公开(公告)号：EP4458808A1

公开(公告)日：2024-11-06

申请号：EP22916031.2

申请日：2022-12-26

Applicant: ADEKA CORPORATION ,  Nihon Nohyaku Co., Ltd.

Inventor： HARA, Kenji ,  SUGIHARA, Kousuke ,  MASUDA, Tsuyoshi ,  FUJII, Kazuki ,  FUKATSU, Kosuke

IPC: C07C235/82 ,  A01N37/22 ,  A01N37/24 ,  A01N43/16 ,  A01N43/30 ,  A01N43/40 ,  A01N43/56 ,  A01N47/02 ,  A01N47/16 ,  A01P5/00 ,  A01P7/04 ,  A61K31/167 ,  A61K31/357 ,  A61K31/44 ,  A61P33/14 ,  C07C317/40 ,  C07C323/40 ,  C07C327/48 ,  C07D213/81 ,  C07D317/66

Abstract: In the production of crops in agriculture, horticulture and the like, the damage caused by insect pests and the like is still large, and the development of a novel pest control agent is desired in view of the factors such as the development of insect pests that are resistant to existing drugs, and the like.
The present invention provides compounds represented by the formula (1)

wherein X and Y are oxygen atoms or sulfur atoms, Z is a hydroxyl group or the like, R 1 and R 2 are alkyl groups and the like, R 4 and R 5 are .alkyl groups and the like, R 3 and R 6 are hydrogen atoms and the like, R 7 is a substituted phenyl group or the like, and Q is an aryl group or the like, or salts thereof, pest control agents containing the compounds as active ingredients, and methods for use thereof.

公开(公告)号：EP4098650A1

公开(公告)日：2022-12-07

申请号：EP21748308.0

申请日：2021-01-29

Applicant: Kumiai Chemical Industry Co., Ltd.

Inventor： TANAKA, Kosuke ,  SAKURAI, Sakae ,  ENOMOTO, Yukihiro ,  TORIYABE, Keiji ,  ARAI, Hirokazu ,  NAKANE, Yuhsuke ,  MATSUDA, Takeshi ,  TAKANEZAWA, Akira ,  KOIKE, Shusuke ,  KITAHARA, Shunsuke ,  MUKAWA, Shigeyuki

IPC: C07C235/46 ,  C07C271/16 ,  C07C311/09 ,  C07C317/18 ,  C07C323/12 ,  C07C323/17 ,  C07C327/48 ,  C07C333/04 ,  A01N37/18 ,  A01P5/00 ,  A01P7/02 ,  A01P7/04 ,  C07F7/12

Abstract: The present invention provides: a 3-alkoxybenzoic acid amide derivative having an excellent pest control effect, or a salt thereof; and a pest control agent and a production intermediate which contain the same as an active ingredient.
Provided are: a 3-alkoxybenzoic acid amide derivative represented by general formula [I]

[In the formula, A represents an oxygen atom or a sulfur atom, G represents a hydrogen atom, a halogen atom, or a C 1 -C 6 alkyl group, R 1 represents a C 1 -C 6 alkyl group, a C 3 -C 6 cycloalkyl group, etc., R 2 represents a hydrogen atom, etc., R 3 represents a halogen atom, C 1 -C 6 alkyl group, etc., R 4 represents a halogen atom, C 1 -C 6 alkyl group, etc., and R 5 represents a C 1 -C 12 alkyl group, etc.], or a salt thereof; and a pest control agent characterized by containing said derivative or salt thereof as an active ingredient.

公开(公告)号：EP2551258B1

公开(公告)日：2018-10-31

申请号：EP11758781.6

申请日：2011-03-21

Applicant: Shenyang Sinochem Agrochemicals R & D Co., Ltd.

Inventor： LIU, Changling ,  LI, Huichao ,  LI, Zhinian ,  HUANG, Guang ,  ZHANG, Hong

IPC: C07C211/56 ,  C07C237/30 ,  C07C237/40 ,  C07C327/48 ,  C07C255/58 ,  C07C317/36 ,  C07C323/36 ,  C07D213/643 ,  C07D213/70 ,  A01N33/18 ,  A01N33/22 ,  A01N37/34 ,  A01N37/44 ,  A01N41/10 ,  A01N43/40

CPC classification number: C07C211/56 ,  A01N33/18 ,  A01N33/22 ,  A01N37/34 ,  A01N37/44 ,  A01N41/10 ,  A01N43/40 ,  C07C237/30 ,  C07C237/40 ,  C07C255/58 ,  C07C317/36 ,  C07C323/36 ,  C07C327/48 ,  C07D213/643 ,  C07D213/70

Abstract: Substituted diphenylamine compounds of general formula I are provided, in which each substituted group is defined as in the description. The compounds of general formula I have broad-spectrum fungicidal activity in the field of agriculture. Furthermore, the preparation methods of the above compounds are simple.

公开(公告)号：EP2493851A2

公开(公告)日：2012-09-05

申请号：EP10773861.9

申请日：2010-11-02

Applicant: Leibniz-Institut für Naturstoff-Forschung und Infektionsbiologie

Inventor： BEHNKEN, Swantje ,  DAHSE, Hans-Martin ,  HERTWECK, Christian ,  ISHIDA, Keishi ,  LINCKE, Thorger ,  ROTH, Martin ,  KLOSS, Florian

IPC: C07C327/48 ,  A61K31/165 ,  A61P31/04 ,  A61P31/10 ,  A61P35/00

CPC classification number: C07C327/48

Abstract: This invention relates to the field of biologically active compounds and specifically to closthioamides, pharmaceutical compositions comprising these compounds, and their use as antibiotic, antifungal, and/or cytotoxic agent.

Abstract translation: 本发明涉及生物活性化合物领域，具体涉及其中B A和E如本文所定义的式（I）的硫代酰胺，包含这些化合物的药物组合物，以及它们作为抗生素，抗真菌剂和/或细胞毒性剂的用途。

公开(公告)号：EP1940787A4

公开(公告)日：2009-07-01

申请号：EP06844228

申请日：2006-10-27

Applicant: LANKENAU INST MEDICAL RES

Inventor： DUHADAWAY JAMES B ,  PRENDERGAST GEORGE C ,  MALACHOWSKI WILLIAM P ,  MULLER ALEXANDER J

IPC: C07D209/14 ,  A61K31/27 ,  A61P31/12 ,  A61P35/00 ,  C07C327/48 ,  C07C333/20 ,  C07C333/22 ,  C07D401/12 ,  C07D417/06

CPC classification number: C07D209/10 ,  C07C333/20 ,  C07C333/22 ,  C07C2602/08 ,  C07C2603/74 ,  C07D333/54 ,  C07D401/12 ,  C07D417/06

公开(公告)号：EP1803706A1

公开(公告)日：2007-07-04

申请号：EP07008232.6

申请日：2002-02-12

Applicant: Ambrilia Biopharma Inc.

Inventor： Stranix, Brent Richard ,  Sauve, Gilles ,  Bouzide, Abderrahim ,  Côté, Alexandre ,  Berube, Gervais ,  Soucy, Patrick ,  Zhao, Yongsen ,  Yelle, Jocelyn

IPC: C07C311/19 ,  C07D209/16 ,  C07C311/46 ,  C07D333/34 ,  C07D333/60 ,  C07C311/42 ,  C07D295/215 ,  C07C327/48 ,  C07D409/12 ,  A61K31/198 ,  A61K31/405 ,  A61K31/381 ,  A61K31/5375 ,  A61P31/18 ,  C07D333/00 ,  C07D209/00

CPC classification number: C07D295/185 ,  A61K38/00 ,  C07C311/19 ,  C07C311/42 ,  C07C311/46 ,  C07C323/60 ,  C07C327/44 ,  C07C327/48 ,  C07C2601/08 ,  C07D209/16 ,  C07D333/34 ,  C07D333/60 ,  C07K5/0215

Abstract: The present application refers to a compound selected from the group consisting of a compound of formula I

wherein the compounds No. 1 to 10, respectively, are defined as follows


The compounds are useful in the treatment of HIV and HTLV infections.

Abstract translation: 本申请是指选自式I化合物的化合物，其中化合物1至10分别定义如下。该化合物可用于治疗HIV和HTLV感染。

公开(公告)号：EP1661886A1

公开(公告)日：2006-05-31

申请号：EP04772372.1

申请日：2004-08-23

Applicant: Mitsui Chemicals, Inc.

Inventor： YOSHIDA, Kei ,  WAKITA, Takeo ,  KATSUTA, Hiroyuki ,  KAI, Akiyoshi ,  CHIBA, Yutaka ,  TAKAHASHI, Kiyoshi ,  KATO, Hiroko ,  KAWAHARA, Nobuyuki ,  NOMURA, Michikazu ,  DAIDO, Hidenori ,  MAKI, Junji ,  BANBA, Shinichi ,  KAWAHARA, Atsuko

IPC: C07C271/28 ,  C07C327/48 ,  C07C333/08 ,  C07D213/81 ,  A01N47/20

CPC classification number: A01N47/20 ,  C07C211/47 ,  C07C211/48 ,  C07C215/68 ,  C07C237/40 ,  C07C265/12 ,  C07C271/28 ,  C07C317/18 ,  C07C317/36 ,  C07C317/40 ,  C07C323/12 ,  C07C323/36 ,  C07C323/42 ,  C07C327/48 ,  C07C333/08 ,  C07C2601/04 ,  C07C2601/08 ,  C07D213/81

Abstract: An object of the present invention is to provide insecticides having high effectiveness. The present invention provides compounds represented by formula (1):

wherein A 1 , A 2 , A 3 , and A 4 independently represent a carbon atom, a nitrogen atom, or an oxidized nitrogen atom; R 1 represents a C1-C6 alkyl group which may be substituted, a phenyl group which may be substituted, or a heterocyclic group which may be substituted; R 2 and R 3 independently represent a hydrogen atom, a C1-C4 alkyl group which may be substituted, or a C1-C4 alkylcarbonyl group which may be substituted; G 1 , G 2 , and G 3 independently represent an oxygen atom or a sulfur atom; Xs may be the same or different and each represent a hydrogen atom, a halogen atom, a C1-C4 alkyl group which may be substituted, or an amino group which may be substituted; n represents an integer of 0 to 4; Q represents a phenyl group which may be substituted, a naphthyl group which may be substituted, a tetrahydronaphthyl group which may be substituted, or a heterocyclic group which may be substituted, insecticides containing the compounds as active ingredients, and a method for producing the compounds.
The compounds represented by formula (1) exhibit an excellent preventive effect as insecticides and also exhibit an excellent preventive effect when being combined with another insecticide, an acaricide, a nematocide, a fungicide, a herbicide, a plant growth regulator, or a biological pesticide.

Abstract translation: 本发明的一个目的是提供具有高效力的杀虫剂。 本发明提供由式（1）表示：其中A 1，A 2，A 3，和A 4独立地表示碳原子，氮原子，或氧化的氮原子; R 1表示可以被取代的，可被取代的苯基，或可被取代的杂环基团的C1-C6烷基; R 2和R 3独立地表示氢原子，可被取代的C1-C4烷基，或可被取代的C1-C4烷基羰基; G 1，G 2，和G 3各自独立地表示在氧原子或硫原子; X可以相同或不同，并且各自表示氢原子，卤原子，其可以是substituiertem，或到的氨基可以是substituiertem基的C1-C4烷基; Ñdarstellt为0至4的整数; Q darstellt哪个可以是substituiertem苯基，其可以是substituiertem萘基，其可以是substituiertem四氢萘基，或可被substituiertem，杀虫剂含有该化合物作为活性成分的杂环基，和一种用于制造所述化合物 ， 由式表示的化合物（1）显示出优良的预防效果作为杀虫剂和当与其它杀虫剂到杀螨剂，杀线虫剂一个，杀真菌剂，除草剂，植物生长调节剂，或生物农药被组合从而表现出优异的预防效果 ，

公开(公告)号：EP1154993B1

公开(公告)日：2004-10-06

申请号：EP00903680.7

申请日：2000-02-10

Applicant: F. HOFFMANN-LA ROCHE AG

Inventor： HULL, Kenneth, Gregory ,  SIDDURI, Achytharao ,  TILLEY, Jefferson, Wright

IPC: C07C327/46 ,  C07C327/48 ,  C07D401/06 ,  C07D213/82 ,  C07D231/08 ,  A61K31/44 ,  A61K31/167 ,  A61P29/00

CPC classification number: C07D213/82 ,  C07C327/46 ,  C07C327/48 ,  C07C2601/04 ,  C07C2601/08 ,  C07D213/56 ,  C07D233/38 ,  C07D239/28 ,  C07D401/06

Abstract: Compounds of formula (1): and the pharmaceutically acceptable salts and esters thereof wherein X and Y are as defined in the specification, inhibit the binding of VCAM-1 to VLA-4 and are useful in treating inflammation associated with chronic inflammatory diseases such as rheumatoid arthritis (RA), multiple sclerosis (MS), asthma, and inflammatory bowel disease (I/BD).

公开(公告)号：EP0866056A4

公开(公告)日：2000-05-24

申请号：EP96935419

申请日：1996-10-24

Applicant: UBE INDUSTRIES

Inventor： FUJII KATSUTOSHI ,  HATANO KOJI ,  SHIKITA SHOJI ,  TANAKA TATSUMI

IPC: A01N37/20 ,  A01N37/40 ,  A01N37/48 ,  A01N39/00 ,  C07C233/69 ,  C07C235/48 ,  C07C235/58 ,  C07C255/57 ,  C07C327/48 ,  A01N37/24 ,  A01N37/34 ,  C07C213/02 ,  C07C217/20 ,  C07C231/02

CPC classification number: C07C327/48 ,  A01N37/20 ,  A01N37/40 ,  A01N37/48 ,  A01N39/00 ,  C07C233/69 ,  C07C235/48 ,  C07C235/58 ,  C07C255/57 ,  Y10S424/10

Abstract: N-[(Fluoroalkoxy)phenoxyalkyl]benzamide compounds represented by general formula (1); and agricultural and horticultural pesticides containing these compounds as the active ingredient which are useful as a nematicide, miticide, insecticide, etc., wherein R and R may be either the same or different and each represents hydrogen, halogeno, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl, C1-4 haloalkoxy, cyano, nitro or hydroxy; R represents hydrogen, halogeno, C1-4 alkyl or C1-4 alkoxy; A represents oxygen or sulfur; x is an integer of from 1 to 4; y is an integer of from 0 to 6; z is an integer of from 2 to 9; and m is an integer of from 0 to 2, provided that 2x + 1 = y + z + m.

Abstract translation: 本发明公开了A N A（氟烷氧基）phenoxyalkylÜbenzamide化合物由式（1）表示： worin - [R <1>和R <3>可以相同或不同，表示氢原子，卤原子，C1 -4烷基，C1-4烷氧基，C 1-4卤代烷基，C 1-4卤代烷氧基，氰基，硝基，或羟基; [R <2>代表氢原子，卤原子，C 1-4烷基，或C 1-4烷氧基; 氧原子，或硫原子的darstellt; n为1至6的整数; x是1至4; y为0至6; z为2至9; m是0至2; 提供确实2X + 1 = Y + Z + M，在中间物，防治有害生物含有上述化合物作为有效成分的所有其可作为一个杀线虫剂，在杀螨剂，杀真菌剂处理它们和的农业和园艺化学 等等。

公开(公告)号：EP0792873A1

公开(公告)日：1997-09-03

申请号：EP97301151.3

申请日：1997-02-21

Applicant: American Cyanamid Company

Inventor： Tomcufcik, Andrew Stephen ,  Hinson, Joseph William

IPC: C07D239/26 ,  A61K31/415 ,  C07D257/04 ,  C07C327/48 ,  C07D277/24 ,  C07C311/08 ,  C07C317/40 ,  C07D207/32 ,  C07D417/12 ,  C07F9/24

CPC classification number: C07D207/333 ,  C07C311/17 ,  C07C317/34 ,  C07C323/49 ,  C07C327/48 ,  C07C327/52 ,  C07D207/325 ,  C07D231/12 ,  C07D233/56 ,  C07D239/26 ,  C07D249/08 ,  C07D257/04 ,  C07D277/24 ,  C07D417/12

Abstract: The present invention relates to substituted ω-[phenoxy, phenylthio, phenylsulfinyl, phenylsulfonyl] [alkyl, alkenyl or alkynyl]amine carboxamides, sulfonamides and phosphonylamides which are useful as antiarrhythmic agents.

Abstract translation: 本发明涉及可用作抗心律不齐剂的取代的ω-苯氧基，苯硫基，苯基亚磺酰基，苯基磺酰基，烷基，烯基或炔基胺胺，酰胺和膦酰基酰胺。