公开(公告)号：US20050272749A1

公开(公告)日：2005-12-08

申请号：US10531981

申请日：2003-11-04

申请人： Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04

摘要： 5-Alkyl-7-aminotriazolopyrimidines of the formula I, where: R1, R2 are hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cycloalkyl, phenyl, naphthyl; 5- or 6-membered saturated, unsaturated or aromatic heterocyclyl which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or R1 and R2 together with the bridging nitrogen atom can form a 5- or 6-membered ring which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 is cycloalkyl or bicycloalkyl; where R1, R2 and R3 may be substituted as outlined in the description; X is alkyl or haloalkyl; and their salts; processes and intermediates for their preparation, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的5-烷基-7-氨基三唑并嘧啶，其中：R 1，R 2是氢，烷基，烯基，炔基，卤代烷基，环烷基，苯基，萘基; 含有1-4个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元饱和，不饱和或芳族杂环基; 或R 1和R 2与桥连氮原子一起可以形成含有1-4个氮原子或一至三个氮原子的5-或6-元环，并且 一个硫或氧原子; R 3是环烷基或双环烷基; 其中R 1，R 2和R 3可以如说明书中概述的那样被取代; X是烷基或卤代烷基; 和它们的盐; 描述了其制备方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20050256138A1

公开(公告)日：2005-11-17

申请号：US10513030

申请日：2003-04-30

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewhr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewhr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07C69/65 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C69/65

摘要： Disclosed are a method for producing fungicidal triazolopyrimidine compounds, agents containing said compounds, and the use thereof for controlling harmful fungi. Also disclosed are triazolopyrimidines of formula (1), in which the substituents have the following meaning: L1 represents alkyl; L2 represents halogen; L3represents hydrogen or halogen; X represents halogen, cyano, alkyl, alkoxy, or haloalkoxy; R1, R2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, alkenyl, alkadienyl, alkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-unit to ten-unit saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group O, N, or S. R1 and R2 can also form a five-unit or six-unit ring along with the nitrogen atom to which they are linked. Said ring can be interrupted and/or substituted by an atom from the group O, N, and S while R1 and/or R2 can be substituted according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing said compounds, and the use thereof for controlling harmful fungi.

摘要翻译： 公开了生产杀真菌三唑并嘧啶化合物的方法，含有所述化合物的试剂及其用于控制​​有害真菌的用途。 还公开了式（1）的三唑并嘧啶，其中取代基具有以下含义：L 1表示烷基; L 2表示卤素; L 3表示氢或卤素; X表示卤素，氰基，烷基，烷氧基或卤代烷氧基; R 1，R 2代表氢，烷基，卤代烷基，环烷基，烯基，链二烯基，炔基或环炔基，苯基，萘基或五个单元至十个单元 饱和的，部分不饱和的或芳族杂环，其含有一至四个O，N或S的杂原子.R 1和R 2也可以形成五单元或 六单元环与它们所连接的氮原子一起。 所述环可以被O，N和S基团的原子中断和/或取代，而R 1和/或R 2可以根据描述被取代 。 本发明还涉及用于生产所述化合物的方法和中间产物，含有所述化合物的试剂及其用于控制​​有害真菌的用途。

公开(公告)号：US20060199801A1

公开(公告)日：2006-09-07

申请号：US10551810

申请日：2004-04-16

申请人： Jordi i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Jordi i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/551 ,  A61K31/541 ,  A61K31/53 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Bicyclic compounds of the formula I in which A1 or A5 is C and the other of the two variables A1, A5 is N, C or C—R3; A2, A3, A4 independently of one another are N or C—R3a, where one of the variables A2, A3 or A4 may also be S or a group N—R4 if A1 and A5 are both C, and where A4 is not N or C—R3a if A1 is N, A3 is C—R3a and A5 is C, and where A1 is attached to A2 and A3 to A4 or A2 is attached to A3 and A4 to A5 or A1 is attached to A5 and A2 to A3 or A1 is attached to A5 and A3 to A4 or A1 is attached to A2 and A4 to A5 by double bonds; n is 0, 1, 2, 3, 4 or 5; Ra is halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R5; R1 is halogen, cyano, C1-C10-alkyl, where a carbon atom of the C1-C10-alkyl radical may be replaced by a silicium atom, C1-C6-haloalkyl, C2-C10-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C4-alkyl, where the cycloalkyl moiety of the two last-mentioned groups may be unsubstituted or contain 1, 2, 3, 4, 5, or 6 radicals selected from the group consisting of C1-C4-alkylidene, C1-C4-alkyl, halogen, C1-C4-haloalkyl and hydroxy and the alkyl moiety of C3-C8-cycloalkyl-C1-C4-alkyl may be unsubstituted or contain 1, 2, 3, or 4 radicals selected from the group consisting of halogen, C1-C4-haloalkyl and hydroxy, C5-C8-cycloalkenyl which may be unsubstituted or contain 1, 2, 3 or 4 radicals selected from the group consisting of C1-C4-alkyl, halogen, C1-C4-haloalkyl and hydroxy, OR6, SR6, NR7R8, a radical of the formula —C(R11)(R12)C(═NOR13)(R14) or a radical of the formula —C(═NOR15)C(═NOR16)(R17); R2 is halogen, cyano, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C5-C8-cycloalkenyl, OR6, SR6 or NR7R8; and the agriculturally acceptable salts of the compounds I, crop protection compositions comprising at least one compound of the formula I and/or an agriculturally acceptable salt of I and at least one solid or liquid carrier and a method for controlling phytopathogenic harmful fungi are described.

公开(公告)号：US20060167017A1

公开(公告)日：2006-07-27

申请号：US10539039

申请日：2003-12-16

申请人： Bernd Muller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Bernd Muller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04

摘要： Triazolopyrimidines of the formula I where the index and the substituents are as defined below: R1 is C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, C3-C10-cycloalkyl, C3-C10-cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon to the triazolopyrimidine and contains one to four heteroatoms from the group consisting of N, O and S; R2 is C1-C4-alkyl which may be substituted by halogen, cyano, nitro or C1-C2-alkoxy; n is 0 or an integer from 1 to 4; R is as defined in the description; X is SOm—Rx, NRxRy or NRx—(C═O)—Ry; m is 0 or an integer from 1 to 3; and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 其中指数和取代基如下定义的式I的三唑并嘧啶：R 1是C 1 -C 10 - 烷基， C 1 -C 10亚烷基，C 2 -C 10 - 炔基，C 3 - 亚烷基 C 1 -C 10 - 环烷基，C 3 -C 10 - 环烯基，苯基，萘基或五至十元饱和的， 部分不饱和或芳族杂环，其通过碳连接到三唑并嘧啶并且包含一至四个由N，O和S组成的组的杂原子; R 2是可以被卤素，氰基，硝基或C 1 H 3取代的C 1 -C 4 - 烷基 -C 2 - 烷氧基; n为0或1至4的整数; R如说明书所定义; X是SO x，x，x，x，y，x，y，x， - （CO）-R y; m为0或1〜3的整数; 并描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US20050272748A1

公开(公告)日：2005-12-08

申请号：US10531980

申请日：2003-11-14

申请人： Jordi Tormo Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 2-Mercapto-substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy or —C(═O)-A; A is hydrogen, hydroxyl, alkyl, alkenyl, alkoxy, haloalkoxy, alkylamino or dialkylamino; m is 0, 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four hetero atoms from the group consisting of O, N and S; R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S; where R1 and/or R2 may be substituted as stated in the description; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 2-巯基取代的式Ⅰ的三唑并嘧啶，其中取代基如下：L是卤素，氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基或-C ）-一个; A是氢，羟基，烷基，烯基，烷氧基，卤代烷氧基，烷基氨基或二烷基氨基; m为0,1,2,3,4或5; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 至10元饱和，部分不饱和或芳族杂环，其含有一个至四个由O，N和S组成的组的杂原子; R 1和R 2与它们所连接的氮原子一起也可以形成五元或六元环，其可被来自基团的原子中断 由O，N和S组成; 其中R 1和/或R 2可以如描述中所述被取代; 描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US06344589B1

公开(公告)日：2002-02-05

申请号：US09830970

申请日：2001-05-03

申请人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Herbert Bayer ,  Norbert Götz ,  Roland Götz

发明人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Herbert Bayer ,  Norbert Götz ,  Roland Götz

IPC分类号： C07C24900

CPC分类号： C07C249/06 ,  C07C249/08 ,  C07C251/40

摘要： A process for preparing bis(oxime) monoethers of the formula I, where: R1 is unsbustituted C1-C4-alkyl or C2-C4-alkenyl-, C2-C4-alkynyl- or phenyl-substituted methyl; R2,R4 independently of one another are hydrogen or methyl; R3,R5 independently of one another are hydrogen or C1-C4-alkyl, trifluoromethyl or phenyl, and intermediates which are obtainable by this process are described.

摘要翻译： 制备式I的双（肟）单醚的方法，其中：R1是未取代的C1-C4-烷基或C2-C4-烯基 - ，C2-C4-炔基或苯基取代的甲基; R2，R4独立地为一 另一个是氢或甲基; R 3，R 5彼此独立地是氢或C 1 -C 4 - 烷基，三氟甲基或苯基，以及可通过该方法获得的中间体。

公开(公告)号：US07488732B2

公开(公告)日：2009-02-10

申请号：US10549936

申请日：2004-03-30

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： C07D239/28 ,  C07D239/34 ,  C07D239/42 ,  C07D239/46 ,  A01N43/54

CPC分类号： A01N43/54 ,  C07D239/28 ,  C07D239/30

摘要： 2-Substituted pyrimidines of the formula I in which the index n and the substituents L, Ra, Rb, Rc, Rz, Ru, Rv, A′, A″ and A′″ are as defined in the description and: R1 is C3-C10-alkyl, C3-C10-alkenyl, C3-C10-alkynyl, C3-C12-cycloalkyl, C3-C10-cycloalkenyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon and contains one to four heteroatoms from the group consisting of O, N and S, R2 is halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy, C3-C4-alkenyloxy or C3-C4-alkynyloxy, where the alkyl, alkenyl and alkynyl radicals of R2 may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl, and R3 is cyano, CO2Ra, C(═O)NRzRb, C(═O)—N—ORb, C(═S)—NRaRb, C(═NORa)NRzRb, C(═NRa)NRzRb, C(═O)NRa—NRzRb, C(═N—NRzRc)NRaRb, C(═O)Ra, C(═NORb)Ra, C(═N—NRzRb)Ra, CRaRb—ORz, CRaRb—NRzRc, ON(═CRaRb), O—C(═O)Ra, NRaRb′, NRa(C(═O)Rb), NRa(C(═O)ORb), NRa(C(═O)—NRzRb), NRa(C(═NRc)Rb), NRa(N═CRcRb), NRa—NRzRb, NRz—ORa, NRa(C(═NRc)—NRzRb), NRa(C(═NORc)Rb), processes for preparing these compounds, compositions comprising these compounds and their pesticidal use are described.

摘要翻译： 其中指数n和取代基L，Ra，Rb，Rc，Rz，Ru，Rv，A'，A“和A”'如说明书中所定义的式I的2-取代的嘧啶：R1 C 3 -C 10 - 烷基，C 3 -C 10 - 烯基，C 3 -C 10 - 炔基，C 3 -C 12 - 环烷基，C 3 -C 10 - 环烯基或五至十元饱和的部分不饱和或芳族杂环，其通过碳 并且含有一至四个由O，N和S组成的组的杂原子，R2是卤素，氰基，C1-C4-烷基，C2-C4-烯基，C2-C4-炔基，C1-C4-烷氧基，C3-C4 - 烯氧基或C 3 -C 4 - 炔氧基，其中R 2的烷基，烯基和炔基可以被卤素，氰基，硝基，C 1 -C 2 - 烷氧基或C 1 -C 4 - 烷氧基羰基取代，并且R 3是氰基，CO 2 R a，C（ -O）NR z R b，C（-O）-N-OR b，C（-S）-NR a R b，C（-NOR a）NR z R b，C（-NR a）NR z R b，C（O）NR a -NR b R b，C -NRaRb，C（-O）Ra，C（-NORb）Ra，C（-N-NRzRb）Ra，CRaRb-ORz，CRaRb-NRzRc，ON（-CRaRb），OC（-O）Ra，NRaRb ，NR a（C（-O）R b），NR a（C（-O）R b），NR a（C（-O）OR b） NRa-N RzRb，NRz-ORa，NRa（C（-NRc）-NRzRb），NRa（C（-NORc）Rb），制备这些化合物的方法，包含这些化合物的组合物及其杀虫剂用途。

公开(公告)号：US07375108B2

公开(公告)日：2008-05-20

申请号：US10564013

申请日：2004-07-15

申请人： Anja Schwögler ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Andreas Gypser ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schäfer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwögler ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Andreas Gypser ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schäfer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： C07D239/42 ,  A01N43/54

CPC分类号： C07D239/42

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents R1 to R3 and L are as defined in the description and R4 corresponds to one of the formulae in which Ra, X and Rb are as defined in the description; and also to processes for preparing these compounds, to pesticidal compositions comprising these compounds and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基R 1至R 3和L如说明书中所定义， SUP> 4 对应于其中R a，S，X和R b的定义之一如说明书中所定义; 以及制备这些化合物的方法，包括这些化合物的农药组合物及其作为农药的用途。

公开(公告)号：US20060211711A1

公开(公告)日：2006-09-21

申请号：US10550571

申请日：2004-03-30

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-alkinylamino-triazolopyrimidins of formula (I), wherein the substituents have the following meanings: L=halogen, alkyl, halogenalkyl, alkoxy, amino, NHR, NR2, cyano, S(O)nA1 or C(O)A2; R=alkyl or alkylcarbonyl, A1=hydrogen, hydroxy, alkyl, alkylamino or aialkylamino; n=0, 1 or 2; A2=alkenyl, alkoxy, halogenalkoxy or one of the groups cited in A1; m=1, 2, 3, 4 or 5, whereby at least one group L is present in an ortho-position to the bond with the triazolopyrimidine skeleton; X=halogen, cyano, alkyl, halogenalkyl or alkoxy; R1=hydrogen or alkyl; R2=alkinyl which can be unsubstituted or substituted according to the description. The invention also relates to methods for the production of said compounds, agents containing said compounds and the use thereof to combat harmful phytopathogenic fungi.

摘要翻译： 式（I）的7-烷基氨基 - 三唑并嘧啶类，其中取代基具有以下含义：L =卤素，烷基，卤代烷基，烷氧基，氨基，NHR，NR 2，氰基，S（O） 或者C（O）A 2 O 2。 R =烷基或烷基羰基，A 1〜H 2，羟基，烷基，烷基氨基或亚烷基氨基; n = 0,1或2; 链烯基，烷氧基，卤代烷氧基或A 1中引用的基团之一; m = 1,2,3,4或5，其中至少一个基团L存在于与三唑并嘧啶骨架的键的邻位; X =卤素，氰基，烷基，卤代烷基或烷氧基; R 1 =氢或烷基; R 2 =炔基，其可以是未取代的或根据描述取代的。 本发明还涉及生产所述化合物的方法，含有所述化合物的试剂及其用于对抗有害植物病原真菌的用途。

公开(公告)号：US07501530B2

公开(公告)日：2009-03-10

申请号：US10548840

申请日：2004-03-20

申请人： Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Andreas Gypser ,  Jordi Tormo i Blasco ,  Anja Schwögler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Frank Schieweck ,  Michael Rack ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether

发明人： Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Andreas Gypser ,  Jordi Tormo i Blasco ,  Anja Schwögler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Frank Schieweck ,  Michael Rack ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether

IPC分类号： C07D333/22 ,  C07C333/32 ,  A01N25/00 ,  C07C335/00 ,  A01N25/32

CPC分类号： C07D333/38

摘要： The invention relates to novel biphenyl carboxamides of formula (I), wherein A, R, Z, X, Y, m and n have the meanings given in the description, to multiple methods for producing these substances, to their use for combating unwanted micro-organisms and to novel intermediate products and the production thereof.

摘要翻译： 本发明涉及式（I）的新型联苯甲酰胺，其中A，R，Z，X，Y，m和n具有与本说明书中给出的含义相同的多种生产这些物质的方法，用于防治不想要的微生物 和新颖的中间产品及其生产。