Isoxazolecarboxylic acid derivatives
    1.
    发明授权
    Isoxazolecarboxylic acid derivatives 失效
    异恶唑羧酸衍生物

    公开(公告)号:US5374605A

    公开(公告)日:1994-12-20

    申请号:US2307

    申请日:1993-01-08

    摘要: The invention relates to isoxazolecarboxylic acid derivatives of the general formula (I) ##STR1## in which A represents alkanediyl,Q represents oxygen, sulphur, imino (NH) or alkylimino (N-alkyl),R.sup.1 represents an in each case optionally substituted radical from the series comprising alkyl, cycloalkyl or phenyl,R.sup.2 represents hydrogen, halogen or optionally substituted alkyl, andR.sup.3 represents in each case optionally substituted cyclohexyl or phenyl,with the exception of the compounds: N-benzyl-5-cyclopropyl-isoxazole-3-carboxamide N-(2-phenyl-ethyl)-5-methyl-isoxazole-3-carboxamide and N-benzyl-5-methyl-isoxazole-3-carboxamide, a process for their preparation, and their use as herbicides.

    摘要翻译: 本发明涉及通式(I)的化合物(I)的异恶唑羧酸衍生物,其中A代表烷二基,Q代表氧,硫,亚氨基(NH)或烷基亚氨基(N-烷基),R1代表每种情况 任选取代的烷基,环烷基或苯基系列的取代基,R 2表示氢,卤素或任选取代的烷基,R 3表示在任何情况下均为任选取代的环己基或苯基,但化合物除外:N-苄基-5-环丙基 - 异恶唑-3-甲酰胺N-(2-苯基 - 乙基)-5-甲基 - 异恶唑-3-甲酰胺和N-苄基-5-甲基 - 异恶唑-3-甲酰胺,其制备方法及其作为除草剂的用途 。

    Substituted triazolinone herbicides and plant growth regulators
    3.
    发明授权
    Substituted triazolinone herbicides and plant growth regulators 失效
    取代的三唑啉酮除草剂和植物生长调节剂

    公开(公告)号:US5523409A

    公开(公告)日:1996-06-04

    申请号:US125975

    申请日:1993-09-23

    摘要: Novel herbicides and plant growth regulants of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, alkoxyalkyl, alkoxy, cycloalkylalkyl or cycloalkyl, or represents in each case optionally substituted aralkyl or aryl,R.sup.2 represents a radical ##STR2## or represents a radical --S(O).sub.n --R.sup.7, R.sup.3 and R.sup.4 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylaminoalkyl, alkoxycarbonylalkyl or alkoxycarbonylalkenyl, or represent in each case optionally substituted cycloalkyl, cycloalkylalkyl, cycloalkenyl or cycloalkenylalkyl, or represent optionally substituted heterocyclylalkyl, or represent in each case optionally substituted aralkyl, aroyl or aryl, or represent alkoxy, alkenyloxy, alkinyloxy, aralkyloxy or aryloxy, or, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical,X represents oxygen or sulphur andY represents oxygen or sulphur,whereinR.sup.5 and R.sup.6 independently of one another each represent alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, alkoxyalkyl, alkoxy, cycloalkyl or cycloalkylalkyl, or represent in each case optionally substituted aryl, aralkyl or heteroaryl, or, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical,R.sup.7 represents alkyl, alkenyl, alkinyl, cycloalkyl or cycloalkylalkyl, or represents in each case optionally substituted aralkyl or aryl andn represents the number 0, 1 or 2,but wherein R.sup.2 only represents a radical --S(O).sub.n --R.sup.7 if R.sup.3 and R.sup.4 do not simultaneously represent methyl.Intermediates therefor where NR.sup.3 R.sup.4 is replaced by Cl are also new.

    摘要翻译: 式(I)的新型除草剂和植物生长调节剂,其中R 1表示氢,烷基,烯基,炔基,卤代烷基,卤代烯基,卤代烷基,烷氧基烷基,烷氧基,环烷基烷基或环烷基,或在每种情况下表示任选取代的芳烷基或 芳基,R 2表示基团,或表示基团-S(O)n -R 7,R 3和R 4彼此独立地表示氢,烷基,烯基,炔基,卤代烷基,卤代烯基,卤代烷基,氰基烷基,羟基烷基,烷氧基烷基 或烷基氨基烷基,烷氧基羰基烷基或烷氧基羰基烯基,或在每种情况下表示任选取代的环烷基,环烷基烷基,环烯基或环烯基烷基,或代表任选取代的杂环基烷基,或在每种情况下表示任选取代的芳烷基,芳酰基或芳基,或代表烷氧基,烯氧基,烷氧基,芳烷氧基 或芳氧基,或者与它们所键合的氮原子一起代表任选的 取代的杂环基,X表示氧或硫,Y表示氧或硫,其中R5和R6彼此独立地表示烷基,烯基,炔基,卤代烷基,卤代烯基,卤代烷基,烷氧基烷基,烷氧基,环烷基或环烷基烷基,或各自表示 任选取代的芳基,芳烷基或杂芳基,或与它们所键合的氮原子一起表示任选取代的杂环基,R 7表示烷基,烯基,炔基,环烷基或环烷基烷基,或在每种情况下表示任选取代的芳烷基或 芳基,n表示数字0,1或2,但如果R3和R4不同时表示甲基,则其中R2仅表示基团-S(O)n-R7。 NR3R4被Cl取代的中间体也是新的。

    Herbicidal substituted sulphonylamidinohydrazones
    8.
    发明授权
    Herbicidal substituted sulphonylamidinohydrazones 失效
    除草取代磺酰脒腙

    公开(公告)号:US5213608A

    公开(公告)日:1993-05-25

    申请号:US916330

    申请日:1992-07-16

    IPC分类号: A01N47/44 C07D521/00

    CPC分类号: C07D521/00 A01N47/44

    摘要: Herbicidal substituted sulphonylamidinohydrazones of the formula ##STR1## in which R.sup.1 represents in each case optionally substituted aryl, aralkyl or heteroaryl,R.sup.2 represents hydrogen, or represents in each case optionally substituted alkyl, aryl or aralkyl,R.sup.3 represents hydrogen, or represents in each case optionally substituted alkyl, alkenyl, alkadienyl, alkinyl, (hetero)aryl, aralkyl, aralkenyl, alkoxy, alkoxycarbonyl or dialkylamino, or together with R.sup.2 represents optionally substituted alkanediyl,R.sup.4 represents hydrogen, halogen, hydroxyl, alkyl, halogenoalkyl, alkoxyalkyl, alkoxy, halogenoalkoxy, alkylthio, halogenoalkylthio, amino, alkylamino or dialkylamino,X represents nitrogen or a --CH group,Y represents nitrogen or a --CR.sup.5 group whereR.sup.5 represents hydrogen, halogen, cyano, alkyl, formyl, alkyl-carbonyl or alkoxy-carbonyl, andZ represents nitrogen or a --CR.sup.6 group whereR.sup.6 represents hydrogen, halogen, hydroxyl, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio, alkylamino or dialkylamino.

    摘要翻译: 式(I)的除草取代的磺酰基脒基腙,其中R 1在每种情况下表示任选取代的芳基,芳烷基或杂芳基,R 2表示氢,或在各种情况下表示任选取代的烷基,芳基或芳烷基,R 3表示氢或表示 在任何情况下,任选取代的烷基,烯基,链二烯基,炔基,(杂)芳基,芳烷基,芳烯基,烷氧基,烷氧基羰基或二烷基氨基,或与R 2表示任选取代的烷二基,R 4表示氢,卤素,羟基,烷基,卤代烷基, 烷氧基,卤代烷氧基,烷硫基,卤代烷硫基,氨基,烷基氨基或二烷基氨基,X表示氮或-CH基,Y表示氮或-CR5基,其中R5表示氢,卤素,氰基,烷基,甲酰基, - 羰基,Z表示氮或-CR 6基团,其中R 6表示氢,卤素,羟基,烷基,卤代烷基,烷氧基,卤代烷氧基,烷硫基, 烷基氨基或二烷基氨基。

    Pesticidal 3-aryl-pyrrolidine-2,4-diones
    10.
    发明授权
    Pesticidal 3-aryl-pyrrolidine-2,4-diones 失效
    杀虫剂3-芳基 - 吡咯烷-2,4-二酮

    公开(公告)号:US5186737A

    公开(公告)日:1993-02-16

    申请号:US678479

    申请日:1991-04-01

    摘要: Insecticidal, acaricidal, herbicidal and antimycotic 3-aryl-pyrrolidine-2,4-diones of the formula ##STR1## in which X represents alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents a number from 0-3,R represents hydrogen or represents the groups --CO--R.sup.1 or --CO--O--R.sup.2, in whichR.sup.1 represents alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, polyalkoxyalkyl or cycloalkyl which can be interrupted by hetero atoms, each of which radicals is optionally substituted by halogen, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl or substituted hetaryloxyalkyl, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl and substituted hetaryloxyalkyl, andR.sup.2 represents alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl or optionally substituted phenyl or cycloalkyl, each of which radicals is optionally substituted by halogen,A represents alkyl, alkenyl, alkinyl, alkoxyalkyl, polyalkoxyalkyl, alkylthioalkyl, or cycloalkyl which is optionally interrupted by a hetero atom, each of which radicals is optionally subsituted by halogen, or represents arylalkyl which is optionally substituted by halogen, alkyl, halogenoalkyl, alkoxy or nitro,B and C* independently of one another represent hydrogen, alkyl or alkoxyalkyl.

    摘要翻译: 式(I)的杀虫,杀螨,除草和抗真菌性3-芳基 - 吡咯烷-2,4-二酮其中X代表烷基,卤素或烷氧基,Y代表氢,烷基,卤素,烷氧基或卤代烷基,Z 表示烷基,卤素或烷氧基,n表示0-3的数,R表示氢或表示基团-CO-R1或-CO-O-R2,其中R1表示烷基,烯基,烷氧基烷基,烷硫基烷基,聚烷氧基烷基或环烷基 任何取代的苯基,取代的杂芳基,取代的苯氧基烷基或取代的噻唑烷基,或代表任意取代的苯基,任选取代的苯基烷基,取代的杂芳基, 取代的苯氧基烷基和取代的硫代氧基烷基,R 2表示烷基,链烯基,烷氧基烷基,聚烷氧基烷基或任选取代的苯基或环烷基,各w 任选被卤素取代的基团,A代表烷基,烯基,炔基,烷氧基烷基,聚烷氧基烷基,烷硫基烷基或环烷基,任选被杂原子中断,每个基团任选被卤素取代,或表示任选取代的芳基烷基 卤素,烷基,卤代烷基,烷氧基或硝基,B和C *彼此独立地表示氢,烷基或烷氧基烷基。