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公开(公告)号:US20100010003A1
公开(公告)日:2010-01-14
申请号:US12373559
申请日:2007-07-17
申请人: Noelle Gauvry , Francois Pautrat , Jacques Bouvier , Jorg Fruchtel , Beatrice Bapst , Sandra Schorderet Weber
发明人: Noelle Gauvry , Francois Pautrat , Jacques Bouvier , Jorg Fruchtel , Beatrice Bapst , Sandra Schorderet Weber
IPC分类号: A61K31/506 , C07D239/46 , A61K31/513 , A61P33/00 , A61K31/496 , C07D413/10 , C07D405/10 , C07D403/10 , C07D401/10 , C07D409/10
CPC分类号: A01N43/54 , A01N43/56 , C07D239/52 , C07D401/04 , C07D403/04 , C07D405/04 , C07D405/10 , C07D409/04
摘要: The invention relates to new pyrimidine compounds of formula (1) wherein the variables have the meaning as indicated in the claims; in free form and in salt form; and optionally the enantiomers and geometrical isomers thereof. The compounds of formula (1) are useful in the control of parasites, in particular ectoparasites, in and on warmblooded animals.
摘要翻译: 本发明涉及式(1)的新的嘧啶化合物,其中变量具有如权利要求中所示的含义; 以自由形式和盐形式; 和任选的其对映体和几何异构体。 式(1)的化合物可用于控制温血动物中和之上的寄生虫,特别是外寄生虫。
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公开(公告)号:US20070155757A1
公开(公告)日:2007-07-05
申请号:US10591624
申请日:2005-03-07
申请人: Jorg Fruchtel , Noelle Gauvry , Sandra Schorderet-Weber , Tania Cavaliero , Jacques Bouvier , Francois Pautrat
发明人: Jorg Fruchtel , Noelle Gauvry , Sandra Schorderet-Weber , Tania Cavaliero , Jacques Bouvier , Francois Pautrat
IPC分类号: A01N43/54
CPC分类号: C07D239/46 , C07D239/50 , C07D239/60
摘要: The invention relates to the use of compounds of the general formula (I), wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11, R12, R13, X1 and X2 have the significances given in claim 1, and optionally the enantiomers and geometrical isomers thereof, for controlling parasites on warm-blooded animals.
摘要翻译: 本发明涉及通式(I)化合物的用途,其中R 1,R 2,R 3,R 3, R 4,R 5,R 6,R 7,R 8,R SUB, R 9,R 10,R 11,R 12,R 13,X 1和X 2具有权利要求1中给出的含义,以及任选的其对映异构体和几何异构体,用于控制温血动物的寄生虫。
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公开(公告)号:US20090197902A1
公开(公告)日:2009-08-06
申请号:US12394112
申请日:2009-02-27
申请人: Jorg Fruchtel , Noelle Gauvry , Sandra Schorderet-Weber , Tania Cavaliero , Jacques Bouvier , Francois Pautrat
发明人: Jorg Fruchtel , Noelle Gauvry , Sandra Schorderet-Weber , Tania Cavaliero , Jacques Bouvier , Francois Pautrat
CPC分类号: C07D239/46 , C07D239/50 , C07D239/60
摘要: The invention relates to the use of compounds of the general formula (I), wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11, R12, R13, X1 and X2 have the significances given in claim 1, and optionally the enantiomers and geometrical isomers thereof, for controlling parasites on warm-blooded animals.
摘要翻译: 本发明涉及通式(I)化合物的用途,其中R1,R2,R3,R4,R5,R6,R7,R8,R9,R10,R11,R12,R13,X1和X2具有给定的含义 在权利要求1中,以及任选的其对映体和几何异构体,用于控制温血动物的寄生虫。
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公开(公告)号:US20110021543A1
公开(公告)日:2011-01-27
申请号:US12598074
申请日:2008-04-29
IPC分类号: A61K31/437 , C07D471/04 , C07D495/04 , A61K31/407 , C07D491/048 , C07D209/52 , A61K31/403 , C07D487/04 , A61K31/519 , A61P33/14 , A61P33/00
CPC分类号: C07D209/12 , C07D209/52 , C07D401/04 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04
摘要: Novel N-aryl substituted heteroindole compounds, processes for their manufacture, veterinary compositions containing such compounds, and methods of controlling ectoparasites are provided. The compounds are believed effective in the control of ectoparasites on warm-blooded productive livestock and domestic animals.
摘要翻译: 提供新的N-芳基取代的杂吲哚化合物,其制备方法,含有这些化合物的兽用组合物和控制外寄生虫的方法。 这些化合物被认为有效地控制温血生产的家畜和家畜的外寄生虫。
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公开(公告)号:US08367682B2
公开(公告)日:2013-02-05
申请号:US12373559
申请日:2007-07-17
申请人: Noëlle Gauvry , François Pautrat , Jacques Bouvier , Jörg Früchtel , Beatrice Bapst , Sandra Schorderet Weber
发明人: Noëlle Gauvry , François Pautrat , Jacques Bouvier , Jörg Früchtel , Beatrice Bapst , Sandra Schorderet Weber
IPC分类号: A01N43/54 , C07D239/52
CPC分类号: A01N43/54 , A01N43/56 , C07D239/52 , C07D401/04 , C07D403/04 , C07D405/04 , C07D405/10 , C07D409/04
摘要: The invention relates to new pyrimidine compounds of formula (1) wherein the variables have the meaning as indicated in the claims; in free form and in salt form; and optionally the enantiomers and geometrical isomers thereof. The compounds of formula (1) are useful in the control of parasites, in particular ectoparasites, in and on warmblooded animals.
摘要翻译: 本发明涉及式(1)的新的嘧啶化合物,其中变量具有如权利要求中所示的含义; 以自由形式和盐形式; 和任选的其对映体和几何异构体。 式(1)的化合物可用于控制温血动物中和之上的寄生虫,特别是外寄生虫。
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公开(公告)号:US20090227538A1
公开(公告)日:2009-09-10
申请号:US12084503
申请日:2006-11-02
IPC分类号: A61K31/695 , C07D209/04 , A61K31/404 , C07D401/02 , A61K31/454 , C07D403/02 , A61K31/496 , C07D413/02 , A61K31/5377 , C07F7/02 , A61P33/00
CPC分类号: C07D403/04 , A01N43/38 , A01N43/40 , A01N47/06 , A01N47/12 , A01N47/18 , A01N47/20 , C07D209/12 , C07D401/04 , C07D401/14 , C07D403/14 , C07D407/04 , C07D407/12 , C07D409/12
摘要: The invention relates to compounds of the general formula (I) wherein R1, R2, R3, R4, R5, R6, A, X, m and n have the significances given in claim 1, and optionally the enantiomers thereof. The active ingredients have advantageous pesticidal properties. They are especially suitable for controlling parasites on warm-blooded animals and plants.
摘要翻译: 本发明涉及通式(I)的化合物,其中R 1,R 2,R 3,R 4,R 5,R 6,A,X,m和n具有权利要求1中给出的含义,以及任选的其对映异构体。 活性成分具有有利的杀虫特性。 它们特别适用于控制温血动物和植物的寄生虫。
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公开(公告)号:US20050059736A1
公开(公告)日:2005-03-17
申请号:US10501495
申请日:2003-01-20
申请人: Pierre Ducray , Thomas Goebel , Jorg Fruchtel , Jacques Bouvier
发明人: Pierre Ducray , Thomas Goebel , Jorg Fruchtel , Jacques Bouvier
IPC分类号: A61P33/10 , A01N37/34 , A01N39/02 , A61K31/277 , A61P33/00 , A61P33/14 , C07C253/30 , C07C255/29 , C07C255/57 , C07C323/56
CPC分类号: C07C255/29 , A01N39/02 , C07C2601/02 , C07C2601/04
摘要: The invention relates to compounds of the general formula (I), in which Ar, R1, R2, R3, R4, R5, R6, R7, R8, W, a, b and n are as defined in claim 1, and to any enantiomers thereof The active ingredients have advantageous pesticidal properties. They are particularly suitable for controlling parasites in warm-blooded animals.
摘要翻译: 本发明涉及通式(I)的化合物,其中Ar,R 1,R 2,R 3,R 4,R 5,R 6,R 7,R 8,W,a,b和n如权利要求1中所定义, 其对映异构体活性成分具有有利的杀虫特性。 它们特别适用于控制温血动物的寄生虫。
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公开(公告)号:US07153814B2
公开(公告)日:2006-12-26
申请号:US10501495
申请日:2003-01-20
申请人: Pierre Ducray , Thomas Goebel , Jorg Fruchtel , Jacques Bouvier
发明人: Pierre Ducray , Thomas Goebel , Jorg Fruchtel , Jacques Bouvier
IPC分类号: A01N37/34 , C07C255/03
CPC分类号: C07C255/29 , A01N39/02 , C07C2601/02 , C07C2601/04
摘要: The invention relates to compounds of the general formula (I), in which Ar, R1, R2, R3, R4, R5, R6, R7, R8, W, a, b and n are as defined in claim 1, and to any enantiomers thereof. The active ingredients have advantageous pesticidal properties. They are particularly suitable for controlling parasites in warm-blooded animals
摘要翻译: 本发明涉及通式(I)的化合物,其中Ar,R 1,R 2,R 3,R 3, R 4,R 5,R 6,R 7,R 8,W,a ,b和n如权利要求1所定义,及其任何对映异构体。 活性成分具有有利的杀虫特性。 它们特别适用于控制温血动物的寄生虫
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公开(公告)号:US08940782B2
公开(公告)日:2015-01-27
申请号:US13679152
申请日:2012-11-16
申请人: Pierre Ducray , Tania Cavaliero , Maike Renner , Jacques Bouvier
发明人: Pierre Ducray , Tania Cavaliero , Maike Renner , Jacques Bouvier
摘要: The present invention is directed to a non-therapeutical process for deterring vermin, which is based on the usage of the largely known beta amino-alcohol derivatives of formula (I) as described herein. Further, the present invention is directed to corresponding vermin-deterring compositions which contain these substances as the active ingredient, compounds of the formula (I) for the preparation of vermin-deterring compositions, and the use of compounds of formula (I) in the defense against vermin.
摘要翻译: 本发明涉及用于抑制害虫的非治疗方法,其基于如本文所述的大量已知的式(I)的β-氨基醇衍生物的用途。 此外,本发明涉及含有这些物质作为活性成分的相应的害虫抑制组合物,用于制备害虫阻止剂组合物的式(I)化合物,以及式(I)化合物在 防御害虫
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公开(公告)号:US07749526B2
公开(公告)日:2010-07-06
申请号:US10537871
申请日:2003-12-16
申请人: Thomas Goebel , Tania Cavaliero , Jacques Bouvier
发明人: Thomas Goebel , Tania Cavaliero , Jacques Bouvier
CPC分类号: A01N37/26 , A01N37/20 , Y10S514/875 , Y10S514/876 , Y10S514/919
摘要: Compounds of formula (I) are described for deterring vermin, wherein R is unbranched or branched C1-C15 alkyl, which is unsubstituted or substituted by halogen, cyano or nitro; R1 and R2 are unbranched or branched C1-C12 alkyl, preferably C1-C6 alkyl, which is unsubstituted or substituted by halogen, cyano or nitro; and X and Y, independently of one another, are a straightchain or branched alkylene bridge with 1 to 20 carbon atoms, preferably an alkylene bridge with 1 to 3 carbon atoms, which is unsubstituted or substituted by halogen, cyano or nitro. Furthermore, an essentially non-therapeutical process for deterring vermin is described, which is based on the usage of these compounds, as well as verminrepellent compositions containing these compounds as the active ingredient, and finally the use of these compounds for producing vermin-deterring compositions and their usage in deterring vermin from animals, humans and objects. New compounds within the scope of formula (I) are also described.
摘要翻译: 描述了式(I)化合物用于阻止害虫,其中R是未被取代或被卤素,氰基或硝基取代的未支链或支链C 1 -C 15烷基; R 1和R 2是未经取代或被卤素,氰基或硝基取代的未支链或支链C 1 -C 12烷基,优选C 1 -C 6烷基; X和Y彼此独立地是具有1至20个碳原子的直链或支链亚烷基桥,优选未取代或被卤素,氰基或硝基取代的具有1至3个碳原子的亚烷基桥。 此外,描述了一种用于抑制害虫的基本上非治疗性的方法,其基于这些化合物的用途,以及含有这些化合物作为活性成分的维生素组合物,最后使用这些化合物来生产害虫抑制剂组合物 以及它们用于阻止动物,人类和物体的害虫。 还描述了式(I)范围内的新化合物。
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