylthio, phenylsulfonyl and the like; G is alkyl, alkenyl, alkynyl, cycloalkyl, C3-C10 cycloalkenyl and the like; Z is O or S; X is H, halogen, CN, NO2, alkyl and the like; Y1 is H, alkyl, alkenyl, phenyl, alkoxyalkyl and the like; Y2 is H, halogen, CN, NO2, OH, mercapto, amino, carboxyl, C1-C6 alkyl, phenyl, phenoxy, heterocycle and the like, m is 1 or 2; and n is 1-3, and salts thereof exhibit a superior effect as agrohorticultural insecticides or acaricides.

摘要翻译： 由式（I）表示的取代的吡唑并苯甲酰胺衍生物，其中R1是H，烷基，烷基羰基，烯基羰基，环烷基，苯基烷基，苯基羰基等; R2是H，卤素，烷基，CN，OH，烷氧基，苯氧基，苯硫基，苯基磺酰基等; G是烷基，烯基，炔基，环烷基，C 3 -C 10环烯基等; Z是O或S; X是H，卤素，CN，NO 2，烷基等; Y1是H，烷基，烯基，苯基，烷氧基烷基等; Y2是H，卤素，CN，NO2，OH，巯基，氨基，羧基，C1-C6烷基，苯基，苯氧基，杂环等，m是1或2; n为1-3，其盐作为农业杀虫剂或杀螨剂具有优异的效果。

公开(公告)号：US08404861B2

公开(公告)日：2013-03-26

申请号：US11990282

申请日：2006-08-11

申请人： Takashi Furuya ,  Hideo Kanno ,  Kozo Machiya ,  Akiyuki Suwa ,  Noriaki Yasokawa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Hideo Kanno ,  Kozo Machiya ,  Akiyuki Suwa ,  Noriaki Yasokawa ,  Shinsuke Fujioka

IPC分类号： C07D231/14

CPC分类号： C07D231/14 ,  A01N43/56 ,  A01N43/78 ,  C07C211/52 ,  C07C217/76 ,  C07D403/12 ,  C07D409/12 ,  C07D417/12

摘要： The substituted pyrazolecarboxanilide derivatives represented by of the formula (I) wherein R1 is H, alkyl, alkylcarbonyl, alkenylcarbonyl, cycloalkyl, phenylalkyl, phenylcarbonyl and the like; R2 is H, halogen, alkyl, CN, OH, alkoxy, phenoxy, phenylthio, phenylsulfonyl and the like; G is alkyl, alkenyl, alkynyl, cycloalkyl, C3-C10 cycloalkenyl and the like; Z is O or S; X is H, halogen, CN, NO2, alkyl and the like; Y1 is H, alkyl, alkenyl, phenyl, alkoxyalkyl and the like; Y2 is H, halogen, CN, NO2, OH, mercapto, amino, carboxyl, C1-C6 alkyl, phenyl, phenoxy, heterocycle and the like, m is 1 or 2; and n is 1-3, and salts thereof exhibit a superior effect as agrohorticultural insecticides or acaricides.

摘要翻译： 由式（I）表示的取代的吡唑并苯甲酰胺衍生物，其中R1是H，烷基，烷基羰基，烯基羰基，环烷基，苯基烷基，苯基羰基等; R2是H，卤素，烷基，CN，OH，烷氧基，苯氧基，苯硫基，苯基磺酰基等; G是烷基，烯基，炔基，环烷基，C 3 -C 10环烯基等; Z是O或S; X是H，卤素，CN，NO 2，烷基等; Y1是H，烷基，烯基，苯基，烷氧基烷基等; Y2是H，卤素，CN，NO2，OH，巯基，氨基，羧基，C1-C6烷基，苯基，苯氧基，杂环等，m是1或2; n为1-3，其盐作为农业杀虫剂或杀螨剂具有优异的效果。

公开(公告)号：US20100311974A1

公开(公告)日：2010-12-09

申请号：US12846235

申请日：2010-07-29

申请人： Takashi FURUYA ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

发明人： Takashi FURUYA ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

IPC分类号： C07D241/12 ,  C07C211/52

CPC分类号： A01N43/60 ,  C07C211/52 ,  C07C217/08 ,  C07C217/10 ,  C07C217/76 ,  C07C233/25 ,  C07C255/25 ,  C07C271/28 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14 ,  C07D241/24

摘要： Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: wherein R1 is H, C1-6 alkyl, halo C1-6 alkyl, or the like; R2 is halogeno, C1-6 alkyl, or the like; G is C2-10 alkyl or the like; Z is oxygen or sulfur; X's are each independently H, halogeno, or the like; Y's are each independently H, halogeno, cyano, or the like; and m and n are each an integer of 1 to 3.

摘要翻译： 由通式（I）表示的取代吡嗪羧酰苯胺衍生物或其盐; 它们的中间体; 用于农业和园艺用途的农药（如杀虫剂和杀螨剂），含有化合物作为活性成分; 及其用途：其中R 1为H，C 1-6烷基，卤代C 1-6烷基等; R2是卤代，C1-6烷基等; G为C 2-10烷基等; Z是氧或硫; X各自独立地为H，卤素等; Y各自独立地为H，卤代，氰基等; m和n分别为1〜3的整数。

公开(公告)号：US08269045B2

公开(公告)日：2012-09-18

申请号：US12846235

申请日：2010-07-29

申请人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

IPC分类号： C07C211/45 ,  C07C211/52 ,  C07D241/24 ,  A01N43/60

CPC分类号： A01N43/60 ,  C07C211/52 ,  C07C217/08 ,  C07C217/10 ,  C07C217/76 ,  C07C233/25 ,  C07C255/25 ,  C07C271/28 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14 ,  C07D241/24

摘要： Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: wherein R1 is H, C1-6 alkyl, halo C1-6 alkyl, or the like; R2 is halogeno, C1-6 alkyl, or the like; G is C2-10 alkyl or the like; Z is oxygen or sulfur; X's are each independently H, halogeno, or the like; Y's are each independently H, halogeno, cyano, or the like; and m and n are each an integer of 1 to 3.

摘要翻译： 由通式（I）表示的取代吡嗪羧酰苯胺衍生物或其盐; 它们的中间体; 用于农业和园艺用途的农药（如杀虫剂和杀螨剂），含有化合物作为活性成分; 及其用途：其中R 1为H，C 1-6烷基，卤代C 1-6烷基等; R2是卤代，C1-6烷基等; G为C 2-10烷基等; Z是氧或硫; X各自独立地为H，卤素等; Y各自独立地为H，卤代，氰基等; m和n分别为1〜3的整数。

公开(公告)号：US07910735B2

公开(公告)日：2011-03-22

申请号：US11597185

申请日：2005-05-26

申请人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

IPC分类号： C07D241/02

CPC分类号： A01N43/60 ,  C07C211/52 ,  C07C217/08 ,  C07C217/10 ,  C07C217/76 ,  C07C233/25 ,  C07C255/25 ,  C07C271/28 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14 ,  C07D241/24

摘要： Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: wherein R1 is H, C1-6 alkyl, halo C1-6 alkyl, or the like; R2 is halogeno, C1-6 alkyl, or the like; G is C2-10 alkyl or the like; Z is oxygen or sulfur; X's are each independently H, halogeno, or the like; Y's are each independently H, halogeno, cyano, or the like; and m and n are each an integer of 1 to 3.

摘要翻译： 由通式（I）表示的取代吡嗪羧酰苯胺衍生物或其盐; 它们的中间体; 用于农业和园艺用途的农药（如杀虫剂和杀螨剂），含有化合物作为活性成分; 及其用途：其中R 1为H，C 1-6烷基，卤代C 1-6烷基等; R2是卤代，C1-6烷基等; G为C 2-10烷基等; Z是氧或硫; X各自独立地为H，卤素等; Y各自独立地为H，卤代，氰基等; m和n分别为1〜3的整数。

公开(公告)号：US20080064708A1

公开(公告)日：2008-03-13

申请号：US11597185

申请日：2005-05-26

申请人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

发明人： Takashi Furuya ,  Kozo Machiya ,  Akiyuki Suwa ,  Shinsuke Fujioka

IPC分类号： A61K31/4965 ,  C07D241/02

CPC分类号： A01N43/60 ,  C07C211/52 ,  C07C217/08 ,  C07C217/10 ,  C07C217/76 ,  C07C233/25 ,  C07C255/25 ,  C07C271/28 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14 ,  C07D241/24

摘要： Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: wherein R1 is H, C1-6 alkyl, halo C1-6 alkyl, or the like; R2 is halogeno, C1-6 alkyl, or the like; G is C2-10 alkyl or the like; Z is oxygen or sulfur; X's are each independently H, halogeno, or the like; Y's are each independently H, halogeno, cyano, or the like; and m and n are each an integer of 1 to 3.

摘要翻译： 由通式（I）表示的取代吡嗪羧酰苯胺衍生物或其盐; 它们的中间体; 用于农业和园艺用途的农药（如杀虫剂和杀螨剂），含有化合物作为活性成分; 及其用途：其中R 1是H，C 1-6烷基，卤代C 1-6烷基等; R 2是卤代，C 1-6烷基等; G是C 2〜C 10烷基等; Z是氧或硫; X各自独立地为H，卤素等; Y各自独立地为H，卤代，氰基等; m和n分别为1〜3的整数。

公开(公告)号：US06559341B2

公开(公告)日：2003-05-06

申请号：US10035132

申请日：2002-01-04

申请人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

发明人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

IPC分类号： C07C2146

CPC分类号： C07D213/40 ,  C07C211/52 ,  C07C233/65 ,  C07C233/66 ,  C07C233/75 ,  C07C233/81 ,  C07C233/91 ,  C07C233/92 ,  C07C235/64 ,  C07C235/84 ,  C07C237/22 ,  C07C251/48 ,  C07C255/57 ,  C07C261/04 ,  C07C271/20 ,  C07C271/64 ,  C07D213/70 ,  C07D263/32 ,  C07D277/30 ,  C07D295/192 ,  C07D307/52 ,  C07D333/20 ,  C07F9/18 ,  C07F9/4021

摘要： The present invention provides a phthalic acid diamide derivative represented by the general formula (I) (wherein R1, R2 and R3 are each H, C3-C6 cycloalkyl group, group of the formula —A1—Ql or the like; X may be the same or different and are each halogen atom, nitro group, phenyl group, group of the formula —A2—R7 or the like; n is 1 to 4; Y may be same or different and are each halogen atom, cyano group, phenyl group, group of the formula —A2—R7 or the like; m is 1 to 5; Z1 and Z2 are each O or S), fluorine-containing aniline compound represented by the general formula (ST-I) as starting material for said phthalic acid diamide derivative (wherein Ra is halogen atom, C1-C6 alkyl group or the like and Rb, Rc and Rd is H or C2-C6 perfluoroalkyl group), and an agricultural and horticultural insecticide containing said phthaldiamide derivative, as well as to provide a method for use of said insecticide. The agricultural and horticultural insecticides of the present invention show excellent activities for controlling injurious insects.

摘要翻译： 本发明提供由通式（I）表示的邻苯二甲酸二酰胺衍生物（其中R1，R2和R3分别为H，C3-C6环烷基，式-A1-Q1等基团等; X可以是 相同或不同，各自为卤原子，硝基，苯基，式-A2-R7等基团; n为1至4; Y可以相同或不同，各自为卤素原子，氰基，苯基 式-A2-R7等基团; m为1〜5; Z 1和Z 2各自为O或S），由通式（ST-I）表示的含氟苯胺化合物作为所述邻苯二甲酸 酸式二酰胺衍生物（其中Ra为卤素原子，C1-C6烷基等，Rb，Rc和Rd为H或C2-C6全氟烷基），以及含有所述邻苯二甲酰胺衍生物的农业和园艺杀虫剂， 一种使用所述杀虫剂的方法。 本发明的农业和园艺杀虫剂显示出控制有害昆虫的优良活性。

公开(公告)号：US06864289B1

公开(公告)日：2005-03-08

申请号：US10088543

申请日：2000-09-22

申请人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

发明人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

IPC分类号： A01N37/22 ,  A01N37/30 ,  A01N37/46 ,  A01N41/10 ,  A01N43/40 ,  C07C233/83 ,  C07C233/85 ,  C07C237/22 ,  C07C251/38 ,  C07C251/40 ,  C07C317/28 ,  C07C317/50 ,  C07C323/12 ,  C07C323/41 ,  C07D213/75 ,  C07D213/81 ,  C07D213/82 ,  C07D239/28 ,  A01N37/50

CPC分类号： C07D213/75 ,  A01N37/22 ,  A01N37/30 ,  A01N37/46 ,  A01N41/10 ,  A01N43/40 ,  C07C233/83 ,  C07C233/85 ,  C07C237/22 ,  C07C251/38 ,  C07C251/40 ,  C07C317/28 ,  C07C317/50 ,  C07C323/12 ,  C07C323/41 ,  C07D213/81 ,  C07D213/82 ,  C07D239/28

摘要： Aromatic diamide derivative represented by the general formula (I) or a salt thereof and agricultural/herticultural composition containing the same as the active ingredient, wherein A1 represents alkylene, alkenylene or alkynylene; B represents, CO— or —C(═N—OR4)— (wherein R4 represents H, etc.); R1 to R3 represent each H, etc.; Q1 to Q5 represent each N or carbon; Y represents halogeno, etc.; m is from 0 to 5; and Z1 and Z2 represent each O or S.

摘要翻译： 由通式（I）表示的芳族二酰胺衍生物或其盐和含有与活性成分相同的农业/农业组合物，其中A 1表示亚烷基，亚烯基或亚炔基; B表示CO-或-C（= N-OR 4） - （其中R 4表示H等）; R 1至R 3代表每个H等; Q 1至Q 5代表每个N或碳; Y代表卤素等; m为0〜5; Z 1和Z 2代表O或S.

公开(公告)号：US06603044B1

公开(公告)日：2003-08-05

申请号：US09449420

申请日：1999-11-29

申请人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

发明人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

IPC分类号： C07C23364

CPC分类号： C07C317/28 ,  A01N37/30 ,  A01N43/10 ,  A01N43/18 ,  A01N43/40 ,  A01N43/54 ,  A01N43/78 ,  A01N43/82 ,  A01N47/02 ,  A01N47/12 ,  C07C317/40 ,  C07C323/42 ,  C07D213/70 ,  C07D239/26 ,  C07D277/36 ,  C07D277/76 ,  C07D285/125 ,  C07D333/36 ,  C07D333/48 ,  C07D335/02

摘要： The present invention provides a phthalamide derivative of the formula (I): wherein A1 is (substituted) C1-C8 alkylene, (substituted) C3-C8 alkenylene, (substituted) C3-C8 alkynylene, etc., R1 is H, (halo) C3-C6 cycloalkyl, (substituted) phenyl, (substituted) heterocycle, —A2—R4, etc., R2 and R3 are H, C3-C6 cycloalkyl, —A2—R4, etc., A2 is —C(═O)—, —C(═S)— or —C(═NR5)—, R4 is H, alkyl, (substituted) phenyl, (substituted) heterocycle, etc., X and Y are halogen, cyano, nitro, (halo) C1-C6 alkyl, (halo) C1-C6 alkoxy, etc., l is 0-4, m is 0-5, n is 0-2; and an agrohorticultural insecticide containing said compound as active ingredient and exhibiting an excellent insecticidal effect.

摘要翻译： 本发明提供式（I）的邻苯二甲酰胺衍生物：其中A 1是（取代的）C 1 -C 8亚烷基，（取代的）C 3 -C 8亚烯基，（取代的）C 3 -C 8亚炔基等，R 1是H ）C3-C6环烷基，（取代）苯基，（取代）杂环，-A2-R4等，R2和R3是H，C3-C6环烷基，-A2-R4等，A2是-C（= O ） - ， - （= S） - 或-C（= NR5） - ，R4是H，烷基，（取代的）苯基，（取代的）杂环等，X和Y是卤素，氰基，硝基，（卤素 ）C 1 -C 6烷基，（卤素）C 1 -C 6烷氧基等，l为0-4，m为0-5，n为0-2; 和含有所述化合物作为活性成分并具有优异杀虫效果的农业杀虫剂。

公开(公告)号：US06362369B1

公开(公告)日：2002-03-26

申请号：US09250261

申请日：1999-02-16

申请人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

发明人： Masanori Tohnishi ,  Hayami Nakao ,  Eiji Kohno ,  Tateki Nishida ,  Takashi Furuya ,  Toshiaki Shimizu ,  Akira Seo ,  Kazuyuki Sakata ,  Shinsuke Fujioka ,  Hideo Kanno

IPC分类号： A01N3718

摘要： The present invention provides a phthalic acid diamide derivative represented by the general formula (I) (wherein R1, R2 and R3 are each H, C3-C6 cycloalkyl group, group of the formula —A1—Ql or the like; X may be the same or different and are each halogen atom, nitro group, phenyl group, group of the formula —A2—R7 or the like; n is 1 to 4; Y may be same or different and are each halogen atom, cyano group, phenyl group, group of the formula —A2—R7 or the like; m is 1 to 5; Z1 and Z2 are each 0 or S), fluorine-containing aniline compound represented by the general formula (ST-I) as starting material for said phthalic acid diamide derivative (wherein Ra is halogen atom, C1-C6 alkyl group or the like and Rb, Rc and Rd is H or C2-C6 perfluoroalkyl group), and an agricultural and horticultural insecticide containing said phthaldiamide derivative, as well as to provide a method for use of said insecticide. The agricultural and horticultural insecticides of the present invention show excellent activities for controlling injurious insects.