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公开(公告)号：EP1617848A2
公开(公告)日：2006-01-25
申请号：EP04750828.8
申请日：2004-04-26
申请人： GILEAD SCIENCES, INC. , Boojamra, Constantine G. , Cannizzaro, Carina E. , Chen, James M. , Chen, Xiaowu , Cho, Aesop
发明人： BOOJAMRA, Constantine, G. , CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , FARDIS, Maria , HUANG, Alan, X. , KIM, Choung, X. , KIRSCHBERG, Thorsten, A. , KRAWCZYK, Steven , LEE, Christopher, P. , LIN, Kuei-Ying , MACKMAN, Richard, L. , MARKEVITCH, David, Y. , NELSON, Peter H. , OARE, David , PRASAD, Vidya K. , PYUN, Hyung-Jung , RAY, Adrian S. , SWAMINATHAN, Sundaramoorthi , WATKINS, Will , ZHANG, Lijun , ZHANG, Jennifer
IPC分类号： A61K31/662
CPC分类号： A61K31/662 , A61K47/548 , C07D205/04 , C07D211/58 , C07D239/94 , C07D409/06 , C07D409/14 , C07D413/14 , C07D475/00 , C07D487/04 , C07F9/4075 , C07F9/5728 , C07F9/582 , C07F9/588 , C07F9/60 , C07F9/65037 , C07F9/650941 , C07F9/653 , C07F9/6539 , C07F9/65515 , C07F9/655354 , C07F9/6561
摘要： The invention is related to phosphorus substituted anti-cancer compounds, compositions containing such compounds, and therapeutic methods that include the administration of such compounds, as well as to processes and intermediates useful for preparing such compounds.
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公开(公告)号：EP4222152A1
公开(公告)日：2023-08-09
申请号：EP21801304.3
申请日：2021-09-29
发明人： CHU, Hang , GUO, Hongyan , JIANG, Lan , LI, Jiayao , LIN, David W. , PYUN, Hyung-Jung , WU, Qiaoyin , YANG, Hong , ZAJDLIK, Adam D. , ZHANG, Jennifer R.
IPC分类号： C07D471/04 , A61P31/18 , A61K31/495
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公开(公告)号：EP4143189A1
公开(公告)日：2023-03-08
申请号：EP21728673.1
申请日：2021-04-28
发明人： CANALES, Eda Y. , CHANG, Weng K. , DEBIEN, Laurent P. , JANSA, Petr , LOYER-DREW, Jennifer A. , MARTINEZ, Luisruben P. , PERREAULT, Stephane , PHILLIPS, Gary B. , PYUN, Hyung-Jung , SAITO, Roland D. , SANGI, Michael S. , SCHRIER, Adam J. , SHATSKIKH, Marina E. , TAYLOR, James G. , TREIBERG, Jennifer A. , VAN VELDHUIZEN, Joshua J.
IPC分类号： C07D471/18 , C07D471/22 , C07D487/08 , C07D491/22 , C07D498/18 , C07D498/22 , C07D513/18 , A61P3/10 , A61P7/02 , A61P19/02 , A61P35/00
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公开(公告)号：EP4122537A1
公开(公告)日：2023-01-25
申请号：EP22179180.9
申请日：2020-03-20
发明人： CHU, Hang , GONZALEZ BUENROSTRO, Ana Z. , GUO, Hongyan , HAN, Xiaochun , JIANG, Lan , LI, Jiayao , MITCHELL, Michael L. , PYUN, Hyung-Jung , SCHROEDER, Scott D. , SCHWARZWALDER, Gregg M. , SHAPIRO, Nathan D. , SHIVAKUMAR, Devleena M. , WU, Qiaoyin , YANG, Hong , ZHANG, Jennifer R.
IPC分类号： A61P31/18 , C07D471/04 , C07D491/06 , A61K31/4375 , C07D487/06 , C07D487/08 , C07D498/08
摘要： Compounds for use in treating or preventing human immunodeficiency virus (HIV) infection are disclosed. The compounds have the following formula (I):
including stereoisomers and pharmaceutically acceptable salts thereof, wherein R 1 , R 2 , L, W 1 , W 2 , X, Y, and Z are as defined herein. Methods associated with the preparation and use of such compounds, as well as pharmaceutical compositions comprising such compounds, are also disclosed.-
公开(公告)号：EP3740209A1
公开(公告)日：2020-11-25
申请号：EP19703916.7
申请日：2019-01-18
IPC分类号： A61K31/553 , A61P31/18
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公开(公告)号：EP3277691B1
公开(公告)日：2019-01-30
申请号：EP16716776.6
申请日：2016-04-01
IPC分类号： C07D491/14 , C07D491/22 , C07D498/14 , C07D498/22 , C07D513/22 , A61K31/4375 , A61P31/18
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7.发明公开POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF HIV INFECTIONS 审中-公开多环甲氨基吡啶酮化合物及其在治疗HIV感染中的应用
公开(公告)号：EP3252058A1
公开(公告)日：2017-12-06
申请号：EP17177433.4
申请日：2014-07-11
IPC分类号： C07D498/14 , C07D471/14 , A61K31/553 , A61K31/4995 , A61P31/18
CPC分类号： A61K31/4985 , A61K31/537 , A61K31/553 , A61K45/06 , C07D471/14 , C07D471/18 , C07D498/14 , C07D498/18
摘要： Compounds for use in the treatment of human immunodeficiency virus (HIV) infection are disclosed. The compounds have the following Formula (I):
including stereoisomers and pharmaceutically acceptable salts thereof, wherein R 1 , X, Y 1 , Y 2 , or L are as defined herein. Methods associated with preparation and use of such compounds, as well as pharmaceutical compositions comprising such compounds, are also disclosed.摘要翻译： 公开了用于治疗人免疫缺陷病毒（HIV）感染的化合物。 该化合物具有下式（I）：包括其立体异构体及其药学上可接受的盐，其中R 1，X，Y 1，Y 2或L如本文所定义。 还公开了与这些化合物的制备和使用有关的方法，以及包含这些化合物的药物组合物。
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8.发明公开POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE 有权多环CARBAMOYLPYRIDONVERBINDUNGEN和它们的药物用途
公开(公告)号：EP2822954A1
公开(公告)日：2015-01-14
申请号：EP13815937.1
申请日：2013-12-19
发明人： JIN, Haolun , LAZERWITH, Scott, E. , MARTIN, Teresa, Alejandra, Trejo , BACON, Elizabeth, M. , COTTELL, Jeromy, J. , CAI, Zhenhong, R. , PYUN, Hyung-Jung , MORGANELLI, Philip, Anthony , JI, Mingzhe , TAYLOR, James, G. , CHEN, Xiaowu , MISH, Michael, R. , DESAI, Manoj, C.
IPC分类号： C07D498/14 , C07D471/04 , C07D471/14 , C07D471/22 , C07D487/04
CPC分类号： C07D498/14 , A61K31/498 , A61K31/4985 , A61K31/529 , A61K31/537 , A61K31/551 , A61K31/553 , A61K45/06 , C07D471/18 , C07D471/22 , C07D487/14 , C07D498/18 , A61K2300/00
摘要： Compounds for use in the treatment of human immunodeficiency virus (HIV) infection are disclosed. The compounds have the following Formula (I): including stereoisomers and pharmaceutically acceptable salts thereof, wherein R 1 , X, W, Y 1 , Y 2 , Z 1 and Z 4 are as defined herein. Methods associated with preparation and use of such compounds, as well as pharmaceutical compositions comprising such compounds, are also disclosed.
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公开(公告)号：EP1663254A2
公开(公告)日：2006-06-07
申请号：EP04750871.8
申请日：2004-04-26
发明人： CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , FARDIS, Maria , GIBBS, Craig , HIRSCHMANN, Ralph, F. , KIRSCHBERG, Thorsten, A. , LEE, Christopher, P. , LIN, Kuei-Ying , MACKMAN, Richard, L. , NELSON, Peter, H. , OARE, David , PYUN, Hyung-Jung , RAY, Adrian, S. , SHERLOCK, Rosemarie , SWAMINATHAN, Sundaramoorthi , WATKINS, Will , ZHANG, Jennifer R. , MILLER, Gerard, D.
IPC分类号： A61K31/662
CPC分类号： A61K31/662 , A61K47/548 , C07D205/04 , C07D211/58 , C07D409/06 , C07D409/14 , C07D413/14 , C07D475/00 , C07D487/04 , C07F9/4075 , C07F9/5728 , C07F9/582 , C07F9/588 , C07F9/60 , C07F9/65037 , C07F9/650941 , C07F9/653 , C07F9/6539 , C07F9/65515 , C07F9/655354 , C07F9/6561 , C07F9/65616
摘要： The invention is related to phosphorus substituted anti-inflammatory compounds, compositions containing such compounds, and therapeutic methods that include the administration of such compounds, as well as to processes and intermediates useful for preparing such compounds.
摘要翻译： 本发明涉及磷取代的抗炎化合物，含有这些化合物的组合物，以及包括给予这些化合物的治疗方法，以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：EP4267587A2
公开(公告)日：2023-11-01
申请号：EP21848379.0
申请日：2021-12-21
发明人： BYUN, Daniel H. , CANALES, Eda Y. , DEBIEN, Laurent P. , JANSA, Petr , LEE, Rick A. , LOYER-DREW, Jennifer A. , PERREAULT, Stephane , PYUN, Hyung-Jung , SAITO, Roland D. , SANGI, Michael S. , SCHRIER, Adam J. , SHATSKIKH, Marina E. , TAYLOR, James G. , TREIBERG, Jennifer A. , VAN VELDHUIZEN, Joshua J. , XU, Lianhong
IPC分类号： C07D519/00 , A61P35/02 , A61K31/437
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