Optically active 2,2′-biphenol derivative and production method of same
    1.
    发明授权
    Optically active 2,2′-biphenol derivative and production method of same 有权
    光活性2,2'-联苯酚衍生物及其制备方法

    公开(公告)号:US08283501B2

    公开(公告)日:2012-10-09

    申请号:US12811805

    申请日:2009-01-06

    IPC分类号: C07C39/15 C07C37/68 C07C37/86

    摘要: Disclosed herein are optically active biphenol derivatives represented by the following formulas (1) and (2), a method for optically resolving a biphenol derivative represented by formula (2′), a production method of an optically active biphenol derivative (1) comprising a step for reacting a Brønsted acid with a biphenol derivative (2), and a production method of an optically active biphenol derivative (3) comprising a step for reacting a Lewis acid with an optically active biphenol derivative (1) or an optically active biphenol derivative (2).

    摘要翻译: 本文公开了由下式(1)和(2)表示的光学活性联苯酚衍生物,用于光学拆分由式(2')表示的联苯酚衍生物的方法,光学活性联苯酚衍生物(1)的制备方法,其包含 使布朗斯台德酸与联苯酚衍生物(2)反应的步骤和光学活性联苯酚衍生物(3)的制备方法包括使路易斯酸与光学活性联苯酚衍生物(1)或光学活性联苯酚衍生物 (2)。

    OPTICALLY ACTIVE 2,2'-BIPHENOL DERIVATIVE AND PRODUCTION METHOD OF SAME
    2.
    发明申请
    OPTICALLY ACTIVE 2,2'-BIPHENOL DERIVATIVE AND PRODUCTION METHOD OF SAME 有权
    具有活性的2,2'-联苯酚衍生物及其制备方法

    公开(公告)号:US20100280284A1

    公开(公告)日:2010-11-04

    申请号:US12811805

    申请日:2009-01-06

    IPC分类号: C07C39/15

    摘要: An optically active 2,2′-biphenol derivative and a production method that enables simple and efficient production of this compound. More specifically, an optically active biphenol derivative represented by the following formulas (1) and (2), a method for optically resolving a biphenol derivative represented by formula (2′), a production method of an optically active biphenol derivative (1) comprising a step for reacting a Brønsted acid with a biphenol derivative (2), and a production method of an optically active biphenol derivative (3) comprising a step for reacting a Lewis acid with an optically active biphenol derivative (1) or an optically active biphenol derivative (2). In the following formulas, R represents, for example, a primary or secondary alkyl group having 1 to 10 carbon atoms, * represents an axially asymmetric center, X represents a halogen atom, and R2 represents a tertiary alkyl group having 4 to 6 carbon atoms.

    摘要翻译: 一种光学活性的2,2'-联苯酚衍生物和能够简单且有效地生产该化合物的制备方法。 更具体地,由下式(1)和(2)表示的光学活性联苯酚衍生物,用于光学拆分由式(2')表示的联苯酚衍生物的方法,光学活性联苯酚衍生物(1)的制备方法,包括 将布朗斯台德酸与联苯酚衍生物(2)反应的步骤和光学活性联苯酚衍生物(3)的制备方法,其包括使路易斯酸与光学活性联苯酚衍生物(1)或光学活性联苯酚 衍生物(2)。 在下式中,R表示例如碳原子数1〜10的伯或仲烷基,*表示轴向不对称中心,X表示卤素原子,R 2表示碳原子数4〜6的叔烷基 。

    OPTICALLY ACTIVE DIBENZAZEPINE DERIVATIVES
    3.
    发明申请
    OPTICALLY ACTIVE DIBENZAZEPINE DERIVATIVES 有权
    光学活性二苯并恶唑衍生物

    公开(公告)号:US20110034688A1

    公开(公告)日:2011-02-10

    申请号:US12936415

    申请日:2009-04-08

    IPC分类号: C07D493/04

    摘要: It is to provide a novel optically active dibenzazepine derivative having a high utility value as an asymmetric phase-transfer catalyst. It is an optically active 6,7-dihydro-5H-dibenzo[c,e]azepine derivative represented by the following formula (1′), (wherein R represents a divalent organic group for cross-linking the 1st position and the 11th position; R1 and R2 are the same or different, and represent a hydrogen atom, halogen atom, or organic group, or R1 and R2 together represent a divalent organic group; R3′and R4′ are the same or different and represent a monovalent organic group, or R3′ and R4′ together form an organic group that forms a cyclic structure comprising an onium nitrogen atom; Ar represents a monovalent organic group; * represents optical activity, i.e., that one axially asymmetric isomer is present in excess of the other axially asymmetric isomer with respect to a bond axis that constitutes the biphenyl structure of the compound; and X− represents a counter anion).

    摘要翻译: 提供作为不对称相转移催化剂的具有高效用价值的新颖的光学活性二苯并氮杂衍生物。 它是由下式(1')表示的光学活性的6,7-二氢-5H-二苯并[c,e]吖庚因衍生物,其中R表示用于交联第1位和第11位的二价有机基 R 1和R 2相同或不同,表示氢原子,卤素原子或有机基团,或者R 1和R 2一起表示二价有机基团; R 3'和R 4'相同或不同,表示一价有机基团 或R3'和R4'一起形成形成包含鎓氮原子的环状结构的有机基团; Ar表示一价有机基团; *表示光学活性,即一种轴向不对称异构体存在于另一种轴向 相对于构成化合物的联苯结构的键轴的不对称异构体; X-表示抗衡阴离子)。

    Optically active dibenzazepine derivatives
    4.
    发明授权
    Optically active dibenzazepine derivatives 有权
    光活性二苯并氮杂衍生物

    公开(公告)号:US08507669B2

    公开(公告)日:2013-08-13

    申请号:US12936415

    申请日:2009-04-08

    IPC分类号: C07D491/16 C07D317/60

    摘要: It is to provide a novel optically active dibenzazepine derivative having a high utility value as an asymmetric phase-transfer catalyst. It is an optically active 6,7-dihydro-5H-dibenzo[c,e]azepine derivative represented by the following formula (1′), (wherein R represents a divalent organic group for cross-linking the 1st position and the 11th position; R1 and R2 are the same or different, and represent a hydrogen atom, halogen atom, or organic group, or R1 and R2 together represent a divalent organic group; R3′ and R4′ are the same or different and represent a monovalent organic group, or R3′ and R4′ together form an organic group that forms a cyclic structure comprising an onium nitrogen atom; Ar represents a monovalent organic group; * represents optical activity, i.e., that one axially asymmetric isomer is present in excess of the other axially asymmetric isomer with respect to a bond axis that constitutes the biphenyl structure of the compound; and X− represents a counter anion).

    摘要翻译: 提供作为不对称相转移催化剂的具有高效用价值的新颖的光学活性二苯并氮杂衍生物。 它是由下式(1')表示的光学活性的6,7-二氢-5H-二苯并[c,e]吖庚因衍生物,其中R表示用于交联第1位和第11位的二价有机基 R1和R2相同或不同,表示氢原子,卤素原子或有机基团,或者R1和R2一起表示二价有机基团; R3'和R4'相同或不同,表示一价有机基团 或R3'和R4'一起形成形成包含鎓氮原子的环状结构的有机基团; Ar表示一价有机基团; *表示光学活性,即一种轴向不对称异构体存在于另一种轴向 相对于构成化合物的联苯结构的键轴的不对称异构体; X-表示抗衡阴离子)。

    NOVEL PHENOL DERIVATIVE
    5.
    发明申请
    NOVEL PHENOL DERIVATIVE 有权
    新颖的酚醛衍生物

    公开(公告)号:US20120184587A1

    公开(公告)日:2012-07-19

    申请号:US13499190

    申请日:2010-09-29

    摘要: Disclosed are a novel compound and a pharmaceutical product, each having a remarkable uricosuric effect. Specifically disclosed are: a novel phenol derivative represented by general formula (1) that is shown in FIG. 1; a pharmaceutically acceptable salt thereof; a hydrate of the derivative or the salt; and a solvate of the derivative or the salt. (In the formula, R1 and R2 may be the same or different and each represents a lower alkyl group, a lower alkenyl group, a lower alkynyl group, a lower alkoxy group, a haloalkyl group, a haloalkoxy group, an alkylsulfanyl group, an alkylsulfinyl group, an alkylsulfonyl group, a lower alkyl-substituted carbamoyl group, a saturated nitrogen-containing heterocyclic N-carbonyl group, a halogen atom, a cyano group or a hydrogen atom; R3 represents a lower alkyl group, a haloalkyl group, a halogen atom, a hydroxy group or a hydrogen atom; and X represents a sulfur atom, an —S(═O)— group or an —S(═O)2— group.)

    摘要翻译: 公开了一种新型化合物和药物,其具有显着的尿酸营养作用。 具体公开的是:图1所示的通式(1)表示的新型苯酚衍生物。 1; 其药学上可接受的盐; 衍生物或盐的水合物; 和衍生物或盐的溶剂化物。 (式中,R 1,R 2可以相同或不同,表示低级烷基,低级烯基,低级炔基,低级烷氧基,卤代烷基,卤代烷氧基,烷基硫烷基, 烷基亚磺酰基,烷基磺酰基,低级烷基取代氨基甲酰基,饱和含氮杂环N-羰基,卤素原子,氰基或氢原子; R3表示低级烷基,卤代烷基, 卤素原子,羟基或氢原子; X表示硫原子,-S(= O) - 基或-S(= O)2 - 基)。

    Display device
    8.
    发明授权
    Display device 失效
    显示设备

    公开(公告)号:US6064453A

    公开(公告)日:2000-05-16

    申请号:US129947

    申请日:1998-08-06

    摘要: Stress exerted on a liquid crystal display element via a case was likely to impede display on the liquid crystal display element, or damage a liquid crystal display device. A front end of a rib 9 protruding toward a case 1 from a peripheral edge portion of a holder 8 supporting a liquid crystal display element 4 is brought into contact with the case 1, whereby stress on the case 1 is imposed on the rib 9. Thus, stress directly acting on the liquid crystal display element 4 via a rubber sheet 7 can be prevented.

    摘要翻译: 经由外壳施加在液晶显示元件上的应力可能阻碍液晶显示元件的显示,或损坏液晶显示装置。 从支撑液晶显示元件4的保持器8的周缘部朝向壳体1突出的肋9的前端与壳体1接触,由此将壳体1上的应力施加在肋9上。 因此,可以防止通过橡胶片7直接作用在液晶显示元件4上的应力。

    Opening and closing mechanism for electronic device
    10.
    发明授权
    Opening and closing mechanism for electronic device 失效
    电子设备开闭机构

    公开(公告)号:US5799079A

    公开(公告)日:1998-08-25

    申请号:US734844

    申请日:1996-10-23

    申请人: Tsutomu Inoue

    发明人: Tsutomu Inoue

    摘要: A portable phone incorporating an opening and closing mechanism comprises a main body, a sub-body, a hinge unit, and distribution cables. The main body and the sub-body respectively include electric circuits. The hinge unit includes a shaft disposed at one end of the sub-body, a cam having a center axis coupled to the shaft and used for regulating opening and closing angles of the sub-body, and a pair of leaf springs for maintaining turning angles of the cam. The distribution cables are connected to the electric circuits, and have their center portions wound around the shaft of the hinge unit. The distribution cables are stretched or compressed when the sub-body is opened or closed.

    摘要翻译: 包括开闭机构的便携式电话机包括主体,子体,铰链单元和分配电缆。 主体和子体分别包括电路。 铰链单元包括设置在子体的一端的轴,具有联接到轴的中心轴并用于调节副体的开闭角度的凸轮和用于保持转向角的一对板簧 的凸轮。 分配电缆连接到电路,并且其中心部分缠绕在铰链单元的轴上。 当子体打开或关闭时,分配电缆被拉伸或压缩。