COMPOUND CONTAINING DIPHENYLMETHANE STRUCTURE AND USE THEREOF

    公开(公告)号:EP3901132A1

    公开(公告)日:2021-10-27

    申请号:EP19909448.3

    申请日:2019-12-13

    Abstract: Disclosed are a compound containing a diphenylmethane structure and a use thereof, belonging to the technical field of compound and polypeptide synthesis. The structure of the compound containing a diphenylmethane structure of the present invention is represented by General Formula (1). The compound containing a diphenylmethane structure of the present invention contains a hydroxyl group, an amino group, a substituted amino group, and an active group, and can be used as an amino acid or peptide C-terminal protection reagent. A peptide synthesis reaction using this protection carrier has a fast reaction speed and a high reagent utilization rate in a suitable solvent system; post-treatment is carried out by means of simple liquid-liquid extraction separation, i.e. effective purification can be carried out, and finally, a product with a high purity can be obtained; and during a synthesis process, the change in solubility is small and an operation process has a strong universality, and therefore, the present method can be developed into a universal production method.

    AMIDE COMPOUND AND USE THEREOF FOR CONTROLLING PLANT DISEASES
    5.
    发明公开
    AMIDE COMPOUND AND USE THEREOF FOR CONTROLLING PLANT DISEASES 审中-公开
    酰胺化合物及其用于控制​​植物病害的用途

    公开(公告)号:EP2154124A1

    公开(公告)日:2010-02-17

    申请号:EP08752106.8

    申请日:2008-04-25

    Abstract: Disclosed is an amide compound represented by the formula (1) below, which has excellent plant disease controlling activity.

    In the formula, X 1 represents a fluorine atom or a methoxy group; X 2 represents a hydrogen atom, a halogen atom, a C 1 -C 4 alkyl group or the like; X 3 represents a halogen atom, a C 1 -C 4 alkyl group or the like; Z represents an oxygen atom or a sulfur atom; and A represents an A 1 -CR 11 R 12 R 13 group, an A 2 -Cy 1 group or an A 3 -Cy 2 group, wherein A 1 represents a CH 2 group or the like, A 2 represents a single bond, a CH 2 group or the like, A 3 represents a C 1 -C 3 haloalkyl group, a C 2 -C 4 alkenyl group or the like, Cy 1 represents a C 3 -C 6 cycloalkyl group substituted with a C 1 -C 6 alkoky group or the like, Cy 2 represents a C 3 -C 6 cycloalkyl group which may be substituted with a halogen atom or the like, R 11 and R 12 independently represent a C 1 -C 4 alkyl group, and R 13 represents a halogen atom, a hydroxyl group or the like.

    Abstract translation: 公开了具有优异的植物病害防治活性的由下式(1)表示的酰胺化合物。 在该式中,X1表示氟原子或甲氧基; X2表示氢原子,卤素原子,C1-C4烷基等; X 3表示卤原子,C 1 -C 4烷基等; Z代表氧原子或硫原子; A表示A1-CR11R12R13基,A2-Cy1基或A3-Cy2基,其中A1表示CH2基等,A2表示单键,CH2基等,A3表示C1-C3 卤代烷基,C2-C4烯基等,Cy1表示被C1-C6烷基等取代的C3-C6环烷基,Cy2表示可以被卤素原子取代的C3-C6环烷基或 例如,R 11和R 12独立地表示C 1 -C 4烷基,并且R 13表示卤素原子,羟基等。

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