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    2-oxoquinoline compounds and pharmaceutical uses thereof
    3.
    发明授权
    2-oxoquinoline compounds and pharmaceutical uses thereof 失效
    2-氧代喹啉化合物及其药物用途

    公开(公告)号：US06806276B2

    公开(公告)日：2004-10-19

    申请号：US10245861

    申请日：2002-09-16

    申请人： Takashi Inaba ,  Tetsudo Kaya ,  Hiroyuki Iwamura

    发明人： Takashi Inaba ,  Tetsudo Kaya ,  Hiroyuki Iwamura

    IPC分类号： A61K3147

    CPC分类号： C07D215/227 ,  C07D215/54 ,  C07D401/12 ,  C07D405/12

    摘要： A 2-oxoquinoline compound or its pharmaceutically acceptable salt of general formula [I]: (wherein each symbol in the formula is as determined in the description), and its pharmaceutical use. The compound [I] of the present invention and its pharmaceutically acceptable salts selectively act on cannabinoid receptors, particularly on peripheral type cannabinoid receptors, and have fewer side effects on the central nervous system, having great immunosuppressive action, anti-inflammatory action or antiallergic action. Therefore, these compounds are useful as cannabinoid receptors (particularly peripheral type cannabinoid receptors) modulator, immunosuppressants, anti-inflammatory agents, and antiallergic agents.

    摘要翻译： 2-氧代喹啉化合物或其通式[I]的药学上可接受的盐：其中式中的每个符号如说明书中所确定）及其药物用途。 本发明的化合物[I]及其药学上可接受的盐选择性地作用于大麻素受体，特别是对外周型大麻素受体，对中枢神经系统具有较少的副作用，具有很大的免疫抑制作用，抗炎作用或抗过敏作用 。 因此，这些化合物可用作大麻素受体（特别是外周型大麻素受体）调节剂，免疫抑制剂，抗炎剂和抗过敏剂。

    2-oxoquinoline compounds and medicinal uses thereof
    4.
    发明授权
    2-oxoquinoline compounds and medicinal uses thereof 失效
    2-氧代喹啉化合物及其药物用途

    公开(公告)号：US06509352B1

    公开(公告)日：2003-01-21

    申请号：US09869895

    申请日：2001-08-29

    申请人： Takashi Inaba ,  Tetsudo Kaya ,  Hiroyuki Iwamura

    发明人： Takashi Inaba ,  Tetsudo Kaya ,  Hiroyuki Iwamura

    IPC分类号： A61K3147

    CPC分类号： C07D215/227 ,  C07D215/54 ,  C07D401/12 ,  C07D405/12

    摘要： A 2-oxoquinoline compound or its pharmaceutically acceptable salt of general formula [I]:   (wherein each symbol in the formula is as determined in the description), and its pharmaceutical use. The compound [I] of the present invention and its pharmaceutically acceptable salts selectively act on cannabinoid receptors, particularly on peripheral type cannabinoid receptors, and have fewer side effects on the central nervous system, having great immunosuppressive action, anti-inflammatory action or antiallergic action. Therefore, these compounds are useful as cannabinoid receptors (particularly peripheral type cannabinoid receptors) modulator, immunosuppressants, anti-inflammatory agents, and antiallergic agents.

    摘要翻译： 2-氧代喹啉化合物或其通式[I]的药学上可接受的盐：其中式中的每个符号如说明书中所确定）及其药物用途。 本发明的化合物[I]及其药学上可接受的盐选择性地作用于大麻素受体，特别是对外周型大麻素受体，对中枢神经系统具有较少的副作用，具有很大的免疫抑制作用，抗炎作用或抗过敏作用 。 因此，这些化合物可用作大麻素受体（特别是外周型大麻素受体）调节剂，免疫抑制剂，抗炎剂和抗过敏剂。