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    Novel ' ' 9'- gonene-11-ones
    1.
    发明授权
    Novel ' ' 9'- gonene-11-ones 失效
    NOVEL''9'- GONENE-11-ONES

    公开(公告)号：US3876637A

    公开(公告)日：1975-04-08

    申请号：US43076974

    申请日：1974-01-04

    Applicant: ROUSSEL UCLAF

    Inventor： COUSSEDIERE DANIEL ,  NEDELEC LUCIEN ,  TORELLI VESPERTO

    IPC: C07J21/00 ,  C07D20060101 ,  C07J1/00 ,  C07J15/00 ,  C07C173/00

    Abstract: Wherein R is alkyl of 1 to 3 carbon atoms, R.sub.1 is selected from the group consisting of =0, ketals and
    R.sub.2 is selected from the group consisting of hydrogen and acyl of an organic carboxylic acid of 1 to 12 carbon atoms and X is selected from the group consisting of hydrogen and hydroxy which are valuable intermediates for the preparation of steroids such as adrenosterone.

    Racemates and optically active isomers of novel .DELTA..sup.9 gonene-11-ones of the formula

    Novel 11beta,18-epoxy steroids
    4.
    发明授权
    Novel 11beta,18-epoxy steroids 失效
    NOET 11BETA，18-EPOXY STEROIDS

    公开(公告)号：US3699100A

    公开(公告)日：1972-10-17

    申请号：US3699100D

    申请日：1971-02-03

    Applicant: ROUSSEL UCLAF

    Inventor： NEDELEC LUCIEN ,  GASC JEAN-CLAUDE

    IPC: A61K31/58 ,  C07J71/00 ,  C07C173/00

    CPC classification number: C07J75/00

    Abstract: NOVEL 11B,18-EPOXY-$4.9-ESTRADIENES OF THE FORMULA

    3-(O=),11,18-(-O-),17-R,17-(R''-O-)ESTRA-4,9-DIENE

    WHEREIN R IS SELECTED FROM THE GROUPS CONSISTING OF HYDROGEN AND ETHYNYL AND R'' IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, ACYL OF AN ORGANIC CARBOXYLIC ACID OF 1 TO 18 CARBON ATOMS, LOWER ALIPHATIC, ARALYALIPHATIC AND HETEROCYCLIC WHICH HAVE ANIT-ANDROGENIC ACTIVITY, THEIR PREPARATION AND INTERMEDIATES THEREFROM.

    Preparation of 7{60 -methyl steroids
    6.
    发明授权
    Preparation of 7{60 -methyl steroids 失效
    制备7种{6-甲基异烟肼

    公开(公告)号：US3697556A

    公开(公告)日：1972-10-10

    申请号：US3697556D

    申请日：1970-07-27

    Applicant: ROUSSEL UCLAF

    Inventor： BOUCOURT ROBERT ,  NEDELEC LUCIEN ,  GASC JEAN-CLAUDE

    IPC: A61K31/565 ,  B65H31/10 ,  C07J1/00 ,  C07J75/00 ,  C07C169/22

    CPC classification number: A61K31/565 ,  B65H31/10 ,  C07J1/00 ,  C07J75/00

    Abstract: WHEREIN R is alkyl of one to four carbon atoms and R'' is selected from the group consisting of hydrogen, acyl of an organic carboxylic acid of one to 18 carbon atoms and an organic ether radical, a novel process for preparing the corresponding Delta 4,9,11-gonatrienes and novel intermediates produced by the said processes.

    A novel process for the preparation of 7 Alpha -methyl- Delta 4,9-gonadienes of the formula

    Abstract translation: 用于制备式WHEREIN R的7个α-甲基-TATA 4,9-基那烯的新方法是1至4个碳原子的烷基，R'选自氢，有机羧酸的酰基， 1至18个碳原子和有机醚基团，一种制备相应的DELTA 4,9,11-三烯的新方法和由所述方法制备的新型中间体。

    Novel 7{60 -methyl-{66 {11 {11 {11 {11 -gonadienes
    7.
    发明授权
    Novel 7{60 -methyl-{66 {11 {11 {11 {11 -gonadienes 失效
    第7号{60 -METHYL- {66 {11 {11}

    公开(公告)号：US3679718A

    公开(公告)日：1972-07-25

    申请号：US3679718D

    申请日：1970-07-27

    Applicant: ROUSSEL UCLAF

    Inventor： BUCOURT ROBERT ,  NEDELEC LUCIEN ,  GASC JEAN-CLAUDE

    IPC: A61K31/565 ,  C07J1/00 ,  C07C169/22

    CPC classification number: A61K31/565 ,  C07J1/00 ,  Y10S514/925

    Abstract: Novel 7 Alpha -methyl- Delta 4,11-gonadiene of the formula

    WHEREIN R is alkyl of one to four carbon atoms and R'' is selected from the group consisting of hydrogen, acyl of an organic carboxylic acid of one to 18 carbon atoms and an organic ether radical which have anabolic and androgenic activities and their preparation.

    Abstract translation: 具有式IV的新型7α-甲基-TATA 4,11-二氢二环，其中R是具有1至4个碳原子的烷基，R'选自氢，1至18个碳原子的有机羧酸的酰基和 具有合成代谢和雄激素活性及其制备的有机醚基团。

    2-oxa-steroid and the production thereof
    8.
    发明授权
    2-oxa-steroid and the production thereof 失效
    2-OXA-STEROID及其生产

    公开(公告)号：US3595877A

    公开(公告)日：1971-07-27

    申请号：US3595877D

    申请日：1968-08-14

    Applicant: ROUSSEL UCLAF

    Inventor： BUCOURT ROBERT ,  NEDELEC LUCIEN

    IPC: C07D295/096 ,  C07D295/116 ,  C07J73/00 ,  C07D7/20

    CPC classification number: C07D295/096 ,  C07C2603/16 ,  C07D295/116 ,  C07J73/003

    Abstract: 2-OXA-13B-R-17A-METHYL-$4,9,11-GONATRIENES OF THE FORMULA

    13-R,16-(R''-O-),16-(CH3-)-2-OXA-GONA-4,9,11-TRIENE

    WHEREIN R IS SELECTED FROM THE GROUP CONSISTING OF METHYL AND ETHYL AND R'' IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, SATRUATED ALKYL OF 1 TO 5 CARBON ATOMS WHICH MAY CONTAIN A HETERO OXYGEN ATOM, UNSATURATED ALKYL OF 2 TO 5 CARBON ATOMS, CYCLOALKYL OF 3 TO 5 CARBON ATOMS WHICH MAY CONTAIN A HETERO OXYGEN ATOM, WITH THE PROVISO THAT R IS ETHYL WHEN R'' IS HYDROGEN WHCIH COMPOUNDS POSSESS ANABLOIC AND ANDROGENIC ACTIVITY. THE INVENTION ALSO RELATES TO A NOVEL PROCESS AND NOVEL INTERMEDIATES FOR THE PREPARATION OF THE COMPOUNDS OF FORMULA I.

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