-
公开(公告)号:US20050065032A1
公开(公告)日:2005-03-24
申请号:US10497627
申请日:2002-11-25
申请人: William Whittingham , Kevin Lawson , Paul Worthington , Charles Russell , Roger Salmon , Leslie May , Mario Jorg , Johannes Pachlatko
发明人: William Whittingham , Kevin Lawson , Paul Worthington , Charles Russell , Roger Salmon , Leslie May , Mario Jorg , Johannes Pachlatko
IPC分类号: A01N25/02 , A01N25/08 , A01N43/40 , C07D213/65 , C07D213/68 , C07D213/70 , C07D213/79 , C07D213/80 , C07D213/81 , C07D213/82 , C07D213/84 , C07D213/85 , A01N25/00 , C07D213/62
CPC分类号: C07D213/70 , A01N43/40 , C07D213/65 , C07D213/68 , C07D213/80 , C07D213/82 , C07D213/85
摘要: Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C1-8 alkyl, C3-6 cycloalkyl, C2-8 alkenyl, C2-8 alkynyl, C1-8 alkoxy, C1-8 alkylthio, nitro, amino, mono- or di-(C1-6)alkylamino, mono- or di-(C2-6)alkenylamino, mono- or di-(C2-6)alkynylamino, formylamino, C1-4 alkyl(formyl)amino, C1-4 alkylcarbonylamino, C1-4 alkyl(C1-4 alkylcarbonyl)amino, cyano, formyl, C1-4 alkylcarbonyl, C1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C1-4)alkylaminocarbonyl, carboxy, C1-4 alkylcarbonyloxy, aryl(C1-4)alkylcarbonyloxy, C1-4 alkylsulphinyl, C1-4 alkylsulphonyl, C1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R1 is phenyl, cyano, C1-4 alkyl, C2-4 alkenyl or C2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or thre halogen atoms, with a cyano group, with a C1-4 alkylcarbonyl group, with a C1-4 alkoxycarbonyl group or with a hydroxy group, or R1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R2 is H, C1-4 alkyl, C1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C1-4 alkoxy; R3 and R4 are independently H, C1-3 alkyl, C2-3 alkenyl or C2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R3 and R4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C1-4 alkyl; and R5 is halo, C1-4 alkyl or C3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C1-6 alkoxy, C1-6 alkylthio, cyano, C1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C1-4)alkylaminocarbonyloxy, or tri(C1-4)alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
-
公开(公告)号:US20070135468A1
公开(公告)日:2007-06-14
申请号:US11623448
申请日:2007-01-16
申请人: William Whittingham , Kevin Lawson , Paul Worthington , Charles Russell , Roger Salmon , Leslie May , Mario Jorg , Johannes Pachlatko
发明人: William Whittingham , Kevin Lawson , Paul Worthington , Charles Russell , Roger Salmon , Leslie May , Mario Jorg , Johannes Pachlatko
IPC分类号: A01N43/54 , A01N43/40 , C07D409/02 , C07D405/02 , C07D403/02 , C07D401/02
CPC分类号: C07D213/70 , A01N43/40 , C07D213/65 , C07D213/68 , C07D213/80 , C07D213/82 , C07D213/85
摘要: Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C1-8 alkyl, C3-6 cycloalkyl, C2-8 alkenyl, C2-8 alkynyl, C1-8 alkoxy, C1-8 alkylthio, nitro, amino, mono- or di-(C1-6)alkylamino, mono- or di-(C2-6)alkenylamino, mono- or di-(C2-6)alkynylamino, formylamino, C1-4 alkyl(formyl)amino, C1-4 alkylcarbonylamino, C1-4 alkyl(C1-4 alkylcarbonyl)amino, cyano, formyl, C1-4 alkylcarbonyl, C1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C1-4)alkylaminocarbonyl, carboxy, C1-4 alkylcarbonyloxy, aryl(C1-4)alkylcarbonyloxy, C1-4 alkylsulphinyl, C1-4 alkylsulphonyl, C1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R1 is phenyl, cyano, C1-4 alkyl, C2-4 alkenyl or C2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C1-4 alkylcarbonyl group, with a C1-4 alkoxycarbonyl group or with a hydroxy group, or R1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R2 is H, C1-4 alkyl, C1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C1-4 alkoxy; R3 and R4 are independently H, C1-3 alkyl, C2-3 alkenyl or C2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R3 and R4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C1-4 alkyl; and R5 is halo, C1-4 alkyl or C3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C1-6 alkoxy, C1-6 alkylthio, cyano, C1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C1-4)alkylaminocarbonyloxy, or tri(C1-4)alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
-
公开(公告)号:US20130043192A1
公开(公告)日:2013-02-21
申请号:US13212861
申请日:2011-08-18
申请人: Ed Smith , Vicente Sanchez , Jeffrey C. Trewella , Stephen J. McGovern , Royce Roemisch , Jennifer Sorrells , Leslie May , Maria Magdalena Ramirez Corredores , Rocio Maria Banda , Lorerz Bauer
发明人: Ed Smith , Vicente Sanchez , Jeffrey C. Trewella , Stephen J. McGovern , Royce Roemisch , Jennifer Sorrells , Leslie May , Maria Magdalena Ramirez Corredores , Rocio Maria Banda , Lorerz Bauer
IPC分类号: B01D17/02
CPC分类号: C10G29/06 , B01D17/02 , B01D17/0208 , B01D17/04 , B01D17/042 , B01D17/044 , B01D17/047 , B01D17/048 , B01D17/06 , C10G3/40 , C10G3/42 , C10G29/10 , C10G29/20 , C10G29/22 , C10G32/02 , C10G33/02 , C10G33/04 , C10G2300/1011 , C10G2300/208 , C10G2300/308 , Y02P30/20
摘要: Disclosed is a process for the alteration of the ratio of the specific gravities of the oil and water phases resulting from the conversion of biomass to liquid products, the reduction of the conductivity and of metals of the product mixture, which each can aid in the removal of solids contained in the oil phase.
摘要翻译: 公开了一种用于改变由生物质转化为液体产物而导致的油相和水相的比重与产物混合物的导电性和金属的降低的比例的方法,其中每一种可以有助于除去 包含在油相中的固体。
-
公开(公告)号:US06699874B2
公开(公告)日:2004-03-02
申请号:US10314594
申请日:2002-12-10
IPC分类号: A01N4354
CPC分类号: A01N43/90 , A01N2300/00
摘要: Fungicidal compositions comprising an acceptable carrier and/or surface active agent and synergistically effective amounts of (a) at least one azolopyrimidine of formula I in which R1, R2, L1, L2 and L3 have the meaning given in claim 1; and (b) at least one fungicidal active ingredient selected from benomyl, carboxin, captan, chlorothalonil, copper oxychloride, cyprodinil, dimethomorph, dithianon, dodine, famoxadone, fenhexamid, fenpiclonil, fenpropimorph, fluazinam, mancozeb, metalaxyl, pyrimethanil, quinoxifen, sulfur, triforine, vinclozolin, a fungicidal triazole derivative, and a synthetic strobilurine derivative. The invention also provides a method of controlling the growth of phytopathogenic fungi at a locus by applying synergistically effective amounts of at least one azolopyrimidine of formula I and at least one fungicidal active ingredient (b) to the locus.
摘要翻译: 包含可接受的载体和/或表面活性剂和协同有效量的(a)至少一种R 1,R 2,L 1,L 2和L 3的式Iin的偶氮嘧啶的杀真菌组合物 >具有权利要求1中给出的含义; 和(b)至少一种杀真菌活性成分,其选自苯菌灵,呋喃丹,克拉曼,百菌清,氯氧化铜,西酞替尼,烯酰吗啉,二噻吩,十二烷,恶唑酮,芬己酰,芬替尼,芬卡芬,氟啶胺,代森锰锌,甲霜灵,嘧霉胺,喹喔啉, ,triperine,长春菌素,杀真菌三唑衍生物和合成次溴酸衍生物。 本发明还提供了一种通过将协同有效量的至少一种式I的偶氮嘧啶和至少一种杀真菌活性成分(b)施用于该基因座来控制植物病原真菌在一个场所生长的方法。
-
公开(公告)号:US06255309B1
公开(公告)日:2001-07-03
申请号:US09272916
申请日:1999-03-19
申请人: Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
发明人: Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
IPC分类号: A61K31505
CPC分类号: C07D487/04 , A01N43/90
摘要: The novel compounds of formula I: wherein (R1, R2, Hal and L1 through L5 are defined in the specification) show selective fungicidal activity. The new compounds may be processed with carriers and adjuvants to produce fungicidal compositions.
摘要翻译: 式I的新化合物:其中(R1,R2,Hal和L1至L5在说明书中定义)表示选择性杀真菌活性。 可以用载体和佐剂处理新的化合物以产生杀真菌组合物。
-
公开(公告)号:US09315739B2
公开(公告)日:2016-04-19
申请号:US13212861
申请日:2011-08-18
申请人: Ed Smith , Vicente Sanchez , Jeffrey C. Trewella , Stephen J. McGovern , Royce Roemisch , Jennifer Sorrells , Leslie May , Maria Magdalena Ramirez Corredores , Rocio Maria Banda , Lorerz Bauer
发明人: Ed Smith , Vicente Sanchez , Jeffrey C. Trewella , Stephen J. McGovern , Royce Roemisch , Jennifer Sorrells , Leslie May , Maria Magdalena Ramirez Corredores , Rocio Maria Banda , Lorerz Bauer
IPC分类号: B01D17/02 , B01D17/04 , C10G29/06 , C10G29/10 , C10G29/20 , C10G29/22 , C10G3/00 , B01D17/06 , C10G32/02 , C10G33/02 , C10G33/04
CPC分类号: C10G29/06 , B01D17/02 , B01D17/0208 , B01D17/04 , B01D17/042 , B01D17/044 , B01D17/047 , B01D17/048 , B01D17/06 , C10G3/40 , C10G3/42 , C10G29/10 , C10G29/20 , C10G29/22 , C10G32/02 , C10G33/02 , C10G33/04 , C10G2300/1011 , C10G2300/208 , C10G2300/308 , Y02P30/20
摘要: Disclosed is a process for the alteration of the ratio of the specific gravities of the oil and water phases resulting from the conversion of biomass to liquid products, the reduction of the conductivity and of metals of the product mixture, which each can aid in the removal of solids contained in the oil phase.
摘要翻译: 公开了一种用于改变由生物质转化为液体产物而导致的油相和水相的比重与产物混合物的导电性和金属的降低的比例的方法,其中每一种可以有助于除去 包含在油相中的固体。
-
公开(公告)号:US06518275B1
公开(公告)日:2003-02-11
申请号:US09809512
申请日:2001-03-15
IPC分类号: A01N3744
CPC分类号: A01N43/90 , A01N61/00 , A01N59/20 , A01N59/02 , A01N47/44 , A01N47/38 , A01N47/40 , A01N47/04 , A01N43/84 , A01N43/76 , A01N43/653 , A01N43/60 , A01N43/54 , A01N43/32 , A01N43/42 , A01N43/40 , A01N37/50 , A01N37/46 , A01N37/38 , A01N37/34 , A01N2300/00
摘要: Fungicidal compositions comprising an acceptable carrier and/or surface active agent and synergistically effective amounts of (a) at least one azolopyrimidine of formula I in which R1, R2, L1, L2 and L3 have the meaning given in claim 1; and (b) at least one fungicidal active ingredient selected from benomyl, carboxin, captan, chlorothalonil, copper oxychloride, cyprodinil, dimethomorph, dithianon, dodine, famoxadone, fenhexamid, fenpiclonil, fenpropimorph, fluazinam, mancozeb, metalaxyl, pyrimethanil, quinoxifen, sulfur, triforine, vinclozolin, a fungicidal triazole derivative, and a synthetic strobilurine derivative. The invention also provides a method of controlling the growth of phytopathogenic fungi at a locus by applying synergistically effective amounts of at least one azolopyrimidine of formula I and at least one fungicidal active ingredient (b) to the locus.
摘要翻译: 包含可接受的载体和/或表面活性剂的杀真菌组合物和协同有效量的(a)至少一种式I的偶氮嘧啶,其中R 1,R 2,L 1,L 2和L 3具有权利要求1中给出的含义; 和(b)至少一种杀真菌活性成分,其选自苯菌灵,呋喃丹,克拉曼,百菌清,氯氧化铜,西酞替尼,烯酰吗啉,二噻吩,十二烷,恶唑酮,芬己酰,芬替尼,芬卡芬,氟啶胺,代森锰锌,甲霜灵,嘧霉胺,喹喔啉, ,triperine,长春菌素,杀真菌三唑衍生物和合成次溴酸衍生物。 本发明还提供了一种通过将协同有效量的至少一种式I的偶氮嘧啶和至少一种杀真菌活性成分(b)施用于该基因座来控制植物病原真菌在一个场所生长的方法。
-
公开(公告)号:US07084146B2
公开(公告)日:2006-08-01
申请号:US09840488
申请日:2001-04-23
申请人: Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
发明人: Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
IPC分类号: C07D487/04 , A01N43/90
CPC分类号: C07D487/04 , A01N43/90
摘要: The novel compounds of formula I: wherein R1 is hydrogen or methyl; R2 is hydrogen, or an optionally substituted alkyl, alkenyl, alkynyl, alkadienyl or phenyl group; Hal is halogen; and L1 through L5 are each hydrogen, halogen, alkyl, alkoxy or nitro, provided that at least one of L1 through L5 represents nitro or alkoxy; show selective fungicidal activity. The new compounds are processed with carriers and adjuvants to fungicidal compositions.
摘要翻译: 式I的新化合物:其中R 1是氢或甲基; R 2是氢或任选取代的烷基,烯基,炔基,链二烯基或苯基; 卤素是卤素; 和L 1至L 5各自为氢,卤素,烷基,烷氧基或硝基,条件是L 1至L 2中的至少一个, SUP> 5表示硝基或烷氧基; 显示选择性杀真菌活性。 新的化合物用载体和佐剂加工成杀真菌剂。
-
公开(公告)号:US6124301A
公开(公告)日:2000-09-26
申请号:US268853
申请日:1999-03-15
申请人: Michael Aven , Henry Van Tuyl Cotter , Leslie May
发明人: Michael Aven , Henry Van Tuyl Cotter , Leslie May
IPC分类号: A01N43/90 , C07D487/04 , A01N43/00
CPC分类号: C07D487/04 , A01N43/90
摘要: Adjuvants selected from liquid polyalkoxylated aliphatic alcohols, solid sodium hydrocarbyl sulfonates and polyalkoxylated trisiloxanes enhance the efficacy of fungicidal triazolopyrimidines. They can be incorporated into formulations of the fungicidal compounds or be added to spray mixtures (tank mix) as separately formulated additives in order to improve the efficacy, systemicity and spectrum of these fungicides.
摘要翻译: 选自液体聚烷氧基化脂族醇,固体烷基磺酸钠和聚烷氧基化三硅氧烷的佐剂增强了杀真菌三唑并嘧啶的功效。 它们可以并入到杀真菌化合物的制剂中,或者作为单独配制的添加剂加入到喷雾混合物(罐混合物)中,以提高这些杀真菌剂的功效,系统性和光谱。
-
公开(公告)号:US06656944B2
公开(公告)日:2003-12-02
申请号:US09832964
申请日:2001-04-11
申请人: Ewald Sieverding , Leslie May
发明人: Ewald Sieverding , Leslie May
IPC分类号: A01N4354
CPC分类号: A01N43/90 , A01N39/04 , A01N39/02 , A01N2300/00
摘要: The invention relates to fungicidal compositions comprising an acceptable carrier and/or surface active agent and synergistically effective amounts of (a) at least one azolopyrimidine of formula I in which R1 through R2, L, A and n have the meaning given in claim 1; (b) and at least one melanin biosynthesis inhibitor (MBI), preferably a phenoxyamide of formula II wherein R5 through R9, Y and m have the meaning given in claim 2; and to a method of controlling the growth of phythopathogenic fungi at a locus which comprises applying synergistically effective amounts of at least one azolopyrimidine of formula I (a) and at least one MBI (b) to the locus.
摘要翻译: 本发明涉及包含可接受的载体和/或表面活性剂和协同有效量的(a)至少一种式Iin的至少一种氮杂嘧啶的杀真菌组合物,其中R 1至R 2,L,A和n具有其含义 在权利要求1中给出;(b)和至少一种黑色素生物合成抑制剂(MBI),优选式VII的苯氧基酰胺,其中R 5至R 9,Y和m具有权利要求2中给出的含义; 以及在一个场所控制植物病原真菌的生长的方法,其包括将协同有效量的至少一种式I(a)的偶氮嘧啶和至少一种MBI(b)施用于该基因座。
-
-
-
-
-
-
-
-
-