-
公开(公告)号：EP3303341B1
公开(公告)日：2020-11-18
申请号：EP16800524.7
申请日：2016-05-20
发明人： YU, Tao , GRAHAM, Thomas, H. , WADDELL, Sherman, T. , MCCAULEY, John, A. , STAMFORD, Andrew, W. , SANDERS, John, M. , HU, Lihong , CAI, Jiaqiang , ZHAO, Lianyun
IPC分类号： C07D487/04 , A61K31/4188 , A61K31/53
-
公开(公告)号：EP2608668B1
公开(公告)日：2016-06-01
申请号：EP11820437.9
申请日：2011-08-22
发明人： MENG, Zhaoyang , REDDY, Panduranga Adulla, P. , SIDDIQUI, M. Arshad , MANDAL, Amit, K. , LIU, Duan , ZHAO, Lianyun , MCRINER, Andrew
IPC分类号： C07D471/14 , C07D519/00 , A61K31/4375 , A61P35/00
CPC分类号： C07D471/14 , C07D498/08 , C07D519/00
-
公开(公告)号：EP2770995B1
公开(公告)日：2019-01-02
申请号：EP12843015.4
申请日：2012-10-26
发明人： LAYTON, Mark, E. , PERO, Joseph, E. , FIJI, Hannah , KELLY, Michael, J., III , DE LEON, Pablo , ROSSI, Michael, A. , GILBERT, Kevin, F. , ROECKER, Anthony, J. , ZHAO, Zhijian , MERCER, Swati Pal , WOLKENBERG, Scott , MULHEARN, James , ZHAO, Lianyun , LI, Dansu
IPC分类号： C07D417/14 , C07D417/12 , C07D451/02 , C07D471/04 , C07D493/10 , C07D491/107 , A61K31/423 , A61P29/00 , A61K31/433 , A61K31/427 , A61K31/55 , A61K31/437 , A61K31/4725 , A61K31/4709
-
公开(公告)号：EP2132178B1
公开(公告)日：2015-08-19
申请号：EP07863005.0
申请日：2007-12-17
发明人： BELANGER, David, B. , SIDDIQUI, M. Arshad , CURRAN, Patrick J. , HAMANN, Blake , ZHAO, Lianyun , REDDY, Panduranga, Adulla, P. , TADIKONDA, Praveen, K. , SHIPPS, Gerald W., Jr. , MANSOOR, Umar, Faruk
IPC分类号： C07D213/81 , C07D401/04 , C07D401/12 , C07D401/14 , C07D405/04 , C07D405/12 , C07D409/04 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14 , C07D471/04 , C07D487/04 , A61K31/44 , A61P29/00
CPC分类号： C07D417/12 , C07D213/81 , C07D401/04 , C07D401/12 , C07D401/14 , C07D405/04 , C07D405/12 , C07D409/04 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/14 , C07D471/04 , C07D487/04
-
公开(公告)号：EP2178861B1
公开(公告)日：2014-08-20
申请号：EP08794560.6
申请日：2008-07-17
发明人： REDDY, Panduranga, Adulla, P. , ZHAO, Lianyun , TADIKONDA, Praveen, K. , WONG, Tzu, Tshin , TANG, Shuyi , TORRES, Luis, E. , CAUBLE, David, F., Jr. , GUZI, Timothy, J. , SIDDIQUI, M. Arshad
IPC分类号： C07D401/14 , C07D413/14 , C07D417/14 , C07D471/04
CPC分类号： C07D401/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D487/04
-
6.发明公开
公开(公告)号：EP3303341A1
公开(公告)日：2018-04-11
申请号：EP16800524.7
申请日：2016-05-20
发明人： YU, Tao , GRAHAM, Thomas, H. , WADDELL, Sherman, T. , MCCAULEY, John, A. , STAMFORD, Andrew, W. , SANDERS, John, M. , HU, Lihong , CAI, Jiaqiang , ZHAO, Lianyun
IPC分类号： C07D487/04 , A61K31/4188 , A61K31/53
CPC分类号： C07D491/147 , A61K31/427 , A61K31/4355 , A61K31/437 , A61K31/4375 , A61K31/4402 , A61K31/505 , A61K31/513 , A61K31/52 , A61K31/635 , A61K31/675 , A61P31/18 , C07D471/14 , A61K2300/00
摘要： The present invention relates to Fused Tricyclic Heterocycle Derivatives of Formula (I): and pharmaceutically acceptable salts thereof, wherein A, B, X, Y, m, R1, R2, R3, R3, R3, R4, R5 and R9 are as defined herein. The present invention also relates to compositions comprising at least one Fused Tricyclic Heterocycle Derivative, and methods of using the Fused Tricyclic Heterocycle Derivatives for treating or preventing HIV infection in a subject.
-
公开(公告)号：EP1931657B1
公开(公告)日：2013-12-25
申请号：EP06801601.3
申请日：2006-08-16
发明人： DENG, Yongqi , CURRAN, Patrick, J. , SHIPPS, Gerald W., Jr. , ZHAO, Lianyun , SIDDIQUI, M. Arshad , POPOVICI-MULLER, Janeta , DUCA, Jose, S. , HRUZA, Alan, W. , FISCHMANN, Thierry, O. , MADISON, Vincent, S. , ZHANG, Rumin , MCNEMAR, Charles, Wayne , MAYHOOD, Todd, W. , WINDSOR, William, T. , LEES, Emma, M. , PARRY, David, A.
IPC分类号： C07D409/04 , C07D215/50 , C07D215/42 , C07D401/12 , C07D401/10 , C07D405/04 , C07D215/48 , C07D413/12 , C07D417/10 , C07D401/06 , C07D409/12 , C07D409/14 , C07D417/04 , C07D417/06 , C07D401/14
CPC分类号： C07D409/04 , C07D215/42 , C07D215/48 , C07D215/50 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/04 , C07D409/12 , C07D409/14 , C07D413/12 , C07D417/04 , C07D417/06 , C07D417/10
-
公开(公告)号：EP2525659A1
公开(公告)日：2012-11-28
申请号：EP11735040.5
申请日：2011-01-18
发明人： SIDDIQUI, M. Arshad , NAN, Yang , PATEL, Mehul, F. , REDDY, Panduranga Adulla P. , MANSOOR, Umar Faruk , MENG, Zhaoyang , VITHARANA, Lalanthi Dilrukshi , ZHAO, Lianyun , MANDAL, Amit, K. , LIU, Duan , TANG, Shuyi , MCRINER, Andrew , BELANGER, David, B. , CURRAN, Patrick, J. , DAI, Chaoyang , ANGELES, Angie, R. , YANG, Liping , DANIELS, Matthew Hersh
IPC分类号： A01N43/90
CPC分类号： C07D471/08 , C07D487/04 , C07D487/08 , C07D491/147 , C07D498/08 , C07D513/08 , C07D519/00
摘要： The present invention provides Pyrazolopyrimidine Compounds of Formula (I): wherein L, T, Z, U, V, W, R3, R6, R7, R8, and m are as defined herein, and pharmaceutically acceptable salts of such Pyrazolopyrimidine Compounds. The Pyrazolopyrimidine Compounds are useful in the treatment of cancer and other diseases or disorders wherein mTOR is deregulated.
-
公开(公告)号：EP4013742A1
公开(公告)日：2022-06-22
申请号：EP20852190.6
申请日：2020-07-21
申请人： Merck Sharp & Dohme Corp. , THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH , MSD R&D (China) Co., Ltd.
发明人： MCCAULEY, John A. , COWMAN, Alan F. , DE LERA RUIZ, Manuel , FAVUZZA, Paola , GUO, Zhuyan , HU, Bin , KELLY III, Michael J. , LEI, Zhiyu , OLSEN, David B. , SLEEBS, Brad , THOMPSON, Jennifer K. , TRIGLIA, Tony , ZHAN, Dongmei , ZHANG, Cailing , ZHAO, Lianyun
IPC分类号： C07D239/22 , C07D405/04 , C07D405/14 , A61K31/513 , A61P33/06
-
公开(公告)号：EP2525659B1
公开(公告)日：2019-02-27
申请号：EP11735040.5
申请日：2011-01-18
发明人： SIDDIQUI, M. Arshad , NAN, Yang , PATEL, Mehul, F. , REDDY, Panduranga Adulla P. , MANSOOR, Umar Faruk , MENG, Zhaoyang , VITHARANA, Lalanthi Dilrukshi , ZHAO, Lianyun , MANDAL, Amit, K. , LIU, Duan , TANG, Shuyi , MCRINER, Andrew , BELANGER, David, B. , CURRAN, Patrick, J. , DAI, Chaoyang , ANGELES, Angie, R. , YANG, Liping , DANIELS, Matthew Hersh
IPC分类号： A01N43/90
-
-
-
-
-
-
-
-
-
搜索结果
19 条记录 (耗时 0.029 秒)
