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1.Substituted indazoles, compositions containing the same, and the preparation and use thereof 失效
标题翻译: 取代的吲唑,含有它们的组合物及其制备和用途公开(公告)号:US07517902B2
公开(公告)日:2009-04-14
申请号:US11566382
申请日:2006-12-04
申请人: Frank Halley , Michel Tabart , Hervé Bouchard , Catherine Souaille , Alain Le Brun , Fabrice Viviani , Laurence Gauzy-Lazo , Pascal Desmazeau , Odile Angouillant-Boniface , Bruno Filoche-Romme
发明人: Frank Halley , Michel Tabart , Hervé Bouchard , Catherine Souaille , Alain Le Brun , Fabrice Viviani , Laurence Gauzy-Lazo , Pascal Desmazeau , Odile Angouillant-Boniface , Bruno Filoche-Romme
IPC分类号: A61K31/541 , A61K31/5377 , C07D417/02 , C07D413/02
CPC分类号: C07D231/56 , C07D403/12 , C07D405/12 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14
摘要: Disclosed are novel substituted indazole compounds, pharmaceutical compositions comprising such compounds, and methods of treatment comprising such compounds.
摘要翻译: 公开了新的取代的吲唑化合物,包含这些化合物的药物组合物和包含这些化合物的治疗方法。
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2.Substituted Indazoles, Compositions Containing The Same, And The Preparation And Use Thereof 失效
标题翻译: 取代的吲唑,含有它的组合物及其制备和使用公开(公告)号:US20070161626A1
公开(公告)日:2007-07-12
申请号:US11566382
申请日:2006-12-04
申请人: Frank Halley , Michel Tabart , Herve Bouchard , Catherine Souaille , Alain Le Brun , Fabrice Viviani , Laurence Gauzy-Lazo , Pascal Desmazeau , Odile Angouillant-Boniface , Bruno Filoche-Romme
发明人: Frank Halley , Michel Tabart , Herve Bouchard , Catherine Souaille , Alain Le Brun , Fabrice Viviani , Laurence Gauzy-Lazo , Pascal Desmazeau , Odile Angouillant-Boniface , Bruno Filoche-Romme
IPC分类号: A61K31/55 , A61K31/541 , A61K31/5377 , A61K31/496 , A61K31/506 , A61K31/4439 , A61K31/427 , A61K31/422 , A61K31/416 , A61K31/4178 , C07D417/02 , C07D413/02 , C07D403/02
CPC分类号: C07D231/56 , C07D403/12 , C07D405/12 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14
摘要: Disclosed are novel substituted indazole compounds, pharmaceutical compositions comprising such compounds, and methods of treatment comprising such compounds.
摘要翻译: 公开了新的取代的吲唑化合物,包含这些化合物的药物组合物和包含这些化合物的治疗方法。
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3.Substituted tetrahydro-1H-pyrazolo [3,4-c] pyridines, compositions comprising them, and use 失效
标题翻译: 取代的四氢-1H-吡唑并[3,4-c]吡啶,包含它们的组合物,并使用公开(公告)号:US07109340B2
公开(公告)日:2006-09-19
申请号:US10888611
申请日:2004-07-09
申请人: Fabienne Thompson , Patrick Mailliet , Teresa Damiano , Marie-Pierre Cherrier , Francois Clerc , Frank Halley , Hervé Bouchard , Laurence Gauzy-Lazo , Bernard Baudoin , Catherine Souaille , Fabrice Viviani , Michel Tabart
发明人: Fabienne Thompson , Patrick Mailliet , Teresa Damiano , Marie-Pierre Cherrier , Francois Clerc , Frank Halley , Hervé Bouchard , Laurence Gauzy-Lazo , Bernard Baudoin , Catherine Souaille , Fabrice Viviani , Michel Tabart
IPC分类号: C07D471/02 , C07D491/02 , C07D498/02 , C07D513/02 , C07D515/02
CPC分类号: C07D471/04
摘要: Substituted tetrahydro-1H-pyrazolo[3,4-c]pyridines, compositions comprising them and use. The present invention relates in particular to novel substituted tetrahydro-1H-pyrazolo[3,4-c]pyridines having therapeutic activity, which can be used in particular in oncology.
摘要翻译: 取代的四氢-1H-吡唑并[3,4-c]吡啶,包含它们的组合物和用途。 本发明特别涉及具有治疗活性的新型取代的四氢-1H-吡唑并[3,4-c]吡啶,其特别可用于肿瘤学。
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4.Substituted tetrahydro-1H-pyrazolo [3,4-c]pyridines compositions comprising them, and use 失效
标题翻译: 包含它们的取代的四氢-1H-吡唑并[3,4-c]吡啶组合物,并使用公开(公告)号:US07435820B2
公开(公告)日:2008-10-14
申请号:US11419794
申请日:2006-05-23
申请人: Fabienne Thompson , Catherine Souaille , Fabrice Viviani , Michel Tabart , Patrick Mailliet , Teresa Damiano , Marie-Pierre Cherrier , Francois Clerc , Frank Halley , Herve Bouchard , Laurence Gauzy-Lazo , Bernard Baudoin
发明人: Fabienne Thompson , Catherine Souaille , Fabrice Viviani , Michel Tabart , Patrick Mailliet , Teresa Damiano , Marie-Pierre Cherrier , Francois Clerc , Frank Halley , Herve Bouchard , Laurence Gauzy-Lazo , Bernard Baudoin
IPC分类号: C07D471/02 , C07D491/02 , C07D498/02 , C07D513/02 , C07D515/02
CPC分类号: C07D471/04
摘要: Substituted tetrahydro-1H-pyrazolo[3,4-c]pyridines, compositions comprising them and use. The present invention relates in particular to novel substituted tetrahydro-1H-pyrazolo[3,4-c]pyridines having therapeutic activity, which can be used in particular in oncology.
摘要翻译: 取代的四氢-1H-吡唑并[3,4-c]吡啶,包含它们的组合物和用途。 本发明特别涉及具有治疗活性的新型取代的四氢-1H-吡唑并[3,4-c]吡啶,其特别可用于肿瘤学。
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5.Substituted tetrahydro-1H-pyrazolo [3,4-c] pyridines, compositions comprising them, and use 失效
标题翻译: 取代的四氢-1H-吡唑并[3,4-c]吡啶,包含它们的组合物,并使用公开(公告)号:US20050096345A1
公开(公告)日:2005-05-05
申请号:US10888611
申请日:2004-07-09
申请人: Fabienne Thompson , Patrick Mailliet , Teresa Damiano , Marie-Pierre Cherrier , Francois Clerc , Frank Halley , Herve Bouchard , Laurence Gauzy-Lazo , Bernard Baudoin , Catherine Souaille , Fabrice Viviani , Michel Tabart
发明人: Fabienne Thompson , Patrick Mailliet , Teresa Damiano , Marie-Pierre Cherrier , Francois Clerc , Frank Halley , Herve Bouchard , Laurence Gauzy-Lazo , Bernard Baudoin , Catherine Souaille , Fabrice Viviani , Michel Tabart
IPC分类号: A61P35/00 , C07D471/04 , C07D471/02 , A61K31/4745
CPC分类号: C07D471/04
摘要: Substituted tetrahydro-1H-pyrazolo[3,4-c]pyridines, compositions comprising them and use. The present invention relates in particular to novel substituted tetrahydro-1H-pyrazolo[3,4-c]pyridines having therapeutic activity, which can be used in particular in oncology.
摘要翻译: 取代的四氢-1H-吡唑并[3,4-c]吡啶,包含它们的组合物和用途。 本发明特别涉及具有治疗活性的新型取代的四氢-1H-吡唑并[3,4-c]吡啶,其特别可用于肿瘤学。
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6.Substituted Pyrrolopyridines, Compositions Containing Them, Manufacturing Process Therefor and Use Thereof 失效
标题翻译: 取代的吡咯并吡啶,其组成物,其制造方法和用途公开(公告)号:US20080139606A1
公开(公告)日:2008-06-12
申请号:US11870640
申请日:2007-10-11
申请人: Michel Tabart , Eric Bacque , Frank Halley , Baptiste Ronan , Pascal Desmazeau , Fabrice Viviani , Catherine Souaille
发明人: Michel Tabart , Eric Bacque , Frank Halley , Baptiste Ronan , Pascal Desmazeau , Fabrice Viviani , Catherine Souaille
IPC分类号: A61K31/437 , C07D471/04 , A61P35/00
CPC分类号: C07D471/04
摘要: The invention relates to compounds of formula (I): wherein Ra, R1, Ar, L, A, W, Y, and Z are as defined in the disclosure; to compositions containing them; and to the preparation and use thereof, in particular as anticancer agents.
摘要翻译: 本发明涉及式(I)化合物:其中R a,R 1,Ar,L,A,W,Y和Z如本公开所定义; 含有它们的组合物; 以及其制备和使用,特别是抗癌剂。
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7.Substituted pyrrolopyridines, compositions containing them, manufacturing process therefor and use thereof 失效
标题翻译: 取代的吡咯并吡啶,含有它们的组合物,其制备方法和用途公开(公告)号:US07947706B2
公开(公告)日:2011-05-24
申请号:US11870640
申请日:2007-10-11
申请人: Michel Tabart , Eric Bacque , Frank Halley , Baptiste Ronan , Pascal Desmazeau , Fabrice Viviani , Catherine Souaille
发明人: Michel Tabart , Eric Bacque , Frank Halley , Baptiste Ronan , Pascal Desmazeau , Fabrice Viviani , Catherine Souaille
IPC分类号: A61K31/437 , C07D471/04 , A61P35/00
CPC分类号: C07D471/04
摘要: The invention relates to compounds of formula (I): wherein Ra, R1, Ar, L, A, W, Y, and Z are as defined in the disclosure; to compositions containing them; and to the preparation and use thereof, in particular as anticancer agents.
摘要翻译: 本发明涉及式(I)化合物:其中R a,R 1,Ar,L,A,W,Y和Z如本公开所定义; 含有它们的组合物; 以及其制备和使用,特别是抗癌剂。
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8.SUBSTITUTED TETRAHYDRO-1H-PYRAZOLO [3,4-C]PYRIDINES COMPOSITIONS COMPRISING THEM, AND USE 失效
标题翻译: 取代的四氢-1H-吡唑并[3,4-C]吡啶类化合物及其用途公开(公告)号:US20060199837A1
公开(公告)日:2006-09-07
申请号:US11419794
申请日:2006-05-23
申请人: Fabienne Thompson , Patrick Mailliet , Teresa Damiano , Marie-Pierre Cherrier , Francois Clerc , Frank Halley , Herve Bouchard , Laurence Gauzy-Lazo , Bernard Baudoin , Catherine Squaille , Fabrice Viviani , Michel Tabart
发明人: Fabienne Thompson , Patrick Mailliet , Teresa Damiano , Marie-Pierre Cherrier , Francois Clerc , Frank Halley , Herve Bouchard , Laurence Gauzy-Lazo , Bernard Baudoin , Catherine Squaille , Fabrice Viviani , Michel Tabart
IPC分类号: C07D471/02 , A61K31/4745
CPC分类号: C07D471/04
摘要: Substituted tetrahydro-1H-pyrazolo[3,4-c]pyridines, compositions comprising them and use. The present invention relates in particular to novel substituted tetrahydro-1H-pyrazolo[3,4-c]pyridines having therapeutic activity, which can be used in particular in oncology.
摘要翻译: 取代的四氢-1H-吡唑并[3,4-c]吡啶,包含它们的组合物和用途。 本发明特别涉及具有治疗活性的新型取代的四氢-1H-吡唑并[3,4-c]吡啶,其特别可用于肿瘤学。
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9.Substituted pyrazolopyridines, compositions containing them, method for the production thereof, and their use 有权
标题翻译: 取代的吡唑并吡啶,含有它们的组合物,其制备方法及其用途公开(公告)号:US08008322B2
公开(公告)日:2011-08-30
申请号:US11778870
申请日:2007-07-17
申请人: Baptiste Ronan , Michel Tabart , Frank Halley , Eric Bacque , Catherine Souaille , Antonio Ugolini , Fabrice Viviani
发明人: Baptiste Ronan , Michel Tabart , Frank Halley , Eric Bacque , Catherine Souaille , Antonio Ugolini , Fabrice Viviani
IPC分类号: A61K31/437 , A61P35/00
CPC分类号: C07D471/04
摘要: The disclosure relates to substituted pyrazolo-pyridines, compositions containing them, methods for the production thereof, and to their use as medicaments, in particular, as anticancer agents.
摘要翻译: 本公开涉及取代的吡唑并吡啶,含有它们的组合物,其制备方法及其作为药物的用途,特别是作为抗癌剂。
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10.Substituted pyrroles and imidazoles, compositions containing same, manufacturing process therefor and use thereof 失效
标题翻译: 取代的吡咯和咪唑,含有它们的组合物,其制备方法和用途公开(公告)号:US07560571B2
公开(公告)日:2009-07-14
申请号:US11832206
申请日:2007-08-01
申请人: Baptiste Ronan , Frank Halley , Catherine Souaille , Fabrice Viviani , Youssef El-Ahmad , Eric Bacque , Michel Tabart
发明人: Baptiste Ronan , Frank Halley , Catherine Souaille , Fabrice Viviani , Youssef El-Ahmad , Eric Bacque , Michel Tabart
IPC分类号: C07D233/64 , C07D207/30 , C07D207/46
CPC分类号: C07D207/34 , C07D233/90
摘要: The disclosure concerns substituted imidazoles and pyrroles, compositions containing the same, the preparation thereof, and the use thereof as medicaments, particularly as anti-cancer agents.
摘要翻译: 本公开涉及取代的咪唑和吡咯,含有它们的组合物,其制备方法及其作为药物的用途,特别是作为抗癌剂。
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