"> Avermectins substituted in the 4
    44.
    发明申请
    Avermectins substituted in the 4" and 4'-positions having pesticidal properties 有权
    在4“和4”位取代的阿维菌素具有杀虫特性

    公开(公告)号:US20060154879A1

    公开(公告)日:2006-07-13

    申请号:US10544274

    申请日:2004-02-03

    IPC分类号: A01N43/04 C07H17/08

    CPC分类号: C07H17/08

    摘要: What is described are a compound of the formula (I) Wherein A-B is —CH═CH— or —CH2—CH2—; n is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 and R3 for instance are either, (i) independently from each other for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; or (ii) together form with the nitrogen atom to which they are bound a three- to seven-membered ring, (iii) together are ═C(R4)R5; R4 and R5 are, independently from each other, for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; Y is O or S; Q is for instance H or unsubstituted or mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions.

    摘要翻译: 描述的是式(I)的化合物,其中A-B是-CH-CH-或-CH 2 -CH 2 - 。 n为0或1; R 1是C 1 -C 12烷基,C 3 -C 8烷基,C 3 -C 12烷基,C 3 -C 12烷基,C 3 -C 12烷基, >环烷基或C 2 -C 12 - 烯基; 例如,R 2和R 3是(i)彼此独立地例如-Q,-C(-Y)-Q或-C( - Y)-OQ; 或(ii)与其结合的氮原子一起形成三至七元环,(iii)一起为-C(R 4)R 5 >; R 4和R 5各自独立地为例如-Q,-C(-Y)-Q或-C(-Y)-O-Q; Y为O或S; Q是例如H或未被取代或单取代或未取代的C 1 -C 12烷基; 或者,如果合适的话,E / Z异构体,E / Z异构体混合物和/或其互变异构体; 制备这些化合物,其异构体和互变异构体的方法以及这些化合物,其异构体和互变异构体的用途; 活性化合物选自这些化合物及其互变异构体的杀虫组合物; 用于制备所述式(I)化合物的中间体,式(I)化合物的制备方法和使用这些组合物来控制害虫的方法。

    "> Avermectin and avermectin monosaccharide derivatives substituted in the 4

    公开(公告)号:US20060140997A1

    公开(公告)日:2006-06-29

    申请号:US10543637

    申请日:2004-01-30

    IPC分类号: A01N25/00 A01N43/04 C07H17/08

    CPC分类号: A01N43/90 C07H17/08

    摘要: What is described are a compound of the formula (I) Wherein U is —N(R2)OR3 or —N+(O−)═C(RE)RZ); n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 and R3 are, for example; independently from each other, -Q, —C(═O)-Z-Q or —CN; RZ and RE are, independently from each other, -Q, —C(═O)-Z-Q or —CN; or RZ and RE together are a three- to seven membered alkylene or alkenylene bridge, which is unsubstituted or mono- to tri-substituted; Z is a bond, O or —NR4—; Q is H, C1-C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12-Cycloalkyl, C5-C12-cycloalkenyl, aryl, or heterocyclyl, which are unsubstituted or mono- to pentasubstituted; R4 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl or C2-C8alkenyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions.

    Diaza-spiro [4.5] decanes useful as pesticides
    48.
    发明授权
    Diaza-spiro [4.5] decanes useful as pesticides 有权
    Diaza-spiro [4.5]癸烷可用作农药

    公开(公告)号:US08110684B2

    公开(公告)日:2012-02-07

    申请号:US12161823

    申请日:2007-01-19

    IPC分类号: C07D217/00 A61K31/44

    CPC分类号: C07D471/10 A01N43/90

    摘要: A method of combating and controlling insects, acarines, nematodes or molluscs which comprises applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, nematicidally or molluscicidally effective amount of a compound of formula (I) wherein Y is a single bond, C═O, C═S or S(O)m where m is 0, 1 or 2; and R1, R3, R2 and R8 are defined organic, groups, p is 0, 1, 2, 3 or 4 or salts or N-oxides thereof; novel compounds and composition's containing them are also provided.

    摘要翻译: 一种防治昆虫,螨虫,线虫或软体动物的方法,其包括将有害生物施用于有害生物的场所或易受害虫攻击的植物,杀虫剂,杀螨剂,杀线虫剂或杀软体动物学上有效量的化合物 其中Y是单键的式(I),C = O,C = S或S(O)m,其中m是0,1或2; R1,R3,R2和R8定义为有机基团,p为0,1,2,3或4或其盐或N-氧化物; 还提供了含有它们的新化合物和组合物。

    Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position
    49.
    发明授权
    Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position 有权
    在4“ - 或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物

    公开(公告)号:US08017589B2

    公开(公告)日:2011-09-13

    申请号:US12768280

    申请日:2010-04-27

    IPC分类号: A61K31/70 C07H17/04

    CPC分类号: C07H17/08 A61K31/7042

    摘要: What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

    摘要翻译: 描述的是下式的化合物,其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基,C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基,C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH,卤素,CN,-N 3,-NO 2,C 3 -C 8 - 环烷基,降冰片基 - ,C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基,C 1 -C 12烷氧基,C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基,C 3 -C 8环烷氧基,C 1 -C 12卤代烷氧基,C 1 -C 12烷硫基,C 3 -C 8环烷硫基, C 1 -C 12烷基亚磺酰基,C 3 -C 8环烷基亚磺酰基,C 1 -C 12卤代烷基亚磺酰基,C 3 -C 8卤代环烷基亚磺酰基,C 1 -C 12烷基磺酰基,C 3 -C 8环烷基磺酰基,C 1 -C 12卤代烷基磺酰基, 卤代环烷基磺酰基,-NR4R6,-X-C(= Y)-R4,-X-C(= Y)-Z-R4,-P(= O)(OC1-C6-烷基)2,芳基,杂环基,芳氧基, 芳硫基和杂环氧基; R3是例如任选取代的H,C 1 -C 12 - 烷基或C 1 -C 12 - 烷基,并且在适用的情况下,E / Z异构体,E / Z异构体和/或互变异构体的混合物,在每种情况下为游离形式或 盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法,以及这些化合物和组合物的用途。

    CHEMICAL COMPOUNDS
    50.
    发明申请
    CHEMICAL COMPOUNDS 失效
    化学化合物

    公开(公告)号:US20110218101A1

    公开(公告)日:2011-09-08

    申请号:US13129063

    申请日:2009-10-27

    摘要: A compound of the formula I or where W, X and Y are for example each CH; R1 is H; R2 is halogen; and R6 is, for formula I, for example, OH, CN, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C6-alkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkenyloxy, C2-C6-alkynyl, C2-C6-haloalkynyl, C2-C6-alkynyloxy, optionally substituted C1 to C3-alkyl, or optionally substituted C1-C6-alkoxy, or R6 is, for formula II, for example, CN, C3-C8-cycloalkyl, or optionally substituted C3-C6-alkyl; and/or salts thereof; and their use as as pesticidal agents.

    摘要翻译: 式I化合物或其中W,X和Y为例如CH; R1是H; R2是卤素; 对于式I,R 6为例如OH,CN,C 3 -C 8 - 环烷基,C 3 -C 8 - 环烷基-C 1 -C 6烷基,C 2 -C 6 - 烯基,C 2 -C 6 - 卤代烯基,C 2 -C 6 - 烯氧基 ,C 2 -C 6炔基,C 2 -C 6 - 卤代炔基,C 2 -C 6 - 炔氧基,任选取代的C 1至C 3 - 烷基或任选取代的C 1 -C 6 - 烷氧基,或R 6为式II,例如CN,C 3 -C 8 - 环烷基或任选取代的C 3 -C 6 - 烷基; 和/或其盐; 以及其作为杀虫剂的用途。