公开(公告)号：US4762830A

公开(公告)日：1988-08-09

申请号：US830430

申请日：1986-02-13

申请人： Elmar Sturm ,  Jean J. Gallay ,  Haukur Kristinsson ,  Georg Pissiotas

发明人： Elmar Sturm ,  Jean J. Gallay ,  Haukur Kristinsson ,  Georg Pissiotas

IPC分类号： C07D263/58 ,  A61K31/496 ,  A61K31/515 ,  A61P33/10 ,  C07D233/70 ,  C07D235/26 ,  C07D239/62 ,  C07D239/66 ,  C07D249/08 ,  C07D249/12 ,  C07D271/06 ,  C07D271/10 ,  C07D271/113 ,  C07D277/24 ,  C07D277/34 ,  C07D277/58 ,  C07D277/68 ,  C07D285/08 ,  C07D285/12 ,  C07D285/13 ,  C07D403/12 ,  C07D413/12 ,  C07D417/12 ,  A61K31/505 ,  C07D403/10

CPC分类号： C07D271/113 ,  C07D233/70 ,  C07D239/62 ,  C07D239/66 ,  C07D249/12 ,  C07D277/34 ,  C07D277/58 ,  C07D277/68 ,  C07D285/08 ,  C07D285/13 ,  C07D413/12 ,  C07D417/12

摘要： The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I ##STR1## wherein X is oxygen or sulfur;R.sub.1 is C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.3 -C.sub.6 cycloalkyl or allyl;R.sub.2 is C.sub.1 -C.sub.6 alkyl or allyl;R.sub.3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; andR.sub.4 and R.sub.5 are each independently of the other hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxy or C.sub.1 -C.sub.6 haloalkoxy;and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.

摘要翻译： 本发明涉及通式I（I）的新的5-（azolyloxyphenylcarbamoyl）巴比土酸衍生物，其中X是氧或硫; R1是C1-C6烷基，C1-C6烷氧基，C3-C6环烷基或烯丙基; R2是C1-C6烷基或烯丙基; R3是通过碳结合的未取代或取代的五元唑环，选自苯并咪唑，苯并恶唑，苯并噻唑，咪唑，恶唑，噻唑，恶二唑，噻二唑和三唑; 并且R 4和R 5各自独立地为另一个氢，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷氧基或C 1 -C 6卤代烷氧基; 和其互变异构体和盐，作为驱肠剂化合物。 与合适的载体和进一步助剂一起，这些化合物可特别用于控制作为动物寄生虫的蠕虫。

公开(公告)号：US4459152A

公开(公告)日：1984-07-10

申请号：US365684

申请日：1982-04-05

申请人： Ernst Fankhauser ,  Elmar Sturm

发明人： Ernst Fankhauser ,  Elmar Sturm

IPC分类号： A01H3/04 ,  A01N33/22 ,  A01N41/10 ,  A01N43/08 ,  A01N47/06 ,  A01N53/00 ,  A01N53/10 ,  C07C317/14 ,  C07C317/22 ,  C07C317/36 ,  C07D307/24 ,  C07D307/68

CPC分类号： C07D307/68 ,  A01N41/10 ,  A01N43/08 ,  A01N47/06 ,  A01N53/00 ,  C07C317/00 ,  C07D307/24 ,  Y10S47/01

摘要： The invention describes gametocidal and microbicidal compositions which contain, as active ingredient, a nitroarylalkylsulfone derivative of the formula I ##STR1## wherein R.sub.1 is alkyl, R.sub.2 and R.sub.3 are each hydrogen, alkyl, alkoxy, haloalkyl, halogen, cyano, nitro or amino or together they complete a naphthalene ring; R.sub.4 is hydrogen or --COR.sub.5, wherein R.sub.5 is alkyl, alkoxy, haloalkoxy, alkenyl, haloalkenyl, alkynyl, cycloalkyl, phenyl, benzyl, furyl or tetrahydrofuryl. The invention relates also to the use of these compositions and compounds for stimulating generative plant growth and for obtaining hybrid seeds, as well as to a method of preparing the hydrazinium and ammonium salts within the scope of the formula I, and to a process for preparing agrochemical compositions which contain compounds of the formula I as active ingredient.

摘要翻译： 本发明描述了含有作为活性成分的式I的硝基芳烷基砜衍生物（I）的灭粉杀微生物组合物，其中R 1是烷基，R 2和R 3各自是氢，烷基，烷氧基，卤代烷基，卤素，氰基，硝基 或氨基或一起它们完成萘环; R4是氢或-COR5，其中R5是烷基，烷氧基，卤代烷氧基，烯基，卤代烯基，炔基，环烷基，苯基，苄基，呋喃基或四氢呋喃基。 本发明还涉及这些组合物和化合物用于刺激生殖植物生长和获得杂种种子的用途，以及制备式I范围内的肼和铵盐的方法以及制备方法 含有式I化合物作为活性成分的农药组合物。

公开(公告)号：US4451279A

公开(公告)日：1984-05-29

申请号：US260536

申请日：1981-05-04

申请人： Elmar Sturm ,  Heinrich Schempp ,  Henry Martin

发明人： Elmar Sturm ,  Heinrich Schempp ,  Henry Martin

IPC分类号： A01N25/32 ,  C07C67/00 ,  C07C313/00 ,  C07C317/28 ,  C07C317/44 ,  C07C317/48 ,  C07C323/12 ,  C07C325/00 ,  C07C327/58 ,  C07C327/60 ,  C07D307/40 ,  C07D307/56 ,  C07D307/68 ,  C07D333/38

CPC分类号： C07D307/68 ,  A01N25/32 ,  C07C327/60 ,  C07D333/38

摘要： Sulfur-containing oxime compounds of the formula I given herein are suitable for protecting cultivated plants against the phytotoxic action of aggressive agricultural chemicals, particularly herbicides. There are described methods for producing sulfur-containing oxime compounds of this type, and examples are given illustrating the application of these compounds.

公开(公告)号：US4382893A

公开(公告)日：1983-05-10

申请号：US260539

申请日：1981-05-04

申请人： Elmar Sturm ,  Heinrich Schempp ,  Henry Martin

发明人： Elmar Sturm ,  Heinrich Schempp ,  Henry Martin

IPC分类号： A01N25/32 ,  C07C67/00 ,  C07C313/00 ,  C07C317/28 ,  C07C317/44 ,  C07C317/48 ,  C07C323/12 ,  C07C325/00 ,  C07C327/58 ,  C07C327/60 ,  C07D307/40 ,  C07D307/56 ,  C07D307/68 ,  C07D333/38 ,  C07C121/80

CPC分类号： C07D307/68 ,  A01N25/32 ,  C07C327/60 ,  C07D333/38

摘要： Sulfur-containing oxime compounds of the formula I given herein are suitable for protecting cultivated plants against the phytotoxic action of aggressive agricultural chemicals, particularly herbicides. There are described methods for producing sulfur-containing oxime compounds of this type, and examples are given illustrating the application of these compounds.

摘要翻译： 本文给出的式I的含硫肟化合物适用于保护栽培植物免受侵蚀性农药，特别是除草剂的植物毒性作用。 描述了这种类型的含硫肟化合物的生产方法，并给出了这些化合物的应用实施例。