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公开(公告)号:US20140155381A1
公开(公告)日:2014-06-05
申请号:US14235512
申请日:2012-07-27
申请人: Erkan Baloglu , Gary J. Bohnert , Shomir Ghosh , Mercedes Lobera , Darby R. Schmidt , Leonard Sung
发明人: Erkan Baloglu , Gary J. Bohnert , Shomir Ghosh , Mercedes Lobera , Darby R. Schmidt , Leonard Sung
IPC分类号: C07D413/14 , C07D407/06 , C07D407/14 , C07D413/06
CPC分类号: C07D413/14 , C07D405/06 , C07D405/14 , C07D407/06 , C07D407/14 , C07D413/06 , C07D491/048
摘要: The present invention relates to novel retinoid-related orphan receptor gamma (RORγ) modulators and their use in the treatment of diseases mediated by RORγ.
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公开(公告)号:US20140155419A1
公开(公告)日:2014-06-05
申请号:US14235481
申请日:2012-07-27
申请人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby R. Schmidt
发明人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby R. Schmidt
IPC分类号: C07D239/52 , C07D213/40 , C07D239/26 , C07D213/30
CPC分类号: C07D239/52 , C07C235/34 , C07D213/30 , C07D213/38 , C07D213/40 , C07D213/65 , C07D239/26 , C07D239/36 , C07D239/54 , C07D401/12 , C07D405/12 , C07D417/12
摘要: The present invention relates to novel retinoid-related orphan receptor gamma (RORγ) modulators and their use in the treatment of diseases mediated by RORγ.
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公开(公告)号:US20120322827A1
公开(公告)日:2012-12-20
申请号:US13522051
申请日:2011-01-13
申请人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
发明人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
IPC分类号: A61K31/4245 , C07D413/12 , A61K31/4196 , A61K31/422 , C07D409/12 , C07D413/14 , A61K31/454
CPC分类号: C07D413/14 , C07D409/12 , C07D413/12 , C07D417/12 , C07D417/14
摘要: Disclosed are compounds having the formula: wherein X1, X2, X3, R1, R2, R3, R4, Y, A, n and L are as defined herein, and methods of making and using the same.
摘要翻译: 公开了具有下式的化合物:其中X1,X2,X3,R1,R2,R3,R4,Y,A,n和L如本文所定义,以及制备和使用它们的方法。
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公开(公告)号:US08981084B2
公开(公告)日:2015-03-17
申请号:US13522070
申请日:2011-01-13
申请人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
发明人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
IPC分类号: C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14 , C07D487/08 , C07D271/06 , C07D409/12 , C07D409/14 , C07D495/04
CPC分类号: C07D487/08 , C07D271/06 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14 , C07D495/04
摘要: Disclosed are compounds having the formula: wherein X1, X2, X3, R1, R2, Y, Q, X, B and L are as defined herein, and methods of making and using the same.
摘要翻译: 公开了具有下式的化合物:其中X1,X2,X3,R1,R2,Y,Q,X,B和L如本文所定义,以及制备和使用它们的方法。
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公开(公告)号:US20130059883A1
公开(公告)日:2013-03-07
申请号:US13522044
申请日:2011-01-13
申请人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
发明人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
IPC分类号: A61K31/4439 , A61K31/4245 , C07D413/12 , C07D417/14 , A61K31/4545 , A61K31/4725 , A61K31/454 , A61P35/00 , A61P3/10 , A61P29/00 , A61P9/00 , A61P3/04 , A61P7/02 , A61P25/08 , A61P25/24 , A61P37/02 , A61P31/12 , A61P31/10 , C07D413/14
CPC分类号: C07D413/12 , A61K31/497 , C07D271/06 , C07D413/14 , C07D417/14 , Y02A50/411 , Y02A50/463
摘要: Disclosed are compounds having the formula: wherein X1, X2, X3, R1, R2, R3, R4, Y, A, Z, L and n are as defined herein, and methods of making and using the same.
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公开(公告)号:US08901156B2
公开(公告)日:2014-12-02
申请号:US13522044
申请日:2011-01-13
申请人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
发明人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
IPC分类号: A01N43/82 , A61K31/41 , A01N43/78 , A61K31/425 , A01N43/76 , A61K31/42 , C07D291/00 , C07D285/08 , C07D271/06 , C07D249/08 , C07D417/14 , A61K31/497 , C07D413/14 , C07D413/12
CPC分类号: C07D413/12 , A61K31/497 , C07D271/06 , C07D413/14 , C07D417/14 , Y02A50/411 , Y02A50/463
摘要: Disclosed are compounds having the formula: wherein X1, X2, X3, R1, R2, R3, R4, Y, A, Z, L and n are as defined herein, and methods of making and using the same.
摘要翻译: 公开了具有下式的化合物:其中X1,X2,X3,R1,R2,R3,R4,Y,A,Z,L和n如本文所定义,以及制备和使用它们的方法。
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公开(公告)号:US20120289495A1
公开(公告)日:2012-11-15
申请号:US13522070
申请日:2011-01-13
申请人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
发明人: Erkan Baloglu , Shomir Ghosh , Mercedes Lobera , Darby Schmidt
IPC分类号: A61K31/4245 , A61K31/5513 , A61K31/5377 , A61K31/506 , C07D413/10 , A61K31/4439 , C07D417/14 , C07D413/14 , C07D487/08 , C07D413/12 , A61K31/427 , A61K31/496
CPC分类号: C07D487/08 , C07D271/06 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14 , C07D495/04
摘要: Disclosed are compounds having the formula: wherein X1, X2, X3, R1, R2, Y, Q, X, B and L are as defined herein, and methods of making and using the same.
摘要翻译: 公开了具有下式的化合物:其中X1,X2,X3,R1,R2,Y,Q,X,B和L如本文所定义,以及制备和使用它们的方法。
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公开(公告)号:US08114894B2
公开(公告)日:2012-02-14
申请号:US12630468
申请日:2009-12-03
申请人: Shomir Ghosh , Gali Golan , Boaz Inbal , Vincent Jacques , Mercedes Lobera
发明人: Shomir Ghosh , Gali Golan , Boaz Inbal , Vincent Jacques , Mercedes Lobera
IPC分类号: A61K31/404 , C07D401/12
CPC分类号: C07D209/24 , C07D401/12 , C07D471/04
摘要: Disclosed herein are compounds that may be modulators of 5-HT receptors, and methods of making and using same.
摘要翻译: 本文公开了可以是5-HT受体的调节剂的化合物,以及制备和使用它们的方法。
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公开(公告)号:US20120088793A1
公开(公告)日:2012-04-12
申请号:US13326836
申请日:2011-12-15
申请人: Shomir Ghosh , Gali Golan , Boaz Inbal , Vincent Jacques , Mercedes Lobera
发明人: Shomir Ghosh , Gali Golan , Boaz Inbal , Vincent Jacques , Mercedes Lobera
IPC分类号: A61K31/454 , A61K31/4545 , A61P25/28 , A61K31/4045
CPC分类号: C07D209/24 , C07D401/12 , C07D471/04
摘要: Disclosed herein are compounds that may be modulators of 5-HT receptors, and methods of making and using same.
摘要翻译: 本文公开了可以是5-HT受体的调节剂的化合物,以及制备和使用它们的方法。
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公开(公告)号:US08586600B2
公开(公告)日:2013-11-19
申请号:US13485037
申请日:2012-05-31
IPC分类号: C07D403/12 , C07D403/14 , C07D401/12 , C07D401/14 , A61K31/506 , A61P35/00 , A61P19/02
CPC分类号: C07D401/04 , A61K31/444 , A61K31/506 , A61K45/06 , C07D401/06 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14
摘要: The present invention provides compounds, pharmaceutically acceptable compositions thereof, and methods of using the same.
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