LYSIN-GLUTAMIC ACID DIPEPTIDE DERIVATIVES
    23.
    发明公开
    LYSIN-GLUTAMIC ACID DIPEPTIDE DERIVATIVES 审中-公开
    赖氨酸 - 谷氨酸二萜衍生物

    公开(公告)号:EP3127604A1

    公开(公告)日:2017-02-08

    申请号:EP16179885.5

    申请日:2013-05-13

    发明人: PUENTENER, KURT

    IPC分类号: B01J19/00 C07C271/22

    摘要: The invention relates to compounds of the formula

    to a process for making same and to the use of the products in the solid phase peptide synthesis.
    The compounds of formula I are versatile peptide intermediates for the solid phase peptide synthesis (SPPS) of peptide drugs which comprise a Glu-fatty alkyl side chain building block attached to a Lys-part of the peptide chain.

    摘要翻译: 本发明涉及下式化合物及其制备方法以及产物在固相肽合成中的用途。 式I化合物是用于肽药物的固相肽合成(SPPS)的多功能肽中间体,其包含与肽链的Lys部分连接的Glu-脂肪烷基侧链结构单元。