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公开(公告)号:US20070293478A1
公开(公告)日:2007-12-20
申请号:US11655589
申请日:2007-01-19
申请人: Holger Zimmermann , Rudolph Schohe-loop , Kerstin Henninger , Daniela Paulsen , Thomas Roelle , Dieter Lang , Kai Thede , Chantal Fuerstner , David Brueckner , Johannes Koebberling , Marcus Bauser
发明人: Holger Zimmermann , Rudolph Schohe-loop , Kerstin Henninger , Daniela Paulsen , Thomas Roelle , Dieter Lang , Kai Thede , Chantal Fuerstner , David Brueckner , Johannes Koebberling , Marcus Bauser
IPC分类号: A61K31/497 , A61K31/5377 , A61K31/5513 , A61P31/22 , C07D243/08 , C07D401/02 , C07D413/14
CPC分类号: C07D215/56 , C07D401/04
摘要: The invention relates to substituted quinolones and to processes for their preparation as well as to their use for the production of medicaments for the treatment and/or prophylaxis of diseases, especially for use as antiviral agents, particularly against cytomegaloviruses.
摘要翻译: 本发明涉及取代的喹诺酮及其制备方法,以及它们用于生产用于治疗和/或预防疾病的药物的用途,特别是用作抗病毒剂,特别是用于巨细胞病毒的药物。
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公开(公告)号:US07867992B2
公开(公告)日:2011-01-11
申请号:US11655589
申请日:2007-01-19
申请人: Holger Zimmermann , Rudolf Schohe-Loop , Kerstin Henninger , Dieter Lang , Kai Thede , Chantal Fuerstner , David Brueckner , Daniela Paulsen , Thomas Roelle , Johannes Koebberling , Marcus Bauser
发明人: Holger Zimmermann , Rudolf Schohe-Loop , Kerstin Henninger , Dieter Lang , Kai Thede , Chantal Fuerstner , David Brueckner , Daniela Paulsen , Thomas Roelle , Johannes Koebberling , Marcus Bauser
IPC分类号: A01N43/62 , A61K31/55 , C07D413/00
CPC分类号: C07D215/56 , C07D401/04
摘要: The invention relates to substituted quinolones and to processes for their preparation as well as to their use for the production of medicaments for the treatment and/or prophylaxis of diseases, especially for use as antiviral agents, particularly against cytomegaloviruses.
摘要翻译: 本发明涉及取代的喹诺酮及其制备方法,以及它们用于生产用于治疗和/或预防疾病的药物的用途,特别是用作抗病毒剂,特别是用于巨细胞病毒的药物。
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公开(公告)号:US07977349B2
公开(公告)日:2011-07-12
申请号:US12188940
申请日:2008-08-08
申请人: Chantal Fuerstner , Kai Thede , Holger Zimmermann , David Brueckner , Kerstin Henninger , Dieter Lang , Rudolf Schohe-Loop
发明人: Chantal Fuerstner , Kai Thede , Holger Zimmermann , David Brueckner , Kerstin Henninger , Dieter Lang , Rudolf Schohe-Loop
IPC分类号: A61K31/4709 , A61P31/12 , C07D401/10 , C07D498/10 , C07D401/14
CPC分类号: C07D401/04 , C07D401/14 , C07D471/10
摘要: The invention relates to substituted quinolones and to methods for their preparation as well as to their use for the production of medicaments for the treatment and/or prophylaxis of diseases, especially for use as antiviral agents, particularly against cytomegaloviruses.
摘要翻译: 本发明涉及取代的喹诺酮类及其制备方法,以及它们用于生产用于治疗和/或预防疾病的药物的用途,特别是用作抗病毒剂,特别是用于巨细胞病毒的药物。
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公开(公告)号:US20080261964A1
公开(公告)日:2008-10-23
申请号:US12006086
申请日:2007-12-28
申请人: Rudolf Schohe-Loop , Holger Zimmermann , Kerstin Henninger , Dieter Lang , Kai Thede , Chantal Fuerstner , David Brueckner
发明人: Rudolf Schohe-Loop , Holger Zimmermann , Kerstin Henninger , Dieter Lang , Kai Thede , Chantal Fuerstner , David Brueckner
IPC分类号: A61K31/5383 , C07D401/02 , A61K31/496 , A61P31/12 , C07D265/38
CPC分类号: C07D215/56
摘要: The invention relates to substituted quinolones of formula (I) and to methods for their preparation as well as their use for the production of medicaments for the treatment and/or prophylaxis of diseases, especially for use as antiviral agents, in particular against cytomegaloviruses.
摘要翻译: 本发明涉及式(I)的取代喹诺酮及其制备方法及其用于生产药物的用途,所述药物用于治疗和/或预防疾病,特别是用作抗病毒剂,特别是用于巨细胞病毒的疾病。
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公开(公告)号:US07569563B2
公开(公告)日:2009-08-04
申请号:US12006086
申请日:2007-12-28
申请人: Rudolf Schohe-Loop , Holger Zimmermann , Kerstin Henninger , Dieter Lang , Kai Thede , Chantal Fuerstner , David Brueckner
发明人: Rudolf Schohe-Loop , Holger Zimmermann , Kerstin Henninger , Dieter Lang , Kai Thede , Chantal Fuerstner , David Brueckner
IPC分类号: A61K31/5365 , A61K31/496 , C07D215/56 , C07D498/061 , A61K31/551
CPC分类号: C07D215/56
摘要: The invention relates to substituted quinolones of formula (I) and to methods for their preparation as well as their use for the production of medicaments for the treatment and/or prophylaxis of diseases, especially for use as antiviral agents, in particular against cytomegaloviruses.
摘要翻译: 本发明涉及式(I)的取代喹诺酮及其制备方法及其用于生产药物的用途,所述药物用于治疗和/或预防疾病,特别是用作抗病毒剂,特别是用于巨细胞病毒的疾病。
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公开(公告)号:US20090181996A1
公开(公告)日:2009-07-16
申请号:US12188940
申请日:2008-08-08
申请人: Chantal Fuerstner , Kai Thede , Holger Zimmermann , David Brueckner , Kerstin Henninger , Dieter Lang , Rudolf Schohe-Loop
发明人: Chantal Fuerstner , Kai Thede , Holger Zimmermann , David Brueckner , Kerstin Henninger , Dieter Lang , Rudolf Schohe-Loop
IPC分类号: A61K31/4709 , C07D401/10 , C07D471/10 , C07D498/10 , C07D401/14 , A61P31/12
CPC分类号: C07D401/04 , C07D401/14 , C07D471/10
摘要: The invention relates to substituted quinolones and to methods for their preparation as well as to their use for the production of medicaments for the treatment and/or prophylaxis of diseases, especially for use as antiviral agents, particularly against cytomegaloviruses.
摘要翻译: 本发明涉及取代的喹诺酮类及其制备方法,以及它们用于生产用于治疗和/或预防疾病的药物的用途,特别是用作抗病毒剂,特别是用于巨细胞病毒的药物。
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公开(公告)号:US07919489B2
公开(公告)日:2011-04-05
申请号:US11894307
申请日:2007-08-20
申请人: Holger Zimmermann , David Brueckner , Kerstin Henninger , Ulrich Rosentreter , Martin Hendrix , Joerg Keldenich , Dieter Lang , Martin Radtke , Daniela Paulsen , Armin Kern
发明人: Holger Zimmermann , David Brueckner , Kerstin Henninger , Ulrich Rosentreter , Martin Hendrix , Joerg Keldenich , Dieter Lang , Martin Radtke , Daniela Paulsen , Armin Kern
IPC分类号: A61P31/12 , A61K31/4178 , A61K31/4164 , C07D401/12 , C07D233/90
CPC分类号: C07D233/90 , C07D401/12
摘要: The invention relates to heterocyclylamide-substituted imidazoles and methods for their preparation, their use for the treatment and/or prophylaxis of diseases as well as their use for the production of medicaments for the treatment and/or prophylaxis of diseases, in particular for the use as antiviral agents, especially against cytomegaloviruses.
摘要翻译: 本发明涉及杂环基酰胺取代的咪唑及其制备方法,它们用于治疗和/或预防疾病及其用于生产用于治疗和/或预防疾病的药物的用途,特别是用于 作为抗病毒剂,特别是针对巨细胞病毒。
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公开(公告)号:US20100105673A1
公开(公告)日:2010-04-29
申请号:US12518717
申请日:2007-12-08
申请人: Adrian Tersteegen , Dirk Heimbach , Kai Thede , Reinhold Welker , Beate Fast , Arnold Paessens , Frank Dittmer , Rudolf Schohe-Loop , Axel Harrenga , Alexander Hillisch , Kerstin Henninger , Walter Hübsch , Marcus Bauser , Susanne Greschat , Dirk Schneider , Tobias Marquardt , Andreas Göller , Andreas Urban , Steffen Wildum , Daniela Paulsen
发明人: Adrian Tersteegen , Dirk Heimbach , Kai Thede , Reinhold Welker , Beate Fast , Arnold Paessens , Frank Dittmer , Rudolf Schohe-Loop , Axel Harrenga , Alexander Hillisch , Kerstin Henninger , Walter Hübsch , Marcus Bauser , Susanne Greschat , Dirk Schneider , Tobias Marquardt , Andreas Göller , Andreas Urban , Steffen Wildum , Daniela Paulsen
IPC分类号: A61K31/365 , A61K31/5377 , A61K31/438 , C07D413/12 , C07D491/107 , C07D307/94 , A61P31/18 , A61P31/12
CPC分类号: C07D307/94 , C07D491/10
摘要: The present invention relates to novel substituted aminofurans, to methods for their preparation, to their use in the treatment and/or prophylaxis of diseases as well as their use in the manufacture of medical products for the treatment and/or prophylaxis of diseases, in particular retroviral disorders, in humans and/or animals.
摘要翻译: 本发明涉及新型取代的氨基呋喃,其制备方法,其用于治疗和/或预防疾病及其在制备用于治疗和/或预防疾病的医药产品中的用途,特别是 逆转录病毒疾病,在人和/或动物中。
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公开(公告)号:US20110172207A1
公开(公告)日:2011-07-14
申请号:US12884113
申请日:2010-09-16
申请人: Rudolf SCHOHE-LOOP , Reinhold Welker , Arnold Paessens , Marcus Bauser , Friederike Stoll , Frank Dittmer , Kerstin Henninger , Daniela Paulsen , Dieter Lang
发明人: Rudolf SCHOHE-LOOP , Reinhold Welker , Arnold Paessens , Marcus Bauser , Friederike Stoll , Frank Dittmer , Kerstin Henninger , Daniela Paulsen , Dieter Lang
IPC分类号: A61K31/4155 , C07D413/06 , C07D403/06 , C07D417/06 , A61K31/5377 , A61K31/553 , A61K31/427 , A61K31/5386 , A61K31/541 , A61K31/496 , A61P31/12 , A61P31/18
CPC分类号: C07D231/14 , A61K31/4155 , C07D401/06 , C07D403/06 , C07D413/06 , C07D417/06 , C07D451/06 , C07D491/08 , C07D498/08
摘要: The present invention relates to novel substituted pyrazolamides, methods for their preparation, their use for the treatment and/or prophylaxis of diseases, as well as their use for the manufacture of medicaments for the treatment and/or prophylaxis of diseases, especially of retroviral diseases, in humans and/or animals.
摘要翻译: 本发明涉及新型取代的吡唑啉酰胺,其制备方法,其用于治疗和/或预防疾病的用途,以及其用于制备用于治疗和/或预防疾病尤其是逆转录病毒疾病的药物的用途 ,在人类和/或动物中。
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公开(公告)号:US08314089B2
公开(公告)日:2012-11-20
申请号:US12884113
申请日:2010-09-16
申请人: Rudolf Schohe-Loop , Reinhold Welker , Arnold Paessens , Marcus Bauser , Friederike Stoll , Frank Dittmer , Kerstin Henninger , Daniela Paulsen , Dieter Lang
发明人: Rudolf Schohe-Loop , Reinhold Welker , Arnold Paessens , Marcus Bauser , Friederike Stoll , Frank Dittmer , Kerstin Henninger , Daniela Paulsen , Dieter Lang
IPC分类号: A61K31/4155 , A61K31/5377 , A61K31/5386 , A61K31/553 , A61K31/496 , C07D413/06 , C07D417/06 , C07D403/06 , A61P31/12
CPC分类号: C07D231/14 , A61K31/4155 , C07D401/06 , C07D403/06 , C07D413/06 , C07D417/06 , C07D451/06 , C07D491/08 , C07D498/08
摘要: The present invention relates to novel substituted pyrazolamides, methods for their preparation, their use for the treatment and/or prophylaxis of diseases, as well as their use for the manufacture of medicaments for the treatment and/or prophylaxis of diseases, especially of retroviral diseases, in humans and/or animals.
摘要翻译: 本发明涉及新型取代的吡唑啉酰胺,其制备方法,其用于治疗和/或预防疾病的用途,以及其用于制备用于治疗和/或预防疾病尤其是逆转录病毒疾病的药物的用途 ,在人类和/或动物中。
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