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公开(公告)号：EP1244641A1
公开(公告)日：2002-10-02
申请号：EP00991169.4
申请日：2000-12-12
发明人： FISCHER, Rüdiger , KLEYMANN, Gerald , BETZ, Ulrich , BAUMEISTER, Judith , BENDER, Wolfgang , ECKENBERG, Peter , HANDKE, Gabriele , HENDRIX, Martin , HENNINGER, Kerstin , JENSEN, Axel , KELDENICH, Jörg , SCHNEIDER, Udo , WEBER, Olaf
IPC分类号： C07D277/54 , C07D417/12 , C07F9/6539 , C07F7/18 , A61K31/426 , A61P31/22
CPC分类号： C07D231/12 , C07D233/56 , C07D249/08 , C07D277/54 , C07D417/12 , C07F7/1856 , C07F9/6539
摘要： The invention relates to novel thiazolyl amide derivatives, to a method for producing them and to their use as medicaments, especially as antiviral medicaments.
摘要翻译： 本发明涉及新的噻唑酰胺衍生物，它们的制备方法以及它们作为药物，特别是作为抗病毒药物的用途。
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公开(公告)号：EP1467723A1
公开(公告)日：2004-10-20
申请号：EP03729422.0
申请日：2003-01-07
发明人： HENDRIX, Martin , BAUMANN, Karlheinz , GROSSER, Rolf , KÖNIG, Gerhard , DÜSTERHUS, Vera , KRÜGER, Joachim
IPC分类号： A61K31/10 , A61K31/4465 , A61K31/4409 , A61K31/496 , A61K31/40 , A61K31/5375 , A61P25/28 , C07C317/22 , C07D295/20 , C07D213/74 , C07D241/08 , C07D211/46 , C07D211/22 , C07D493/10 , C07D211/52
CPC分类号： C07D239/42 , C07C317/18 , C07C2601/14 , C07D207/06 , C07D207/46 , C07D211/22 , C07D211/46 , C07D211/52 , C07D213/74 , C07D241/08 , C07D295/205 , C07D491/10
摘要： The invention relates to the phenyl sulfoxides and phenyl sulfones of formula (I) and to methods for producing the same as well as to their use in the production of drugs for the treatment and/or prophylaxis of diseases, especially Alzheimer's disease. The inventive compounds inhibit η secretase.
摘要翻译： 本发明涉及苯基亚砜和砜及其制备方法，以及它们用于生产药物用于治疗和/或预防疾病，特别是阿尔茨海默氏病的用途。
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公开(公告)号：EP1363912A1
公开(公告)日：2003-11-26
申请号：EP02704706.7
申请日：2002-02-11
发明人： NIEWÖHNER, Ulrich , SCHAUSS, Dagmar , KÖNIG, Gerhard , HENDRIX, Martin , BÖSS, Frank-Gerhard , VAN DER STAAY, Franz-Josef , SCHREIBER, Rudy , SCHLEMMER, Karl-Heinz , MORIWAKI, Toshiya , NIEWÖHNER, Maria Theresia
IPC分类号： C07D487/04 , A61K31/53 , A61P25/00 , C07D253/06
CPC分类号： C07D253/07 , C07D487/04
摘要： The invention relates to novel substituted imidazotriazinones, to a method for their production and to the use thereof for producing medicaments, in particular to improve perception, powers of concentration, learning capacity and/or memory retentiveness.
摘要翻译： 本发明涉及新型取代的咪唑并三嗪酮，其制备方法及其用于制备药物的用途，特别是改善知觉，注意力，学习能力和/或记忆保持力的能力。
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公开(公告)号：EP1319185A1
公开(公告)日：2003-06-18
申请号：EP00945756.5
申请日：2000-06-15
发明人： KLEYMANN, Gerald , BETZ, Ulrich , FISCHER, Rüdiger , HENDRIX, Martin , HEWLETT, Guy , PEVZNER, Veniamin
IPC分类号： G01N33/569 , G01N33/50
CPC分类号： G01N33/502 , C07D277/54 , C07D417/12 , G01N33/5008 , G01N2333/035
摘要： The invention relates to a method for identifying compounds with antiviral activity, characterized in that those compounds are selected in the presence of which resistant viral mutants can be selected, wherein at least one selected viral mutant carries at least one mutation in the primase gene and another selected viral mutant carries at least one mutation in the helicase gene or a selected viral mutant carries at least one mutation in the helicase and at least one mutation in the primase gene.
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5.发明公开
公开(公告)号：EP1307201A2
公开(公告)日：2003-05-07
申请号：EP01969511.3
申请日：2001-07-19
发明人： BÖSS, Frank-Gerhard , HENDRIX, Martin , KÖNIG, Gerhard , NIEWÖHNER, Ulrich , SCHLEMMER, Karl-Heinz , SCHREIBER, Rudy , VAN DER STAAY, Franz-Josef , SCHAUSS, Dagmar
CPC分类号： A61K31/505
摘要： The invention relates to the use of selective phosphodiesterase 2, (PDE 2), inhibitors for producing medicaments to improve cognition, powers of concentration, learning capability and/or memory retention.
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公开(公告)号：EP1181267A1
公开(公告)日：2002-02-27
申请号：EP00931134.1
申请日：2000-05-08
发明人： ARLT, Dieter , HENDRIX, Martin , ELBE, Hans-Ludwig , HÄNSSLER, Gerd , KUCK, Karl-Heinz , ERDELEN, Christoph , SAWADA, Haruko
IPC分类号： C07C233/15 , C07C233/09 , C07C57/42 , C07C233/20 , C07C259/06 , C07C233/52 , C07C233/47 , C07C69/003 , C07C233/54 , C07C251/66 , C07C259/08 , C07D295/16 , C07D213/40 , C07D213/75 , C07D213/61
CPC分类号： C07D213/40 , A01N37/06 , A01N37/18 , A01N37/22 , C07C57/60 , C07C69/65 , C07C233/13 , C07C233/14 , C07C233/15 , C07C233/22 , C07C233/51 , C07C233/55 , C07C239/10 , C07C239/12 , C07C251/66 , C07C255/60 , C07C259/06 , C07C259/10 , C07C2601/14 , C07D213/61 , C07D213/75 , C07D217/18 , C07D277/28 , C07D295/185
摘要： The invention relates to novel halogen compounds, to a method for producing them and to their use for treating plants for protecting them against attack from phytopathogenic microorganisms and insects. The invention also relates to novel intermediate products and to methods for producing the same.
摘要翻译： 本发明涉及新型卤素化合物，其制备方法及其用于处理植物以防止植物病原微生物和昆虫侵袭的用途。 本发明还涉及新的中间产物及其制备方法。
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7.发明公开
公开(公告)号：EP1347978A1
公开(公告)日：2003-10-01
申请号：EP01271375.6
申请日：2001-12-10
发明人： NIEWÖHNER, Ulrich , SCHAUSS, Dagmar , HENDRIX, Martin , KÖNIG, Gerhard , BÖSS, Frank-Gerhard , VAN DER STAAY, Franz-Josef , SCHREIBER, Rudy , SCHLEMMER, Karl-Heinz , GROSSER, Rolf
IPC分类号： C07D487/04 , C07D253/06 , A61K31/53 , A61P25/28
CPC分类号： C07D487/04 , A61K31/53
摘要： The invention relates to novel substituted imidazotriazinones (I), methods for the production thereof, and the use thereof for producing medicaments particularly for improving perception, concentration capacity, learning capacity and/or memory capacity.
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8.发明公开THIAZOLYLHARNSTOFF-DERIVATE UND IHRE VERWENDUNG ALS ANTIVIRALE MITTEL 有权THIAZOLYLHARNSTOFF衍生物及其作为抗病毒剂
公开(公告)号：EP1161423A1
公开(公告)日：2001-12-12
申请号：EP00907614.2
申请日：2000-02-24
发明人： FISCHER, Rüdiger , KLEYMANN, Gerald , BAUMEISTER, Judith , BENDER, Wolfgang , BETZ, Ulrich , ECKENBERG, Peter , HANDKE, Gabriele , HENDRIX, Martin , SCHNEIDER, Udo , WEBER, Olaf , HENNINGER, Kerstin , JENSEN, Axel , KELDENICH, Jörg
IPC分类号： C07D277/54 , C07D417/12 , C07D487/04 , A61K31/426 , A61K31/427 , A61P31/12
CPC分类号： C07D231/12 , C07D233/56 , C07D249/08 , C07D277/54 , C07D417/12 , C07D487/04
摘要： The invention relates to thiazolyl urea derivatives of formula (I), to a method for the production thereof, and to their use as medicaments, in particular, as antiviral medicaments.
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