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1.发明公开SELECTIVE ESTROGEN RECEPTOR MODULATORS FOR THE TREATMENT OF VASOMOTOR SYMPTOMS 有权用于治疗血管舒缩症状，雌激素受体的选择性调节剂
公开(公告)号：EP1709021A1
公开(公告)日：2006-10-11
申请号：EP05704874.6
申请日：2005-01-18
Applicant: ELI LILLY AND COMPANY
Inventor： DALLY, Robert, Dean , DODGE, Jeffrey, Alan , FRANK, Scott, Alan , HINKLIN, Ronald, Jay , SHEPHERD, Timothy, Alan , WALLACE, Owen, Brendan
IPC: C07D295/08 , C07D311/78 , C07D335/04 , C07D221/18 , A61K31/4453 , A61K31/4523 , A61K31/55 , A61P15/12
CPC classification number: C07D295/088 , C07D221/18 , C07D311/78 , C07D335/04
Abstract: The present invention relates to a selective estrogen receptor modulator of formula I or Ia: (I) (Ia); or a pharmaceutical acid addition salt thereof; useful for treating vasomotor symptoms, in particular hot flashes, night sweats and other symptoms that affect women around menopause.
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2.发明授权SELECTIVE ESTROGEN RECEPTOR MODULATORS CONTAINING A PHENYLSULFONYL GROUP 有权选择性雌激素受体调节剂，AN苯磺酰基CONTAIN
公开(公告)号：EP1530470B9
公开(公告)日：2010-04-07
申请号：EP03765254.2
申请日：2003-07-16
Applicant: ELI LILLY AND COMPANY
Inventor： DALLY, Robert, Dean , DODGE, Jeffrey, Alan , FRANK, Scott, Alan , JONES, Scott, Alan , SHEPHERD, Timothy, Alan , WALLACE, Owen, Brendan , FONG, Kin, Chiu , HUMMEL, Conrad, Wilson , LEWIS, Geroge, Sal
IPC: A61K31/4453 , A61P5/32 , C07D295/08 , C07D333/56 , C07D333/72 , C07D295/12 , C07D333/64
CPC classification number: C07D295/088 , C07D295/13 , C07D333/56 , C07D333/64 , C07D333/72 , C07D409/02
Abstract: The present invention relates to a selective estrogen receptor modulator of formula I or a pharmaceutical acid addition salt thereof; useful, e.g., for treating endometriosis and/or uterine leiomyoma/leiomyomata.
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公开(公告)号：EP1740575A2
公开(公告)日：2007-01-10
申请号：EP05778064.5
申请日：2005-04-08
Applicant: ELI LILLY AND COMPANY
Inventor： DALLY, Robert, Dean , SHEPHERD, Timothy, Alan , BENDER, David, Michael , ROJO GARCIA, Maria, Isabel
IPC: C07D401/12 , C07D413/14 , C07D207/08 , C07D207/12 , C07D403/12 , C07D413/04 , A61K31/401 , A61P25/00
CPC classification number: C07D413/04 , C07D207/08 , C07D207/12 , C07D211/26 , C07D211/42 , C07D217/18 , C07D241/04 , C07D241/08 , C07D401/12 , C07D403/12 , C07D409/12 , C07D413/14 , C07D417/12 , C07D471/08
Abstract: The present invention provides BACE inhibitors of Formula (I): methods for their use and preparation, and intermediates for their preparation.
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公开(公告)号：EP2358710A1
公开(公告)日：2011-08-24
申请号：EP09744896.3
申请日：2009-11-03
Applicant: Eli Lilly and Company
Inventor： DALLY, Robert, Dean , JOSEPH, Sajan , SHEPHERD, Timothy, Alan
IPC: C07D473/00 , A61K31/52 , A61P35/00
CPC classification number: C07D487/04 , C07D473/34
Abstract: The present invention provides AKT and p70 S6 kinase inhibitors of Formula (I). The present invention also provides pharmaceutical compositions comprising compounds of Formula (I), uses of compounds of Formula (I) and methods of using compounds of Formula (I).
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5.发明授权SELECTIVE ESTROGEN RECEPTOR MODULATORS CONTAINING A PHENYLSULFONYL GROUP 有权选择性雌激素受体调节剂，AN苯磺酰基CONTAIN
公开(公告)号：EP1530470B1
公开(公告)日：2009-06-10
申请号：EP03765254.2
申请日：2003-07-16
Applicant: ELI LILLY AND COMPANY
Inventor： DALLY, Robert, Dean , DODGE, Jeffrey, Alan , FRANK, Scott, Alan , JONES, Scott, Alan , SHEPHERD, Timothy, Alan , WALLACE, Owen, Brendan , FONG, Kin, Chiu , HUMMEL, Conrad, Wilson , LEWIS, Geroge, Sal
IPC: A61K31/4453 , A61P5/32 , C07D295/08 , C07D333/56 , C07D333/72 , C07D295/12 , C07D333/64
CPC classification number: C07D295/088 , C07D295/13 , C07D333/56 , C07D333/64 , C07D333/72 , C07D409/02
Abstract: The present invention relates to a selective estrogen receptor modulator of formula I or a pharmaceutical acid addition salt thereof; useful, e.g., for treating endometriosis and/or uterine leiomyoma/leiomyomata.
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Patent Agency Ranking
公开(公告)号：EP1554272B1
公开(公告)日：2006-10-25
申请号：EP03784749.8
申请日：2003-07-31
Applicant: ELI LILLY AND COMPANY
Inventor： BONJOUKLIAN, Rosanne , DE DIEGO GOMEZ, Jose, Eugenio Lilly, S. A. , DE DIOS, Alfonso Lilly, S. A. , HAMDOUCHI, Chafiq, Hamdouchi , LI, Tiechao , LOPEZ DE URALDE GARMENDIA, Beatriz Lilly, S. A. , VIETH, Michal , YORK, Jeremy, Schulenburg , DALLY, Robert, Dean , DEL PRADO CATALINA, Miriam, Filadelfa Lilly, S. A. , JARAMILLO, Carlos Lilly, S. A. , MARTIN CABREJAS, Luisa, Maria Lilly, S. A. , MONTERO SALGADO, Carlos Lilly, S. A. , PLEITE, Sheila Lilly, S. A. , SANCHEZ-MARTINEZ, Concepcion Lilly, S. A. , SHEPHERD, Timothy, Alan , WIKEL, James, Howard
IPC: C07D409/14 , C07D403/04 , C07D401/14 , C07D405/14 , C07D403/14 , C07D413/14 , C07D471/04 , C07D487/04 , C07D409/04 , C07D417/04 , A61K31/41 , A61P35/04
CPC classification number: C07D403/04 , C07D413/04 , C07D413/14 , C07D417/04 , C07D513/04
Abstract: The present invention provides kinase inhibitors of Formula I: wherein W represents inter alia imidazol, oxazol, pyrazol, thiazol as triazol, which are substituted by phenyl or thienyl. The disclosed compounds inhibit p-38 kinase and are useful in the treatment of metastasis or rheumatoid arthritis.
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公开(公告)号：EP2148880B1
公开(公告)日：2014-05-28
申请号：EP08747285.8
申请日：2008-05-01
Applicant: ELI LILLY AND COMPANY
Inventor： DALLY, Robert, Dean , HUANG, Jianping , JOSEPH, Sajan , SHEPHERD, Timothy, Alan , HOLST, Christian L.
IPC: C07D487/04 , A61K31/437 , A61P35/00
CPC classification number: C07D487/04
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公开(公告)号：EP2358710B1
公开(公告)日：2012-08-15
申请号：EP09744896.3
申请日：2009-11-03
Applicant: Eli Lilly and Company
Inventor： DALLY, Robert, Dean , JOSEPH, Sajan , SHEPHERD, Timothy, Alan
IPC: C07D473/00 , A61K31/52 , A61P35/00
CPC classification number: C07D487/04 , C07D473/34
Abstract: The present invention provides AKT and p70 S6 kinase inhibitors of Formula (I). The present invention also provides pharmaceutical compositions comprising compounds of Formula (I), uses of compounds of Formula (I) and methods of using compounds of Formula (I).
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9.发明授权SELECTIVE ESTROGEN RECEPTOR MODULATORS FOR THE TREATMENT OF VASOMOTOR SYMPTOMS 有权用于治疗血管舒缩症状，雌激素受体的选择性调节剂
公开(公告)号：EP1709021B1
公开(公告)日：2010-08-04
申请号：EP05704874.6
申请日：2005-01-18
Applicant: ELI LILLY AND COMPANY
Inventor： DALLY, Robert, Dean , DODGE, Jeffrey, Alan , FRANK, Scott, Alan , HINKLIN, Ronald, Jay , SHEPHERD, Timothy, Alan , WALLACE, Owen, Brendan
IPC: C07D295/08 , C07D311/78 , C07D335/04 , C07D221/18 , A61K31/4453 , A61K31/4523 , A61K31/55 , A61P15/12
CPC classification number: C07D295/088 , C07D221/18 , C07D311/78 , C07D335/04
Abstract: The present invention relates to a selective estrogen receptor modulator of formula I or Ia: (I) (Ia); or a pharmaceutical acid addition salt thereof; useful for treating vasomotor symptoms, in particular hot flashes, night sweats and other symptoms that affect women around menopause.
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公开(公告)号：EP2148880A1
公开(公告)日：2010-02-03
申请号：EP08747285.8
申请日：2008-05-01
Applicant: ELI LILLY AND COMPANY
Inventor： DALLY, Robert, Dean , HUANG, Jianping , JOSEPH, Sajan , SHEPHERD, Timothy, Alan , HOLST, Christian L.
IPC: C07D487/04 , A61K31/437 , A61P35/00
CPC classification number: C07D487/04
Abstract: The present invention provides p70 S6 kinase inhibitors of the formula: pharmaceutical formulations comprising them, and methods for their use.
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