公开(公告)号：US3769425A

公开(公告)日：1973-10-30

申请号：US3769425D

申请日：1972-06-07

Applicant: ROUSSEL UCLAF

Inventor： ROUSSEAU G ,  POITTEVIN A

IPC: C07C69/738 ,  A61K31/19 ,  A61K31/215 ,  A61P25/04 ,  A61P29/00 ,  C07C15/20 ,  C07C49/385 ,  C07C51/00 ,  C07C53/08 ,  C07C57/38 ,  C07C57/46 ,  C07C57/50 ,  C07C57/62 ,  C07C59/54 ,  C07C59/86 ,  C07C59/88 ,  C07C67/00 ,  C07C405/00 ,  C07D309/06 ,  C07D309/36 ,  C07D311/04 ,  C07D311/96 ,  C07D335/02 ,  A61K27/00

CPC classification number: C07C57/50 ,  C07C57/46 ,  C07C57/62 ,  C07C59/54 ,  C07C59/86 ,  C07C59/88 ,  C07D309/06 ,  C07D311/04 ,  C07D311/96

Abstract: NOVEL SPIRO BENZOCYCLANE ACETIC ACID COMPOUNDS OF THE FORMULA

(-(CH2)2-Y-(CH2)2-)>C
1,2-PHENYLENE)-)

WHEREIN R IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN AND LINEAR AND BRANCHED ALKLY OF 1 TO 4 CARBON ATOMS. R1 IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, CHLORINE, TRIFLUOROMETHYL AND LOWER ALKOXY, Y IS SELECTED FROM THE GROUP CONSISTING OF METHYLENE, OXYGEN AND SULFUR, N IS 2, 3 OR 4 AND R2 IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN SUBSTITUTED OR UNSUBSTITUTED ALKYL OF 1 TO 6 CARBON ATOMS AND CATION OF NON-TOXIC, PHARMACEUTICALLY ACCEPTABLE MINERAL AND ORGANIC BASES, PROCESSES FOR THEIR PREPRATION AND NOVEL INTERMEDIATES. THE COMPOUNDS OF FORMULA I HAVE ANALGESIC AND ANTI-INFLAMMATORY PROPERTIES.

公开(公告)号：US3857838A

公开(公告)日：1974-12-31

申请号：US28839372

申请日：1972-09-12

Applicant: ROUSSEL UCLAF

Inventor： PERRONNET J ,  POITTEVIN A

IPC: A01N57/08 ,  C07D471/04 ,  C07D487/04 ,  C07F9/6561 ,  C07D51/46

CPC classification number: C07D471/04 ,  C07D487/04 ,  C07F9/6561

Abstract: An organophosphate ester having the formula

WHEREIN A represents a divalent radical selected from the group consisting of alkylene having three to five carbon atoms, aza substitued alkylene having three to five carbon atoms in the chain and thia substituted alkylene having three to five carbon atoms in the chain, Y'' represents a member selected from the group consisting of hydrogen, alkyl having one to six carbon atoms, cyano, halo and alkylthio having one to six carbon atoms, X represents a member selected from the group consisting of sulfur and oxygen, R1'''' represents an alkyl having one to four carbon atoms, R2'''' represents a member selected from the group consisting of alkyl having one to four carbon atoms, alkoxy having one to four carbon atoms, alkoxyalkoxy having one to four carbon atoms in each alk, and

WHERE R1'' and R2'' are members selected from the group consisting of hydrogen and alkyl having one to three carbon atoms; as well as the process of producing said organophosphate esters. The compounds have insecticidal and acaricidal properties.

Abstract translation: 具有下式的有机磷酸酯取代为WHEREIN A表示选自具有3-5个碳原子的亚烷基的二价基团，链中具有3-5个碳原子的氮杂取代的亚烷基和具有3至5个碳原子的取代的亚烷基 该链Y表示选自氢，碳原子数1〜6的烷基，氰基，卤代和碳原子数1〜6的烷硫基，X表示选自硫和氧的成员， R 1“表示碳原子数为1〜4的烷基，R 2”表示选自碳原子数1〜4的烷基，碳原子数1〜4的烷氧基，碳原子数1〜4的烷氧基烷氧基， 烷基和其中R 1'和R 2'是选自氢和具有1至3个碳原子的烷基的成员; 以及生产所述有机磷酸酯的方法。 这些化合物具有杀虫和杀螨的特性。

公开(公告)号：US3799974A

公开(公告)日：1974-03-26

申请号：US25456872

申请日：1972-05-18

Applicant: ROUSSEL UCLAF

Inventor： ROUSSEAU G ,  ALLAIS A ,  POITTEVIN A

IPC: C07C49/675 ,  C07C49/697 ,  C07C57/46 ,  C07C57/50 ,  C07C57/62 ,  C07C59/54 ,  C07C59/86 ,  C07C59/88 ,  C07C69/157 ,  C07D311/96 ,  C07C63/00 ,  C07C65/20

CPC classification number: C07C59/88 ,  C07C49/675 ,  C07C49/697 ,  C07C57/46 ,  C07C57/50 ,  C07C57/62 ,  C07C59/54 ,  C07C59/86 ,  C07D311/96

Abstract: NOVEL SPRIO BENZOCYCLANE ACETIC ACID COMPOUND OF THE FORMULA
WHEREIN R IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN AND LINEAR AND BRANCHED ALKYL OF 1 TO 4 CARBON ATOMS R1 IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, CHLORINE, TRIFLUOROMETHYL AND LOWER ALKOXY, Y IS SELECTED FROM THE GROUP CONSISTING OF METHYLENE, OXYGEN AND SULFUR, N IS 2,3, OR 4 AND R2 IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, SUBSTITUTED OR UNSUBSTITUTED ALKYL OF 1 TO 6 CARBON ATOMS AND CATION OF NONTOXIC, PHARMACEUTICALLY ACCEPTABLE MINERAL AND ORGANIC BASES. PROCESSES FOR THEIR PREPARATION AND NOVEL INTERMEDIATES. THE COMPOUNDS OF FORMULA 1 HAVE ANALGESIC AND ANTI-INFLAMMATORY PROPERTIES.

-)-)BENZENE

1-R1,3-(R2-OOC-CH(-R)-),5,6-(-(CH2)N-C

公开(公告)号：US3830884A

公开(公告)日：1974-08-20

申请号：US28947472

申请日：1972-09-15

Applicant: ROUSSEL UCLAF

Inventor： PERRONNET J ,  POITTEVIN A ,  DEMOUTE J

IPC: A01N57/12 ,  C07F9/165 ,  C07F9/16

CPC classification number: A01N57/12 ,  C07F9/1651

Abstract: DIALKYLSULFOXIMINOCARBONYLMETHYL THIOPHOSPHATES HAVING THE FORMULA

R1-O-P(=X)(-O-R2)-S-CH2-CO-N=S(=O)(-R3)-R4

WHEREIN R1, R2, R3 AND R4 ARE ALKYL HAVING FROM 1 TO 7 CARBON ATOMS AND X REPRESENTS A MEMBER SELECTED FROM THE GROUP CONSISTING OF OXYGEN AND SULFUR; THE PROCESS OF MANUFACTURE, PESTICIDAL COMPOSITIONS AND THE ACARICIDAL METHOD. THE SAID THIOPHOSPHATES POSSESS ACARICIDAL PROPERTIES.