公开(公告)号：US20110319665A1

公开(公告)日：2011-12-29

申请号：US13254946

申请日：2010-03-08

申请人： Alexander Korte ,  Jan Klaas Lohmann ,  Thomas Grote ,  Klaus Ebel ,  Thomas Zierke ,  Horst Mayer ,  Ralf Wazulek

发明人： Alexander Korte ,  Jan Klaas Lohmann ,  Thomas Grote ,  Klaus Ebel ,  Thomas Zierke ,  Horst Mayer ,  Ralf Wazulek

IPC分类号： C07C205/06 ,  C07C211/52

CPC分类号： C07C205/11 ,  C07C205/09 ,  C07C205/10 ,  C07C2601/16

摘要： The present invention relates to a process for preparing substituted 2-nitrobiphenyls and to specific 2-nitrobiphenyls. The invention further relates to a process for preparing 2-aminobiphenyls from such 2-nitrobiphenyls and to a process for preparing (het)arylamides of such 2-aminobiphenyls.

摘要翻译： 本发明涉及制备取代的2-硝基联苯和特定2-硝基联苯的方法。 本发明还涉及从这种2-硝基联苯制备2-氨基联苯的方法和制备这种2-氨基联苯的（het）芳基酰胺的方法。

公开(公告)号：US07550471B2

公开(公告)日：2009-06-23

申请号：US10531981

申请日：2003-11-04

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A61K31/519 ,  C07D487/00

CPC分类号： C07D487/04

摘要： The invention relates to 5-alkyl-7-aminotriazolopyrimidines of the formula (I) and to the salts thereof. In said formula substituents have the following meanings: R1 and R2 each is a hydrogen atom or a group of alkyl, alcenyl, haloalkyl, cycloalky, phenyl or naphtyle, saturated, unstaturated or aromatic heterocycle having from five to six members which contain from one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can from together with a connecting them nitrogen atom a cycle of 5 to 6 members containing from one to four nitrogen atoms or from one to three nitrogen atoms and one sulfur or oxygen atom, R3 is a cycloalkyl or bicycloalkyl group, R1, R2 and R3 can be substituted in conformity with a description, and X is an alkyl or alkyl halide group. The inventive methods and intermediary products necessary for producing said compounds, agents containing them and the use therefore for fighting against harmful mushroom are also disclosed.

摘要翻译： 本发明涉及式（I）的5-烷基-7-氨基三唑并嘧啶及其盐。 在所述式中，取代基具有以下含义：R 1和R 2各自为氢原子或具有5至6个成员的烷基，烯基，卤代烷基，环烷基，苯基或萘杂，饱和的，不饱和的或芳族杂环的基团， 四个氮原子或一个至三个氮原子和一个硫或氧原子，或者R 1和R 2可以连同它们的氮原子一起包含5至6个含有1-4个氮原子或1-3个氮原子的成员 和一个硫或氧原子，R 3为环烷基或双环烷基，R 1，R 2和R 3可以根据说明书进行取代，X为烷基或卤代烷基。 还公开了生产所述化合物所需的创造性方法和中间产物，含有它们的试剂和用于防止有害蘑菇的用途。

公开(公告)号：US20080221177A1

公开(公告)日：2008-09-11

申请号：US12101175

申请日：2008-04-11

申请人： Wassilios GRAMMENOS ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Wassilios GRAMMENOS ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A01N43/40 ,  A01P3/00

CPC分类号： C04B35/632 ,  C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

摘要： Sulfonamides of the formula I where the substituents are as follows: R1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R2, R3, R4, R5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R2′ and R3′, R2′, R3′ are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R2, R3, R4 and R5 are hydrogen: X is phenyl substituted by a group C(R6)═NOR7, where R6 is alkyl and R7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R2, R3, R4 and R5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的磺酰胺，其中取代基如下：R 1是氢，烷基，烷氧基，烯基或炔基; R 2，R 3，R 4，R 5是氢，卤素，烷基，烷氧基或卤代甲基 ; R 2和R 3一起也可以形成苯基，环戊基或环己基环，这些环可以携带两个基团R 2， '和R 3'，R 2'，R 3'是氢，卤素，烷基，烷氧基或卤代甲基; 在a）情况下，如果R 2，R 3，R 4和R 5是氢：X是 被C（R 6） - - NOR 7取代的苯基，其中R 6是烷基，R 7是 烷基，苄基，烯基，卤代烷基，卤代烯基，炔基或卤代炔基; 并且在情况b）中，如果R 2，R 3，R 4和R 5中的至少一个， SUP>不是氢：X是苯基，萘基或五或六元饱和或部分不饱和或芳族杂环，其通过碳原子连接并含有一至四个由O，N和S组成的组的杂原子 ，其中X可以根据描述被替代; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080032889A1

公开(公告)日：2008-02-07

申请号：US11630558

申请日：2005-06-14

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A01C1/06 ,  C07D487/04

CPC分类号： A01N43/90 ,  C07D487/04

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, halocycloalkyl, alkenyl, cycloalkyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen, alkyl or one of the groups mentioned under R1; R1 and/or R2 may carry one to four identical or different groups Ra: Ra is chlorine, bromine, iodine, cyano, nitro, hydroxyl, alkyl, alkylcarbonyl, cycloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, alkylthio, alkylamino, dialkyl-amino, alkenyl, cycloalkenyl, alkenyloxy, haloalkenyloxy, alkynyl, halo-alkynyl, alkynyloxy, haloalkynyloxy, cycloalkoxy, cycloalkenyloxy, oxyalkylenoxy, naphthyl, a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, where these aliphatic, alicyclic or aromatic groups for their part may be substituted according to the description; and X is halogen; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义的式I的取代三唑并嘧啶：R 1是烷基，卤代环烷基，烯基，环烷基，环烯基，卤代环烯基，炔基，卤代炔基或萘基，或五或六元环， 包含一至四个由O，N和S组成的组的杂原子的2-元饱和的，部分不饱和的或芳族的杂环，R 2是氢，烷基或R 1上提到的基团之一， / SUP>; R 1和/或R 2可以携带一至四个相同或不同的基团R a是：R a是 氯，溴，碘，氰基，硝基，羟基，烷基，烷基羰基，环烷基，烷氧基，卤代烷氧基，烷氧基羰基，烷硫基，烷基氨基，二烷基氨基，烯基，环烯基，烯氧基，卤代烯氧基，炔基，卤代炔基，炔氧基，卤代炔氧基， 环烷氧基，环烯氧基，氧亚烷基氧基，萘基，五至十元饱和的部分不饱和或芳族杂环，其包含一至四个由O，N和S组成的组的杂原子，其中这些脂族，脂环族或芳族基团可以 根据描述进行替代; X为卤素; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080027085A1

公开(公告)日：2008-01-31

申请号：US11632342

申请日：2005-07-22

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hunger ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Ulrich Schofl ,  Harald Kohle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hunger ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Ulrich Schofl ,  Harald Kohle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

IPC分类号： A01N43/54 ,  A01P3/00 ,  C07D471/00

CPC分类号： C07D401/04

摘要： The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type, whereby: k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

公开(公告)号：US20070299115A1

公开(公告)日：2007-12-27

申请号：US11661679

申请日：2005-09-05

申请人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Shwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

发明人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Shwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

IPC分类号： A01N37/48 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01P3/00 ,  C07C233/00 ,  C07D213/82 ,  C07D231/14 ,  C07D277/56

CPC分类号： C07D213/82 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  C07D231/14 ,  C07D277/56

摘要： The invention relates to (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I) and to salts of said anilides that can be used for agricultural purposes for controlling pathogenic fungi. In said formula, the variables are defined as follows: A represents a phenyl or at least a monounsaturated 5- or 6-membered heterocycle comprising 1, 2 or 3 heteroatoms, selected from N, O, S, S(═O) and S(═O)2 as ring members, whereby phenyl and the monounsaturated 5- or 6-membered heterocycle can be unsubstituted or can be substituted according to the description; B represents a group of general formula (II), in which the variables R3, R4, R5 and the index m are defined as cited in the claims and the description; Y represents oxygen or sulphur, R1 represents H, OH, alkyl, cycloalkyl, alkoxy, haloalkyl, halocycloalkyl or haloalkoxy; R2 represents halogen, nitro, CN, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, haloalkyl, halocycloalkyl, haloalkenyl, haloalkynyl or haloalkoxy; and n represents 0, 1, 2, 3 or 4; and salts that can be used for agricultural purposes. The invention also relates to the use of the (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I), to a method for controlling pathogenic fungi and to a crop protection agent containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound.

摘要翻译： 本发明涉及通式（I）的（杂）环（硫代）羧酸酰苯胺和可用于农业目的的用于控制致病真菌的所述酰苯胺的盐。 在所述式中，变量定义如下：A表示苯基或至少一个单不饱和的5-或6-元杂环，其包含1,2或3个选自N，O，S，S（-O）和S （-O）2，作为环成员，由此苯基和单不饱和的5-或6-元杂环可以是未取代的或可以根据描述被取代; B表示通式（II）的基团，其中定义了变量R 3，R 4，R 5和指数m， 如权利要求和说明书所引用的; Y表示氧或硫，R 1表示H，OH，烷基，环烷基，烷氧基，卤代烷基，卤代环烷基或卤代烷氧基; R 2表示卤素，硝基，CN，烷基，环烷基，烯基，炔基，烷氧基，卤代烷基，卤代环烷基，卤代烯基，卤代炔基或卤代烷氧基。 并且n表示0,1,2,3或4; 和可用于农业目的的盐。 本发明还涉及通式（I）的（杂）环（硫代）羧酸二酰苯胺用于控制致病真菌的方法和含有至少一种通式（I）的化合物的作物保护剂， 和/或所述化合物的农业上相容的盐。

公开(公告)号：US07300908B2

公开(公告)日：2007-11-27

申请号：US10482216

申请日：2002-07-03

申请人： Bernd Müller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

发明人： Bernd Müller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/48

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n=0 or a whole number of 1-5; R=halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R1=alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R1 being able to be substituted according to the description; R2=alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi

摘要翻译： 式（I）的三唑并嘧啶，其中指数和取代基具有以下含义：n = 0或整数1-5; 环烷氧基，烷氧基羰基，链烯氧基羰基，烷氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰基，肟基烷基，链烯基肟基羰基，烷氧基羰基，烷氧基羰基， 烷基羰基，链烯基羰基，炔基羰基，环烷基羰基或五至十元饱和，部分不饱和或芳族杂环，含有一至四个O，N或S基团的杂原子; R 1 =烷基，烯基，炔基，环烷基，环烯基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环，其含有一至四个O，N或S ，R和/或R 1能够根据描述进行取代; 可以被卤素，氰基，硝基，烷氧基或烷氧基羰基取代的烷基，烯基或炔基。 本发明还涉及生产所述化合物的方法，含有该化合物的试剂及其在控制有害真菌中的用途

公开(公告)号：US20070259919A1

公开(公告)日：2007-11-08

申请号：US11630569

申请日：2005-06-18

申请人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/40 ,  A01N43/86 ,  A01P3/00 ,  C07D213/22 ,  C07D401/04 ,  C07D417/04

CPC分类号： C07D401/04 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/78 ,  C07D213/61 ,  C07D213/70 ,  C07D213/74 ,  C07D213/78 ,  C07D213/84 ,  C07D213/86 ,  C07D417/04

摘要： The invention relates to 2-substituted pyridines of the formula I in which the index n and the substituents R1 to R4 and L are as defined in the description and in each case one of the two ring members X1, X2 is N, the other is C—H or C-halogen; Y is a group —CH—R1—, —N—R1—, —O— or —S— and  is five- or six-membered hetaryl comprising 1 to 3 heteroatoms selected from the group consisting of O, N and S or is phenyl, and to processes for their preparation, intermediates for their preparation, pesticidal compositions and methods for controlling harmful fungi and animal pests using the compounds according to the invention.

摘要翻译： 本发明涉及式I中的2-取代吡啶，其中指数n和取代基R 1至R 4和L如说明书和每一个中所定义 两个环成员X 1，X 2中的一个是N，另一个是CH或C-卤素; Y是基团-CH-R 1 - ，-NR 1 - ， - O-或-S-，并且是包含1至3个的五元或六元杂芳基 选自O，N和S的杂原子或为苯基，并且其制备方法，其制备中间体，杀虫组合物和使用本发明化合物控制有害真菌和动物害虫的方法。

公开(公告)号：US20070208038A1

公开(公告)日：2007-09-06

申请号：US10594738

申请日：2005-03-26

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04 ,  A01N43/90

CPC分类号： A01N43/90 ,  C07D487/04

摘要： 6-(2-Fluorophenyl)-triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is C4-C8-alkyl, C4-C8-haloalkyl, substituted C3-C8-cycloalkyl, C3-C8-halocycloalkyl, C5-C8-alkenyl, C2-C8-haloalkenyl, C3-C6-cycloalkenyl, C3-C6-halocycloalkenyl, C2-C8-alkynyl, C2-C8-haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen, C1-C3-alkyl or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and contain one to three further heteroatoms from the group consisting of O, N and S as ring member, except for piperidin-1-yl optionally substituted by methyl groups; R1 and/or R2 may be substituted according to the description; L1 is chlorine or fluorine; L2 is hydrogen, is, if L1 is fluorine, also fluorine; X is alkyl; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

公开(公告)号：US20070149551A1

公开(公告)日：2007-06-28

申请号：US11677862

申请日：2007-02-22

申请人： Andreas GYPSER ,  Thomas Grote ,  Anja Schwogler ,  Joachim Rheiheimer ,  Frank Schieweck ,  Jordi Blasco ,  Ingo Rose ,  Peter Schafer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Eberhard Ammernann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas GYPSER ,  Thomas Grote ,  Anja Schwogler ,  Joachim Rheiheimer ,  Frank Schieweck ,  Jordi Blasco ,  Ingo Rose ,  Peter Schafer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Eberhard Ammernann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A61K31/506 ,  C07D403/02

CPC分类号： C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D403/12

摘要： 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRNaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC (═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC (═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C (═O)NRaRb or —C(═O) Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.