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    Isoxazoline derivatives as insecticidal compounds
    21.
    发明授权
    Isoxazoline derivatives as insecticidal compounds 有权
    异恶唑啉衍生物作为杀虫剂

    公开(公告)号：US09307766B2

    公开(公告)日：2016-04-12

    申请号：US14240052

    申请日：2012-08-24

    申请人： Jerome Yves Cassayre ,  Peter Renold ,  Thomas Pitterna ,  Myriem El Qacemi

    发明人： Jerome Yves Cassayre ,  Peter Renold ,  Thomas Pitterna ,  Myriem El Qacemi

    IPC分类号： A01N43/80 ,  A01N43/40 ,  C07D413/14 ,  C07D413/12 ,  A01N37/42 ,  A01N37/50 ,  A01N43/42 ,  C07F7/18 ,  A01N43/20

    CPC分类号： A01N43/80 ,  A01N37/42 ,  A01N37/50 ,  A01N43/20 ,  A01N43/40 ,  A01N43/42 ,  C07D413/12 ,  C07D413/14 ,  C07F7/1804

    摘要： The present invention provides compounds of formula (I) wherein G1 is oxygen; R1 is hydrogen; R2 is group (P) L is a bond, methylene or ethylene; one of A1 and A2 is S, SO or SO2 and the other is —C(R4)R4—; R3 is hydrogen or methyl; each R4 is independently hydrogen or methyl; Y2 and Y3 are independently CH or nitrogen, wherein Y2 and Y3 are not both nitrogen; X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X1, X3 and X6 are not hydrogen; X4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).

    摘要翻译： 本发明提供其中G1是氧的式（I）化合物; R1是氢; R2是基团（P），L是键，亚甲基或亚乙基; A1和A2之一是S，SO或SO2，另一个是-C（R 4）R 4 - ; R3是氢或甲基; 每个R 4独立地是氢或甲基; Y2和Y3独立地是CH或氮，其中Y2和Y3不都是氮; X2是C-X6或氮; X1，X3和X6独立地为氢，卤素或三卤代甲基，其中X 1，X 3和X 6中的至少两个不是氢; X4是三氟甲基，二氟甲基或氯二氟甲基。 本发明还提供了可用于制备式（I）化合物的中间体，以及使用式（I）化合物控制昆虫，螨虫，线虫或软体动物的方法。

    ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS
    23.
    发明申请
    ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS 有权
    异辛唑衍生物作为杀虫剂化合物

    公开(公告)号：US20140194376A1

    公开(公告)日：2014-07-10

    申请号：US14240052

    申请日：2012-08-24

    申请人： Jerome Yves Cassayre ,  Peter Renold ,  Thomas Pitterna ,  Myriem El Qacemi

    发明人： Jerome Yves Cassayre ,  Peter Renold ,  Thomas Pitterna ,  Myriem El Qacemi

    IPC分类号： A01N43/80 ,  A01N43/40 ,  A01N43/42 ,  A01N43/20

    CPC分类号： A01N43/80 ,  A01N37/42 ,  A01N37/50 ,  A01N43/20 ,  A01N43/40 ,  A01N43/42 ,  C07D413/12 ,  C07D413/14 ,  C07F7/1804

    摘要： The present invention provides compounds of formula (I) wherein G1 is oxygen; R1 is hydrogen; R2 is group (P) L is a bond, methylene or ethylene; one of A1 and A2 is S, SO or SO2 and the other is —C(R4)R4—; R3 is hydrogen or methyl; each R4 is independently hydrogen or methyl; Y2 and Y3 are independently CH or nitrogen, wherein Y2 and Y3 are not both nitrogen; X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X1, X3 and X6 are not hydrogen; X4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).

    摘要翻译： 本发明提供其中G1是氧的式（I）化合物; R1是氢; R2是基团（P），L是键，亚甲基或亚乙基; A1和A2之一是S，SO或SO2，另一个是-C（R 4）R 4 - ; R3是氢或甲基; 每个R 4独立地是氢或甲基; Y2和Y3独立地是CH或氮，其中Y2和Y3不都是氮; X2是C-X6或氮; X1，X3和X6独立地为氢，卤素或三卤代甲基，其中X 1，X 3和X 6中的至少两个不是氢; X4是三氟甲基，二氟甲基或氯二氟甲基。 本发明还提供了可用于制备式（I）化合物的中间体，以及使用式（I）化合物控制昆虫，螨虫，线虫或软体动物的方法。

    PROCESS FOR THE PREPARATION OF DIHYDROPYRROLE DERIVATIVES
    25.
    发明申请
    PROCESS FOR THE PREPARATION OF DIHYDROPYRROLE DERIVATIVES 有权
    制备二氢衍生物衍生物的方法

    公开(公告)号：US20130237583A1

    公开(公告)日：2013-09-12

    申请号：US13703630

    申请日：2011-06-14

    申请人： Myriem El Qacemi ,  Helmars Smits ,  Jerome Yves Cassayre ,  Nicholas Phillip Mulholland ,  Peter Renold ,  Edouard Godineau ,  Thomas Pitterna

    发明人： Myriem El Qacemi ,  Helmars Smits ,  Jerome Yves Cassayre ,  Nicholas Phillip Mulholland ,  Peter Renold ,  Edouard Godineau ,  Thomas Pitterna

    IPC分类号： C07D207/46 ,  C07D207/20

    CPC分类号： C07D207/46 ,  A01N43/36 ,  C07D207/20 ,  C07D401/04 ,  C07D413/12 ,  C07D413/14 ,  C07D417/14

    摘要： The present invention provides stereoselective processes for the preparation of compounds of formula (I) wherein P is phenyl, naphthyl, a 6-membered heteroaryl group containing one or two nitrogen atoms as ring members, or a 10-membered bicyclic heteroaryl group containing one or two nitrogen atoms as ring members, and wherein the phenyl, naphthyl and heteroaryl groups are optionally substituted; R1 is chlorodifluoromethyl or trifluoromethyl; R2 is optionally substituted aryl or optionally substituted heteroaryl; n is 0 or 1; including the process comprising (a-i) reacting a compound of formula II wherein P, R1 and R2 are as defined for the compound of formula I; with nitromethane in the presence a chiral catalyst to give a compound of formula III Wherein P, R1 and R2 are as defined for the compound of formula I; and (a-ii) reductively cyclising the compound of formula III to give the compound of formula I. The invention also provides intermediates useful for processes for the synthesis of compounds of formula (I).

    摘要翻译： 本发明提供了制备式（I）化合物的立体选择性方法，其中P是苯基，萘基，含有一个或两个氮原子作为环成员的6元杂芳基或含有一个或多个氮原子的10元双环杂芳基 两个氮原子作为环成员，并且其中苯基，萘基和杂芳基任选被取代; R1是氯二氟甲基或三氟甲基; R2是任选取代的芳基或任选取代的杂芳基; n为0或1; 包括（a-i）使式II化合物与式Ⅰ化合物反应的方法，其中P，R 1和R 2如对式I化合物所定义; 在硝基甲烷中存在手性催化剂，得到式III化合物，其中P，R 1和R 2如式I化合物所定义; 和（a-ii）还原性环化式III化合物以得到式I化合物。本发明还提供了可用于合成式（I）化合物的方法的中间体。

    Insecticidal compounds
    27.
    发明授权
    Insecticidal compounds 失效
    杀虫化合物

    公开(公告)号：US08193221B2

    公开(公告)日：2012-06-05

    申请号：US12738035

    申请日：2008-10-13

    申请人： Werner Zambach ,  Peter Renold

    发明人： Werner Zambach ,  Peter Renold

    IPC分类号： A01N43/00 ,  A01N43/80 ,  C07D413/12 ,  C07D261/04

    CPC分类号： C07D261/04 ,  C07D261/08 ,  C07D413/12 ,  C07D417/12

    摘要： A compound of formula (I) wherein A1, A2, A3, A4, R1, R2, R3 and R4 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal or molluscicidal compositions comprising them and to methods of using them to combat and control insect, acarine, nematode or mollusc pests.

    摘要翻译： 其中A1，A2，A3，A4，R1，R2，R3和R4如权利要求1所定义的式（I）化合物; 或其盐或N-氧化物。 此外，本发明涉及制备式（I）化合物的方法和中间体，其包含它们的杀虫，杀螨，杀线虫或杀软体动物的组合物以及使用它们来对抗和控制昆虫，螨虫，线虫或软体动物害虫的方法。

    3-AMINO-BENZO [D] ISOTHIAZOLE DIOXIDE DERIVATIVES AND THEIR USE AS PESTICIDES
    30.
    发明申请
    3-AMINO-BENZO [D] ISOTHIAZOLE DIOXIDE DERIVATIVES AND THEIR USE AS PESTICIDES 失效
    3-氨基苯并[D]异噻唑二酮衍生物及其作为杀虫剂的用途

    公开(公告)号：US20110071200A1

    公开(公告)日：2011-03-24

    申请号：US12993983

    申请日：2009-05-18

    申请人： Werner Zambach ,  Ottmar Franz Hueter ,  Peter Renold ,  Thomas Pitterna ,  Peter Maienfisch

    发明人： Werner Zambach ,  Ottmar Franz Hueter ,  Peter Renold ,  Thomas Pitterna ,  Peter Maienfisch

    IPC分类号： A61K31/428 ,  C07D275/06 ,  A01N43/80 ,  A01C1/06 ,  A01P7/00 ,  A61P33/14

    CPC分类号： C07D275/06

    摘要： A compound of Formula (I) or Formula (II) where W is C—R3; X is C—R4; Y is C—R5; R1 and R6, independently of each other, is, for example, H, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl or C1-C6-alkyl-C(═O); R2 is H; and R3, R4 and R5, independently of each other, are, for example, H, halogen, cyano, nitro, C1-C6-alkyl, or C1-C6-haloalkyl; provided that in formula II R1 is H and R6 is as defined above; and in formula I that (a) at least one of R1 and R3 to R6 is other than hydrogen, (b) R3 or R4 is other than C1 when in each instance the remaining five groups of R1 to R6 are hydrogen, and (c) (i) R3 is other than methyl, (ii) R4 is other than C1, (iii) R5 is other than C1 and (iv) R3 is not C1 when R5 is methoxy, when in each instance (i) to (iv) R1 is H, R6 is MeC(═O), and remaining groups of R2 to R5 are hydrogen; and/or salts thereof; and their use as as pesticidal agents.

    摘要翻译： 式（I）或式（II）的化合物，其中W是C-R 3; X是C-R4; Y为C-R5; R 1和R 6彼此独立地是例如H，C 1 -C 6 - 烷基，C 2 -C 6 - 烯基，C 2 -C 6 - 炔基，C 3 -C 8 - 环烷基或C 1 -C 6 - 烷基-C（= O ）; R2为H; 和R 3，R 4和R 5彼此独立地是例如H，卤素，氰基，硝基，C 1 -C 6烷基或C 1 -C 6卤代烷基; 条件是式Ⅱ中R 1为H且R 6如上定义; （a）R1和R3至R6中的至少一个不是氢，（b）R 3或R 4不同于C 1，当R 5至R 6的剩余五个基团为氢时，和（c ）（i）R 3不是甲基，（ⅱ）R 4不是C 1，（ⅲ）R 5不是C 1，（ⅳ）当R 5是甲氧基时，R 3不是C 1，当（i）〜 ）R1为H，R6为MeC（= O），R2至R5的其余基团为氢; 和/或其盐; 以及其作为杀虫剂的用途。