Novel benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides
    2.
    发明申请
    Novel benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides 失效
    新型苄基偕胺肟衍生物,其生产和使用的中间产物和方法作为杀真菌剂

    公开(公告)号:US20050187265A1

    公开(公告)日:2005-08-25

    申请号:US11061470

    申请日:2005-02-22

    摘要: Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described. In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1-C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1-C6-alkyl, thienyl-C1-C4-alkyl, or pyrazolyl-C1-C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy, C1-C6-alkylcarbonyl; n is 0-5; p is, depending on the number of free valencies, 0-4.

    摘要翻译: 描述了新的苯甲酰胺肟衍生物,其制备方法和中间体及其作为杀真菌剂的用途。 在本发明的上下文中,苯甲酰胺肟衍生物是式I的化合物,其中:A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基,其中一个碳可被氧,氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团:氢,卤素,C 1 -C 6 C 1 -C 6烷基,C 1 -C 6 - 烷氧基,C 1 -C 4 - 卤代烷基 ,C 1 -C 4 - 卤代烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基,噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基,R 3 - (CH 3)3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团:氢,卤素,C 1 -C 6 - 烷基,C 1 - C 1 -C 6 - 烷氧基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 卤代烷氧基 C 1 -C 4 - 烷硫基,C 1 -C 4 - 烷氧基烷氧基,C 1 -C 4烷基硫基,C 1 -C 4 - -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量,0-4。

    Fungicides containing pyrrolidones as their active agents
    4.
    发明授权
    Fungicides containing pyrrolidones as their active agents 失效
    杀真菌剂含有吡咯烷酮作为其活性剂

    公开(公告)号:US06476061B1

    公开(公告)日:2002-11-05

    申请号:US09831406

    申请日:2001-05-09

    IPC分类号: A61N4336

    CPC分类号: C07D207/50 A01N43/36

    摘要: The invention relates to fungicides containing compounds of formula (I) as their active agents, the radicals in said formula (I) having the following meanings: R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-halogenalkylcarbonyl; R2 is hydrogen, C1-C6-alkyl or C1-C6-halogenalkyl; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, C1-C6-halogenalkyl, C1-C6-alkoxy, C1-C6-halogenalkoxy, C1-C6-alkylsulfonyl, C1-C6-halogenalkylsulfonyl, formyl, cyano, C1-C6-alkylthio or phenyl which can optionally be substituted by halogen atoms, C1-C6-alkyl or C1-C6-halogenalkyl groups, and to their agriculturally usable salts. The invention also relates to methods for combating fungi in plants using these fungicides.

    摘要翻译: 本发明涉及含有式(I)化合物作为其活性剂的杀真菌剂,所述式(I)中的基团具有以下含义:R 1是氢,C 1 -C 6 - 烷基,C 1 -C 6 - 烷基羰基,甲酰基或C 1 -C 6烷基, C6-卤代烷基羰基; R2是氢,C1-C6-烷基或C1-C6-卤代烷基; R3-R12是氢,卤素,C1-C8-环烷基,C1-C6-烷基,C1-C6-卤代烷基,C1-C6-烷氧基,C1-C6-卤代烷氧基,C1-C6-烷基磺酰基,C1-C6-卤代烷基磺酰基, 甲酰基,氰基,C 1 -C 6 - 烷硫基或可以被卤素原子,C 1 -C 6烷基或C 1 -C 6 - 卤代烷基取代的苯基,以及它们的农业上可用的盐。 本发明还涉及使用这些杀真菌剂防治植物中真菌的方法。

    Fungicidal compositions comprising as active compounds pyrrolidones, and their use in the treatment of plants
    5.
    发明授权
    Fungicidal compositions comprising as active compounds pyrrolidones, and their use in the treatment of plants 失效
    包含作为活性化合物吡咯烷酮的杀真菌组合物及其在处理植物中的用途

    公开(公告)号:US06680283B1

    公开(公告)日:2004-01-20

    申请号:US10410788

    申请日:2003-04-11

    IPC分类号: A01N4336

    摘要: Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula I where R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl; R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl, R13 is hydrogen, C1-C6-alkyl, R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group consisting of nitrogen and oxygen, and their agriculturally useful salts are described.

    摘要翻译: 具有杀真菌作用的农药组合物包含作为活性化合物的式I其中R 1为氢,C 1 -C 6烷基,C 1 -C 6烷基羰基,甲酰基或C 1 -C 6卤代烷基羰基; R 2为卤素, C 1 -C 6烷氧基,C 1 -C 6烷氧基,C 1 -C 6烷氧基,C 1 -C 6烷氧基,C 1 -C 6烷氧基, C 6 - 烷基亚磺酰基,卤代-C 1 -C 6 - 烷基磺酰基,氰基或基团NR 13 R 14; R 3 -R 12是氢,卤素,C 1 -C 8 - 环烷基,C 1 -C 6 - 烷基 卤代-C 1 -C 6 - 烷基,C 1 -C 6 - 烷氧基,卤代-C 1 -C 6 - 烷氧基,C 1 -C 6烷基磺酰基,卤代-C 1 -C 6烷基磺酰基,甲酰基,C 1 -C 6烷基羰基,氰基,C 1 -C 6 - 烷硫基或苯基,其可以是未取代的或被卤素,C 1 -C 6 - 烷基或卤代-C 1 -C 6烷基取代,R 13是氢,C 1 -C 6烷基,R 14是C 1 -C 6 - 烷基,C 1 -C 8 - 环烷基或与R 13和它们所连接的氮原子一起是饱和或不饱和的杂环五元或六元环,其含有一个或两个选自以下的杂原子: 描述了由氮和氧组成的组及其农业上有用的盐。

    Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides
    6.
    发明授权
    Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides 失效
    苄基偕胺肟衍生物,中间产物及其生产和用作杀真菌剂的方法

    公开(公告)号:US07101900B2

    公开(公告)日:2006-09-05

    申请号:US11061470

    申请日:2005-02-22

    摘要: Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described.In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1–C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1–C6-alkyl, C1–C6-alkoxy, C1–C4-haloalkyl, C1–C4-haloalkoxy, C1–C4-alkylthio, C1–C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1–C6-alkyl, thienyl-C1–C4-alkyl, or pyrazolyl-C1–C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1–C6-alkyl, C1–C6-alkoxy, C1–C4-haloalkyl, C1–C4-haloalkoxy, C1–C4-alkylthio, C1–C4-alkoxyalkoxy, C1–C6-alkylcarbonyl; n is 0–5; p is, depending on the number of free valencies, 0–4.

    摘要翻译: 描述了新的苯甲酰胺肟衍生物,其制备方法和中间体及其作为杀真菌剂的用途。 在本发明的上下文中,苯甲酰胺肟衍生物是式I的化合物,其中:A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基,其中一个碳可被氧,氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团:氢,卤素,C 1 -C 6 C 1 -C 6烷基,C 1 -C 6 - 烷氧基,C 1 -C 4 - 卤代烷基 ,C 1 -C 4 - 卤代烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基,噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基,R 3 - (CH 3)3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团:氢,卤素,C 1 -C 6 - 烷基,C 1 - C 1 -C 6 - 烷氧基,C 1 -C 4 - 卤代烷基,C 1 -C 3 > 4个 - 卤代烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4 - - 烷氧基烷氧基,C 1 -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量,0-4。

    Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides
    7.
    发明授权
    Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides 失效
    苄基偕胺肟衍生物,中间产物及其生产和用作杀真菌剂的方法

    公开(公告)号:US06881742B1

    公开(公告)日:2005-04-19

    申请号:US10089148

    申请日:2000-10-05

    摘要: Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described.In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1-C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1-C6-alkyl, thienyl-C1-C4-alkyl, or pyrazolyl-C1-C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy, C1-C6-alkylcarbonyl; n is 0-5; p is, depending on the number of free valencies, 0-4.

    摘要翻译: 描述了新的苯甲酰胺肟衍生物,其制备方法和中间体及其作为杀真菌剂的用途。 在本发明的上下文中,苯甲酰胺肟衍生物是式I的化合物,其中:A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基,其中一个碳可被氧,氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团:氢,卤素,C 1 -C 6 C 1 -C 6烷基,C 1 -C 6 - 烷氧基,C 1 -C 4 - 卤代烷基 ,C 1 -C 4 - 卤代烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基,噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基,R 3 - (CH 3)3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团:氢,卤素,C 1 -C 6 - 烷基,C 1 - C 1 -C 6 - 烷氧基,C 1 -C 4 - 卤代烷基,C 1 -C 3 > 4个 - 卤代烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4 - - 烷氧基烷氧基,C 1 -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量,0-4。

    Fungicidal agents containing pyrrolidones as their active agents and use thereof for treating plants
    8.
    发明授权
    Fungicidal agents containing pyrrolidones as their active agents and use thereof for treating plants 失效
    含有吡咯烷酮作为其活性剂的杀真菌剂及其用于处理植物的用途

    公开(公告)号:US06586369B1

    公开(公告)日:2003-07-01

    申请号:US10204349

    申请日:2002-08-20

    IPC分类号: C07D20718

    摘要: Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula I where R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl; R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl, R13 is hydrogen, C1-C6-alkyl, R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group consisting of nitrogen and oxygen, and their agriculturally useful salts are described.

    摘要翻译: 具有杀真菌作用的农药组合物,包含作为活性化合物的式I化合物,其中R 1是氢,C 1 -C 6烷基,C 1 -C 6烷基羰基,甲酰基或C 1 -C 6卤代烷基羰基; R 2是卤素,C 1 -C 6烷硫基, C 1 -C 6烷氧基,C 1 -C 6烷氧基,C 1 -C 6烷氧基,C 1 -C 6 - 烷基亚磺酰基, C 1 -C 6 - 烷基磺酰基,氰基或NR 13 R 14基; R 3 -R 12是氢,卤素,C 1 -C 8 - 环烷基,C 1 -C 6烷基,卤代-C 1 -C 6 - 烷基,C 1 -C 6 - 烷氧基, C 1 -C 6 - 烷基磺酰基,卤代-C 1 -C 6 - 烷基磺酰基,甲酰基,C 1 -C 6 - 烷基羰基,氰基,C 1 -C 6 - 烷硫基或苯基,其可以是未取代的或被卤素取代, 或卤代-C 1 -C 6烷基,R 13是氢,C 1 -C 6烷基,R 14是C 1 -C 6 - 烷基,C 1 -C 8 - 环烷基,或者与R 13和它们所连接的氮原子一起是饱和或 不饱和杂环五元或六元环,其含有一个或两个选自组的杂原子 描述了氮和氧及其农业上有用的盐。