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公开(公告)号:US07038043B1
公开(公告)日:2006-05-02
申请号:US09482235
申请日:2000-01-13
IPC分类号: C07D273/00
CPC分类号: C07D498/22 , C07C45/68
摘要: Indolocarbazoles are furanosylated (e.g., 7) with acetals (e.g., 8) or their open chain congeners (e.g., 9) under conditions known to promote acetal exchange or formation, such as protic or Lewis acids. Furanosylated indolocarbazoles (e.g., 10) are also prepared via ring contraction of pyranosylated indolocarbazoles (e.g., 11) under conditions know to effect oxidation and benzylic acid type rearrangements, and pyranosylated indolocarbazoles (e.g., 11) are prepared via ring expansion of the furanosylated congeners (e.g., 10)
摘要翻译: 在已知可促进乙缩醛交换或形成的条件下,例如质子酸或路易斯酸,吲哚并吡唑类化合物(例如7)具有缩醛(例如8)或其开链同系物(例如9)。 呋喃糖基化吲哚并唑(例如,10)也是通过吡喃糖基化吲哚并唑(例如11)在已知有效氧化和苄酸型重排的条件下通过环收缩来制备的,吡喃糖基化的吲哚并唑(例如,11)是通过呋喃糖基化同系物 (例如10)
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公开(公告)号:US06182176B2
公开(公告)日:2001-01-30
申请号:US08201185
申请日:1994-02-24
申请人: Michael L. Ziegler , Robert J. Brooks , William R. Bryg , Craig R. Frink , Thomas R. Hotchkiss , Robert D. Odineal , James B. Williams , John L. Wood
发明人: Michael L. Ziegler , Robert J. Brooks , William R. Bryg , Craig R. Frink , Thomas R. Hotchkiss , Robert D. Odineal , James B. Williams , John L. Wood
IPC分类号: G06F1314
CPC分类号: G06F13/36
摘要: A shared bus system having a bus and a set of client modules coupled to the bus. Each client module is capable of sending transactions on the bus to other client modules and receiving transactions on the bus from other client modules for processing. Each module has a queue for storing transactions received by the module for processing. A bus controller limits the types of transactions that can be sent on the bus to prevent any module's queue from overflowing.
摘要翻译: 共享总线系统,其具有总线和耦合到总线的一组客户端模块。 每个客户端模块都能够将总线上的事务发送到其他客户端模块,并从其他客户端模块接收总线上的事务处理。 每个模块都有一个队列,用于存储由模块接收的事务处理。 总线控制器限制可以在总线上发送的事务的类型,以防止任何模块的队列溢出。
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公开(公告)号:US5519838A
公开(公告)日:1996-05-21
申请号:US201186
申请日:1994-02-24
申请人: Michael L. Ziegler , Robert J. Brooks , William R. Bryg , Kenneth K. Chan , Thomas R. Hotchkiss , Robert E. Naas , Robert D. Odineal , Brendan A. Voge , James B. Williams , John L. Wood
发明人: Michael L. Ziegler , Robert J. Brooks , William R. Bryg , Kenneth K. Chan , Thomas R. Hotchkiss , Robert E. Naas , Robert D. Odineal , Brendan A. Voge , James B. Williams , John L. Wood
IPC分类号: G06F13/368 , G06F13/00
CPC分类号: G06F13/368
摘要: A bus system having a bus arbitration scheme. The bus system includes a bus and a plurality of client modules coupled to the bus. Each of the client modules is capable of transmitting information on the bus to another of client module, and only one client module is entitled to transmit information on the bus at any time. A module entitled to transmit information on the bus has control of the bus for a minimum period of time defining a cycle. To determine which module is entitled to use the bus, each client module generates an arbitration signal when it seeks to transmit information on the bus. Each client module has an arbitration signal processor responsive to the arbitration signals for determining whether the module is entitled to transmit information on said bus. The system preferably also contains a host module that informs the client modules what types of transactions allowed on the bus in a given cycle. Each arbitration signal processor preferably is also responsive to the client option signals sent by the host module during an earlier cycle.
摘要翻译: 具有总线仲裁方案的总线系统。 总线系统包括总线和耦合到总线的多个客户端模块。 每个客户端模块能够将总线上的信息发送到客户端模块的另一个,只有一个客户端模块有权在任何时候在总线上传输信息。 有权在总线上传输信息的模块可以控制总线最短时间来定义一个周期。 为了确定哪个模块有权使用总线,当客户端模块试图在总线上传输信息时,每个客户端模块都会产生仲裁信号。 每个客户端模块具有响应于仲裁信号的仲裁信号处理器,用于确定模块是否有权在所述总线上发送信息。 系统还优选地还包括主机模块,其向客户端模块通知在给定周期中在总线上允许的交易类型。 每个仲裁信号处理器优选地还响应于在较早的周期期间由主机模块发送的客户端选项信号。
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公开(公告)号:US4088289A
公开(公告)日:1978-05-09
申请号:US772048
申请日:1977-02-25
申请人: John L. Wood , Thomas C. Wenrich
发明人: John L. Wood , Thomas C. Wenrich
CPC分类号: E21B7/023
摘要: A portable rock drill rig includes a pair of telescoping struts for supporting and positioning a mast or feed beam. The struts are connected at their upper ends to a support bracket which is connected to an elongated mast support member by a hydraulic cylinder to provide relative sliding movement between the bracket and support member. The drill rig includes a crawler undercarriage having spaced apart and pivotally mounted crawler assemblies. The lower ends of the struts are each connected to an arm which is fixed to the main frame of the undercarriage. The arms are also connected to respective track oscillation cylinders. The mounting arrangement of the struts provides for improved positioning of the mast for drilling, tramming and transport operations.
摘要翻译: 便携式凿岩钻机包括一对伸缩支柱,用于支撑和定位桅杆或进给梁。 支柱在其上端连接到支撑托架,支撑托架通过液压缸连接到细长的桅杆支撑构件,以在支架和支撑构件之间提供相对的滑动运动。 钻机包括履带式起落架,其具有间隔开的和可枢转地安装的履带组件。 支柱的下端各自连接到固定到起落架的主框架上的臂。 臂也连接到相应的轨道振荡筒。 支柱的安装布置提供了用于钻孔,电车和运输操作的桅杆的改进的定位。
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公开(公告)号:US06364424B1
公开(公告)日:2002-04-02
申请号:US09491687
申请日:2000-01-26
IPC分类号: B60B310
CPC分类号: B60B3/001 , B60B3/002 , B60B3/14 , B60B21/025 , B60B21/062 , B60B27/0094 , B60B27/023 , B62K15/00
摘要: A portable wheel assembly for use with bicycles and other wheeled vehicles. The wheel assembly comprises a centrally positioned hub which is adapted for rotatable movement about an axis. A plurality of pie shaped disk segments are coupled together along their radial side edges to form a circular support disk with a central opening. Each disk segment is adapted to removably couple with the hub at its innermost radial edge and extends radially outwardly to form a portion of a circular rim at its outermost radial edge. The rim is adapted for supporting a tire. The tire comprises a non-pneumatic tire with an annular ridge which is adapted to couple with the circular rim formed by the disk. During assembly, each of the pie shaped disk segments is coupled together and then coupled to the hub assembly at the inside radial edge or central opening. As the disk segments are coupled to the hub, the tire is assembled onto the outer radial edge or rim. Securing the supporting disk structure to the hub also secures the tire to the rim.
摘要翻译: 一种用于自行车和其他轮式车辆的便携式车轮组件。 车轮组件包括中心定位的毂,其适于围绕轴线的可旋转运动。 多个饼形盘段沿其径向侧边缘联接在一起以形成具有中心开口的圆形支撑盘。 每个盘段适于在其最内径向边缘处可拆卸地与轮毂相连,并且径向向外延伸以在其最外径向边缘处形成圆形边缘的一部分。 轮辋适用于支撑轮胎。 轮胎包括具有环形脊的非充气轮胎,其适于与由盘形成的圆形边缘联接。 在组装期间,每个饼形盘片段联接在一起,然后在内部径向边缘或中心开口处联接到轮毂组件。 当盘段联接到轮毂时,轮胎被组装到外径向边缘或边缘上。 将支撑盘结构固定到轮毂还将轮胎固定到轮辋上。
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公开(公告)号:US5770732A
公开(公告)日:1998-06-23
申请号:US285027
申请日:1994-08-02
申请人: Ralph F. Hirschmann , Amos B. Smith, III , Paul Sprengeler , Ryan C. Holcomb , Terence Keenan , John L. Wood , Mark Guzman , Alexander Pasternak
发明人: Ralph F. Hirschmann , Amos B. Smith, III , Paul Sprengeler , Ryan C. Holcomb , Terence Keenan , John L. Wood , Mark Guzman , Alexander Pasternak
IPC分类号: C07D401/12 , A61K31/40 , A61K31/4015 , A61K31/4025 , A61P43/00 , C07D207/36 , C07D207/38 , C07D405/12 , C07D409/12 , C07D413/00 , C07D207/00
CPC分类号: C07D207/38 , C07D207/36
摘要: Novel pyrrolinone-based compounds mimic or inhibit the biological and/or chemical activity of peptides, including peptide .beta.-strand conformations. Certain compounds contain functionalized pyrrolinone units in place of one or more amino acids of a target peptide.
摘要翻译: 新的基于吡咯啉酮的化合物模拟或抑制肽的生物和/或化学活性,包括肽β-链构象。 某些化合物含有官能化的吡咯啉酮单元代替目标肽的一个或多个氨基酸。
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公开(公告)号:US4997196A
公开(公告)日:1991-03-05
申请号:US429089
申请日:1989-10-30
申请人: John L. Wood
发明人: John L. Wood
CPC分类号: A63C17/015 , A63C17/01 , A63C17/26 , A63C2203/14 , Y10S362/80
摘要: Improvements to a skateboard comprise a board having a complete string of LED's embedded in a groove around the periphery of the skateboard in the first embodiment, powered by a microcontroller and a battery mounted to the underside of the board. In the second embodiment, along the same lines, a kit is provided wherein skid bars have the LED's mounted in them, connected by wiring leading to the microcontroller and battery. The kit can be sold for after-market use, and may consist of just the two side boards, or the rear skid board as well, often called the kick board.
摘要翻译: 对滑板的改进包括在第一实施例中具有嵌入在滑板周边的凹槽中的完整的LED串的板,其由微控制器和安装到板的下侧的电池供电。 在第二实施例中,沿着相同的线,提供了一个套件,其中滑杆具有安装在其中的LED,通过引导到微控制器和电池的布线连接。 该套件可以出售用于售后市场,可能只包括两个侧板,也可能由后挡板组成,通常称为踢脚板。
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公开(公告)号:USD247428S
公开(公告)日:1978-03-07
申请号:US638400
申请日:1975-12-08
申请人: John L. Wood
设计人: John L. Wood
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公开(公告)号:US6037468A
公开(公告)日:2000-03-14
申请号:US206082
申请日:1998-12-04
申请人: John L. Wood , Brian M. Stoltz
发明人: John L. Wood , Brian M. Stoltz
IPC分类号: C07C45/68 , C07D498/22
CPC分类号: C07D498/22 , C07C45/68
摘要: Tertiary alcohols containing the structural features illustrated in 3 or 4 below (Scheme I) are prepared by reacting at least one diazo carbonyl compound, e.g., 1 in Scheme I) and at least one allylic alcohol (e.g., 2 in Scheme I) in a coupling reaction run under conditions that produce carbene or carbenoid intemediates from the diazo containing substrate such as transition metal catalysis or either thermal or photochemical decomposition. In some preferred embodiments, Rh.sub.2 (OAc).sub.4 is employed to catalyze the coupling reaction. ##STR1## Indolocarbazoles (e.g., 7 below) are prepared by coupling of diazo carbonyl compounds (e.g., 5) and biindoles (e.g., 6). Indolocarbazoles are furanosylated (e.g., 7) with acetals (e.g., 8) or their open chain congeners (e.g., 9) under conditions known to promote acetal exchange or formation, such as protic or Lewis acids. Furanosylated indolocarbazoles (e.g., 10) are also prepared via ring contraction of pyranosylated indolocarbazoles (e.g., 11) under conditions know to effect oxidation and benzylic acid type rearrangements, and pyranosylated indolocarbazoles (e.g., 11) are prepared via ring expansion of the furanosylated congeners (e.g., 10). ##STR2##
摘要翻译: 通过使至少一种重氮羰基化合物,例如方案I中的1)与至少一种烯丙醇(例如方案I中的2)反应制备含有下面3或4中所示结构特征的三元醇(方案I) 偶联反应在从含重氮基质产生卡宾或卡宾中间体的条件下进行,例如过渡金属催化或热或光化学分解。 在一些优选的实施方案中,使用Rh 2(OAc)4催化偶联反应。 吲哚并恶唑(如下文7)是通过重氮羰基化合物(例如5)和双吲哚(例如6)的偶联来制备的。 在已知可促进乙缩醛交换或形成的条件下,例如质子酸或路易斯酸,吲哚并吡唑类化合物(例如7)具有缩醛(例如8)或其开链同系物(例如9)。 呋喃糖基化吲哚并唑(例如,10)也是通过吡喃糖基化吲哚并唑(例如11)在已知有效氧化和苄酸型重排的条件下通过环收缩来制备的,吡喃糖基化的吲哚并唑(例如,11)是通过呋喃糖基化同系物 (例如10)。
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公开(公告)号:US5489692A
公开(公告)日:1996-02-06
申请号:US18696
申请日:1993-02-17
申请人: Ralph Hirschmann , Amos B. Smith, III , Paul Sprengeler , Ryan C. Holcomb , Terence Keenan , John L. Wood , Mark Guzman
发明人: Ralph Hirschmann , Amos B. Smith, III , Paul Sprengeler , Ryan C. Holcomb , Terence Keenan , John L. Wood , Mark Guzman
IPC分类号: C07D207/36 , C07D207/38 , C07D207/00 , C07D413/00
CPC分类号: C07D207/38 , C07D207/36
摘要: Novel pyrrolinone-based compounds mimic or inhibit the biological and/or chemical activity of peptides, including peptide .beta.-strand conformations. Certain compounds contain functionalized pyrrolinone units in place of one or more amino acids of a target peptide.
摘要翻译: 新的基于吡咯啉酮的化合物模拟或抑制肽的生物和/或化学活性,包括肽β-链构象。 某些化合物含有官能化的吡咯啉酮单元代替目标肽的一个或多个氨基酸。
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