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公开(公告)号:US20110152535A1
公开(公告)日:2011-06-23
申请号:US13039137
申请日:2011-03-02
申请人: Joachim Rheinheimer , Wolfgang von Deyn , Joachim Gebhardt , Michael Rack , Rene Lochtman , Norbert Götz , Michael Keil , Matthias Witschel , Helmut Hagen , Ulf Mißlitz , Ernst Baumann
发明人: Joachim Rheinheimer , Wolfgang von Deyn , Joachim Gebhardt , Michael Rack , Rene Lochtman , Norbert Götz , Michael Keil , Matthias Witschel , Helmut Hagen , Ulf Mißlitz , Ernst Baumann
IPC分类号: C07D261/04
CPC分类号: C07C249/06 , C07C201/10 , C07C201/12 , C07C205/44 , C07C209/62 , C07C251/48 , C07C253/00 , C07C255/50 , C07C315/04 , C07C319/14 , C07D261/04 , C07D413/10 , C07C323/09 , C07C317/24 , C07C317/32 , C07C205/06 , C07C211/52
摘要: A process is described for preparing isoxazoles of the formula I where the substituents are as defined below: R1 is hydrogen, C1-C6-alkyl, R2 is C1-C6-alkyl, R3, R4, R5 are hydrogen, C1-C6-alkyl, or R4 and R5 together form a bond, R6 is a heterocyclic ring, n is 0, 1 or 2; which comprises preparing an intermediate of the formula VI where R1, R3, R4 and R5 are as defined above, followed by halogenation, thiomethylation, oxidation and acylation to give compounds of the formula I. Also novel intermediates for preparing the compounds of the formula I and novel processes for preparing the intermediates are described.
摘要翻译: 描述了制备式I的异恶唑的方法,其中取代基如下所定义:R 1是氢,C 1 -C 6烷基,R 2是C 1 -C 6烷基,R 3,R 4,R 5是氢,C 1 -C 6 - 烷基 ,或R4和R5一起形成键,R6是杂环,n是0,1或2; 其包括制备式VI的中间体,其中R 1,R 3,R 4和R 5如上定义,然后进行卤化,硫甲基化,氧化和酰化,得到式I化合物。还有用于制备式I化合物的中间体 并描述了制备中间体的新方法。
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公开(公告)号:US06528455B1
公开(公告)日:2003-03-04
申请号:US10148909
申请日:2002-06-05
申请人: Gerhard Hamprecht , Michael Puhl , Robert Reinhard , Ingo Sagasser , Cyrill Zagar , Karl-Otto Westphalen , Matthias Witschel , Helmut Walter
发明人: Gerhard Hamprecht , Michael Puhl , Robert Reinhard , Ingo Sagasser , Cyrill Zagar , Karl-Otto Westphalen , Matthias Witschel , Helmut Walter
IPC分类号: C07D23954
CPC分类号: C07D209/48 , C07C205/37 , C07C217/84 , C07C265/12 , C07C331/28 , C07D239/54 , C07D239/56 , C07D251/38
摘要: Phenoxy- and thiophenoxyacrylic acid compounds of the formula I in which Het, R1, R2, R3, V, W and Z are as defined in claim 1 and processes for their preparation, intermediates for their preparation, herbicidally active compositions comprising the compounds of the formula I and a method for controlling harmful fungi are described.
摘要翻译: 其中Het,R1,R2,R3,V,W和Z如权利要求1所定义的式Iin的苯氧基和硫代苯氧基丙烯酸化合物及其制备方法,其制备中间体,除草活性组合物,其包含式 描述了一种控制有害真菌的方法。
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公开(公告)号:US20090186766A1
公开(公告)日:2009-07-23
申请号:US12300884
申请日:2007-05-11
申请人: Matthias Witschel , Cyrill Zagar , Eike Hupe , Toralf Kühn , William Karl Moberg , Liliana Parra Rapado , Frank Stelzer , Andrea Vescovi , Michael Rack , Robert Reinhard , Bernd Sievernich , Klaus Grossmann , Thomas Ehrhardt
发明人: Matthias Witschel , Cyrill Zagar , Eike Hupe , Toralf Kühn , William Karl Moberg , Liliana Parra Rapado , Frank Stelzer , Andrea Vescovi , Michael Rack , Robert Reinhard , Bernd Sievernich , Klaus Grossmann , Thomas Ehrhardt
IPC分类号: A01N43/56 , C07D231/12 , A01P13/00
CPC分类号: C07D231/14 , A01N43/10 , A01N43/56 , C07D405/12
摘要: The present invention relates to heteroaroyl-substituted alanines of the formula I in which the variables A and R1 to R8 are as defined in the description, and to their agriculturally useful salts, to processes and intermediates for their preparation, and to the use of these compounds or of compositions comprising these compounds for controlling unwanted plants.
摘要翻译: 本发明涉及式I中的杂芳酰基取代的丙氨酸,其中变量A和R 1至R 8如说明书中所定义,以及其农业上有用的盐,其制备方法和中间体以及这些 化合物或包含这些化合物的组合物以控制不想要的植物。
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公开(公告)号:US20070270312A1
公开(公告)日:2007-11-22
申请号:US11662586
申请日:2005-09-14
申请人: Matthias Witschel , Frank Stelzer , Toralf Kuhn , Liliana Rapado , Michael Rack , Eike Hupe , Cyrill Zagar , Robert Reinhard , Bernd Sievernich , Thomas Ehrhardt
发明人: Matthias Witschel , Frank Stelzer , Toralf Kuhn , Liliana Rapado , Michael Rack , Eike Hupe , Cyrill Zagar , Robert Reinhard , Bernd Sievernich , Thomas Ehrhardt
IPC分类号: A01N43/10 , A01N43/42 , A01N43/48 , A01N43/56 , A01P13/00 , C07D215/38 , C07D231/00 , C07D333/22 , C07D401/00
CPC分类号: A01N43/56 , A01N43/10 , A01N43/38 , A01N43/40 , A01N43/42 , A01N43/78 , C07D307/68 , C07D333/38 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D417/12
摘要: The present invention relates to heteroaroyl-substituted serinamides of the formula I in which the variables A, Het and R1 to R5 are as defined in the description, and to their agriculturally useful salts, to processes and intermediates for their preparation, and to the use of these compounds or of the compositions comprising these compounds for controlling unwanted plants.
摘要翻译: 本发明涉及式I的杂芳酰取代的丝氨酰胺,其中变量A,Het和R 1至R 5如描述中所定义,并且与它们 农业上有用的盐,其制备方法和中间体,以及这些化合物或包含这些化合物的组合物用于防治有害植物的用途。
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公开(公告)号:US07851411B2
公开(公告)日:2010-12-14
申请号:US10499522
申请日:2002-12-17
申请人: Peter Plath , Norbert Götz , Michael Rack , Andreas Landes , Cyrill Zagar , Matthias Witschel , Klaus Groβmann
发明人: Peter Plath , Norbert Götz , Michael Rack , Andreas Landes , Cyrill Zagar , Matthias Witschel , Klaus Groβmann
IPC分类号: A01N43/36 , A01N37/00 , A01N37/34 , C07D295/104 , C07D305/06 , C07C255/07
CPC分类号: C07D295/185 , A01N37/44 , A01N43/08 , A01N43/16 , C07C255/30 , C07C323/60 , C07C327/22 , C07C2601/02 , C07C2601/08 , C07C2601/14 , C07D305/08 , C07D307/18 , C07D307/20 , C07D307/22 , C07D309/14 , C07D319/06 , C07D331/04
摘要: α-Cyanoacrylates of the formula I, where: R1 is ORa wherein Ra is hydrogen, substituted alkyl, branched alkyl, branched alkenyl, cycloloalkyl, heterocyclyl, aryl, phenylalkyl or alkylimino; is NRbRc wherein Rb is hydrogen, alkyl which may be substituted, alkenyl, alkynyl; Rc is hydrogen, alkyl which may be substituted alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, phenylalkyl or alkylimino; or Rb and Rc form an alkandiyl-chain which may be substituted; or is SRd wherein Rd is hydrogen, alkyl which may be substituted, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, phenylalkyl or alkylimino; R2 is alkyl which may be substituted; is alkenyl or alkynyl; R3 is alkyl may be substituted; is alkenyl or alkynyl; R4 is hydrogen, halogen, cyano or alkyl; and their agriculturally useful salts, processes and intermediates for their preparation; and the use of these compounds or of compositions comprising these compounds for controlling undesirable plants are described.
摘要翻译: 式I的α-氰基丙烯酸酯,其中:R 1是OR a,其中R a是氢,取代的烷基,支链烷基,支链烯基,环烷基,杂环基,芳基,苯基烷基或烷基亚氨基; 是NRbRc,其中Rb是氢,可以被取代的烷基,烯基,炔基; Rc是氢,可以被取代的烯基,炔基,环烷基,杂环基,芳基,苯基烷基或烷基亚氨基的烷基; 或R b和R c形成可被取代的烷撑二链; 或者是其中Rd为氢的SRd,可以被取代的烷基,烯基,炔基,环烷基,杂环基,芳基,苯基烷基或烷基亚氨基; R2是可被取代的烷基; 是烯基或炔基; R3是烷基可以被取代; 是烯基或炔基; R4是氢,卤素,氰基或烷基; 及其农业上有用的盐,其制备方法和中间体; 并且描述了这些化合物或包含这些化合物的组合物用于防治不期望的植物的用途。
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公开(公告)号:US20090137396A1
公开(公告)日:2009-05-28
申请号:US12159686
申请日:2007-01-04
申请人: Eike Hupe , Cyrill Zagar , Matthias Witschel , Toralf Kuehn , William Karl Moberg , Liliana Parra Rapado , Frank Stelzer , Andrea Vescovi , Robert Reinhard , Bernd Sievernich , Klaus Grossmann , Thomas Ehrhardt
发明人: Eike Hupe , Cyrill Zagar , Matthias Witschel , Toralf Kuehn , William Karl Moberg , Liliana Parra Rapado , Frank Stelzer , Andrea Vescovi , Robert Reinhard , Bernd Sievernich , Klaus Grossmann , Thomas Ehrhardt
IPC分类号: A01N43/84 , A01N43/60 , C07D241/04 , A01P21/00 , C07D413/08
CPC分类号: C07D241/18 , A01N43/60 , A01N43/653 , A01N43/713 , A01N43/80 , A01N55/00 , C07D241/08 , C07D403/06 , C07D409/06 , C07D413/06 , C07D417/06
摘要: The present invention relates to the use of piperazine compounds of the formula I or of the agriculturally useful salts of piperazine compounds of the formula I as herbicides, where in formula I the variables are as defined in the claims and the description.Moreover, the invention relates to compositions comprising, in addition to auxiliaries customary for formulating crop protection agents, piperazine compounds of the formula I or agriculturally useful salts of I, and to a process for preparing these compositions. Furthermore, the invention relates to certain piperazine compounds of the formula I, a process for preparing piperazine compounds of the formula I and a method for controlling unwanted vegetation which comprises treating plants, their seeds and/or their habitat with at least one piperazine compound of the formula I.
摘要翻译: 本发明涉及式I的哌嗪化合物或式I的哌嗪化合物的农业上可用的盐作为除草剂的用途,其中在式I中,变量如权利要求和说明书所定义。 此外,本发明涉及除了常规用于配制作物保护剂的助剂,式I的哌嗪化合物或I的农业上有用的盐以及制备这些组合物的方法之外,本发明涉及组合物。 此外,本发明涉及式I的某些哌嗪化合物,一种制备式I的哌嗪化合物的方法和一种防治有害植物的方法,其包括用至少一种哌嗪化合物处理植物,其种子和/或其栖息地 公式一
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公开(公告)号:US20090054240A1
公开(公告)日:2009-02-26
申请号:US12279425
申请日:2007-02-07
申请人: Matthias Witschel , Cyrill Zagar , Eike Hupe , Toralf Kuhn , William Karl Moberg , Liliana Parra Rapado , Frank Stelzer , Andrea Vescovi , Michael Rack , Robert Reinhard , Bernd Sievernich , Klaus Grossmann , Thomas Ehrhardt
发明人: Matthias Witschel , Cyrill Zagar , Eike Hupe , Toralf Kuhn , William Karl Moberg , Liliana Parra Rapado , Frank Stelzer , Andrea Vescovi , Michael Rack , Robert Reinhard , Bernd Sievernich , Klaus Grossmann , Thomas Ehrhardt
IPC分类号: A01N43/56 , C07D231/14 , C07D333/24 , C07D307/68 , A01N43/10 , C07D405/02 , A01P13/00
CPC分类号: C07D231/12 , C07D333/06 , C07D401/12 , C07D403/12 , C07D407/12
摘要: The present invention relates to heteroaroyl-substituted alanines of the formula I in which the variables A and R1 to R7 are as defined in the description, and to their agriculturally useful salts, to processes and intermediates for their preparation, and to the use of these compounds or of compositions comprising these compounds for controlling unwanted plants.
摘要翻译: 本发明涉及式I的杂芳酰基取代的丙氨酸,其中变量A和R 1至R 7如说明书中所定义,并且其农业上有用的盐,其制备方法和中间体以及这些 化合物或包含这些化合物的组合物以控制不想要的植物。
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公开(公告)号:US20090036311A1
公开(公告)日:2009-02-05
申请号:US12279351
申请日:2007-02-07
申请人: Matthias Witschel , Cyrill Zagar , Eike Hupe , Toralf Kuhn , William Karl Moberg , Liliana Parra Rapado , Frank Stelzer , Andrea Vescovi , Robert Reinhard , Bernd Sievernich , Klaus Grossmann , Thomas Ehrhardt
发明人: Matthias Witschel , Cyrill Zagar , Eike Hupe , Toralf Kuhn , William Karl Moberg , Liliana Parra Rapado , Frank Stelzer , Andrea Vescovi , Robert Reinhard , Bernd Sievernich , Klaus Grossmann , Thomas Ehrhardt
IPC分类号: A01N37/18 , C07C237/34 , C07C229/34 , A01N37/44 , A01P13/00
CPC分类号: C07D307/14 , C07C237/22 , C07C271/22 , C07C275/16 , C07C311/06 , C07C311/58 , C07C335/08 , C07C335/10 , C07D309/04 , C07D309/20
摘要: The present invention relates to benzoyl-substituted alanines of the formula I in which the variables R1 to R12 are as defined in the description, and to their agriculturally useful salts, to processes and intermediates for their preparation, and to the use of these compounds or of compositions comprising these compounds for controlling unwanted plants.
摘要翻译: 本发明涉及式I的苯甲酰基取代的丙氨酸,其中变量R1至R12如说明书中所定义,及其农业上有用的盐,其制备方法和中间体以及这些化合物或 包含这些化合物的组合物用于防治有害植物。
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公开(公告)号:US20070093390A1
公开(公告)日:2007-04-26
申请号:US10548733
申请日:2004-03-10
申请人: Matthias Witschel , Cyrill Zagar , Andreas Landes , Peter Dombo
发明人: Matthias Witschel , Cyrill Zagar , Andreas Landes , Peter Dombo
IPC分类号: A01N43/60
CPC分类号: C07D487/04 , A01N43/90 , A01N61/00 , A01N2300/00
摘要: A synergistic herbicidal mixture comprising A) [N-(5,7-Dimethoxy(1,2,4)triazolo[1,5-a]pyrimidin-2-yl)-2-methoxy-4-(trifluoro methyl)]-3-pyridinesulfonamide (I) or one of its environmentally compatible salts; B) at least a synergistically effective amount of a herbicidal compound from the group of the p-hydroxyphenylpyruvatdioxygenase (HPPD)-inhibitors; and, if desired, C) at least a safener selected from the group of dichlormid, benoxacor, LAB 145, 138, MG-191, furilazole, cyometrinil, oxabetrinil, fluoxfenim, flurazole, naphtalic acid anhydride, fenclorim, fenchlorazole, mefenpyr, isoxadifen, cloquintocet, 1-ethyl-4-hydroxy-3-(1H-tetrazol-5-yl)-1H-quinolin-2-one, 4-carboxy methyl-chroman-4carboxylic acid, N-(2-methoxy-benzoyl)-4-(3-methylureido)benzenesulfonamide, (3-oxo-isothiochroman-4ylidenemethoxy)-acetic acid methyl ester; or their environmentally compatible salts, amides, esters and hydrates. Compositions comprising these mixtures, processes for the preparation of these compositions and their use for controlling undesired plants.
摘要翻译: 一种协同除草混合物,其包含A)[N-(5,7-二甲氧基(1,2,4)三唑并[1,5-a]嘧啶-2-基)-2-甲氧基-4-(三氟甲基)] - 3-吡啶磺酰胺(I)或其与环境相容的盐之一; B)至少一种协同有效量的来自对羟基苯基丙酮酸加氧酶(HPPD)抑制剂的除草化合物; 如果需要,C)至少一种选自二倍体,benoxacor,LAB 145,138,MG-191,氟唑,cyometrinil,oxabetrinil,氟西芬,氟尿嘧啶,萘酸酐,芬舍林,芬氯唑,mefenpyr,异恶唑 ,1-乙基-4-羟基-3-(1H-四唑-5-基)-1H-喹啉-2-酮,4-羧基甲基 - 苯并二氢吡喃-4-羧酸,N-(2-甲氧基 - 苯甲酰基) -4-(3-甲基脲基)苯磺酰胺,(3-氧代 - 异硫苯并二氢吡喃-4-基亚甲基乙氧基) - 乙酸甲酯; 或其环境相容的盐,酰胺,酯和水合物。 包含这些混合物的组合物,用于制备这些组合物的方法及其用于防治不想要的植物的用途。
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公开(公告)号:US20060293187A1
公开(公告)日:2006-12-28
申请号:US10548815
申请日:2004-03-05
申请人: Cyrill Zagar , Matthias Witschel , Andreas Landes
发明人: Cyrill Zagar , Matthias Witschel , Andreas Landes
CPC分类号: A01N43/54 , A01N2300/00 , A01N43/40
摘要: A herbicidal mixture comprising 3-Phenyluracils of the formula (I) in which the variables R1-R7 are as defined below: R1 is methyl or NH2; R2 is haloalkyl; R3 is hydrogen or halogen; R4 is halogen or cyano; R5 is hydrogen, cyano, alkyl, alkoxy, alkoxyalkyl, cyclo-alkyl, alkenyl, alkynyl or optionally substituted benzyl; R6, R7 are hydrogen, optionally substituted alkyl, alkoxy, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, phenyl or benzyl; or R6, R7 together with the nitrogen atom form a 3- to 7-membered saturated or unsaturated optionally substituted hetero-cycle, including their agriculturally acceptable salts; and at least one further herbicide B; and optionally at least one safener C.
摘要翻译: 包含式(I)的3-苯基尿嘧啶的除草混合物,其中变量R 1〜R 7如下所定义:R 1〜 是甲基或NH 2; R 2是卤代烷基; R 3是氢或卤素; R 4是卤素或氰基; R 5是氢,氰基,烷基,烷氧基,烷氧基烷基,环烷基,烯基,炔基或任选取代的苄基; R 6,R 7是氢,任选取代的烷基,烷氧基,烯基,炔基,环烷基,环烯基,苯基或苄基; 或R 6,R 7与氮原子一起形成3-至7-元饱和或不饱和的任选取代的杂环,包括其农业上可接受的盐; 和至少一种另外的除草剂B; 和任选的至少一种安全剂C.
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