Carboxamides
    11.
    发明授权

    公开(公告)号:US5201932A

    公开(公告)日:1993-04-13

    申请号:US877365

    申请日:1992-05-04

    摘要: Carboxamides Ia, Ib, Ic and Id ##STR1## (X=O, S; R.sup.1 =H, halogen, substituted or unsubstituted alkyl, substituted or unsubstituted benzyl, alkoxy, alkylthio, haloalkoxy, haloalkylthio, substituted or unsubstituted phenyl, substituted or unsubstituted phenoxy or phenylthio, a substituted or unsubstituted 5- or 6-membered heterocyclic radical containing one or two heteroatoms, cycloalkyl-substituted alkyl, substituted or unsubstituted alkenyl which may be epoxidized, substituted or unsubstituted alkynyl, substituted or unsubstituted cycloalkyl or cycloalkenyl; R.sup.1 '=cycloalkyl-substituted alkyl, substituted or unsubstituted alkenyl which may be epoxidized, substituted or unsubstituted cycloalkenyl; R.sup.2 =CHO, 4,5-dihydrooxazol-2-yl, COYR.sup.5, CONR.sup.6 R.sup.7 ; Y=O, S; R.sup.5 =H, substituted or unsubstituted alkyl, cycloalkyl, substituted or unsubstituted alkenyl, substituted or unsubstituted cycloalkenyl, substituted or unsubstituted alkynyl, substituted or unsubstituted phenyl, a 5- or 6-membered heterocyclic radical containing up to 3 heteroatoms, benzotriazole, N-phthalimido, tetrahydrophthalimido, succinimido, maleiimido, 2,2-dimethyl-1,3-dioxolan-4-ylmethyl, 1,3-dioxolan-2-on-4-ylmethyl, and when Y.dbd.O: one equivalent of a cation from the group of the alkali or alkaline earth metals, Mn, Cu, Fe ammonium and substituted ammonium, a radical --N.dbd.CR.sup.8 R.sup.9 or --W--Z; R.sup.8, R.sup.9 .dbd.H, substituted or unsubstituted alkyl, substituted or unsubstituted haloalkyl, cycloalkyl, alkoxy, furanyl, substituted or unsubstituted phenyl; R.sup.8 +R.sup.9 =4-7-membered methylene chain; W=alkylene chain, ethoxyethylene chain, butylene, butynylene chain; Z=a molecular moiety bonded to W in the .omega.-position and is the same as that linked to W in the .alpha.-position of W; R.sup.6 .dbd.H, alkyl, cycloalkyl; R.sup.7 .dbd.H; alkyl; --C(O-alkyl).dbd.N--H or --(O--alkyl).dbd.N--alkyl; R.sup.6 +R.sup.7 =4-5-membered methylene chain; R.sup.3 .dbd.H, substituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl; R.sup.4 .dbd.H, OH, alkoxy, subsituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted alkenyl, substituted or unsubstituted alkynyl, di-(C.sub.1 -C.sub.4)-alkylamino, a substituted or unsubstituted 5- or 6-membered heterocyclic radical containing one or two heteroatoms, substituted or unsubstituted phenyl, substituted or unsubstituted naphthyl; R.sub.3 +R.sub.4 =4-7-membered methylene chain which may be interrupted by O, S or N--CH.sub.3, or --(CH.sub.2).sub.3 --CO--)and their environmentally tolerated salts.The compounds Ia to Id are suitable as herbicides.

    Sulfonamides
    12.
    发明授权
    Sulfonamides 失效
    磺胺

    公开(公告)号:US5171353A

    公开(公告)日:1992-12-15

    申请号:US521032

    申请日:1990-05-09

    摘要: Sulfonamides of the general formula I ##STR1## where R.sup.1 is hydrogen of C.sub.1 -C.sub.4 -alkyl,R.sup.2 is hydrogen or substituted or unsubstituted C.sub.1 -C.sub.6 -alkyl; C.sub.3 -C.sub.4 -alkenyl; C.sub.3 -C.sub.4 -alkynyl or substituted or unsubstituted saturated or singly unsaturated 5- to 7- membered heteroaryl;R.sup.3 and R.sup.4 are halogen; substituted or unsubstituted C.sub.1 -C.sub.4 -alkoxy C.sub.1 -C.sub.4 -alkylthio, C.sub.2 -C.sub.6 -alkenyl, C.sub.2 -C.sub.6 -alkenyloxy, C.sub.2 -C.sub.6 -alkenylthio, C.sub.2 -C.sub.6 -alkynyl, C.sub.2 -C.sub.6 -alkynyloxy, C.sub.2 -C.sub.6 -alkynylthio, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -cycloalkylthio, C.sub.5 -C.sub.6 -cycloalkenyl, C.sub.3 -C.sub.6 -cycloalkoxy, C.sub.5 -C.sub.6 -cycloalkenyloxy, C.sub.5 -C.sub.6 -cycloalkenylthio, phenyl, phenoxy, phenylthio, benzyl, benzyloxy or benzylthio;the group given for R.sup.2, or NR.sup.7 R.sup.8, where R.sup.7 and R.sup.8 are hydrogen, C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.5 -C.sub.6 -cycloalkenyl, substituted or unsubstituted phenyl and/or benzyl bedeuten, or issubstituted or unsubstituted C.sub.4 -C.sub.6 -alkylene which may be interrupted or oxygen, sulfur or nitrogen;X is nitrogen or .dbd.CR.sup.5 14 ,where R.sup.5 is one of the radicals R.sup.3,n is 0 or 1 andA is substituted or unsubstituted mono- or dinuclear aryl containing one or two nitrogen, oxygen and/or sulfur atoms,and their agriculturally useful salts, and herbicidal and growth-regulating agents containing them.

    摘要翻译: 其中R 1是C 1 -C 4 - 烷基的氢,R 2是氢或被取代或未被取代的C 1 -C 6 - 烷基的磺酰胺, C3-C4-烯基; C3-C4-炔基或取代或未取代的饱和或单不饱和5-至7-元杂芳基; R3和R4是卤素; 取代或未取代的C 1 -C 4 - 烷氧基C 1 -C 4 - 烷硫基,C 2 -C 6 - 链烯基,C 2 -C 6 - 烯氧基,C 2 -C 6 - 烯硫基,C 2 -C 6炔基,C 2 -C 6 - 炔氧基,C 2 -C 6 - 炔硫基, C 3 -C 6环烷基,C 3 -C 6环烷硫基,C 5 -C 6环环烯基,C 3 -C 6环烷氧基,C 5 -C 6环环烯氧基,C 5 -C 6环环硫基,苯基,苯氧基,苯硫基,苄基,苄氧基或苄硫基; R2或NR7R8的基团,其中R7和R8是氢,C1-C6-烷基,C3-C6-烯基,C3-C6-炔基,C3-C6-环烷基,C5-C6-环烯基,取代或未取代的苯基 或/或苄基叔丁基醚,或者是可被中断的取代或未取代的C 4 -C 6亚烷基或氧,硫或氮; X是氮或= CR514,其中R5是基团R3之一,n是0或1,A是含有一个或两个氮,氧和/或硫原子的取代或未取代的单核或二核芳基及其农业上有用的盐 ,和含有它们的除草和生长调节剂。

    N-aryltetrahydrophthalimides and herbicidal compositions thereof
    13.
    发明授权
    N-aryltetrahydrophthalimides and herbicidal compositions thereof 失效
    N-三氟甲磺酰嘧啶及其除草剂组合物

    公开(公告)号:US5133799A

    公开(公告)日:1992-07-28

    申请号:US697036

    申请日:1991-05-08

    摘要: R.sup.1 is C.sub.1 -C.sub.4 -alkyl which may carry from one to five halogen atoms or one of the groups stated for X;R.sup.2 is a heteroaromatic structure bonded via a nitrogen atom, which has a 5-membered ring and contains, in addition to carbon ring members, from one to three nitrogen atoms, andR.sup.3 is halogen, C.sub.1 -C.sub.4 -alkylthio, one of the groups stated for R.sup.2 or phenylthio which in turn may carry from one to three of the following radicals: halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy or C.sub.1 -C.sub.4 -alkylthio, and where the phenylthio group may also carry halogen atoms such that the total number of radicals is 4 or 5,and salts thereof which can be used in agriculture, are suitable as herbicides. 2

    摘要翻译: 其中X是氢或卤素; R 1是可以携带1至5个卤素原子的C1-C4-烷基或为X表示的基团之一; R2是通过氮原子键合的杂芳族结构,其具有5元环,并且除了碳环成员之外还含有一个至三个氮原子,并且R 3是卤素,C 1 -C 4 - 烷硫基,其中一个基团 对于R2或苯硫基,其又可以携带1-3个以下基团:卤素,C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 卤代烷氧基或C 1 -C 4 - 烷硫基 并且苯硫基也可以携带卤素原子使得基团的总数为4或5,并且其可用于农业的盐适用作除草剂。

    Pyrimido(5,4-e)-as-triazine-5,7(6H,8H)-diones
    15.
    发明授权
    Pyrimido(5,4-e)-as-triazine-5,7(6H,8H)-diones 失效
    嘧啶并(5,4-e)-as-三嗪-5,7(6H,8H) - 二酮

    公开(公告)号:US5069708A

    公开(公告)日:1991-12-03

    申请号:US547160

    申请日:1990-07-03

    IPC分类号: A01N43/90 C07D487/04

    CPC分类号: A01N43/90

    摘要: Herbicidal agents containing a pyrimido[5,4-e]-as-triazine-5,7-(6H,8H)-dione Ia ##STR1## (R.sup.1, R.sup.2 .dbd.H, C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.2 -C.sub.8 -alkenyl, phenyl or benzyl, R.sup.3 .dbd.H, halogen, nitro, C.sub.1 -C.sub.8 -alkyl which may carry up to three further substituents, C.sub.2 -C.sub.6 -alkenyl, phenyl-C.sub.2 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -cycloalkyl which may carry up to 3 C.sub.1 -C.sub.4 -alkyl substituents, a 5- or 6-membered heterocyclic structure where up to 2 of the ring members are O, S or NR.sup.4 ; --CO--R.sup.4 or --CO--O--R.sup.4 ; phenyl or hetaryl, which may carry up to 3 further substituents; or ZR.sup.6 ; R.sup.4 .dbd.H, C.sub.1 -C.sub.6 -alkyl; Z.dbd.O, S or --N(R.sup.7)--; R.sup.6 .dbd.H, C.sub.1 -C.sub.6 -alkyl, phenyl or benzyl, which may carry up to 3 further substituents; R.sup.7 .dbd.H, C.sub.1 -C.sub.6 -alkyl or R.sup.6 and R.sup.7 together with nitrogen form a 5- or 6-membered ring which may contain O; n=0 or 1) or a salt of Ia with a mineral acid.

    摘要翻译: 含有嘧啶并[5,4-e] -as-三嗪-5,7-(6H,8H) - 二酮Ia(Ia)(R1,R2 = H,C1-C6-烷基,C3- C 2 -C 6环烷基,C 2 -C 8 - 烯基,苯基或苄基,R 3 = H,卤素,硝基,可带有至多三个其它取代基的C 1 -C 8烷基,C 2 -C 6 - 链烯基,苯基-C 2 -C 6 - 烯基, 可含有3个C 1 -C 4烷基取代基的C 3 -C 6环烷基,其中至多2个环成员为O,S或NR 4的5或6元杂环结构; -CO-R 4或-CO- R 4 = H,C 1 -C 6 - 烷基; Z = O,S或-N(R 7) - ; R 6 = H,C 1 -C 6烷基; - 烷基,苯基或苄基,其可以带有多达3个其它取代基; R 7 = H,C 1 -C 6 - 烷基或者R 6和R 7与氮一起形成5-或6-元环,其可以含有O; n = 0或 1)或Ia与无机酸的盐。

    Herbicidal 3-(3,4,5,6-tetrahydrophthalimido)-cinnamic esters
    20.
    发明授权
    Herbicidal 3-(3,4,5,6-tetrahydrophthalimido)-cinnamic esters 失效
    除草剂3-(3,4,5,6-四氢邻苯二甲酰亚胺基) - 肉桂酯

    公开(公告)号:US5296452A

    公开(公告)日:1994-03-22

    申请号:US525035

    申请日:1990-05-18

    CPC分类号: C07D209/48 A01N37/46

    摘要: 3-(N-3,4,5,6-Tetrahydrophthalimido)-cinnamic esters of the general formula I ##STR1## where n is 1 or 2 and the substituents have the following meanings:R.sup.1 is hydrogen or fluorine,R.sup.2 is halogen,R.sup.3 is hydrogen, halogen or C.sub.1 -C.sub.4 -alkyl,R.sup.4 is hydrogen, substituted or unsubstituted C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.7 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl or benzyl,R is C.sub.1 -C.sub.4 -alkyl,processes for their manufacture, and herbicidal agents containing them.

    摘要翻译: 3-(N-3,4,5,6-四氢邻苯二甲酰亚氨基) - 肉桂酸酯,其中n为1或2,并且取代基具有以下含义:R 1为氢或氟,R 2为卤素 R3是氢,卤素或C1-C4-烷基,R4是氢,取代或未取代的C1-C6-烷基,C3-C7-环烷基,C3-C6-烯基,C3-C6-炔基或苄基,R是C1- C4烷基,其制备方法和含有它们的除草剂。