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公开(公告)号:US06469047B1
公开(公告)日:2002-10-22
申请号:US09669779
申请日:2000-09-25
IPC分类号: A61K31535
CPC分类号: C07D213/75 , C07C233/87 , C07C271/22 , C07C271/44 , C07C271/48 , C07C271/54 , C07C271/56 , C07C271/58 , C07C311/06 , C07C311/09 , C07C311/58 , C07C323/43 , C07C323/59 , C07D207/16 , C07D207/22 , C07D207/28 , C07D211/46 , C07D211/60 , C07D211/62 , C07D215/36 , C07D217/06 , C07D217/14 , C07D217/22 , C07D231/16 , C07D235/06 , C07D235/26 , C07D249/18 , C07D277/12 , C07D277/56 , C07D295/205 , C07D317/58 , C07D333/20 , C07D333/34 , C07D333/38 , C07D333/62 , C07D333/72 , C07D471/10
摘要: The compounds of the invention are inhibitors of alpha4 containing integrin-mediated binding to ligands such as VCAM-1 and MAdCAM.
摘要翻译: 本发明的化合物是含有整合素介导的与配体如VCAM-1和MAdCAM结合的α4的抑制剂。
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公开(公告)号:US07595399B2
公开(公告)日:2009-09-29
申请号:US10772678
申请日:2004-02-04
IPC分类号: C07D211/06 , C07D295/027 , C07D217/12
CPC分类号: C07D213/75 , C07C233/87 , C07C271/22 , C07C271/44 , C07C271/48 , C07C271/54 , C07C271/56 , C07C271/58 , C07C311/06 , C07C311/09 , C07C311/58 , C07C323/43 , C07C323/59 , C07D207/16 , C07D207/22 , C07D207/28 , C07D211/46 , C07D211/60 , C07D211/62 , C07D215/36 , C07D217/06 , C07D217/14 , C07D217/22 , C07D231/16 , C07D235/06 , C07D235/26 , C07D249/18 , C07D277/12 , C07D277/56 , C07D295/205 , C07D317/58 , C07D333/20 , C07D333/34 , C07D333/38 , C07D333/62 , C07D333/72 , C07D471/10
摘要: The compounds of the invention are inhibitors of alpha4 containing integrin-mediated binding to ligands such as VCAM-1 and MAdCAM.
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公开(公告)号:US20090325962A1
公开(公告)日:2009-12-31
申请号:US12545671
申请日:2009-08-21
IPC分类号: A61K31/5375 , C07C271/40 , A61K31/27 , C07D263/58 , A61K31/421 , C07D217/00 , A61K31/47 , C07D215/00 , C07D265/30 , C07D241/04 , A61K31/495 , C07C229/00 , A61K31/195 , A61P19/02 , A61P11/06 , A61P17/00 , A61P1/00
CPC分类号: C07D213/75 , C07C233/87 , C07C271/22 , C07C271/44 , C07C271/48 , C07C271/54 , C07C271/56 , C07C271/58 , C07C311/06 , C07C311/09 , C07C311/58 , C07C323/43 , C07C323/59 , C07D207/16 , C07D207/22 , C07D207/28 , C07D211/46 , C07D211/60 , C07D211/62 , C07D215/36 , C07D217/06 , C07D217/14 , C07D217/22 , C07D231/16 , C07D235/06 , C07D235/26 , C07D249/18 , C07D277/12 , C07D277/56 , C07D295/205 , C07D317/58 , C07D333/20 , C07D333/34 , C07D333/38 , C07D333/62 , C07D333/72 , C07D471/10
摘要: The compounds of the invention are inhibitors of alpha4 containing integrin-mediated binding to ligands such as VCAM-1 and MAdCAM.
摘要翻译: 本发明的化合物是含有整合素介导的与配体如VCAM-1和MAdCAM结合的α4的抑制剂。
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