Method for increasing the address space for mobile terminals in a wireless network
    12.
    发明授权
    Method for increasing the address space for mobile terminals in a wireless network 有权
    一种用于增加无线网络中的移动终端的地址空间的方法

    公开(公告)号:US09271304B2

    公开(公告)日:2016-02-23

    申请号:US14363148

    申请日:2011-12-09

    摘要: A method, in a base station subsystem (10), of allocating radio resources to mobile stations (20) in a wireless communication system (1) involves the base station subsystem (10) assigning a respective Temporary Block Flow (TBF) to each mobile station (20) in a cell (40) in the communication system (1), and then assigning to each TBF a Temporary Flow Identity (TFI), at least one Packet Data Channel (PDCH), and an Uplink State Flag (USF) if the TBF is an uplink TBF. The base station subsystem (10) then selects different training sequences from a plurality of available training sequences and assigns a respective different selected training sequence to two or more TBFs wherein these two or more TBFs share the same assigned Temporary Flow Identity (TFI), the same assigned Packet Data Channel (PDCH), and/or the same assigned Uplink State Flag (USF) if the TBF is an uplink TBF.

    摘要翻译: 一种在基站子系统(10)中向无线通信系统(1)中的移动台(20)分配无线电资源的方法,其特征在于,所述基站子系统(10)将相应的临时块流(TBF)分配给每个移动台 在通信系统(1)中的小区(40)中的站(20),然后向每个TBF分配临时流标识(TFI),至少一个分组数据信道(PDCH)和上行链路状态标志(USF) 如果TBF是上行链路TBF。 然后,基站子系统(10)从多个可用的训练序列中选择不同的训练序列,并将相应不同的选择的训练序列分配给两个或更多个TBF,其中这两个或更多TBF共享相同的分配临时流标识(TFI), 相同的分配数据信道(PDCH),和/或相同的分配的上行链路状态标志(USF),如果TBF是上行链路TBF。

    Processes for producing benzophenone derivatives
    13.
    发明授权
    Processes for producing benzophenone derivatives 有权
    二苯甲酮衍生物的制备方法

    公开(公告)号:US09085519B2

    公开(公告)日:2015-07-21

    申请号:US13521910

    申请日:2011-01-19

    IPC分类号: C07C41/30 C07C41/34 C07C45/72

    摘要: There is provided a process for the preparation of a compound of formula I, wherein X, R1, R2a, R2b, R2c, R2d, R2e, R3a, R3b, R3c, R3d and R3e are as described in the description. Such compounds may, for example, be useful medicament (or intermediates for medicaments).

    摘要翻译: 提供了制备式I化合物的方法,其中X,R1,R2a,R2b,R2c,R2d,R2e,R3a,R3b,R3c,R3d和R3e如说明书所述。 这样的化合物可以是例如有用的药物(或药物的中间体)。

    NEW PROCESSES FOR PRODUCING BENZOPHENONE DERIVATIVES
    15.
    发明申请
    NEW PROCESSES FOR PRODUCING BENZOPHENONE DERIVATIVES 有权
    生产苯并噻吩衍生物的新工艺

    公开(公告)号:US20130035514A1

    公开(公告)日:2013-02-07

    申请号:US13521910

    申请日:2011-01-19

    IPC分类号: C07C41/30 C07C41/34

    摘要: There is provided a process for the preparation of a compound of formula I, wherein X, R1, R2a, R2b, R2c, R2d, R2e, R3a, R3b, R3c, R3d and R3e are as described in the description. Such compounds may, for example, be useful medicament (or intermediates for medicaments).

    摘要翻译: 提供了制备式I化合物的方法,其中X,R1,R2a,R2b,R2c,R2d,R2e,R3a,R3b,R3c,R3d和R3e如说明书所述。 这样的化合物可以是例如有用的药物(或药物的中间体)。

    Certain arylaliphatic and heteroaryl-aliphatic piperazinyl pyrazines and their use in the treatment of serotonin-related diseases
    16.
    发明授权
    Certain arylaliphatic and heteroaryl-aliphatic piperazinyl pyrazines and their use in the treatment of serotonin-related diseases 失效
    某些芳基脂族和杂芳基 - 脂族哌嗪基吡嗪及其在治疗5-羟色胺相关疾病中的应用

    公开(公告)号:US07534794B2

    公开(公告)日:2009-05-19

    申请号:US10269670

    申请日:2002-10-11

    摘要: The invention relates to compounds of the general formula (I): wherein Ar is optionally substituted aryl or heteroaryl; A is (i) —O—, —S—, —SO2—, —NH—, (ii) a C1-4-alkyl- or C1-6-acyl-substituted nitrogen atom or (iii) a C1-8-alkylene chain or a heteroalkylene chain having 2 to 8 chain atoms, which optionally contains at least one unsaturation, and which may be substituted and/or contain a bridge to form a saturated or partially or fully unsaturated ring having 3-8 ring members; B is —C(R4)(R5)—, —OC(R4)(R5)—, —N(R6)C(R4)(R5)—, —N(R6)—, —O—, —S— or —SO2—; R is optionally substituted C3-8-cycloalkyl, aryl or heteroaryl; R1 is (i) a saturated or unsaturated azacyclic or aminoazacyclic ring, or a saturated diazacyclic or aminodiazacyclic ring, which has 4 to 7 ring members, or a saturated aminoazabicyclic, azabicyclic or diazabicyclic ring which has 7 to 10 ring members, which rings optionally are substituted in one or more positions, or a group —[C(R4)(R5)]xN(R2a)(R3a)]; R2a, R3a, R4, R5, R6 and x are as defined in the claims, and n is 0 or 1; and pharmaceutically acceptable salts, hydrates and prodrug forms thereof. The compounds may be prepared by per se conventional methods and can be used for treating a human or animal subject suffering from a serotonin-related disorder, such as eating disorders, especially obesity, memory disorders, schizophrenia, mood disorders, anxiety disorders, pain, sexual dysfunctions, and urinary disorders The invention also relates to such use as well as to pharmaceutical compositions comprising a compound of formula (I).

    摘要翻译: 本发明涉及通式(I)的化合物:其中Ar为任选取代的芳基或杂芳基; A是(ⅰ)-O - , - S - , - SO 2 - , - NH - ,(ⅱ)C 1-4 - 烷基 - 或C 1-6 - 酰基取代的氮原子或(ⅲ) 亚烷基链或具有2至8个链原子的杂亚烷基链,其任选地包含至少一个不饱和键,并且其可以被取代和/或含有桥以形成具有3-8个环成员的饱和或部分或完全不饱和的环; B是-C(R 4)(R 5) - , - OC(R 4)(R 5) - , - N(R 6) 或-SO 2 - ; R是任选取代的C 3-8 - 环烷基,芳基或杂芳基; R1是(i)饱和或不饱和的氮杂环或氨基氮杂环或饱和的二氮环或氨基二氮环,其具有4至7个环成员,或具有7至10个环成员的饱和氨基氮杂双环,氮杂双环或二氮杂双环,其任选地环 在一个或多个位置被取代,或基团 - [C(R 4)(R 5)] x N(R 2a)(R 3a)]; R2a,R3a,R4,R5,R6和x如权利要求中所定义,n为0或1; 及其药学上可接受的盐,水合物和前药形式。 化合物可以通过本身的常规方法制备,并且可以用于治疗患有5-羟色胺相关病症的人或动物受试者,例如进食障碍,特别是肥胖,记忆障碍,精神分裂症,情绪障碍,焦虑症,疼痛, 性功能障碍和尿失调本发明还涉及这样的用途以及包含式(I)化合物的药物组合物。

    New compounds
    17.
    发明申请
    New compounds 审中-公开
    新化合物

    公开(公告)号:US20080221129A1

    公开(公告)日:2008-09-11

    申请号:US11825431

    申请日:2007-07-06

    CPC分类号: C07D487/04

    摘要: The present invention relates to compounds of the formula (I): including pharmaceutically acceptable salts, solvates, hydrates, geometrical isomers, tautomers, optical isomers, and N-oxides thereof, said compounds being useful as inhibitors of stearoyl-CoA desaturase (SCD). The invention further relates to the use of compounds of the formula (I) for treatment of medical conditions in which the modulation of SCD activity is beneficial, such as cardiovascular diseases, obesity, non-insulin-dependent diabetes mellitus, hypertension, neurological diseases, immune disorders, cancer, essential fatty acid deficiency, acne, psoriasis, rosacea or other skin conditions.

    摘要翻译: 本发明涉及式(I)化合物:其药学上可接受的盐,溶剂化物,水合物,几何异构体,互变异构体,旋光异构体及其N-氧化物,所述化合物可用作硬脂酰辅酶A去饱和酶(SCD) 。 本发明还涉及式(I)化合物用于治疗其中SCD活性调节有益的医学病症,例如心血管疾病,肥胖症,非胰岛素依赖性糖尿病,高血压,神经系统疾病, 免疫疾病,癌症,必需脂肪酸缺乏症,痤疮,牛皮癣,酒渣鼻或其他皮肤病症。

    Filling assembly, gasket for use in said filling assembly, and a method for filling liquid
    18.
    发明授权
    Filling assembly, gasket for use in said filling assembly, and a method for filling liquid 有权
    填充组件,用于所述填充组件的垫圈,以及用于填充液体的方法

    公开(公告)号:US09238515B2

    公开(公告)日:2016-01-19

    申请号:US13515998

    申请日:2010-12-15

    CPC分类号: B65B9/20 B65B31/045

    摘要: A filling assembly for filling of a tube of packaging material having a seal starting at a first level, comprises a conduit arranged to lead liquid into the tube of packaging material below said first level and a passage arranged to eject gas through openings into the tube of packaging material below said first level. The filling assembly is characterized in that a gasket is arranged to provide a seal between said filling assembly and said tube of packaging material upstream said openings such that the overpressure P1 downstream the gasket may exceed an ambient pressure Pa upstream the gasket.

    摘要翻译: 一种用于填充具有从第一层开始的密封剂的包装材料管的填充组件,包括布置成将液体引导到所述第一水平面以下的包装材料管中的导管,以及设置成将气体通过开口喷射到管 包装材料低于第一级。 填充组件的特征在于,垫圈布置成在所述填充组件和所述开口之上的所述包装材料管之间提供密封,使得垫圈下游的超压P1可以超过垫圈上游的环境压力Pa。

    Method for Increasing the Address Space for Mobile Terminals in a Wireless Network
    19.
    发明申请
    Method for Increasing the Address Space for Mobile Terminals in a Wireless Network 有权
    用于增加无线网络中移动终端的地址空间的方法

    公开(公告)号:US20150103759A1

    公开(公告)日:2015-04-16

    申请号:US14363148

    申请日:2011-12-09

    IPC分类号: H04W72/12 H04L5/00

    摘要: A method, in a base station subsystem (10), of allocating radio resources to mobile stations (20) in a wireless communication system (1) involves the base station subsystem (10) assigning a respective Temporary Block Flow (TBF) to each mobile station (20) in a cell (40) in the communication system (1), and then assigning to each TBF a Temporary Flow Identity (TFI), at least one Packet Data Channel (PDCH), and an Uplink State Flag (USF) if the TBF is an uplink TBF. The base station subsystem (10) then selects different training sequences from a plurality of available training sequences and assigns a respective different selected training sequence to two or more TBFs wherein these two or more TBFs share the same assigned Temporary Flow Identity (TFI), the same assigned Packet Data Channel (PDCH), and/or the same assigned Uplink State Flag (USF) if the TBF is an uplink TBF.

    摘要翻译: 一种在基站子系统(10)中向无线通信系统(1)中的移动台(20)分配无线电资源的方法,其特征在于,所述基站子系统(10)将相应的临时块流(TBF)分配给每个移动台 在通信系统(1)中的小区(40)中的站(20),然后向每个TBF分配临时流标识(TFI),至少一个分组数据信道(PDCH)和上行链路状态标志(USF) 如果TBF是上行链路TBF。 然后,基站子系统(10)从多个可用的训练序列中选择不同的训练序列,并将相应不同的选择的训练序列分配给两个或更多个TBF,其中这两个或更多TBF共享相同的分配临时流标识(TFI), 相同的分配数据信道(PDCH),和/或相同的分配的上行链路状态标志(USF),如果TBF是上行链路TBF。